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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(1S)-1-ethoxyethyl]-5-[[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C21H19FN4O2S
3-[(1S)-1-ethoxyethyl]-5-[[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— 1-[5-[(3,7-diphenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)oxymethyl]-2-methyl-1,2,4-triazol-3-yl]-N,N-dimethylmethanamine —— C24H24N8O
1-[5-[(3,7-diphenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)oxymethyl]-2-methyl-1,2,4-triazol-3-yl]-N,N-dimethylmethanamine
—— 4-[(3-Chloro-4-methoxyphenyl)methylamino]-1-(4-methoxyphenyl)phthalazine-6-carbonitrile —— C24H19ClN4O2
4-[(3-Chloro-4-methoxyphenyl)methylamino]-1-(4-methoxyphenyl)phthalazine-6-carbonitrile
—— 1-{N-[2-(amidinoaminooxy)ethyl]amino}carbonylmethyl-6-methyl-3-(1-phenylcyclobutyl)methylamino-pyrazinone 252271-03-7 C21H29N7O3
1-{N-[2-(amidinoaminooxy)ethyl]amino}carbonylmethyl-6-methyl-3-(1-phenylcyclobutyl)methylamino-pyrazinone
—— N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(2-oxopyrimidin-1-yl)acetamide —— C14H19N5O3
N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(2-oxopyrimidin-1-yl)acetamide
—— [2-(dimethylamino)-4-methylpyrimidin-5-yl]-[(2S)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]methanone —— C15H22N4O
[2-(dimethylamino)-4-methylpyrimidin-5-yl]-[(2S)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]methanone
—— N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(2-oxopyrimidin-1-yl)acetamide —— C14H19N5O3
N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(2-oxopyrimidin-1-yl)acetamide
—— Methyl 4-[5-cyano-2-[4-(2-imidazol-1-ylethyl)anilino]pyrimidin-4-yl]benzoate —— C24H20N6O2
Methyl 4-[5-cyano-2-[4-(2-imidazol-1-ylethyl)anilino]pyrimidin-4-yl]benzoate
—— (Z)-N-[2-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]ethyl]-3-thiophen-2-ylprop-2-enamide —— C20H19N3O3S
(Z)-N-[2-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]ethyl]-3-thiophen-2-ylprop-2-enamide
—— (Z)-3-(2-chlorophenyl)-N-[2-[3-(4-fluorophenyl)-6-oxopyridazin-1-yl]ethyl]prop-2-enamide —— C21H17ClFN3O2
(Z)-3-(2-chlorophenyl)-N-[2-[3-(4-fluorophenyl)-6-oxopyridazin-1-yl]ethyl]prop-2-enamide
—— 2-pyridin-4-yl-4-[(3S)-3-[(sulfamoylamino)methyl]piperidin-1-yl]-6-(trifluoromethyl)pyrimidine —— C16H19F3N6O2S
2-pyridin-4-yl-4-[(3S)-3-[(sulfamoylamino)methyl]piperidin-1-yl]-6-(trifluoromethyl)pyrimidine
—— [2-(dimethylamino)-4-methylpyrimidin-5-yl]-[(2R)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]methanone —— C15H22N4O
[2-(dimethylamino)-4-methylpyrimidin-5-yl]-[(2R)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]methanone
—— (Z)-3-(furan-2-yl)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]prop-2-enamide —— C19H17N3O3
(Z)-3-(furan-2-yl)-N-[2-(6-oxo-3-phenylpyridazin-1-yl)ethyl]prop-2-enamide
—— 2-pyridin-4-yl-4-[(3R)-3-[(sulfamoylamino)methyl]piperidin-1-yl]-6-(trifluoromethyl)pyrimidine —— C16H19F3N6O2S
2-pyridin-4-yl-4-[(3R)-3-[(sulfamoylamino)methyl]piperidin-1-yl]-6-(trifluoromethyl)pyrimidine
—— (2R)-N-[3-[[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]phenyl]oxolane-2-carboxamide —— C22H20F3N5O2
(2R)-N-[3-[[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]phenyl]oxolane-2-carboxamide
—— (2S,6S)-2-methyl-6-phenyl-4-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C21H19F3N4O
(2S,6S)-2-methyl-6-phenyl-4-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— 4-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]sulfanyl-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine —— C16H14F3N7OS
4-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]sulfanyl-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine
—— 4-[(2R)-2-(1,3-benzodioxol-5-yl)pyrrolidin-1-yl]-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine —— C21H17F3N4O2
4-[(2R)-2-(1,3-benzodioxol-5-yl)pyrrolidin-1-yl]-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine
—— (1S)-1-(2,5-dimethoxyphenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol —— C20H19F3N4O3
(1S)-1-(2,5-dimethoxyphenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol
—— (1S)-1-(2-fluorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol —— C18H14F4N4O
(1S)-1-(2-fluorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol
—— (2S)-N-[3-[[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]phenyl]oxolane-2-carboxamide —— C22H20F3N5O2
(2S)-N-[3-[[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]phenyl]oxolane-2-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-5-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]sulfanyl-1,3,4-thiadiazol-2-amine —— C17H15F3N6OS2
N-[[(2S)-oxolan-2-yl]methyl]-5-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]sulfanyl-1,3,4-thiadiazol-2-amine
—— (2R,6S)-2-methyl-6-phenyl-4-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine —— C21H19F3N4O
(2R,6S)-2-methyl-6-phenyl-4-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]morpholine
—— (1R)-1-cyclohexyl-N,N-dimethyl-N'-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]ethane-1,2-diamine —— C20H26F3N5
(1R)-1-cyclohexyl-N,N-dimethyl-N'-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]ethane-1,2-diamine
—— 1-[(3R)-1-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-yl]imidazolidin-2-one —— C18H19F3N6O
1-[(3R)-1-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-yl]imidazolidin-2-one
—— N-[[(2R)-oxolan-2-yl]methyl]-5-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]sulfanyl-1,3,4-thiadiazol-2-amine —— C17H15F3N6OS2
N-[[(2R)-oxolan-2-yl]methyl]-5-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]sulfanyl-1,3,4-thiadiazol-2-amine
—— (1R)-1-(2,5-dimethoxyphenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol —— C20H19F3N4O3
(1R)-1-(2,5-dimethoxyphenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol
—— (1R)-1-(2-fluorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol —— C18H14F4N4O
(1R)-1-(2-fluorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol
—— (3S)-3-cyclohexyl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol —— C19H23F3N4O
(3S)-3-cyclohexyl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol
—— 5-chloro-N-(2,2,2-trifluoro-1-methylethyl)-6-(2,4,6-trifluorophenyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C14H8ClF6N5
5-chloro-N-(2,2,2-trifluoro-1-methylethyl)-6-(2,4,6-trifluorophenyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— N-[(2S)-2-hydroxypropyl]-3-[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]oxybenzamide —— C20H17F3N4O3
N-[(2S)-2-hydroxypropyl]-3-[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]oxybenzamide
—— 4-[7-(2,4-Dichlorophenyl)-2-ethylpyrazolo[1,5-a]pyrimidin-3-yl]pentanamide —— C19H20Cl2N4O
4-[7-(2,4-Dichlorophenyl)-2-ethylpyrazolo[1,5-a]pyrimidin-3-yl]pentanamide
—— N-[(2R)-2-hydroxypropyl]-3-[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]oxybenzamide —— C20H17F3N4O3
N-[(2R)-2-hydroxypropyl]-3-[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]oxybenzamide
—— (1R)-1-(4-chlorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol —— C18H14ClF3N4O
(1R)-1-(4-chlorophenyl)-2-[[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]ethanol
—— 4-[(2S)-2-(1,3-benzodioxol-5-yl)pyrrolidin-1-yl]-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine —— C21H17F3N4O2
4-[(2S)-2-(1,3-benzodioxol-5-yl)pyrrolidin-1-yl]-2-pyridin-4-yl-6-(trifluoromethyl)pyrimidine
—— (3R)-3-cyclohexyl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol —— C19H23F3N4O
(3R)-3-cyclohexyl-3-[[2-pyridin-2-yl-6-(trifluoromethyl)pyrimidin-4-yl]amino]propan-1-ol
—— (1S)-1-cyclohexyl-N,N-dimethyl-N'-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]ethane-1,2-diamine —— C20H26F3N5
(1S)-1-cyclohexyl-N,N-dimethyl-N'-[2-pyridin-4-yl-6-(trifluoromethyl)pyrimidin-4-yl]ethane-1,2-diamine
—— 4-[6-(4-Fluorophenyl)pyridazin-3-yl]-1,4-diazabicyclo[3.2.2]nonane —— C17H19FN4
4-[6-(4-Fluorophenyl)pyridazin-3-yl]-1,4-diazabicyclo[3.2.2]nonane
—— 2-(6-Methyl-2-oxo-3-phenethylamino-2H-pyrazin-1-yl)-N-pyridin-2-ylmethyl-acetamide —— C21H23N5O2
2-(6-Methyl-2-oxo-3-phenethylamino-2H-pyrazin-1-yl)-N-pyridin-2-ylmethyl-acetamide
—— N-benzyl-4-(fluoromethyl)-6-(4-methylsulfonylphenyl)pyrimidin-2-amine —— C19H18FN3O2S
N-benzyl-4-(fluoromethyl)-6-(4-methylsulfonylphenyl)pyrimidin-2-amine
—— 6-(4-fluoro-3-methylphenyl)-2-isobutyl-4-(4-methyl-1-piperazinyl)methyl-2H-pyridazin-3-one —— C21H29FN4O
6-(4-fluoro-3-methylphenyl)-2-isobutyl-4-(4-methyl-1-piperazinyl)methyl-2H-pyridazin-3-one
—— 2-[cyclopropyl-[4-(4-methoxyphenyl)-6-methylimidazo[4,5-c]pyridazin-7-yl]methyl]-4-methyl-3H-1,2-oxazole —— C21H23N5O2
2-[cyclopropyl-[4-(4-methoxyphenyl)-6-methylimidazo[4,5-c]pyridazin-7-yl]methyl]-4-methyl-3H-1,2-oxazole
—— 2-[[(1R,2R)-2-(dimethylamino)cyclopentyl]amino]-4-(3-methylanilino)-6-oxo-1H-pyrimidine-5-carboxamide —— C19H26N6O2
2-[[(1R,2R)-2-(dimethylamino)cyclopentyl]amino]-4-(3-methylanilino)-6-oxo-1H-pyrimidine-5-carboxamide
—— N-[3-(2,6-difluorophenyl)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]methanesulfonamide —— C14H13F2N5O3S
N-[3-(2,6-difluorophenyl)-1-methyl-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]methanesulfonamide
—— Ethyl 4-(2-chlorophenyl)-6-methyl-2-(thiazol-2-yl)-1,4-dihydropyrimidine-5-carboxylate —— C17H16ClN3O2S
Ethyl 4-(2-chlorophenyl)-6-methyl-2-(thiazol-2-yl)-1,4-dihydropyrimidine-5-carboxylate
—— 1-[4-[[2-Amino-5-[(3-fluorophenyl)methyl]-6-methylpyrimidin-4-yl]amino]oxan-4-yl]ethanone —— C19H23FN4O2
1-[4-[[2-Amino-5-[(3-fluorophenyl)methyl]-6-methylpyrimidin-4-yl]amino]oxan-4-yl]ethanone
—— (Z)-2-phenyl-N-[3-(6-pyrrolidin-1-ylpyridazin-3-yl)phenyl]ethenesulfonamide —— C22H22N4O2S
(Z)-2-phenyl-N-[3-(6-pyrrolidin-1-ylpyridazin-3-yl)phenyl]ethenesulfonamide
—— 4-[4-[4-[(1R)-1-methoxyethyl]phenyl]-6-methylpyrimidin-2-yl]morpholine —— C18H23N3O2
4-[4-[4-[(1R)-1-methoxyethyl]phenyl]-6-methylpyrimidin-2-yl]morpholine
—— 4-[6-[4-[(1S)-1-piperidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine —— C21H28N4S
4-[6-[4-[(1S)-1-piperidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine
—— 4-[4-[4-[(1S)-1-methoxyethyl]phenyl]-6-methylpyrimidin-2-yl]morpholine —— C18H23N3O2
4-[4-[4-[(1S)-1-methoxyethyl]phenyl]-6-methylpyrimidin-2-yl]morpholine