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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3R)-7-({2-chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)-1,2,3,4-tetrahydroisoquinolin-3-yl]methanol 1049810-55-0 C32H38ClN5O4S
[(3R)-7-({2-chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)-1,2,3,4-tetrahydroisoquinolin-3-yl]methanol
—— 2-[[(5-methyl-4-phenyl-1H-pyrazol-3-yl)amino]diazenyl]ethanol 82823-56-1 C12H15N5O
2-[[(5-methyl-4-phenyl-1H-pyrazol-3-yl)amino]diazenyl]ethanol
—— 5-(2-methoxy-4-methylpentyl)-1,3-thiazole-4-carboxylic acid 865776-73-4 C11H17NO3S
5-(2-methoxy-4-methylpentyl)-1,3-thiazole-4-carboxylic acid
—— 2-(4-(2-piperidin-1-yl-eth-1-ylamino)-phenyl)-imidazo[1,2-a]-pyridine-8-carboxamide 1092689-76-3 C21H25N5O
2-(4-(2-piperidin-1-yl-eth-1-ylamino)-phenyl)-imidazo[1,2-a]-pyridine-8-carboxamide
—— 2-[3-Phenyl-5-(trifluoromethyl)indazol-1-yl]-1,3-thiazole-4-carboxylic acid 1204771-73-2 C18H10F3N3O2S
2-[3-Phenyl-5-(trifluoromethyl)indazol-1-yl]-1,3-thiazole-4-carboxylic acid
—— 5-(2,6-Dimethoxyphenyl)-1-[4-[N-methyl-N-[3-[N'-methyl-N'-(benzyloxycarbonyl)amino]propyl]carbamoyl]-2-isopropylphenyl]-3-pyrazolecarboxylic acid 184165-32-0 C35H40N4O7
5-(2,6-Dimethoxyphenyl)-1-[4-[N-methyl-N-[3-[N'-methyl-N'-(benzyloxycarbonyl)amino]propyl]carbamoyl]-2-isopropylphenyl]-3-pyrazolecarboxylic acid
—— 8-(4-Chlorobenzyl)-3-mesityl-2,5-dimethyl-7-propyl-8H-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidine 344291-55-0 C29H31ClN4
8-(4-Chlorobenzyl)-3-mesityl-2,5-dimethyl-7-propyl-8H-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidine
—— 2-(3-(2-(5-methyl-2-(furan-2-yl)oxazol-4-yl)ethoxy)phenyl)acetic acid 244152-44-1 C18H17NO5
2-(3-(2-(5-methyl-2-(furan-2-yl)oxazol-4-yl)ethoxy)phenyl)acetic acid
—— N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide 1416309-83-5 C24H34N6O3
N-{5-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-2,2-dimethylcyclohexyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
—— 3-{3-chloro-4-[5-(5-chloro-6-isopropoxypyridin-3-yl)-[1,2,4]oxadiazol-3-yl]-phenoxy}-cyclobutanecarboxylic acid potassium salt 1394000-47-5 C21H18Cl2N3O5*K
3-{3-chloro-4-[5-(5-chloro-6-isopropoxypyridin-3-yl)-[1,2,4]oxadiazol-3-yl]-phenoxy}-cyclobutanecarboxylic acid potassium salt
—— 77584-60-2 C48H42CoN8O6S2
—— 4-ethyl-2-methyl-[1,2,4]oxadiazolidine-3,5-dione 5302-12-5 C5H8N2O3
4-ethyl-2-methyl-[1,2,4]oxadiazolidine-3,5-dione
—— (2RS)-[1-(2-methyl-5-m-tolylthiazole-4-carbonyl)azetidin-2-ylmethyl]carbamic acid tert-butyl ester 1007874-00-1 C21H27N3O3S
(2RS)-[1-(2-methyl-5-m-tolylthiazole-4-carbonyl)azetidin-2-ylmethyl]carbamic acid tert-butyl ester
—— 1-(3-chlorophenyl)-3-[(tetrahydro-2H-pyran-4-ylamino)carbonyl]imidazo[1,5-a]pyridin-2-ium trifluoroacetate 1039350-32-7 C2HF3O2*C19H18ClN3O2
1-(3-chlorophenyl)-3-[(tetrahydro-2H-pyran-4-ylamino)carbonyl]imidazo[1,5-a]pyridin-2-ium trifluoroacetate
—— N-{3-[4-[1-ethyl-3-(4-{[(phenylamino)-carbonyl]amino}phenyl)-1H-pyrazol-4-yl]-1-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl}acetamide 942919-56-4 C39H33N7O4S
N-{3-[4-[1-ethyl-3-(4-{[(phenylamino)-carbonyl]amino}phenyl)-1H-pyrazol-4-yl]-1-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl}acetamide
—— 1-(6,8-dichloro-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-pyrrolidin-2-one 1197847-59-8 C19H17Cl2N3O
1-(6,8-dichloro-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-pyrrolidin-2-one
—— (R)-N-(3,5-dichloro-4-(2-(3,4-difluorobenzylamino)-9-(piperidin-3-ylmethyl)-9H-purin-8-yl)-phenyl)acetamide 1021697-24-4 C26H25Cl2F2N7O
(R)-N-(3,5-dichloro-4-(2-(3,4-difluorobenzylamino)-9-(piperidin-3-ylmethyl)-9H-purin-8-yl)-phenyl)acetamide
—— 1-methyl-3-oxo-2-phenyl-5-(pyrazin-2-yl)-2,3-dihydro-1H-pyrazole-4-carbaldehyde 1361236-23-8 C15H12N4O2
1-methyl-3-oxo-2-phenyl-5-(pyrazin-2-yl)-2,3-dihydro-1H-pyrazole-4-carbaldehyde
—— compound 94 842128-73-8 C26H29N9O
compound 94
—— 4-({4-[2-(tert-butylamino)-4-methyl-1,3-thiazol-5-yl]pyrimidin-2-yl}amino)benzonitrile 930583-74-7 C19H20N6S
4-({4-[2-(tert-butylamino)-4-methyl-1,3-thiazol-5-yl]pyrimidin-2-yl}amino)benzonitrile
—— 1-(4-hydroxyphenyl)-6-[4-(4-methylpiperazin-1-ylmethyl)phenyl]-1,3-dihydroimidazo[4,5-b]pyrazin-2-one 1351477-03-6 C23H24N6O2
1-(4-hydroxyphenyl)-6-[4-(4-methylpiperazin-1-ylmethyl)phenyl]-1,3-dihydroimidazo[4,5-b]pyrazin-2-one
—— 4-(cyclohexylsulfanyl)-1-(2,4-dinitrophenyl)-3-(3-methoxyphenyl)-1H-pyrazole 1309878-24-7 C22H22N4O5S
4-(cyclohexylsulfanyl)-1-(2,4-dinitrophenyl)-3-(3-methoxyphenyl)-1H-pyrazole
—— 6-iodo-5-(4-(2-methoxyethoxy)-4-(1H-tetrazol-5-yl)cyclohexyl)-3-(1-phenyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine 1361450-79-4 C25H27IN10O2
6-iodo-5-(4-(2-methoxyethoxy)-4-(1H-tetrazol-5-yl)cyclohexyl)-3-(1-phenyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(dimethylamino)-3-methyl-N-phenyl-1H-pyrazole-1-carboxamide 1256934-37-8 C13H16N4O
5-(dimethylamino)-3-methyl-N-phenyl-1H-pyrazole-1-carboxamide
—— 2-chloro-4-[3,5-dimethyl-4-(pyridin-3-ylmethoxy)-1H-pyrazol-1-yl]benzonitrile trifluoroacetate 1189139-60-3 C2HF3O2*C18H15ClN4O
2-chloro-4-[3,5-dimethyl-4-(pyridin-3-ylmethoxy)-1H-pyrazol-1-yl]benzonitrile trifluoroacetate
—— (R)-4-(4-methylthiazol-2-yl)oxazolidin-2-one 1269649-51-5 C7H8N2O2S
(R)-4-(4-methylthiazol-2-yl)oxazolidin-2-one
—— (5-trifluoromethyl-[1,3,4]thiadiazol-2-yl)-dithiocarbamic acid ethyl ester 41793-68-4 C6H6F3N3S3
(5-trifluoromethyl-[1,3,4]thiadiazol-2-yl)-dithiocarbamic acid ethyl ester
—— (S)-ethyl 4-(1-(3-(3-chloro-4-cyano-2-methylphenyl)-1H-pyrazol-1-yl)propan-2-ylcarbamoyl)thiazole-2-carboxylate 1297542-04-1 C21H20ClN5O3S
(S)-ethyl 4-(1-(3-(3-chloro-4-cyano-2-methylphenyl)-1H-pyrazol-1-yl)propan-2-ylcarbamoyl)thiazole-2-carboxylate
—— 1-(3,4-dichloro-phenyl)-1H-indazole-4-carboxylic acid [2-(3-trifluoromethyl-phenyl)-ethyl]-amide 1194017-62-3 C23H16Cl2F3N3O
1-(3,4-dichloro-phenyl)-1H-indazole-4-carboxylic acid [2-(3-trifluoromethyl-phenyl)-ethyl]-amide
—— 2-(6-ethoxy-pyridin-3-yl)-pyrimidine-5-carboxylic acid cyclopropyl-[1-(3-phenyl[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]amide 1415835-34-5 C28H29N7O3
2-(6-ethoxy-pyridin-3-yl)-pyrimidine-5-carboxylic acid cyclopropyl-[1-(3-phenyl[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]amide
—— 3,4-Bis-(4-fluoro-phenyl)-1-(toluene-4-sulfonyl)-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one 76058-90-7 C25H19F2N3O3S2
3,4-Bis-(4-fluoro-phenyl)-1-(toluene-4-sulfonyl)-4,8-dihydro-1H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-Phenylthiocarbamoyl-3-methyl-5-<furyl-(2)>-Δ<sup>2</sup>-pyrazolin 109506-09-4 C15H15N3OS
1-Phenylthiocarbamoyl-3-methyl-5-<furyl-(2)>-Δ<sup>2</sup>-pyrazolin
—— 4-benzyl-1-({[4-(4-bromophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)thiosemicarbazide 1355732-91-0 C18H17BrN6OS2
4-benzyl-1-({[4-(4-bromophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)thiosemicarbazide
—— 2-(1-Amino-ethyl)-5-cyclohexylmethylsulfanyl-3-methyl-3H-imidazole-4-carboxylic acid amide 330438-45-4 C14H24N4OS
2-(1-Amino-ethyl)-5-cyclohexylmethylsulfanyl-3-methyl-3H-imidazole-4-carboxylic acid amide
—— 1267583-39-0 C22H18N8
—— 4-[5-Mercapto-4-(4-methoxy-phenyl)-4H-[1,2,4]triazol-3-yl]-2-methoxy-phenol 122772-17-2 C16H15N3O3S
4-[5-Mercapto-4-(4-methoxy-phenyl)-4H-[1,2,4]triazol-3-yl]-2-methoxy-phenol
—— 1-benzyloxymethyl-3-(2-cyanobenzyl)-2-(3-cyclopropoxy-4-difluoromethoxyphenyl)-1,5-dihydropyrrolo[2,3-d]-pyridazin-4-one 944332-19-8 C32H26F2N4O4
1-benzyloxymethyl-3-(2-cyanobenzyl)-2-(3-cyclopropoxy-4-difluoromethoxyphenyl)-1,5-dihydropyrrolo[2,3-d]-pyridazin-4-one
—— 1-benzyloxymethyl-3-(3-cyanobenzyl)-2-(3-cyclopropoxy-4-difluoromethoxyphenyl)-1,5-dihydropyrrolo[2,3-d]-pyridazin-4-one 944332-22-3 C32H26F2N4O4
1-benzyloxymethyl-3-(3-cyanobenzyl)-2-(3-cyclopropoxy-4-difluoromethoxyphenyl)-1,5-dihydropyrrolo[2,3-d]-pyridazin-4-one
—— 1-(3,5-dichloro-4-hydroxyphenyl)-N-(3,4-dichlorobenzyl)-N-(3,3-dimethylbutyl)-1H-1,2,4-triazole-3-carboxamide 1219013-24-7 C22H22Cl4N4O2
1-(3,5-dichloro-4-hydroxyphenyl)-N-(3,4-dichlorobenzyl)-N-(3,3-dimethylbutyl)-1H-1,2,4-triazole-3-carboxamide
—— 5-amino-4-[2',3'-bi(tert-butoxycarbonyl)-guanidino]-1-ethylpyrazole 689293-93-4 C16H28N6O4
5-amino-4-[2',3'-bi(tert-butoxycarbonyl)-guanidino]-1-ethylpyrazole
—— 1-{2-[-5-(4-chlorophenyl)-3-methyl-1H-pyrazol-1-yl]acetyl}-4-(4-methoxyphenyl)thiosemicarbazide 1322724-62-8 C20H20ClN5O2S
1-{2-[-5-(4-chlorophenyl)-3-methyl-1H-pyrazol-1-yl]acetyl}-4-(4-methoxyphenyl)thiosemicarbazide
—— N-(4-methoxyphenyl)-2-{[(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]acetyl}hydrazinecarboselenoamide 1449684-42-7 C26H25N5O2SSe
N-(4-methoxyphenyl)-2-{[(1-methyl-4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]acetyl}hydrazinecarboselenoamide
—— N-(4-(4-chloro-1H-imidazol-1-yl)-3,5-difluorophenyl)-9-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[1,5-a]azepin-2-amine 1235494-39-9 C22H18ClF3N6
N-(4-(4-chloro-1H-imidazol-1-yl)-3,5-difluorophenyl)-9-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[1,5-a]azepin-2-amine
—— 2-cyano-N'-[(1,3-diphenyl-1H-pyrazol-4-yl)methylene]acetohydrazide 864669-72-7 C19H15N5O
2-cyano-N'-[(1,3-diphenyl-1H-pyrazol-4-yl)methylene]acetohydrazide
—— 5-(cyclohexylmethoxy)-1-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazole-4-carboxamide 937743-60-7 C21H36N4O2
5-(cyclohexylmethoxy)-1-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrazole-4-carboxamide
—— 5-(4-Chloro-phenyl)-3-oxo-2-phenyl-3,5-dihydro-2H-pyrazolo[3,4-d]pyridazine-7-carboxylic acid ethyl ester 137201-93-5 C20H15ClN4O3
5-(4-Chloro-phenyl)-3-oxo-2-phenyl-3,5-dihydro-2H-pyrazolo[3,4-d]pyridazine-7-carboxylic acid ethyl ester
—— 3-(4-fluorophenyl)-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-dien-5-carboxylic acid 916591-86-1 C15H13FN2O2
3-(4-fluorophenyl)-3,4-diazatricyclo[5.2.1.0(2,6)]deca-2(6),4-dien-5-carboxylic acid
—— 5-(3-dimethylaminoprop-2-en-1-oyl)-1-cyclopentyl-2-methylimidazole 600699-69-2 C14H21N3O
5-(3-dimethylaminoprop-2-en-1-oyl)-1-cyclopentyl-2-methylimidazole
—— isothiazole-3,4,5-tricarboxylic acid 3-ethyl ester 4,5-dimethyl ester 67049-09-6 C10H11NO6S
isothiazole-3,4,5-tricarboxylic acid 3-ethyl ester 4,5-dimethyl ester
—— 3-({4-[2-(dimethylamino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]pyrimidin-2-yl}amino)phenol 930582-74-4 C16H14F3N5OS
3-({4-[2-(dimethylamino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]pyrimidin-2-yl}amino)phenol