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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]ethanone 1440952-15-7 C25H24FN5OS
1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-fluoro-3-methylphenyl)-5-phenylpyrazol-1-yl]ethanone
—— 3-[5-(1-methyl-5-{[(5-methylpyridin-2-yl)oxy]methyl}-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide 1359027-93-2 C19H18N6O4S
3-[5-(1-methyl-5-{[(5-methylpyridin-2-yl)oxy]methyl}-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
—— (2S)-2-[1-(2-chloro-6-cyano-phenyl)pyrazolo[3,4-d]pyrimidin-4-yl]oxy-N-(5-chloro-2-pyridyl)-3-(3-hydroxyazetidin-1-yl)propanamide 1207830-95-2 C23H18Cl2N8O3
(2S)-2-[1-(2-chloro-6-cyano-phenyl)pyrazolo[3,4-d]pyrimidin-4-yl]oxy-N-(5-chloro-2-pyridyl)-3-(3-hydroxyazetidin-1-yl)propanamide
—— 2-[2-(4-chloro-phenyl)-oxazol-4-yl]-ethanol 27473-19-4 C11H10ClNO2
2-[2-(4-chloro-phenyl)-oxazol-4-yl]-ethanol
—— Acetic acid 2-methoxy-4-(2-phenyl-5-p-tolyl-2H-pyrazol-3-yl)-phenyl ester 76455-77-1 C25H22N2O3
Acetic acid 2-methoxy-4-(2-phenyl-5-p-tolyl-2H-pyrazol-3-yl)-phenyl ester
—— 5-(but-3-ynyl)-3-(2-(trifluoromethyl)phenyl)-1,2,4-oxadiazole 872362-56-6 C13H9F3N2O
5-(but-3-ynyl)-3-(2-(trifluoromethyl)phenyl)-1,2,4-oxadiazole
—— 1-methyl-3-(5-(1-methyl-1H-pyrazol-5-yl)-4-(2,4,6-trifluorophenoxy)pyridin-2-yl)urea 1442666-45-6 C17H14F3N5O2
1-methyl-3-(5-(1-methyl-1H-pyrazol-5-yl)-4-(2,4,6-trifluorophenoxy)pyridin-2-yl)urea
—— 1-[2-({[3-chloro-5-fluoro-4-({[5-{1-[4-fluoro-3-(methyloxy)phenyl]-1-methylethyl}-1-(4-fluorophenyl)-1H-imidazol-2-yl]thio}methyl)phenyl]carbonyl}amino)ethyl]-4-aza-1-azoniabicyclo[2.2.2]octane chloride 1311371-08-0 C35H38ClF3N5O2S*Cl
1-[2-({[3-chloro-5-fluoro-4-({[5-{1-[4-fluoro-3-(methyloxy)phenyl]-1-methylethyl}-1-(4-fluorophenyl)-1H-imidazol-2-yl]thio}methyl)phenyl]carbonyl}amino)ethyl]-4-aza-1-azoniabicyclo[2.2.2]octane chloride
—— 1354909-08-2 C22H20ClFN2O4
—— 1-(3-tert-butyl-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)-2,2-dimethylpropan-1-one 932727-51-0 C18H26N2O
1-(3-tert-butyl-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl)-2,2-dimethylpropan-1-one
—— 2-(β-Piperidinoethylamino)-4-(2'-thienyl)-thiazol 33853-34-8 C14H19N3S2
2-(β-Piperidinoethylamino)-4-(2'-thienyl)-thiazol
—— 1-(3-fluorophenyl)-N-[(3S)-1-pyrrolo[1,2-a]pyrazin-1-ylpyrrolidin-3-yl]pyrazole-3-carboxamide 1613021-56-9 C21H19FN6O
1-(3-fluorophenyl)-N-[(3S)-1-pyrrolo[1,2-a]pyrazin-1-ylpyrrolidin-3-yl]pyrazole-3-carboxamide
—— ethyl 2-methyl-1'-[4-(trifluoromethyl)phenyl]-1'H,2H-3,4'-bipyrazole-4-carboxylate 1359029-63-2 C17H15F3N4O2
ethyl 2-methyl-1'-[4-(trifluoromethyl)phenyl]-1'H,2H-3,4'-bipyrazole-4-carboxylate
—— 2-[(1S)-1-({[2-(methoxycarbonyl)-3-thienyl]sulfonyl}amino)-7-oxooctyl]-5-phenyl-1H-imidazol-3-ium trifluoroacetate 891260-21-2 C2HF3O2*C23H27N3O5S2
2-[(1S)-1-({[2-(methoxycarbonyl)-3-thienyl]sulfonyl}amino)-7-oxooctyl]-5-phenyl-1H-imidazol-3-ium trifluoroacetate
—— 2-[3-(4-Fluoro-3-methylphenyl)-5-methyl-1,2,4-triazol-1-yl]acetic acid 1443257-55-3 C12H12FN3O2
2-[3-(4-Fluoro-3-methylphenyl)-5-methyl-1,2,4-triazol-1-yl]acetic acid
—— 2-[5-Ethyl-3-(4-fluoro-3-methylphenyl)pyrazol-1-yl]-1-(2-methyl-4,5,7,8-tetrahydro-[1,3]oxazolo[4,5-d]azepin-6-yl)ethanone 1440952-60-2 C22H25FN4O2
2-[5-Ethyl-3-(4-fluoro-3-methylphenyl)pyrazol-1-yl]-1-(2-methyl-4,5,7,8-tetrahydro-[1,3]oxazolo[4,5-d]azepin-6-yl)ethanone
—— 2-ethylamino-5-((6-(4-bromophenyl)imidazo[2,1-b]thiazol-3-yl)methyl)-1,3,4-thiadiazole 1212415-59-2 C16H14BrN5S2
2-ethylamino-5-((6-(4-bromophenyl)imidazo[2,1-b]thiazol-3-yl)methyl)-1,3,4-thiadiazole
—— tert-butyl 3-[({4-[7-(aminocarbonyl)-2H-indazol-2-yl]benzyl}amino)carbonyl]azetidine-1-carboxylate 952479-89-9 C24H27N5O4
tert-butyl 3-[({4-[7-(aminocarbonyl)-2H-indazol-2-yl]benzyl}amino)carbonyl]azetidine-1-carboxylate
—— 3-[4-(4-Methoxy-phenyl)-1H-imidazol-2-yl]-benzylamine hydrochloride 321196-72-9 C17H17N3O*ClH
3-[4-(4-Methoxy-phenyl)-1H-imidazol-2-yl]-benzylamine hydrochloride
—— 2-[4-(1-Methylethoxy)phenyl]-3-[(4-methyl-1-piperazinyl)methyl]imidazo[1,2-a]pyridin-6-amine 1216474-78-0 C22H29N5O
2-[4-(1-Methylethoxy)phenyl]-3-[(4-methyl-1-piperazinyl)methyl]imidazo[1,2-a]pyridin-6-amine
—— 1-(3,5-dimethoxybenzoyl)-3-({5-[4-(trifluoromethyl)phenyl]-2H-tetrazol-2-yl}methyl)azetidine-3-carboxylic acid 1154098-65-3 C22H20F3N5O5
1-(3,5-dimethoxybenzoyl)-3-({5-[4-(trifluoromethyl)phenyl]-2H-tetrazol-2-yl}methyl)azetidine-3-carboxylic acid
—— 1242559-28-9 C23H22ClFN4O2
—— 3-[2-(4-chloro-phenyl)-2H-pyrazol-3-yl]-1-(3-trifluoromethoxy-phenyl)-1H-pyridazin-4-one 1228532-70-4 C20H12ClF3N4O2
3-[2-(4-chloro-phenyl)-2H-pyrazol-3-yl]-1-(3-trifluoromethoxy-phenyl)-1H-pyridazin-4-one
—— 4-[1-ethyl-3-(4-nitrophenyl)-1H-pyrazol-4-yl]-N-[2-(4-morpholinyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide 942920-56-1 C25H27N7O4
4-[1-ethyl-3-(4-nitrophenyl)-1H-pyrazol-4-yl]-N-[2-(4-morpholinyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
—— 4-methyl-5-oxazol-4-yl-2,4-dihydro[1,2,4]triazol-3-one 1182358-76-4 C6H6N4O2
4-methyl-5-oxazol-4-yl-2,4-dihydro[1,2,4]triazol-3-one
—— 4-{[4-(3-chloro-4-cyanophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]methyl}-2-fluorobenzamide 1126772-42-6 C20H16ClFN4O
4-{[4-(3-chloro-4-cyanophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]methyl}-2-fluorobenzamide
—— N-tert-butyl-3-{[1-(3-chloro-4-cyanophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}benzamide 1189137-52-7 C24H25ClN4O
N-tert-butyl-3-{[1-(3-chloro-4-cyanophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}benzamide
—— 4-{3,5-dimethyl-4-[(2,4,6-trifluorophenoxy)methyl]-1H-pyrazol-1-yl}benzonitrile 1189136-03-5 C19H14F3N3O
4-{3,5-dimethyl-4-[(2,4,6-trifluorophenoxy)methyl]-1H-pyrazol-1-yl}benzonitrile
—— (R)-ethyl 2-(3-(4-fluorobenzyl)-5-methyl-2-oxoimidazolidin-1-yl)-4-methylthiazole-5-carboxylate 1184958-39-1 C18H20FN3O3S
(R)-ethyl 2-(3-(4-fluorobenzyl)-5-methyl-2-oxoimidazolidin-1-yl)-4-methylthiazole-5-carboxylate
—— 4-{1-[3-(benzyloxy)benzyl]-3,5-dimethyl-1H-pyrazol-4-yl}-2-chlorobenzonitrile 1126776-00-8 C26H22ClN3O
4-{1-[3-(benzyloxy)benzyl]-3,5-dimethyl-1H-pyrazol-4-yl}-2-chlorobenzonitrile
—— 4-(3,5-dimethyl-4-{[(3,5,6-trifluoropyridin-2-yl)oxy]methyl}-1H-pyrazol-1-yl)benzonitrile 1189136-08-0 C18H13F3N4O
4-(3,5-dimethyl-4-{[(3,5,6-trifluoropyridin-2-yl)oxy]methyl}-1H-pyrazol-1-yl)benzonitrile
—— 1469778-83-3 C28H23BrN6O
—— 3-<4-Methoxy-phenyl>-5-<4-(1,3-diphenyl-pyrazol-5-yl)-stilben-4'-yl>-<1.2.4>oxadiazol 71944-59-7 C38H28N4O2
3-<4-Methoxy-phenyl>-5-<4-(1,3-diphenyl-pyrazol-5-yl)-stilben-4'-yl>-<1.2.4>oxadiazol
—— (2E)-3-(2-Dibenzylamino-4-phenyl-5-thiazolyl)acrylsaeure-methylester 139564-84-4 C27H24N2O2S
(2E)-3-(2-Dibenzylamino-4-phenyl-5-thiazolyl)acrylsaeure-methylester
—— (1R,2R)-1-(6-fluoro-1-phenyl-1H-benzoimidazol-2-yl)-1-(7H-purin-6-ylamino)propan-2-ol 1393181-17-3 C21H18FN7O
(1R,2R)-1-(6-fluoro-1-phenyl-1H-benzoimidazol-2-yl)-1-(7H-purin-6-ylamino)propan-2-ol
—— (2S)-N-(5-methylpyridin-2-yl)-2-(1-(4-methylthiophen-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)-3-((R)-1-(triisopropylsilyloxy)propan-2-yloxy)propanamide 1207833-60-0 C31H44N6O4SSi
(2S)-N-(5-methylpyridin-2-yl)-2-(1-(4-methylthiophen-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)-3-((R)-1-(triisopropylsilyloxy)propan-2-yloxy)propanamide
—— 2-(3-{4-carbamoyl-5-[3-(4-chlorophenyl)ureido]-1H-imidazol-2-yl}phenoxy)-2-methylpropionic acid 1143506-89-1 C21H20ClN5O5
2-(3-{4-carbamoyl-5-[3-(4-chlorophenyl)ureido]-1H-imidazol-2-yl}phenoxy)-2-methylpropionic acid
—— 2-(3-bromophenyl)-3-{2-[(3-fluorophenyl)amino]-4-pyrimidinyl}-N,N-dimethylpyrazolo[1,5-a]pyridin-7-amine 895637-31-7 C25H20BrFN6
2-(3-bromophenyl)-3-{2-[(3-fluorophenyl)amino]-4-pyrimidinyl}-N,N-dimethylpyrazolo[1,5-a]pyridin-7-amine
—— [3-(2,4-dimethyl-phenyl)-2,6-dimethyl-pyrazolo[5,1-b]oxazol-7-ylmethyl]-dipropyl-amine 1207258-00-1 C22H31N3O
[3-(2,4-dimethyl-phenyl)-2,6-dimethyl-pyrazolo[5,1-b]oxazol-7-ylmethyl]-dipropyl-amine
—— 5-methyl-3-oxo-3<i>H</i>-isothiazole-2-carboxylic acid methylamide 26533-96-0 C6H8N2O2S
5-methyl-3-oxo-3<i>H</i>-isothiazole-2-carboxylic acid methylamide
—— 4-methyl-pyridine-2-carboxylic acid {1-[1-benzyl-5-(4-fluoro-phenyl)-1H-[1,2,4]triazol-3-ylcarbamoyl]-1-methyl-ethyl}-amide 1205602-41-0 C26H25FN6O2
4-methyl-pyridine-2-carboxylic acid {1-[1-benzyl-5-(4-fluoro-phenyl)-1H-[1,2,4]triazol-3-ylcarbamoyl]-1-methyl-ethyl}-amide
—— 2-(2,5-diphenyl-2<i>H</i>-[1,2,4]triazol-3-yl)-pentane-1,4-diol 34924-41-9 C19H21N3O2
2-(2,5-diphenyl-2<i>H</i>-[1,2,4]triazol-3-yl)-pentane-1,4-diol
—— 4-(5-phenyl-3-pyridin-2-yl-pyrazol-1-yl)-benzoic acid ethyl ester 37738-33-3 C23H19N3O2
4-(5-phenyl-3-pyridin-2-yl-pyrazol-1-yl)-benzoic acid ethyl ester
—— (R)-4-((4-(5-chloro-2-(6-methoxypyridin-3-yl)phenyl)-5-fluorothiazol-2-yl)(cyclopropyl)amino)-4-oxo-3-((tetrahydro-2H-pyran-4-yl)methyl)butanoic acid 1229368-03-9 C28H29ClFN3O5S
(R)-4-((4-(5-chloro-2-(6-methoxypyridin-3-yl)phenyl)-5-fluorothiazol-2-yl)(cyclopropyl)amino)-4-oxo-3-((tetrahydro-2H-pyran-4-yl)methyl)butanoic acid
—— N-(3-chloro-4-{5-[8-chloro-6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,2,4-oxadiazol-3-yl}phenyl)ethenesulfonamide 1228372-18-6 C18H10Cl2F3N5O3S
N-(3-chloro-4-{5-[8-chloro-6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,2,4-oxadiazol-3-yl}phenyl)ethenesulfonamide
—— (4-methylpiperazin-1-yl){3-[(5-methyl-3-{3-[4-(tetrahydro-2H-pyran-4-yl)phenyl]-1,2,4-oxa-diazol-5-yl}-1H-pyrazol-1-yl)methyl]phenyl}methanone 1227159-40-1 C30H34N6O3
(4-methylpiperazin-1-yl){3-[(5-methyl-3-{3-[4-(tetrahydro-2H-pyran-4-yl)phenyl]-1,2,4-oxa-diazol-5-yl}-1H-pyrazol-1-yl)methyl]phenyl}methanone
—— 5-[1-(2,4-dichloro-benzyl)-1H-[1,2,4]triazol-3-ylamino]-2-(4-methyl-imidazol-1-yl)-benzonitrile 1225444-96-1 C20H15Cl2N7
5-[1-(2,4-dichloro-benzyl)-1H-[1,2,4]triazol-3-ylamino]-2-(4-methyl-imidazol-1-yl)-benzonitrile
—— (2S)-(-)-2-(2-Aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl)propanoic acid 570397-59-0 C11H19N3O3
(2S)-(-)-2-(2-Aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl)propanoic acid
—— 3,5-Bis-(hexan-1-sulfinyl)-4-cyanisothiazol 31891-95-9 C16H26N2O2S3
3,5-Bis-(hexan-1-sulfinyl)-4-cyanisothiazol
—— 3-{3-[5-(adamantan-1-yloxymethyl)-2-cyclohexyl-1H-imidazol-4-yl]-[1,2,4]oxadiazol-5-yl}-benzoic acid methyl ester 373649-36-6 C30H36N4O4
3-{3-[5-(adamantan-1-yloxymethyl)-2-cyclohexyl-1H-imidazol-4-yl]-[1,2,4]oxadiazol-5-yl}-benzoic acid methyl ester