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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-methoxy-2-(1H-pyrazol-1-yl)phenol 1616057-74-9 C10H10N2O2
3-methoxy-2-(1H-pyrazol-1-yl)phenol
—— 2-phenyl-5-trifluoromethyl-oxazole-4-carboxylic acid (6-bromo-pyridin-3-yl)-amide 1085841-97-9 C16H9BrF3N3O2
2-phenyl-5-trifluoromethyl-oxazole-4-carboxylic acid (6-bromo-pyridin-3-yl)-amide
—— [2-(1H-tetrazol-5-yl)phenoxy]acetic acid 893770-65-5 C9H8N4O3
[2-(1H-tetrazol-5-yl)phenoxy]acetic acid
—— 5-{3-[2-chloro-4-({4-[(1-methylethyl)amino]butyl}oxy)phenyl]-1,2,4-oxadiazol-5-yl}-2-[(1-methylethyl)oxy]benzonitrile 1259517-21-9 C25H29ClN4O3
5-{3-[2-chloro-4-({4-[(1-methylethyl)amino]butyl}oxy)phenyl]-1,2,4-oxadiazol-5-yl}-2-[(1-methylethyl)oxy]benzonitrile
—— (S)-N-(3-(2-ethyl-6-methyl-4-(5-(6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl)phenoxy)-2-hydroxypropyl)-2-hydroxyacetamide 1516901-63-5 C22H26N4O5
(S)-N-(3-(2-ethyl-6-methyl-4-(5-(6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl)phenoxy)-2-hydroxypropyl)-2-hydroxyacetamide
—— N-3-[5-(2-methyl-6-[(2-morpholinoethyl)amino]-4-pyrimidinylamino)-1H-3-pyrazolyl]phenyl-1-benzenesulfonamide 1327167-12-3 C26H30N8O3S
N-3-[5-(2-methyl-6-[(2-morpholinoethyl)amino]-4-pyrimidinylamino)-1H-3-pyrazolyl]phenyl-1-benzenesulfonamide
—— 1-phenylpyrazolo[4',3':5,6]pyrano[3,2-c]pyridin-4(1H)-one 929569-04-0 C15H9N3O2
1-phenylpyrazolo[4',3':5,6]pyrano[3,2-c]pyridin-4(1H)-one
—— 2-(1-(5-(2-(piperidin-1-yl)-4-(trifluoromethyl)oxazole-5-carboxamido)pyridin-2-yl)piperidin-4-yl)acetic acid 1228001-75-9 C22H26F3N5O4
2-(1-(5-(2-(piperidin-1-yl)-4-(trifluoromethyl)oxazole-5-carboxamido)pyridin-2-yl)piperidin-4-yl)acetic acid
—— Ro 41-1049 127917-66-2 C12H12FN3OS*ClH
Ro 41-1049
—— Ethyl 5-(6-methylpyridin-3-yl)-1,3-oxazole-4-carboxylate 136591-86-1 C12H12N2O3
Ethyl 5-(6-methylpyridin-3-yl)-1,3-oxazole-4-carboxylate
—— {4-[3-(3-amino-2,6-difluoro-phenyl)-1H-pyrazol-4-yl]-pyridin-2-yl}-methyl-amine 1206835-69-9 C15H13F2N5
{4-[3-(3-amino-2,6-difluoro-phenyl)-1H-pyrazol-4-yl]-pyridin-2-yl}-methyl-amine
—— 5-(3-{4-[(4-bromobutyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259518-13-2 C24H26BrN3O3
5-(3-{4-[(4-bromobutyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(2-chloro-4-{[4-(ethylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-23-1 C24H27ClN4O3
5-[3-(2-chloro-4-{[4-(ethylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 5-(3-{4-[(2-bromoethyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259518-08-5 C22H22BrN3O3
5-(3-{4-[(2-bromoethyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 1-methyl-4-phenyl-3-(trifluoromethyl)-1H-pyrazole 96256-50-7 C11H9F3N2
1-methyl-4-phenyl-3-(trifluoromethyl)-1H-pyrazole
—— (3-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}propyl)methylamine 1259517-38-8 C23H28ClN3O3
(3-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}propyl)methylamine
—— 5-(3-{4-[(2-bromoethyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259518-11-0 C20H17BrClN3O3
5-(3-{4-[(2-bromoethyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(Cyclopentylamino)-6-phenoxy-imidazo[1,2-a]pyridin-2-yl]-2-methoxy-phenol 1187590-36-8 C25H25N3O3
5-[3-(Cyclopentylamino)-6-phenoxy-imidazo[1,2-a]pyridin-2-yl]-2-methoxy-phenol
—— 2-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-methylphenyl]oxy}-N-methylethanamine 1259517-08-2 C21H24ClN3O3
2-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-methylphenyl]oxy}-N-methylethanamine
—— 5-[3-(2-chloro-4-{[4-(propylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-22-0 C25H29ClN4O3
5-[3-(2-chloro-4-{[4-(propylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(2-ethyl-4-{[2-(methylamino)ethyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-36-6 C23H26N4O3
5-[3-(2-ethyl-4-{[2-(methylamino)ethyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(2-ethyl-4-{[4-(methylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-41-3 C25H30N4O3
5-[3-(2-ethyl-4-{[4-(methylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 3-{4-[(3-bromopropyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole 1259518-10-9 C22H24BrClN2O3
3-{4-[(3-bromopropyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole
—— 5-[3-(2-chloro-4-{[4-(dimethylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-20-8 C24H27ClN4O3
5-[3-(2-chloro-4-{[4-(dimethylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— N-3-[5-(2-methyl-6-[(3-morpholinopropyl)amino]-4-pyrimidinylamino)-1H-3-pyrazolyl]phenyl-1-benzenesulfonamide 1327167-13-4 C27H32N8O3S
N-3-[5-(2-methyl-6-[(3-morpholinopropyl)amino]-4-pyrimidinylamino)-1H-3-pyrazolyl]phenyl-1-benzenesulfonamide
—— 5-(3-{4-[(3-bromopropyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259518-12-1 C21H19BrClN3O3
5-(3-{4-[(3-bromopropyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 2-(4-chlorophenyl)-3-(hydroxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide 1228303-48-7 C22H25ClN4O2
2-(4-chlorophenyl)-3-(hydroxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— 2-phenoxy-6-N-[4-(trifluoromethoxy)phenyl]-4-N-[1-[3-(trifluoromethyl)phenyl]imidazol-2-yl]pyrimidine-4,6-diamine 1238312-53-2 C27H18F6N6O2
2-phenoxy-6-N-[4-(trifluoromethoxy)phenyl]-4-N-[1-[3-(trifluoromethyl)phenyl]imidazol-2-yl]pyrimidine-4,6-diamine
—— N-[3-(5-[6-(4-hydroxypiperidino)-2-methyl-4-pyrimidinyl]amino-1H-3-pyrazolyl)phenyl]-1-benzenesulfonamide 1327167-09-8 C25H27N7O3S
N-[3-(5-[6-(4-hydroxypiperidino)-2-methyl-4-pyrimidinyl]amino-1H-3-pyrazolyl)phenyl]-1-benzenesulfonamide
—— (2-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}ethyl)methylamine 1259517-29-7 C22H26ClN3O3
(2-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}ethyl)methylamine
—— 5-[3-(2-chloro-4-{[4-(methylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-24-2 C23H25ClN4O3
5-[3-(2-chloro-4-{[4-(methylamino)butyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— (3-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-methylphenyl]oxy}propyl)methylamine 1259517-43-5 C22H26ClN3O3
(3-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-methylphenyl]oxy}propyl)methylamine
—— N-(3-(5-[(6-[2-(dimethylamino)ethyl]amino-2-methyl-4-pyrimidinyl)amino]-1H-3-pyrazolyl)phenyl)-1-benzenesulfonamide 1327167-11-2 C24H28N8O2S
N-(3-(5-[(6-[2-(dimethylamino)ethyl]amino-2-methyl-4-pyrimidinyl)amino]-1H-3-pyrazolyl)phenyl)-1-benzenesulfonamide
—— 3-{4-[(4-bromobutyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole 1259518-09-6 C23H26BrClN2O3
3-{4-[(4-bromobutyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole
—— 5-(3-{4-[(4-bromobutyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259517-90-2 C22H21BrClN3O3
5-(3-{4-[(4-bromobutyl)oxy]-2-chlorophenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 5-(3-{4-[(3-bromopropyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile 1259518-14-3 C23H24BrN3O3
5-(3-{4-[(3-bromopropyl)oxy]-2-ethylphenyl}-1,2,4-oxadiazol-5-yl)-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(2-chloro-4-{[2-(methylamino)ethyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-39-9 C21H21ClN4O3
5-[3-(2-chloro-4-{[2-(methylamino)ethyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 3-{4-[(2-bromoethyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole 1259517-99-1 C21H22BrClN2O3
3-{4-[(2-bromoethyl)oxy]-2-ethylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole
—— 3-{4-[(2-bromoethyl)oxy]-2-methylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-l,2,4-oxadiazole 1259517-54-8 C20H20BrClN2O3
3-{4-[(2-bromoethyl)oxy]-2-methylphenyl}-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-l,2,4-oxadiazole
—— 5-[3-(2-ethyl-4-{[3-(methylamino)propyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile 1259517-42-4 C24H28N4O3
5-[3-(2-ethyl-4-{[3-(methylamino)propyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2-[(1-methylethyl)oxy]benzonitrile
—— 5-[3-(2-chloro-4-{[3-(methylamino)propyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2[(1-methylethyl)oxy]benzonitrile 1259517-40-2 C22H23ClN4O3
5-[3-(2-chloro-4-{[3-(methylamino)propyl]oxy}phenyl)-1,2,4-oxadiazol-5-yl]-2[(1-methylethyl)oxy]benzonitrile
—— 3-(4-[(3-bromopropyl)oxy]-2-methylphenyl)-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole 1259518-16-5 C21H22BrClN2O3
3-(4-[(3-bromopropyl)oxy]-2-methylphenyl)-5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazole
—— (4-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}butyl)methylamine 1259517-37-7 C24H30ClN3O3
(4-{[4-(5-{3-chloro-4-[(1-methylethyl)oxy]phenyl}-1,2,4-oxadiazol-3-yl)-3-ethylphenyl]oxy}butyl)methylamine
—— (S)-3-{[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-3-(2-methanesulfonyl-pyridin-4-yl)-propionic acid 1220166-17-5 C22H18FN5O5S
(S)-3-{[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-3-(2-methanesulfonyl-pyridin-4-yl)-propionic acid
—— (S)-3-{[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-3-(2-methanesulfonyl-pyridin-4-yl)-propionic acid methyl ester 1220169-83-4 C23H20FN5O5S
(S)-3-{[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-3-(2-methanesulfonyl-pyridin-4-yl)-propionic acid methyl ester
—— [2-(4-chlorophenyl)-6-(morpholin-4-ylcarbonyl)imidazo[1,2-a]pyridin-3-yl]methanol 1228303-45-4 C19H18ClN3O3
[2-(4-chlorophenyl)-6-(morpholin-4-ylcarbonyl)imidazo[1,2-a]pyridin-3-yl]methanol
—— {2-(4-chlorophenyl)-6-[(4-methoxypiperidin-1-yl)carbonyl]imidazo[1,2-a]pyridin-3-yl}methanol 1228303-42-1 C21H22ClN3O3
{2-(4-chlorophenyl)-6-[(4-methoxypiperidin-1-yl)carbonyl]imidazo[1,2-a]pyridin-3-yl}methanol
—— 1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [(S)-1-(2-methanesulfonyl-6-methylamino-pyridin-4-yl)-propyl]-amide 1220167-96-3 C23H23FN6O3S
1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [(S)-1-(2-methanesulfonyl-6-methylamino-pyridin-4-yl)-propyl]-amide
—— 1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [(S)-1-(2-methanesulfonyl-pyridin-4-yl)-2-methylcarbamoyl-ethyl]-amide 1220169-85-6 C23H21FN6O4S
1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [(S)-1-(2-methanesulfonyl-pyridin-4-yl)-2-methylcarbamoyl-ethyl]-amide
—— 1-{[2-(4-chlorophenyl)-3-(hydroxymethyl)imidazo[1,2-a]pyridin-6-yl]carbonyl}pyrrolidin-3-ol 1228303-59-0 C19H18ClN3O3
1-{[2-(4-chlorophenyl)-3-(hydroxymethyl)imidazo[1,2-a]pyridin-6-yl]carbonyl}pyrrolidin-3-ol