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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4-benzyl-piperazin-1-yl)-(3-methyl-2-nitro-3<i>H</i>-imidazol-4-ylmethylene)-amine 40647-59-4 C16H20N6O2
(4-benzyl-piperazin-1-yl)-(3-methyl-2-nitro-3<i>H</i>-imidazol-4-ylmethylene)-amine
—— [4-(2-methoxy-phenyl)-5-(3,4,5-trimethoxy-phenyl)-4<i>H</i>-[1,2,4]triazol-3-ylsulfanyl]-acetic acid ethyl ester 70452-59-4 C22H25N3O6S
[4-(2-methoxy-phenyl)-5-(3,4,5-trimethoxy-phenyl)-4<i>H</i>-[1,2,4]triazol-3-ylsulfanyl]-acetic acid ethyl ester
—— 4-<4-Chlor-1-(4-chlor-phenyl)-pyrazol-3-yl>-benzaldehyd 71945-35-2 C16H10Cl2N2O
4-<4-Chlor-1-(4-chlor-phenyl)-pyrazol-3-yl>-benzaldehyd
—— 2-Phenyl-3-chlor-7-dibrommethylpyrazol<1,5-a>-pyrimidin-5-carbonsaeure 72197-36-5 C14H8Br2ClN3O2
2-Phenyl-3-chlor-7-dibrommethylpyrazol<1,5-a>-pyrimidin-5-carbonsaeure
—— [2-(3-chloro-phenoxymethyl)-4-methyl-thiazol-5-yl]-acetic acid 59865-75-7 C13H12ClNO3S
[2-(3-chloro-phenoxymethyl)-4-methyl-thiazol-5-yl]-acetic acid
—— 1-(<i>N</i>-<i>tert</i>-butyl-formimidoyl)-2-methyl-1<i>H</i>-imidazole 53630-79-8 C9H15N3
1-(<i>N</i>-<i>tert</i>-butyl-formimidoyl)-2-methyl-1<i>H</i>-imidazole
—— 4-[2-(2-Cyclohexyl-5-methyl-oxazol-4-yl)-ethoxy]-phenylamine 141399-44-2 C18H24N2O2
4-[2-(2-Cyclohexyl-5-methyl-oxazol-4-yl)-ethoxy]-phenylamine
—— 5-[5-(Trifluoromethyl)-3-isoxazolyl]-2-furansulfonyl chloride 1268334-87-7 C8H3ClF3NO4S
5-[5-(Trifluoromethyl)-3-isoxazolyl]-2-furansulfonyl chloride
—— 2-((3S,4R)-4-(3-bromo-4-chloro-5-methyl-1H-pyrrole-2-carboxamido)-3-fluoropiperidin-1-yl)-4-(1-(cyclopropylmethyl)-1H-1,2,4-triazol-5-yl)thiazole-5-carboxylic acid 1229425-70-0 C21H22BrClFN7O3S
2-((3S,4R)-4-(3-bromo-4-chloro-5-methyl-1H-pyrrole-2-carboxamido)-3-fluoropiperidin-1-yl)-4-(1-(cyclopropylmethyl)-1H-1,2,4-triazol-5-yl)thiazole-5-carboxylic acid
—— 2-({[4-({[5-{1-[4-chloro-3-(methyloxy)phenyl]-1-methylethyl}-1-(4-fluorophenyl)-1H-imidazol-2-yl]thio}methyl)-3,5-difluorophenyl]sulfonyl}amino)-N,N,N-triethylethanaminium 2,2,2-trifluoroacetate 1311371-73-9 C2F3O2*C35H43ClF3N4O3S2
2-({[4-({[5-{1-[4-chloro-3-(methyloxy)phenyl]-1-methylethyl}-1-(4-fluorophenyl)-1H-imidazol-2-yl]thio}methyl)-3,5-difluorophenyl]sulfonyl}amino)-N,N,N-triethylethanaminium 2,2,2-trifluoroacetate
—— 1197340-81-0 C20H14F3N5O3S
—— 4-cyano-N-(1-{4-[3-(2-methylpyrrolidin-1-yl)propoxy]phenyl}-1H-pyrazol-4-yl)benzamide 1152748-50-9 C25H27N5O2
4-cyano-N-(1-{4-[3-(2-methylpyrrolidin-1-yl)propoxy]phenyl}-1H-pyrazol-4-yl)benzamide
—— N-(3-{4-[5-(2-dimethylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2,6-dimethyl-phenoxy}-2-hydroxy-propyl)-2-hydroxy-acetamide 1150645-36-5 C22H28N6O5
N-(3-{4-[5-(2-dimethylamino-6-methyl-pyrimidin-4-yl)-[1,2,4]oxadiazol-3-yl]-2,6-dimethyl-phenoxy}-2-hydroxy-propyl)-2-hydroxy-acetamide
—— (1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid [1-(6-methyl-pyridin-2-yl)-ethyl]-amide 1268876-21-6 C22H20F2N4O
(1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid [1-(6-methyl-pyridin-2-yl)-ethyl]-amide
—— 3-(1-methyl-3-trifluoromethyl-1H-pyrazole-5-yl)phenylsulphonic acid N-methyl-N-[4-(3-phenylureido)phenyl]amide 1259029-49-6 C25H22F3N5O3S
3-(1-methyl-3-trifluoromethyl-1H-pyrazole-5-yl)phenylsulphonic acid N-methyl-N-[4-(3-phenylureido)phenyl]amide
—— DHK2-2 1071472-92-8 C25H25N5O3S
DHK2-2
—— (4-phenylamino-5-phenyl-1,2,4-triazol-3-yl)-N-phenyl-benzenecarbothiohydrazonate 1333972-76-1 C27H22N6S
(4-phenylamino-5-phenyl-1,2,4-triazol-3-yl)-N-phenyl-benzenecarbothiohydrazonate
—— (4,5-Diphenyl-1H-imidazol-2-ylsulfanyl)-acetic acid [1-(2-nitro-phenyl)-meth-(E)-ylidene]-hydrazide 129585-76-8 C24H19N5O3S
(4,5-Diphenyl-1H-imidazol-2-ylsulfanyl)-acetic acid [1-(2-nitro-phenyl)-meth-(E)-ylidene]-hydrazide
—— 2-[3-(2-methoxy-ethoxy)-phenyl]-5-phenyl-2<i>H</i>-tetrazole 21423-45-0 C16H16N4O2
2-[3-(2-methoxy-ethoxy)-phenyl]-5-phenyl-2<i>H</i>-tetrazole
—— 5-(3-fluoro-2-methyl-phenyl)-2-methyl-thiazole-4-carboxylic acid 1038509-07-7 C12H10FNO2S
5-(3-fluoro-2-methyl-phenyl)-2-methyl-thiazole-4-carboxylic acid
—— 6-Hydroxy-2,3-dimethyl-5-<3-phenyl-pyrazol-5-yl>-benzofuran 4196-64-9 C19H16N2O2
6-Hydroxy-2,3-dimethyl-5-<3-phenyl-pyrazol-5-yl>-benzofuran
—— 2-butyl-5-[4-methoxy-benzyl-thio]-1H-imidazole-4-carboxylaldehyde 162649-05-0 C16H20N2O2S
2-butyl-5-[4-methoxy-benzyl-thio]-1H-imidazole-4-carboxylaldehyde
—— 7-chloro-2-(4-fluorophenyl)-5-methyloxazolo[5,4-d]pyrimidine 1245318-93-7 C12H7ClFN3O
7-chloro-2-(4-fluorophenyl)-5-methyloxazolo[5,4-d]pyrimidine
—— N-{5-[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2,3-triazol-1-yl]-6-methyl-pyridin-3-yl}-3-[methyl-(1-methyl-pyrrolidin-3-yl)amino]-5-trifluoromethoxy-benzamide 1219947-62-2 C27H30F3N9O2
N-{5-[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2,3-triazol-1-yl]-6-methyl-pyridin-3-yl}-3-[methyl-(1-methyl-pyrrolidin-3-yl)amino]-5-trifluoromethoxy-benzamide
—— 5-(3-methoxyphenyl)-N-((5-phenyl-1H-pyrazol-3-yl)methyl)-1,2,4-triazin-3-amine 1224743-61-6 C20H18N6O
5-(3-methoxyphenyl)-N-((5-phenyl-1H-pyrazol-3-yl)methyl)-1,2,4-triazin-3-amine
—— [5-cyclopropyl-3-methyl-1-(3-trifluoromethoxy-phenyl)-1H-pyrazol-4-yl]-[4-((2R,3S)-3-hydroxy-2-methyl-pyrrolidin-1-yl)-piperidin-1-yl]-methanone 1107658-12-7 C25H31F3N4O3
[5-cyclopropyl-3-methyl-1-(3-trifluoromethoxy-phenyl)-1H-pyrazol-4-yl]-[4-((2R,3S)-3-hydroxy-2-methyl-pyrrolidin-1-yl)-piperidin-1-yl]-methanone
—— [2-(3-hexyl-phenyl)-3-methyl-5-pyridin-4-yl-3H-imidazol-4-yl]-(4-pyrrolidin-1-yl-piperidin-1-yl)-methanone 1097066-97-1 C31H41N5O
[2-(3-hexyl-phenyl)-3-methyl-5-pyridin-4-yl-3H-imidazol-4-yl]-(4-pyrrolidin-1-yl-piperidin-1-yl)-methanone
—— (5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-[4-[2-(3-fluorophenyl)tetrazole-5-carbonyl]-3,3-dimethylpiperazin-1-yl]methanone 1443757-46-7 C23H22ClFN6O4
(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-[4-[2-(3-fluorophenyl)tetrazole-5-carbonyl]-3,3-dimethylpiperazin-1-yl]methanone
—— 4-(3-(4-ethynylphenyl)-1-methyl-1H-pyrazol-4-yl)morpholine 1443362-84-2 C16H17N3O
4-(3-(4-ethynylphenyl)-1-methyl-1H-pyrazol-4-yl)morpholine
—— 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-{(1S,4R)-4-[3-((S)-3-hydroxymethyl-piperidin-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy]-1,2,3,4-tetrahydro-naphthalen-1-yl}-urea 1443240-63-8 C37H44N8O3
1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-{(1S,4R)-4-[3-((S)-3-hydroxymethyl-piperidin-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy]-1,2,3,4-tetrahydro-naphthalen-1-yl}-urea
—— 2-[3-(3-Fluoro-4-methylphenyl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone 1440954-71-1 C24H21FN4OS
2-[3-(3-Fluoro-4-methylphenyl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone
—— 1313819-33-8 C21H25N7O3S
—— 4-(4-ethylphenyl)-1-(3-nitrophenyl)-1H-1,2,3-triazole 1599462-32-4 C16H14N4O2
4-(4-ethylphenyl)-1-(3-nitrophenyl)-1H-1,2,3-triazole
—— 2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-methylpiperidin-1-yl]-4-(pyrazin-2-yl)-1,3-thiazole-5-carboxylic acid 1229571-39-4 C20H20Cl2N6O3S
2-[(3S,4R)-4-{[(3,4-dichloro-5-methyl-1H-pyrrol-2-yl)carbonyl]amino}-3-methylpiperidin-1-yl]-4-(pyrazin-2-yl)-1,3-thiazole-5-carboxylic acid
—— 2-phenyl-3-(trifluoromethyl)benzo[d]imidazo[2,1-b]thiazole 1268167-80-1 C16H9F3N2S
2-phenyl-3-(trifluoromethyl)benzo[d]imidazo[2,1-b]thiazole
—— 2-cyclopropyl-5-(3-fluoro-phenyl)-thiazole-4-carboxylic acid methyl ester 1038508-86-9 C14H12FNO2S
2-cyclopropyl-5-(3-fluoro-phenyl)-thiazole-4-carboxylic acid methyl ester
—— 33533-16-3 C21H24N4OS
—— 3-({(tert-butoxycarbonyl)[(1S,3R)-3-fluorocyclopentyl]amino}methyl)-5-(3,5-difluorophenyl)-4-formyl-1-methyl-1H-pyrazole 932706-35-9 C22H26F3N3O3
3-({(tert-butoxycarbonyl)[(1S,3R)-3-fluorocyclopentyl]amino}methyl)-5-(3,5-difluorophenyl)-4-formyl-1-methyl-1H-pyrazole
—— 5-[(2S,3R)-3-nitro-2-phenylbutyl]sulfonyl-1-phenyltetrazole 1580477-12-8 C17H17N5O4S
5-[(2S,3R)-3-nitro-2-phenylbutyl]sulfonyl-1-phenyltetrazole
—— 1-<i>tert</i>-butylamino-3-{4-[4-(4-chloro-phenyl)-1(3)<i>H</i>-imidazol-2-yl]-phenoxy}-propan-2-ol 60963-67-9 C22H26ClN3O2
1-<i>tert</i>-butylamino-3-{4-[4-(4-chloro-phenyl)-1(3)<i>H</i>-imidazol-2-yl]-phenoxy}-propan-2-ol
—— N-cyclohexyl-N-(2-hydroxyethyl)-4-[4-(1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]benzamide 1383703-28-3 C24H26N6O2
N-cyclohexyl-N-(2-hydroxyethyl)-4-[4-(1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]benzamide
—— 3-cyclohexyl-1-[4-(3,5-dimethyl-pyrazol-1-yl)-benzenesulfonyl]-2-thioxo-imidazolidin-4-one 69203-74-3 C20H24N4O3S2
3-cyclohexyl-1-[4-(3,5-dimethyl-pyrazol-1-yl)-benzenesulfonyl]-2-thioxo-imidazolidin-4-one
—— (2R)-2-phenyl-1-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-phenyl-2-piperidin-1-ylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-piperidin-1-ylethanone 1228965-35-2 C54H58N8O2
(2R)-2-phenyl-1-[(2S)-2-[5-[4-[2-[4-[2-[(2S)-1-[(2R)-2-phenyl-2-piperidin-1-ylacetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]phenyl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-piperidin-1-ylethanone
—— 3-Methyl-4-methylthio-1-phenylpyrazol-5-yl-methylcarbamat 25838-10-2 C13H15N3O2S
3-Methyl-4-methylthio-1-phenylpyrazol-5-yl-methylcarbamat
—— N-[(3R,5R)-1-azabicyclo[3.2.1]oct-3-yl]-5-(2-hydroxyphenyl)-1,3-thiazole-2-carboxamide 524014-02-6 C17H19N3O2S
N-[(3R,5R)-1-azabicyclo[3.2.1]oct-3-yl]-5-(2-hydroxyphenyl)-1,3-thiazole-2-carboxamide
—— 2-[3-[5-(5-phenyl-1H-1,2,4-triazol-3-yl)pyridin-2-yl]-3-azaspiro[5.5]undecan-9-yl]acetic acid 1445205-50-4 C25H29N5O2
2-[3-[5-(5-phenyl-1H-1,2,4-triazol-3-yl)pyridin-2-yl]-3-azaspiro[5.5]undecan-9-yl]acetic acid
—— 4-Amino-N,N-dibenzyl-2-ethylthio-5-thiazolcarboxamid 63238-09-5 C20H21N3OS2
4-Amino-N,N-dibenzyl-2-ethylthio-5-thiazolcarboxamid
—— {1-[4-(6-ethoxy-3-phenyl-imidazo[1,2-a]pyrimidin-2-yl)-phenyl]-cyclobutyl}-carbamic acid tert-butyl ester 1355999-80-2 C29H32N4O3
{1-[4-(6-ethoxy-3-phenyl-imidazo[1,2-a]pyrimidin-2-yl)-phenyl]-cyclobutyl}-carbamic acid tert-butyl ester
—— N-(7-cyclobutyl-3-phenyl-1,2,4-triazolo[4,3-b]pyridazin-6-yl)-N-[3-(imidazol-1-yl)propyl]amine 233278-46-1 C21H23N7
N-(7-cyclobutyl-3-phenyl-1,2,4-triazolo[4,3-b]pyridazin-6-yl)-N-[3-(imidazol-1-yl)propyl]amine
—— (R)-2-[2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-phenyl]-1,4-oxazepan-4-yl]-3-methyl-6-(pyrimidin-4-yl)pyrimidin-4(3H)-one 1246455-03-7 C23H23N7O3
(R)-2-[2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-phenyl]-1,4-oxazepan-4-yl]-3-methyl-6-(pyrimidin-4-yl)pyrimidin-4(3H)-one