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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(benzylthio)carbonyl-3-amino-4-oxo-5-(5-(2,6-dichloro-4-methylphenylthio)tetrazol-2-yl)pentanoic acid 192455-80-4 C21H19Cl2N5O4S2
N-(benzylthio)carbonyl-3-amino-4-oxo-5-(5-(2,6-dichloro-4-methylphenylthio)tetrazol-2-yl)pentanoic acid
—— 3-chloro-N-cyclohexyl-4-(2-(3,4-difluorobenzylamino)-9-((R)-piperidine-3-ylmethyl)-9H-purin-8-yl)benzamide 1021697-63-1 C31H34ClF2N7O
3-chloro-N-cyclohexyl-4-(2-(3,4-difluorobenzylamino)-9-((R)-piperidine-3-ylmethyl)-9H-purin-8-yl)benzamide
—— 3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-N-(thiazol-2-yl)-3-o-tolylpropanamide 1025760-31-9 C28H25FN4OS
3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-N-(thiazol-2-yl)-3-o-tolylpropanamide
—— N-(6-(1-(1-(2-amino-2-oxoethyl)piperidin-4-yl)-4-(4-fluorophenyl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)-4-methyl-2-(pyridin-3-yl)thiazole-5-carboxamide 1615721-73-7 C32H29FN10O2S
N-(6-(1-(1-(2-amino-2-oxoethyl)piperidin-4-yl)-4-(4-fluorophenyl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)-4-methyl-2-(pyridin-3-yl)thiazole-5-carboxamide
—— 4-(1-methyl-3-(4-((1-methyl-1H-pyrazol-4-yl)ethynyl)phenyl)-1H-pyrazole-4-yl)pyridine 1610785-67-5 C21H17N5
4-(1-methyl-3-(4-((1-methyl-1H-pyrazol-4-yl)ethynyl)phenyl)-1H-pyrazole-4-yl)pyridine
—— 3-(3-fluorophenyl)-3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-N-(1,3,4-thiadiazol-2-yl)propanamide 1025760-44-4 C26H21F2N5OS
3-(3-fluorophenyl)-3-(1-(4-fluorophenyl)-1H-indazol-5-yl)-2,2-dimethyl-N-(1,3,4-thiadiazol-2-yl)propanamide
—— 3-[[(4-bromo-2-methylphenyl)carbonyl]-(1-methylethyl)amino]-5-(4-imidazo[1,2-a]pyridin-2-ylphenyl)-2-thiophenecarboxylic acid 1019337-25-7 C29H24BrN3O3S
3-[[(4-bromo-2-methylphenyl)carbonyl]-(1-methylethyl)amino]-5-(4-imidazo[1,2-a]pyridin-2-ylphenyl)-2-thiophenecarboxylic acid
—— 4-[5-(1-benzyl-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-oxadiazol-3-yl]benzoic acid 1233243-66-7 C25H24N4O3
4-[5-(1-benzyl-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-oxadiazol-3-yl]benzoic acid
—— 8-fluoro-3-(morpholin-4-ylcarbonyl)-1-[4-(morpholin-4-ylmethyl)phenyl]-1,4-dihydrothiochromeno[4,3-c]pyrazole 5,5-dioxide 1305267-42-8 C26H27FN4O5S
8-fluoro-3-(morpholin-4-ylcarbonyl)-1-[4-(morpholin-4-ylmethyl)phenyl]-1,4-dihydrothiochromeno[4,3-c]pyrazole 5,5-dioxide
—— 928825-32-5 C21H15Cl2F3N6O3
—— <i>N</i>-butyl-<i>N</i>-(5-methoxy-4-methyl-oxazol-2-yl)-isobutyramide 57068-97-0 C13H22N2O3
<i>N</i>-butyl-<i>N</i>-(5-methoxy-4-methyl-oxazol-2-yl)-isobutyramide
—— 4-{6-[6-(4-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-benzonitrile 1029525-93-6 C24H13FN6O
4-{6-[6-(4-fluorophenyl)-imidazo[2,1-b]oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-benzonitrile
—— 5-(3,3-dimethyl-triaz-1-enyl)-2-phenyl-1(3)<i>H</i>-imidazole-4-carboxylic acid benzyl ester 37116-39-5 C19H19N5O2
5-(3,3-dimethyl-triaz-1-enyl)-2-phenyl-1(3)<i>H</i>-imidazole-4-carboxylic acid benzyl ester
—— N-[1-(3-{1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-N'-propylsulfamide 1289201-70-2 C24H29F3N4O3S
N-[1-(3-{1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-N'-propylsulfamide
—— 4-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-but-3-yn-1-ol 1049807-95-5 C24H31ClN4O4S
4-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-but-3-yn-1-ol
—— ethyl [2-(5-chloro-2-{[(2,4,6-trifluorophenyl)methyl]oxy}phenyl)-1,3-oxazol-4-yl]acetate 913651-00-0 C20H15ClF3NO4
ethyl [2-(5-chloro-2-{[(2,4,6-trifluorophenyl)methyl]oxy}phenyl)-1,3-oxazol-4-yl]acetate
—— [3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazol-4-yl][2-(3-methyl-benzyl)pyrrolidin-1-yl]methanone 1373536-42-5 C18H20F3N3O
[3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazol-4-yl][2-(3-methyl-benzyl)pyrrolidin-1-yl]methanone
—— 4-Amino-2-[(2-fluorophenyl)methyl]-7-(hydroxymethyl)-[1,2,4]triazolo[4,3-a]quinoxalin-1-one 1305263-39-1 C17H14FN5O2
4-Amino-2-[(2-fluorophenyl)methyl]-7-(hydroxymethyl)-[1,2,4]triazolo[4,3-a]quinoxalin-1-one
—— N-{3-[3-(2-{[3-(pyrrolidin-l-ylmethyl)phenyl]amino}pyrimidin-4-yl)imidazo[l,2-a]pyridin-2-yl]phenyl}-2-(thiophen-2-yl)acetamide 1301135-62-5 C34H31N7OS
N-{3-[3-(2-{[3-(pyrrolidin-l-ylmethyl)phenyl]amino}pyrimidin-4-yl)imidazo[l,2-a]pyridin-2-yl]phenyl}-2-(thiophen-2-yl)acetamide
—— N-{1-[3-(1-ethyl-5-{4-[(tetrahydro-2H-pyran-3-ylamino)methyl]phenoxy}-1H-pyrazol-3-yl)phenyl]-1-methylethyl}-2,2,2-trifluoroethanesulfonamide 1289202-67-0 C28H35F3N4O4S
N-{1-[3-(1-ethyl-5-{4-[(tetrahydro-2H-pyran-3-ylamino)methyl]phenoxy}-1H-pyrazol-3-yl)phenyl]-1-methylethyl}-2,2,2-trifluoroethanesulfonamide
—— 5-(3-chloro-2-(2-cyclohexylethoxy)phenyl)-1H-imidazole 1300729-25-2 C17H21ClN2O
5-(3-chloro-2-(2-cyclohexylethoxy)phenyl)-1H-imidazole
—— 6-(4-(1H-pyrazol-1-yl)phenylamino)-4-(benzylamino)nicotinamide 1374212-94-8 C22H20N6O
6-(4-(1H-pyrazol-1-yl)phenylamino)-4-(benzylamino)nicotinamide
—— 9,10-dioxa-syn-(carboethoxy,methyl)bimane 79746-76-2 C14H16N2O6
9,10-dioxa-syn-(carboethoxy,methyl)bimane
—— 1-methyl-3-[(1S,4S)-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)sulfonyl]-3(H)-imidazol-1-ium trifluoromethane-sulfonate 1187160-72-0 CF3O3S*C9H14N3O3S
1-methyl-3-[(1S,4S)-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)sulfonyl]-3(H)-imidazol-1-ium trifluoromethane-sulfonate
—— 1393096-35-9 C26H19ClF8N6O
—— 1-[2-[[5-[[2-Methyl-4-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrrol-1-yl]methyl]pyridin-2-yl]amino]ethyl]piperidin-4-ol 1226861-10-4 C27H29F3N6O3
1-[2-[[5-[[2-Methyl-4-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrrol-1-yl]methyl]pyridin-2-yl]amino]ethyl]piperidin-4-ol
—— 1449704-59-9 C11H13FN2S*ClH
—— EC011 1135429-16-1 C18H22N6O
EC011
—— 1-(4-(5-(5-chloro-1-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 1236148-68-7 C22H18ClN5O3
1-(4-(5-(5-chloro-1-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid
—— 3-((1H-1,2,4-triazol-1-yl)methyl)-2-(4-bromophenyl)-imidazo[1,2-a]pyridine 1197846-80-2 C16H12BrN5
3-((1H-1,2,4-triazol-1-yl)methyl)-2-(4-bromophenyl)-imidazo[1,2-a]pyridine
—— 4-tert-butyl-N-(4-chloro-2-(7H-purin-7-yl)phenyl)benzenesulfonamide 1094757-31-9 C21H20ClN5O2S
4-tert-butyl-N-(4-chloro-2-(7H-purin-7-yl)phenyl)benzenesulfonamide
—— 4-(5-cyano-7-propan-2-yl-1,3-benzoxazol-2-yl)-N-[[(5R)-3-[5-(2-fluoro-6-propan-2-yloxyphenyl)pyridin-2-yl]-2-oxo-1,3-oxazolidin-5-yl]methyl]benzamide 1093752-71-6 C36H32FN5O5
4-(5-cyano-7-propan-2-yl-1,3-benzoxazol-2-yl)-N-[[(5R)-3-[5-(2-fluoro-6-propan-2-yloxyphenyl)pyridin-2-yl]-2-oxo-1,3-oxazolidin-5-yl]methyl]benzamide
—— N-(2-(1H-[1,2,3]triazolo[4,5-b]pyridin-1-yl)-5-methylpyridin-3-yl)-4-tert-butylbenzenesulfonamide 1094758-14-1 C21H22N6O2S
N-(2-(1H-[1,2,3]triazolo[4,5-b]pyridin-1-yl)-5-methylpyridin-3-yl)-4-tert-butylbenzenesulfonamide
—— 5-(5-chloromethyl-4-methoxymethyl-thiazol-2-yl)-2-trifluoromethyl-pyridine 933781-48-7 C12H10ClF3N2OS
5-(5-chloromethyl-4-methoxymethyl-thiazol-2-yl)-2-trifluoromethyl-pyridine
—— 3-(2-(chloromethyl)-5-(5-methyl-1H-pyrazol-3-ylamino)imidazo[1,2-f]pyrimidin-7-yl)-N-cyclopropylbenzamide 883736-43-4 C21H20ClN7O
3-(2-(chloromethyl)-5-(5-methyl-1H-pyrazol-3-ylamino)imidazo[1,2-f]pyrimidin-7-yl)-N-cyclopropylbenzamide
—— (5-(4,6-dimethoxypyrimidin-2-yl)hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)(2-fluoro-6-(2H-1 ,2,3-triazol-2-yl)phenyl)methanone 1293282-96-8 C21H22FN7O3
(5-(4,6-dimethoxypyrimidin-2-yl)hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)(2-fluoro-6-(2H-1 ,2,3-triazol-2-yl)phenyl)methanone
—— 1-isopropyl-3-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)urea 1041395-31-6 C28H36N6O3
1-isopropyl-3-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)urea
—— 2-chloro-N-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)benzamide 1041395-62-3 C31H32ClN5O3
2-chloro-N-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)benzamide
—— N-[(1S,2R,4R)-7-azabicyclo[2.2.1]hept-2-yl]-5-(4-aminophenyl)-1,3-oxazole-2-carboxamide 500612-74-8 C16H18N4O2
N-[(1S,2R,4R)-7-azabicyclo[2.2.1]hept-2-yl]-5-(4-aminophenyl)-1,3-oxazole-2-carboxamide
—— [rac]-3-(4-{2-[2-(4-chloro-phenyl)-5-methyl-oxazol-4-yl]-ethoxy}-5,6,7,8-tetrahydro-naphthalen-1-yl)-2-ethoxy-propionic acid 475480-67-2 C27H30ClNO5
[rac]-3-(4-{2-[2-(4-chloro-phenyl)-5-methyl-oxazol-4-yl]-ethoxy}-5,6,7,8-tetrahydro-naphthalen-1-yl)-2-ethoxy-propionic acid
—— 2-(tert-butyldimethylsilyl)-5-(10-bromodecyl)-1-(N,N-dimethylsulfamoyl)-imidazole 841261-22-1 C21H42BrN3O2SSi
2-(tert-butyldimethylsilyl)-5-(10-bromodecyl)-1-(N,N-dimethylsulfamoyl)-imidazole
—— 3-(2,4-difluorophenyl)-6-(1-methyl-1H-1,2,4-triazol-3-ylmethoxy)-7-(pyrrolidin-1-yl)-1,2,4-triazolo[4,3-b]pyridazine 233275-88-2 C19H18F2N8O
3-(2,4-difluorophenyl)-6-(1-methyl-1H-1,2,4-triazol-3-ylmethoxy)-7-(pyrrolidin-1-yl)-1,2,4-triazolo[4,3-b]pyridazine
—— 3-chloro-4-[2-[(3,4-difluorophenyl)methylamino]-9-[[(3R)-piperidin-3-yl]methyl]purin-8-yl]benzamide 1021697-04-0 C25H24ClF2N7O
3-chloro-4-[2-[(3,4-difluorophenyl)methylamino]-9-[[(3R)-piperidin-3-yl]methyl]purin-8-yl]benzamide
—— 8-[2,6-dichloro-4-(2-methoxyethoxy)phenyl]-N-[(3,4-difluorophenyl)methyl]-9-[[(3R)-piperidin-3-yl]methyl]purin-2-amine 1021697-16-4 C27H28Cl2F2N6O2
8-[2,6-dichloro-4-(2-methoxyethoxy)phenyl]-N-[(3,4-difluorophenyl)methyl]-9-[[(3R)-piperidin-3-yl]methyl]purin-2-amine
—— 1-[5-(Cyclopropylmethylsulfinyl)-2-fluoro-4-methylphenyl]-3-(difluoromethyl)-1,2,4-triazole 1267994-90-0 C14H14F3N3OS
1-[5-(Cyclopropylmethylsulfinyl)-2-fluoro-4-methylphenyl]-3-(difluoromethyl)-1,2,4-triazole
—— 8-(2,6-dichlorophenyl)-N-[(3,4-difluorophenyl)methyl]-9-(pyrrolidin-3-ylmethyl)purin-2-amine 1021694-01-8 C23H20Cl2F2N6
8-(2,6-dichlorophenyl)-N-[(3,4-difluorophenyl)methyl]-9-(pyrrolidin-3-ylmethyl)purin-2-amine
—— 4,5-dibromo-1-((2-(trimethylsilyl)ethoxy)methyl)-2-(2-tolyl)-1H-imidazole 1448032-46-9 C16H22Br2N2OSi
4,5-dibromo-1-((2-(trimethylsilyl)ethoxy)methyl)-2-(2-tolyl)-1H-imidazole
—— methyl N-cyano-N'-[8-[[(cyanoamino)-[2-[(5-methyl-1H-imidazol-4-yl)methylsulfanyl]ethylamino]methylidene]amino]octyl]carbamimidothioate 66169-59-3 C20H33N9S2
methyl N-cyano-N'-[8-[[(cyanoamino)-[2-[(5-methyl-1H-imidazol-4-yl)methylsulfanyl]ethylamino]methylidene]amino]octyl]carbamimidothioate
—— 1-benzyl-2-(4-methoxyphenyl)-4,5-di(3-nitrophenyl)-1H-imidazole 1448032-56-1 C29H22N4O5
1-benzyl-2-(4-methoxyphenyl)-4,5-di(3-nitrophenyl)-1H-imidazole
—— 2-{2-[(4aR,5R)-4a-cyclopropyl-1-(4-fluorophenyl)-5-hydroxy-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-N-(2-hydroxyethyl)benzamide 1299473-64-5 C30H32FN3O3
2-{2-[(4aR,5R)-4a-cyclopropyl-1-(4-fluorophenyl)-5-hydroxy-1,4,4a,5,6,7-hexahydrocyclopenta[f]indazol-5-yl]ethyl}-N-(2-hydroxyethyl)benzamide