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—— 5-ethyl-N-[(2R)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]-1H-pyrazole-3-carboxamide —— C13H22N4O2
5-ethyl-N-[(2R)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(2S)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]-1H-pyrazole-3-carboxamide —— C13H22N4O2
5-ethyl-N-[(2S)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-(methoxymethyl)-N-[(2S)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]furan-2-carboxamide —— C14H22N2O4
5-(methoxymethyl)-N-[(2S)-4-methyl-1-(methylamino)-1-oxopentan-2-yl]furan-2-carboxamide
—— 5-[(1R)-1-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C23H21N7OS
5-[(1R)-1-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1S)-1-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C21H21N7S
5-[(1S)-1-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1R)-1-[[4-(furan-2-ylmethyl)-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C23H21N7OS
5-[(1R)-1-[[4-(furan-2-ylmethyl)-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1S)-1-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C23H21N7OS
5-[(1S)-1-[[4-(furan-2-ylmethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1R)-1-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C21H21N7S
5-[(1R)-1-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1R)-1-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-1-phenyltetrazole —— C23H19N7S
5-[(1R)-1-[(4,5-diphenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1R)-1-[(2-methylphenyl)methylsulfanyl]ethyl]-1-phenyltetrazole —— C17H18N4S
5-[(1R)-1-[(2-methylphenyl)methylsulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(1R)-1-[[4-methyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C19H19N7S
5-[(1R)-1-[[4-methyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-N-(3-methoxypropyl)-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide —— C22H30N4O4
5-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-N-(3-methoxypropyl)-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide
—— 5-[(1S)-1-[[4-(furan-2-ylmethyl)-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole —— C23H21N7OS
5-[(1S)-1-[[4-(furan-2-ylmethyl)-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1-phenyltetrazole
—— 5-ethyl-N-[(1S)-1-[3-methoxy-4-(2-methoxyethoxy)phenyl]ethyl]-1H-pyrazole-3-carboxamide —— C18H25N3O4
5-ethyl-N-[(1S)-1-[3-methoxy-4-(2-methoxyethoxy)phenyl]ethyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[[3-[[(2R)-2-methylbutanoyl]amino]phenyl]methyl]-1H-pyrazole-3-carboxamide —— C18H24N4O2
5-ethyl-N-[[3-[[(2R)-2-methylbutanoyl]amino]phenyl]methyl]-1H-pyrazole-3-carboxamide
—— 5-(methoxymethyl)-N-[[3-[[(2R)-2-methylbutanoyl]amino]phenyl]methyl]furan-2-carboxamide —— C19H24N2O4
5-(methoxymethyl)-N-[[3-[[(2R)-2-methylbutanoyl]amino]phenyl]methyl]furan-2-carboxamide
—— 5-ethyl-N-[(1R)-1-[3-methoxy-4-(2-methoxyethoxy)phenyl]ethyl]-1H-pyrazole-3-carboxamide —— C18H25N3O4
5-ethyl-N-[(1R)-1-[3-methoxy-4-(2-methoxyethoxy)phenyl]ethyl]-1H-pyrazole-3-carboxamide
—— 5-(methoxymethyl)-N-[[3-[[(2S)-2-methylbutanoyl]amino]phenyl]methyl]furan-2-carboxamide —— C19H24N2O4
5-(methoxymethyl)-N-[[3-[[(2S)-2-methylbutanoyl]amino]phenyl]methyl]furan-2-carboxamide
—— 5-ethyl-N-[[3-[[(2S)-2-methylbutanoyl]amino]phenyl]methyl]-1H-pyrazole-3-carboxamide —— C18H24N4O2
5-ethyl-N-[[3-[[(2S)-2-methylbutanoyl]amino]phenyl]methyl]-1H-pyrazole-3-carboxamide
—— 5-(3-imidazol-1-ylpropyl)-3-[(3S)-oxolan-3-yl]-1-propyl-1,2,4-triazole —— C15H23N5O
5-(3-imidazol-1-ylpropyl)-3-[(3S)-oxolan-3-yl]-1-propyl-1,2,4-triazole
—— 5-ethyl-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]-1H-pyrazole-3-carboxamide —— C18H22N4O2
5-ethyl-N-[(1S)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]-1H-pyrazole-3-carboxamide —— C18H22N4O2
5-ethyl-N-[(1R)-2-(2-oxopyrrolidin-1-yl)-1-phenylethyl]-1H-pyrazole-3-carboxamide
—— 5-ethyl-N-[(2R)-2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide —— C21H29N3O2
5-ethyl-N-[(2R)-2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5-chloro-1H-indol-2-yl)-[(6R)-6-hydroxy-4-methyl-1,4-diazepan-1-yl]methanone —— C15H18ClN3O2
(5-chloro-1H-indol-2-yl)-[(6R)-6-hydroxy-4-methyl-1,4-diazepan-1-yl]methanone
—— [(5S)-9-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C23H30FN3O
[(5S)-9-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— [5-[[(2S)-2-(1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol —— C22H27N3O2
[5-[[(2S)-2-(1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol
—— 5-(3-imidazol-1-ylpropyl)-3-[(3R)-oxolan-3-yl]-1-propyl-1,2,4-triazole —— C15H23N5O
5-(3-imidazol-1-ylpropyl)-3-[(3R)-oxolan-3-yl]-1-propyl-1,2,4-triazole
—— 5-ethyl-N-[(2S)-2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide —— C21H29N3O2
5-ethyl-N-[(2S)-2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
—— [5-[[(2R)-2-(1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol —— C22H27N3O2
[5-[[(2R)-2-(1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol
—— 5-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide —— C27H34N6O2
5-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide
—— (5-chloro-1H-indol-2-yl)-[(6S)-6-hydroxy-4-methyl-1,4-diazepan-1-yl]methanone —— C15H18ClN3O2
(5-chloro-1H-indol-2-yl)-[(6S)-6-hydroxy-4-methyl-1,4-diazepan-1-yl]methanone
—— [(5R)-5-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(oxan-4-yl)methanone —— C20H32N4O3
[(5R)-5-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(oxan-4-yl)methanone
—— [(5R)-9-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol —— C23H30FN3O
[(5R)-9-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-5-yl]methanol
—— 5-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide —— C29H37N5O2
5-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-3-carboxamide
—— [(5S)-5-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(oxan-4-yl)methanone —— C20H32N4O3
[(5S)-5-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-(oxan-4-yl)methanone
—— 5-tert-butyl-N-[3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]propyl]-1H-pyrazole-3-carboxamide —— C18H32N4O
5-tert-butyl-N-[3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]propyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-1H-pyrazole-3-carboxamide —— C18H32N4O
5-tert-butyl-N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-1H-pyrazole-3-carboxamide
—— [5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-4-ylpyrrolidin-1-yl]methanone —— C17H22N4O
[5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-4-ylpyrrolidin-1-yl]methanone
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(2R)-2-pyridin-4-ylpyrrolidin-1-yl]methanone —— C17H22N4O
(5-tert-butyl-1H-pyrazol-3-yl)-[(2R)-2-pyridin-4-ylpyrrolidin-1-yl]methanone
—— [5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2R)-2-pyridin-4-ylpyrrolidin-1-yl]methanone —— C17H22N4O
[5-(2-methylpropyl)-1H-pyrazol-3-yl]-[(2R)-2-pyridin-4-ylpyrrolidin-1-yl]methanone
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(2S)-2-pyridin-4-ylpyrrolidin-1-yl]methanone —— C17H22N4O
(5-tert-butyl-1H-pyrazol-3-yl)-[(2S)-2-pyridin-4-ylpyrrolidin-1-yl]methanone
—— 5-tert-butyl-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-1H-pyrazole-3-carboxamide —— C17H21N3O2
5-tert-butyl-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-3-carboxamide —— C18H33N5O
5-tert-butyl-N-[(2R)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-3-carboxamide —— C18H33N5O
5-tert-butyl-N-[(2S)-3-methyl-2-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2S)-2-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)propyl]-1H-pyrazole-3-carboxamide —— C18H26N4OS
5-tert-butyl-N-[(2S)-2-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)propyl]-1H-pyrazole-3-carboxamide
—— 5-bromo-N-[(2S)-2-(diethylamino)-4-methylpentyl]furan-3-carboxamide —— C15H25BrN2O2
5-bromo-N-[(2S)-2-(diethylamino)-4-methylpentyl]furan-3-carboxamide
—— 5-tert-butyl-N-[(2R)-2-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)propyl]-1H-pyrazole-3-carboxamide —— C18H26N4OS
5-tert-butyl-N-[(2R)-2-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)propyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide —— C21H30N4O2
5-tert-butyl-N-[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-tert-butyl-N-[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide —— C21H30N4O2
5-tert-butyl-N-[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-bromo-N-[(2R)-2-(diethylamino)-4-methylpentyl]furan-3-carboxamide —— C15H25BrN2O2
5-bromo-N-[(2R)-2-(diethylamino)-4-methylpentyl]furan-3-carboxamide