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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[(2-chlorophenyl)carbonyl]-3-(4-fluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazine 1254072-33-7 C18H14ClFN4O
7-[(2-chlorophenyl)carbonyl]-3-(4-fluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazine
—— 6-[3-[2-methoxy-5-(benzoxazole-2-yl)phenyl]-3-(methyl)ureido]hexanoic acid hydroxyamide 738589-18-9 C22H26N4O5
6-[3-[2-methoxy-5-(benzoxazole-2-yl)phenyl]-3-(methyl)ureido]hexanoic acid hydroxyamide
—— 5-methoxycarbonylmethyl-4-methoxycarbonyl-1-methyl-2-oxo-1H,3H-imidazole 155499-52-8 C9H12N2O5
5-methoxycarbonylmethyl-4-methoxycarbonyl-1-methyl-2-oxo-1H,3H-imidazole
—— N-Difluorphosphoryl-pyrrol 54981-23-6 C4H4F2NOP
N-Difluorphosphoryl-pyrrol
—— 10-cyclopentyl-9-ethyl-7-methyl-3-[[3-(4-methyl-1,2,4-triazol-3-yl)phenyl]amino]-2,4,7,9,10-pentazabicyclo[4.4.0]deca-1,3,5-trien-8-one 1018316-25-0 C22H27N9O
10-cyclopentyl-9-ethyl-7-methyl-3-[[3-(4-methyl-1,2,4-triazol-3-yl)phenyl]amino]-2,4,7,9,10-pentazabicyclo[4.4.0]deca-1,3,5-trien-8-one
—— 4-Hydroxy-8-[4-(3,4,5-trichlorophenylaminosulfonyl)phenyl]pyrazolo[1,5-a]-1,3,5-triazine 117413-76-0 C17H10Cl3N5O3S
4-Hydroxy-8-[4-(3,4,5-trichlorophenylaminosulfonyl)phenyl]pyrazolo[1,5-a]-1,3,5-triazine
—— N,N-Bis-(2-hydroxyethyl)-3-(5-oxo-6-pentyl-6,9-dihydro-5H-[1,2,4]triazolo[3,4-i]purin-8-yl)-4-propoxybenzenesulfonamide 321889-87-6 C24H33N7O6S
N,N-Bis-(2-hydroxyethyl)-3-(5-oxo-6-pentyl-6,9-dihydro-5H-[1,2,4]triazolo[3,4-i]purin-8-yl)-4-propoxybenzenesulfonamide
—— 3-(cyclopentylmethoxy)-2-(2-fluorophenyl)-2H-pyrazolo[4,3-c]quinoline 1118098-93-3 C22H20FN3O
3-(cyclopentylmethoxy)-2-(2-fluorophenyl)-2H-pyrazolo[4,3-c]quinoline
—— 13a-ethyl-7-(4-phenyl-1H-1,2,3-triazol-5-yl)-10,11,13,13a-tetrahydro-[1,4]oxazino[3,4-h][1,2,4]triazolo[4,3-f]pteridine 1371625-90-9 C20H19N9O
13a-ethyl-7-(4-phenyl-1H-1,2,3-triazol-5-yl)-10,11,13,13a-tetrahydro-[1,4]oxazino[3,4-h][1,2,4]triazolo[4,3-f]pteridine
—— (4-Chloro-phenyl)-[5-(2-methyl-4-phenyl-thiazol-5-yl)-[1,3,4]thiadiazol-2-yl]-amine 112979-22-3 C18H13ClN4S2
(4-Chloro-phenyl)-[5-(2-methyl-4-phenyl-thiazol-5-yl)-[1,3,4]thiadiazol-2-yl]-amine
—— 4-Amino-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 1305262-81-0 C16H12FN5O
4-Amino-2-[(4-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one
—— (R)-3-{(S)-2-cyclohexyl-1-[5-(2-fluoro-4-iodophenyl)-1H-imidazol-2-yl]ethyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione 1165869-85-1 C28H30FIN4O4
(R)-3-{(S)-2-cyclohexyl-1-[5-(2-fluoro-4-iodophenyl)-1H-imidazol-2-yl]ethyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione
—— tert-butyl (4-{[4-(2-ethyl-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]amino}benzyl)carbamate 930582-36-8 C22H27N5O2S
tert-butyl (4-{[4-(2-ethyl-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]amino}benzyl)carbamate
—— (3-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)-(tetrahydro-pyran-4-ylmethyl)-amine 908300-51-6 C16H18N6O
(3-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)-(tetrahydro-pyran-4-ylmethyl)-amine
—— 3-[2-(3-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-ylamino)-ethyl]-phenol 908300-61-8 C18H16N6O
3-[2-(3-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-ylamino)-ethyl]-phenol
—— 1-Allyl-3-methyl-1-{1-[5-methyl-2-(4-trifluoromethyl-phenyl)-1H-imidazol-4ylmethyl]-piperidin-4-yl}-urea 466665-34-9 C22H28F3N5O
1-Allyl-3-methyl-1-{1-[5-methyl-2-(4-trifluoromethyl-phenyl)-1H-imidazol-4ylmethyl]-piperidin-4-yl}-urea
—— N-(4-Cyano-2-nitrophenyl)-pyrazol 19005-65-3 C10H6N4O2
N-(4-Cyano-2-nitrophenyl)-pyrazol
—— 4-[2-(tert-butylamino)-4-methyl-1,3-thiazol-5-yl]-N-(3,4-difluorophenyl)pyrimidine-2-amine 930584-52-4 C18H19F2N5S
4-[2-(tert-butylamino)-4-methyl-1,3-thiazol-5-yl]-N-(3,4-difluorophenyl)pyrimidine-2-amine
—— compound 57 842128-47-6 C23H21N9O
compound 57
—— 4-[2-(dimethylamino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]-N-phenylpyrimidine-2-amine 930581-08-1 C16H14F3N5S
4-[2-(dimethylamino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]-N-phenylpyrimidine-2-amine
—— 3-methyl-but-2-enoic acid 5-(5-methanesulfonyl-1-{3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzylamide monotrifluoroacetate 1048690-33-0 C2HF3O2*C32H43F3N6O4S
3-methyl-but-2-enoic acid 5-(5-methanesulfonyl-1-{3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzylamide monotrifluoroacetate
—— 1-methyl-3-(1,1,2,3,3,3-hexafluoropropyl)imidazolium hexafluorophosphate 943523-33-9 C7H7F6N2*F6P
1-methyl-3-(1,1,2,3,3,3-hexafluoropropyl)imidazolium hexafluorophosphate
—— 1607426-64-1 C15H18F3N5OS
—— 2-[5-[3-(Difluoromethyl)-1,2,4-triazol-1-yl]-4-fluoro-2-methylphenyl]sulfanylacetonitrile 1267994-81-9 C12H9F3N4S
2-[5-[3-(Difluoromethyl)-1,2,4-triazol-1-yl]-4-fluoro-2-methylphenyl]sulfanylacetonitrile
—— ethyl 1-((2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl)methyl)-5-(furan-2-yl)-1H-pyrazole-3-carboxylate 1197846-37-9 C24H19ClN4O3
ethyl 1-((2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl)methyl)-5-(furan-2-yl)-1H-pyrazole-3-carboxylate
—— (2-chloro-4-imidazo[4,5-b]pyridin-3-yl-phenyl)-acetic acid 913173-57-6 C14H10ClN3O2
(2-chloro-4-imidazo[4,5-b]pyridin-3-yl-phenyl)-acetic acid
—— (S)-3-(3-(4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-isopropyl-1-(piperidin-4-yl)imidazolidin-2-one hydrochloride 1269644-22-5 C25H29N9O*ClH
(S)-3-(3-(4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-isopropyl-1-(piperidin-4-yl)imidazolidin-2-one hydrochloride
—— 2-(prop-2-yl)-5-trifluoromethyl-2H-[1,2,3]triazole-4-carboxylic acid ethyl ester 942060-39-1 C9H12F3N3O2
2-(prop-2-yl)-5-trifluoromethyl-2H-[1,2,3]triazole-4-carboxylic acid ethyl ester
—— 1-[4-(1-pyrrolidinylcarbonyl)phenyl]-3-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridine 1092459-33-0 C18H15F3N4O
1-[4-(1-pyrrolidinylcarbonyl)phenyl]-3-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridine
—— 5-(3-Methoxy-4-methylphenyl)-3-(5-methylpyridin-3-yl)-1,2,4-oxadiazole 1201443-64-2 C16H15N3O2
5-(3-Methoxy-4-methylphenyl)-3-(5-methylpyridin-3-yl)-1,2,4-oxadiazole
—— (S)-3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-(2-methylthiazol-4-yl)oxazolidin-2-one 1269645-18-2 C21H15FN8O2S
(S)-3-(3-(3-fluoro-4-(1H-1,2,4-triazol-3-yl)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)-4-(2-methylthiazol-4-yl)oxazolidin-2-one
—— 5-(2-fluorophenyl)-2-[5-methyl-1-(4-methylbenzyl)-1H-pyrazol-3-yl]-1,3-benzoxazole 1085451-22-4 C25H20FN3O
5-(2-fluorophenyl)-2-[5-methyl-1-(4-methylbenzyl)-1H-pyrazol-3-yl]-1,3-benzoxazole
—— 2-[1-(2,3-dimethyl-phenyl)-1H-tetrazol-5-ylsulfanyl]-N-[2-(3-methoxy-phenyl)-2H-pyrazol-3-yl]-acetamide 1200439-66-2 C21H21N7O2S
2-[1-(2,3-dimethyl-phenyl)-1H-tetrazol-5-ylsulfanyl]-N-[2-(3-methoxy-phenyl)-2H-pyrazol-3-yl]-acetamide
—— 2-chloro-5-(2-methyl-4-phenyl-oxazol-5-yl)-pyridine 459447-85-9 C15H11ClN2O
2-chloro-5-(2-methyl-4-phenyl-oxazol-5-yl)-pyridine
—— N-cyclopropyl-4-{8-[(2-methylpropyl)amino]-6-[(4-sulfamoylphenyl)ethynyl]imidazo[1,2-a]pyrazin-3-yl}benzamide 1351374-11-2 C28H28N6O3S
N-cyclopropyl-4-{8-[(2-methylpropyl)amino]-6-[(4-sulfamoylphenyl)ethynyl]imidazo[1,2-a]pyrazin-3-yl}benzamide
—— 3-Isopropyl-1-(3-methoxy-phenyl)-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one 650628-95-8 C15H16N4O2
3-Isopropyl-1-(3-methoxy-phenyl)-1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one
—— [2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-5-(6-methylpyridin-3-yl)-1,3-thiazol-4-yl]methanamine 1309444-02-7 C16H22N4OS
[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-5-(6-methylpyridin-3-yl)-1,3-thiazol-4-yl]methanamine
—— potassium trifluoro(1-methyl-5-phenyl-1H-pyrazol-3-yl)borate 1402242-70-9 C10H9BF3N2*K
potassium trifluoro(1-methyl-5-phenyl-1H-pyrazol-3-yl)borate
—— 2-[6-(3-Methylbutan-2-ylsulfanyl)-3-phenylpyrazolo[3,4-b]pyridin-1-yl]-1,3-thiazole-4-carboxylic acid 1204772-65-5 C21H20N4O2S2
2-[6-(3-Methylbutan-2-ylsulfanyl)-3-phenylpyrazolo[3,4-b]pyridin-1-yl]-1,3-thiazole-4-carboxylic acid
—— 5-(4-chlorophenyl)-3-[1-(1-naphthylmethyl)piperidin-4-yl]pyrazole 156337-40-5 C25H24ClN3
5-(4-chlorophenyl)-3-[1-(1-naphthylmethyl)piperidin-4-yl]pyrazole
—— 1-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-tetrazolyl)phenyl]-2,5-imidazolidinedione 377079-08-8 C22H19F2N9O3
1-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-tetrazolyl)phenyl]-2,5-imidazolidinedione
—— 6-benzyloxy-4-chloro-2-phenyl-2H-pyrazolo[3,4-c]quinoline 1315307-88-0 C23H16ClN3O
6-benzyloxy-4-chloro-2-phenyl-2H-pyrazolo[3,4-c]quinoline
—— 1-{4-[2-(1-methyl-1H-pyrazol-5-yl)-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-3-yl]phenyl}cyclobutanamine 1374261-88-7 C28H25N7
1-{4-[2-(1-methyl-1H-pyrazol-5-yl)-9H-imidazo[1,2-d]pyrido[2,3-b][1,4]benzodiazepin-3-yl]phenyl}cyclobutanamine
—— 4-Amino-2-[[2-(trifluoromethyl)phenyl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 1305262-86-5 C17H12F3N5O
4-Amino-2-[[2-(trifluoromethyl)phenyl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-1-one
—— 1-(2-phenyl-2-trimethylsilanyloxy-ethyl)-1<i>H</i>-[1,2,3]triazole-4,5-dicarboxylic acid dimethyl ester 55848-62-9 C17H23N3O5Si
1-(2-phenyl-2-trimethylsilanyloxy-ethyl)-1<i>H</i>-[1,2,3]triazole-4,5-dicarboxylic acid dimethyl ester
—— 4-{4-(4-(furan-2-yl)-1H-imidazol-1-yl)-3-isopropyl-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-(4-hydroxycyclohexylamino)benzamide 1260533-08-1 C29H31N7O3
4-{4-(4-(furan-2-yl)-1H-imidazol-1-yl)-3-isopropyl-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-(4-hydroxycyclohexylamino)benzamide
—— 1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [1-(3-fluorophenyl)cyclopropyl]amide 1295298-45-1 C22H16F2N4O
1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [1-(3-fluorophenyl)cyclopropyl]amide
—— 4-{4-(4-(1-(hydroxyethyl)-1H-pyrazol-4-yl)-1H-imidazol-1-yl)-3-isopropyl-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-(isopropyl)benzamide 1260534-32-4 C27H30N8O2
4-{4-(4-(1-(hydroxyethyl)-1H-pyrazol-4-yl)-1H-imidazol-1-yl)-3-isopropyl-1H-pyrazolo[3,4-b]pyridin-1-yl}-2-(isopropyl)benzamide
—— 5-cyclopropyl-8-(difluoromethoxy)-1-(5-phenyloxazole-4-carbonyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307894-55-8 C24H21F2N3O4
5-cyclopropyl-8-(difluoromethoxy)-1-(5-phenyloxazole-4-carbonyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one
—— (6,8-dichloro-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-(1H-imidazol-2-yl)-amine 1197848-45-5 C18H15Cl2N5
(6,8-dichloro-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-(1H-imidazol-2-yl)-amine