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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(3-chlorophenyl)methyl]-2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)acetamide —— C16H15ClN4O2
N-[(3-chlorophenyl)methyl]-2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)acetamide
—— 5,6-Dimethyl-3-oxo-2-[(2,3,4,5,6-pentafluorophenyl)methyl]pyridazine-4-carbonitrile —— C14H8F5N3O
5,6-Dimethyl-3-oxo-2-[(2,3,4,5,6-pentafluorophenyl)methyl]pyridazine-4-carbonitrile
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(S)-(4-fluorophenyl)-thiophen-2-ylmethyl]acetamide —— C20H17FN4O2S
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(S)-(4-fluorophenyl)-thiophen-2-ylmethyl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide —— C17H24N4O4S
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methylpropyl)acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-di(propan-2-yl)acetamide —— C15H22N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-di(propan-2-yl)acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-methyl-N-(thiophen-2-ylmethyl)acetamide —— C15H16N4O2S
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-methyl-N-(thiophen-2-ylmethyl)acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(4-methylphenyl)methyl]-N-propylacetamide —— C20H24N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(4-methylphenyl)methyl]-N-propylacetamide
—— 5,6-Dimethyl-2-[(3-methylphenyl)methyl]-3-oxopyridazine-4-carbonitrile —— C15H15N3O
5,6-Dimethyl-2-[(3-methylphenyl)methyl]-3-oxopyridazine-4-carbonitrile
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1S)-3-methyl-1-phenylbutyl]acetamide —— C20H24N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1S)-3-methyl-1-phenylbutyl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(4-ethylphenyl)methyl]-N-methylacetamide —— C19H22N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(4-ethylphenyl)methyl]-N-methylacetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(2S)-2-ethylhexyl]acetamide —— C17H26N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(2S)-2-ethylhexyl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-methyl-N-[(1S)-1-phenylethyl]acetamide —— C18H20N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-methyl-N-[(1S)-1-phenylethyl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide —— C16H18N4O2S2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide
—— 2-[2-[(3S)-3-(furan-2-yl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C23H21N5O3
2-[2-[(3S)-3-(furan-2-yl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— 2-(3-fluorophenyl)-4-(4-fluorophenyl)-6-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]pyrazolo[3,4-d]pyrimidin-3-amine —— C29H27F2N7O
2-(3-fluorophenyl)-4-(4-fluorophenyl)-6-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]pyrazolo[3,4-d]pyrimidin-3-amine
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C14H18N4O3
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclopentyl-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C18H24N4O4S
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclopentyl-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-bis(2-methoxyethyl)acetamide —— C15H22N4O4
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-bis(2-methoxyethyl)acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclohexyl-N-ethylacetamide —— C17H24N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclohexyl-N-ethylacetamide
—— (Z)-N-cyclopropyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-(thiophen-2-ylmethyl)prop-2-enamide —— C17H19N3O3S
(Z)-N-cyclopropyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-(thiophen-2-ylmethyl)prop-2-enamide
—— N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C28H33N5O6
N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H33N5O5S
N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (Z)-N-cyclopropyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-(furan-2-ylmethyl)prop-2-enamide —— C17H19N3O4
(Z)-N-cyclopropyl-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-(furan-2-ylmethyl)prop-2-enamide
—— N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C28H33N5O6
N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H33N5O5S
N-[2-[4-[6-(3,4-dimethoxyphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (5Z)-5-(anilinomethylidene)-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C14H13N3O2S
(5Z)-5-(anilinomethylidene)-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C24H32FN5O2S
(5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]sulfanylacetic acid —— C16H15N3O4S2
2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]sulfanylacetic acid
—— (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C24H32FN5O2S
(5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]acetic acid —— C16H15N3O4S
2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]acetic acid
—— 2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]sulfanylacetate —— C16H14N3O4S2-
2-[4-[[(E)-(4,6-dioxo-1-prop-2-enyl-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]phenyl]sulfanylacetate
—— (5Z)-5-[(4-butylanilino)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H21N3O2S
(5Z)-5-[(4-butylanilino)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[(3-ethylanilino)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H17N3O2S
(5Z)-5-[(3-ethylanilino)methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-methyl-N-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H25ClN4O2S
(5S)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-methyl-N-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-methyl-N-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C26H25ClN4O2S
(5R)-5-(4-chlorophenyl)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-methyl-N-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— ethyl (4S)-6-[[[4-(dimethylamino)phenyl]methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H30N4O3
ethyl (4S)-6-[[[4-(dimethylamino)phenyl]methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (1R,4R)-2-(2-chloropyrimidin-5-yl)sulfonyl-2-azabicyclo[2.2.1]heptane —— C10H12ClN3O2S
(1R,4R)-2-(2-chloropyrimidin-5-yl)sulfonyl-2-azabicyclo[2.2.1]heptane
—— ethyl (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C20H26N4O3S2
ethyl (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C20H26N4O3S2
ethyl (5S)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-7-methyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C31H38N4O4S
ethyl (3R)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C31H38N4O4S
ethyl (3S)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C24H29FN4O2S
(5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C24H29FN4O2S
(5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-fluorophenyl)-N,7-dimethyl-N-propan-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— [(4R)-5-ethoxycarbonyl-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C19H28N4O5S
[(4R)-5-ethoxycarbonyl-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— 1-(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-3-[(4-fluorophenyl)methyl]-1-(2-methylpropyl)thiourea —— C20H28FN5O2S
1-(6-Amino-1-butyl-2,4-dioxopyrimidin-5-yl)-3-[(4-fluorophenyl)methyl]-1-(2-methylpropyl)thiourea
—— N-[2-[4-[6-(4-methylphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C30H33N5O5
N-[2-[4-[6-(4-methylphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclopropanecarboxamide —— C28H29Cl2N5O2
N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1S)-1-phenylethyl]cyclopropanecarboxamide
—— N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]-1,3-benzodioxole-5-carboxamide —— C32H29Cl2N5O4
N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]-1,3-benzodioxole-5-carboxamide
—— N-[2-[4-[6-(4-methylphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C30H33N5O5
N-[2-[4-[6-(4-methylphenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]thiophene-2-carboxamide —— C29H27Cl2N5O2S
N-[2-[4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]piperazin-1-yl]-2-oxoethyl]-N-[(1R)-1-phenylethyl]thiophene-2-carboxamide