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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)-N-[(Z)-[(2S)-2-phenylcyclohexylidene]amino]acetamide —— C18H20N4O2S
2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)-N-[(Z)-[(2S)-2-phenylcyclohexylidene]amino]acetamide
—— N-[(Z)-[(Z)-2-bromo-3-phenylprop-2-enylidene]amino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C15H13BrN4O2S
N-[(Z)-[(Z)-2-bromo-3-phenylprop-2-enylidene]amino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N-[(Z)-[(2R)-2-methylcyclohexylidene]amino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C13H18N4O2S
N-[(Z)-[(2R)-2-methylcyclohexylidene]amino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— (Z)-N-benzyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-ethylprop-2-enamide —— C18H21N3O3
(Z)-N-benzyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-ethylprop-2-enamide
—— N-[(Z)-1-(3-bromophenyl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C14H13BrN4O2S
N-[(Z)-1-(3-bromophenyl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— 2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)-N-[(Z)-1-(2,4,5-trimethylphenyl)ethylideneamino]acetamide —— C17H20N4O2S
2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)-N-[(Z)-1-(2,4,5-trimethylphenyl)ethylideneamino]acetamide
—— N-[(Z)-(3-chlorophenyl)methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C13H11ClN4O2S
N-[(Z)-(3-chlorophenyl)methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N-[(Z)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C17H18N4O4S
N-[(Z)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N-[(Z)-[2,5-dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C16H16N6O2S2
N-[(Z)-[2,5-dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— (Z)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-ethyl-N-[(3-fluorophenyl)methyl]prop-2-enamide —— C18H20FN3O3
(Z)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-ethyl-N-[(3-fluorophenyl)methyl]prop-2-enamide
—— N-[(Z)-[(1S)-cyclohex-3-en-1-yl]methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C13H16N4O2S
N-[(Z)-[(1S)-cyclohex-3-en-1-yl]methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N-[(Z)-1-(furan-2-yl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C12H12N4O3S
N-[(Z)-1-(furan-2-yl)ethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N-[(Z)-(4-fluorophenyl)methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C13H11FN4O2S
N-[(Z)-(4-fluorophenyl)methylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— N'-[1-(2,4-dimethylpyrrol-3-ylidene)ethyl]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetohydrazide —— C14H17N5O2S
N'-[1-(2,4-dimethylpyrrol-3-ylidene)ethyl]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetohydrazide
—— N-[(Z)-furan-2-ylmethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide —— C11H10N4O3S
N-[(Z)-furan-2-ylmethylideneamino]-2-(4-oxo-2-sulfanylidene-1H-pyrimidin-6-yl)acetamide
—— (Z)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)prop-2-enoic acid —— C9H10N2O4
(Z)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)prop-2-enoic acid
—— N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1R)-1-phenylethyl]acetamide —— C33H34ClN5O2
N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1R)-1-phenylethyl]acetamide
—— N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C31H35N5O6
N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C31H35N5O6
N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— 3-[(E)-2-[2,5-dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]ethenyl]-4-methyl-6-oxo-1H-pyridazine-5-carbonitrile —— C17H15N5OS
3-[(E)-2-[2,5-dimethyl-1-(1,3-thiazol-2-yl)pyrrol-3-yl]ethenyl]-4-methyl-6-oxo-1H-pyridazine-5-carbonitrile
—— N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-2-phenylacetamide —— C31H37N5O4
N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-2-phenylacetamide
—— N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-2-phenylacetamide —— C31H37N5O4
N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-2-phenylacetamide
—— 4-methoxy-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide —— C29H35N5O6S
4-methoxy-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide
—— methyl 4-[3-(3,5-dimethylphenoxy)propylsulfanyl]-6-methyl-2-oxo-1H-pyrimidine-5-carboxylate —— C18H22N2O4S
methyl 4-[3-(3,5-dimethylphenoxy)propylsulfanyl]-6-methyl-2-oxo-1H-pyrimidine-5-carboxylate
—— methyl 4-[2-(1-adamantyl)-2-oxoethyl]sulfanyl-6-methyl-2-oxo-1H-pyrimidine-5-carboxylate —— C19H24N2O4S
methyl 4-[2-(1-adamantyl)-2-oxoethyl]sulfanyl-6-methyl-2-oxo-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[3-chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17ClF3N3O4
ethyl (4R)-6-[[3-chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-3-[(6-chloropyridazin-3-yl)amino]urea —— C16H21Cl2N5O
1-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-3-[(6-chloropyridazin-3-yl)amino]urea
—— N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]thiophene-2-carboxamide —— C29H28ClN5O2S
N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]thiophene-2-carboxamide
—— 1-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-3-[(6-chloropyridazin-3-yl)amino]urea —— C16H21Cl2N5O
1-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-3-[(6-chloropyridazin-3-yl)amino]urea
—— N-[(2R)-butan-2-yl]-4-chloro-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]benzenesulfonamide —— C27H32ClN5O4S
N-[(2R)-butan-2-yl]-4-chloro-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]benzenesulfonamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-3-methyl-N-[(1S)-1-phenylethyl]butanamide —— C32H41N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-3-methyl-N-[(1S)-1-phenylethyl]butanamide
—— [2-[(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-ethylamino]-2-oxoethyl] 2-(4-methylphenyl)acetate —— C21H28N4O5
[2-[(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-ethylamino]-2-oxoethyl] 2-(4-methylphenyl)acetate
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]cyclopropanecarboxamide —— C31H37N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]cyclopropanecarboxamide
—— N-[(2S)-butan-2-yl]-4-chloro-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]benzenesulfonamide —— C27H32ClN5O4S
N-[(2S)-butan-2-yl]-4-chloro-N-[2-[4-[6-(3-methoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]benzenesulfonamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-methyl-N-[(1S)-1-phenylethyl]propanamide —— C31H39N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-methyl-N-[(1S)-1-phenylethyl]propanamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1S)-1-phenylethyl]acetamide —— C35H39N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1S)-1-phenylethyl]acetamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-methoxy-N-[(1R)-1-phenylethyl]acetamide —— C30H37N5O5
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-methoxy-N-[(1R)-1-phenylethyl]acetamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1R)-1-phenylethyl]acetamide —— C35H39N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-2-phenyl-N-[(1R)-1-phenylethyl]acetamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-3-methyl-N-[(1R)-1-phenylethyl]butanamide —— C32H41N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-3-methyl-N-[(1R)-1-phenylethyl]butanamide
—— N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]thiophene-2-carboxamide —— C29H28ClN5O2S
N-[2-[4-[6-(2-chlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]thiophene-2-carboxamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclobutanecarboxamide —— C32H39N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclobutanecarboxamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclopropanecarboxamide —— C31H37N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclopropanecarboxamide
—— N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]cyclobutanecarboxamide —— C32H39N5O4
N-[2-[4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]-1,4-diazepan-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]cyclobutanecarboxamide
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(5-phenylfuran-2-yl)propanoate —— C20H17N3O4S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(5-phenylfuran-2-yl)propanoate
—— (5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C30H34ClN5O3S
(5R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-methyl-3-[2-(2-morpholin-4-ylethylamino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— ethyl (6R)-4-[[4-(cyclopentanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H36Cl2N4O4
ethyl (6R)-4-[[4-(cyclopentanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (5R)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30ClN5O3S
(5R)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C26H37Cl2N5O4
ethyl (6S)-4-[[4-(tert-butylcarbamoyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (5S)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C28H30ClN5O3S
(5S)-5-(3-chlorophenyl)-N-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— ethyl (6S)-4-[[4-(cyclopentanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C27H36Cl2N4O4
ethyl (6S)-4-[[4-(cyclopentanecarbonyl)-1,4-diazepan-1-yl]methyl]-6-(3,4-dichlorophenyl)-3-ethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate