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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-2-propan-2-ylpyrimidine-5-carboxamide —— C14H22N4O4S
N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-2-propan-2-ylpyrimidine-5-carboxamide
—— 2-(dimethylamino)-4-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]pyrimidine-5-carboxamide —— C14H23N5O4S
2-(dimethylamino)-4-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]pyrimidine-5-carboxamide
—— 2-(cyclobutylmethyl)-3-ethyl-5-[2-(2-methoxyethoxy)-5-(4-methylpiperazin-1-yl)sulfonylpyridin-3-yl]-6H-pyrazolo[4,3-d]pyrimidin-7-one —— C25H35N7O5S
2-(cyclobutylmethyl)-3-ethyl-5-[2-(2-methoxyethoxy)-5-(4-methylpiperazin-1-yl)sulfonylpyridin-3-yl]-6H-pyrazolo[4,3-d]pyrimidin-7-one
—— 2-methyl-4-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-1H-pyrimidin-6-one —— C19H27N3O2
2-methyl-4-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-1H-pyrimidin-6-one
—— 5-[2-butyl-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-3-yl]-N-methylpyrimidin-2-amine —— C15H22N6O
5-[2-butyl-5-[(3S)-oxolan-3-yl]-1,2,4-triazol-3-yl]-N-methylpyrimidin-2-amine
—— 5-[2-butyl-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-3-yl]-N-methylpyrimidin-2-amine —— C15H22N6O
5-[2-butyl-5-[(3R)-oxolan-3-yl]-1,2,4-triazol-3-yl]-N-methylpyrimidin-2-amine
—— N-cyclopropyl-6-[3-[(1S)-1-methoxyethyl]phenyl]pyridazin-3-amine —— C16H19N3O
N-cyclopropyl-6-[3-[(1S)-1-methoxyethyl]phenyl]pyridazin-3-amine
—— 6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N-propan-2-ylpyridazin-3-amine —— C17H24N4
6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N-propan-2-ylpyridazin-3-amine
—— 2-methyl-4-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-1H-pyrimidin-6-one —— C19H27N3O2
2-methyl-4-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-1H-pyrimidin-6-one
—— (6R)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one —— C8H11N3O
(6R)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one
—— 5-methyl-pyridine-2-sulfonic acid [2-[2-(2-hydroxy-ethoxy)-pyridin-4-yl]-6-methoxy-5-(2-methoxy-phenoxy)-pyrimidin-4-yl]-amide —— C25H25N5O7S
5-methyl-pyridine-2-sulfonic acid [2-[2-(2-hydroxy-ethoxy)-pyridin-4-yl]-6-methoxy-5-(2-methoxy-phenoxy)-pyrimidin-4-yl]-amide
—— 4-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]-6-propan-2-yloxypyrimidin-2-amine —— C19H26N4O2
4-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]-6-propan-2-yloxypyrimidin-2-amine
—— (6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine —— C8H9ClN2
(6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine
—— 4-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]-6-propan-2-yloxypyrimidin-2-amine —— C19H26N4O2
4-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]-6-propan-2-yloxypyrimidin-2-amine
—— 4-[(3R)-1-(4-methyl-2-pyridin-3-ylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H20N6O2
4-[(3R)-1-(4-methyl-2-pyridin-3-ylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 4-[(3S)-1-(4-methyl-2-pyridin-3-ylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H20N6O2
4-[(3S)-1-(4-methyl-2-pyridin-3-ylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— N-cyclopropyl-6-[3-[(1R)-1-methoxyethyl]phenyl]pyridazin-3-amine —— C16H19N3O
N-cyclopropyl-6-[3-[(1R)-1-methoxyethyl]phenyl]pyridazin-3-amine
—— (6R)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine —— C8H9ClN2
(6R)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine
—— (6R)-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one —— C8H10N2O
(6R)-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one
—— (6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-amine —— C8H10ClN3
(6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-amine
—— (6S)-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one —— C8H10N2O
(6S)-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one
—— (6S)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one —— C8H11N3O
(6S)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one
—— N-[(4-carbamimidoylphenyl)methyl]-2-[6-oxo-5-(propan-2-ylamino)-2-pyridin-3-ylpyrimidin-1-yl]acetamide;2,2,2-trifluoroacetic acid —— 2C2HF3O2*C22H25N7O2
N-[(4-carbamimidoylphenyl)methyl]-2-[6-oxo-5-(propan-2-ylamino)-2-pyridin-3-ylpyrimidin-1-yl]acetamide;2,2,2-trifluoroacetic acid
—— 2-piperazin-1-yl-4-o-tolyl-pyrimidine-5-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide —— C26H25F6N5O
2-piperazin-1-yl-4-o-tolyl-pyrimidine-5-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide
—— N-[(4-carbamimidoylphenyl)methyl]-2-[6-oxo-5-(propan-2-ylamino)-2-pyridin-3-ylpyrimidin-1-yl]acetamide —— C22H25N7O2
N-[(4-carbamimidoylphenyl)methyl]-2-[6-oxo-5-(propan-2-ylamino)-2-pyridin-3-ylpyrimidin-1-yl]acetamide
—— 4-[6-[3-[(1S)-1-pyrrolidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine —— C20H26N4S
4-[6-[3-[(1S)-1-pyrrolidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine
—— 2-[2-(aminomethyl)-4-methoxyphenyl]-5-ethyl-N-[5-(2-sulfamoylphenyl)pyrimidin-2-yl]pyrazole-3-carboxamide —— C24H25N7O4S
2-[2-(aminomethyl)-4-methoxyphenyl]-5-ethyl-N-[5-(2-sulfamoylphenyl)pyrimidin-2-yl]pyrazole-3-carboxamide
—— 4-[6-[3-[(1R)-1-pyrrolidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine —— C20H26N4S
4-[6-[3-[(1R)-1-pyrrolidin-1-ylethyl]phenyl]pyridazin-3-yl]thiomorpholine
—— 6-[[Benzyl(methyl)amino]methyl]-1-[(2-fluorophenyl)methyl]-3-(3-methoxyphenyl)-2-methylimidazo[1,5-a]pyrimidin-4-one —— C30H29FN4O2
6-[[Benzyl(methyl)amino]methyl]-1-[(2-fluorophenyl)methyl]-3-(3-methoxyphenyl)-2-methylimidazo[1,5-a]pyrimidin-4-one
—— (4S)-5-bromo-4-ethyl-1,4-dihydropyrimidine —— C6H9BrN2
(4S)-5-bromo-4-ethyl-1,4-dihydropyrimidine
—— (4R)-5-bromo-4-ethyl-1,4-dihydropyrimidine —— C6H9BrN2
(4R)-5-bromo-4-ethyl-1,4-dihydropyrimidine
—— (3S)-1-methyl-3-propan-2-yl-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one —— C18H21N5O2
(3S)-1-methyl-3-propan-2-yl-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one
—— 2-pyridin-4-yl-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]pyrimidine-5-carboxamide —— C17H12F3N5O
2-pyridin-4-yl-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]pyrimidine-5-carboxamide
—— 2-pyridin-4-yl-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]pyrimidine-5-carboxamide —— C17H12F3N5O
2-pyridin-4-yl-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]pyrimidine-5-carboxamide
—— 2-cyclopropyl-6-oxo-N-[(3R)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide —— C18H20N4O3S
2-cyclopropyl-6-oxo-N-[(3R)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide
—— (3R)-1-methyl-3-propan-2-yl-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one —— C18H21N5O2
(3R)-1-methyl-3-propan-2-yl-4-(2-pyridin-4-ylpyrimidine-5-carbonyl)piperazin-2-one
—— N-[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C20H21N5O2
N-[(2R)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— 2-(methylamino)-N-[(1R)-1-(4-propylphenyl)ethyl]pyrimidine-5-carboxamide —— C17H22N4O
2-(methylamino)-N-[(1R)-1-(4-propylphenyl)ethyl]pyrimidine-5-carboxamide
—— N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]imidazo[1,2-a]pyrimidine-2-carboxamide —— C21H25N5O
N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
—— 2-(propan-2-ylamino)-N-[(3S)-thiolan-3-yl]pyrimidine-5-carboxamide —— C12H18N4OS
2-(propan-2-ylamino)-N-[(3S)-thiolan-3-yl]pyrimidine-5-carboxamide
—— 2-cyclopropyl-6-oxo-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide —— C18H20N4O3S
2-cyclopropyl-6-oxo-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrimidine-5-carboxamide
—— N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide —— C17H22N6O
N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
—— N-[[(2S)-morpholin-2-yl]methyl]-4-propylpyrimidine-5-carboxamide —— C13H20N4O2
N-[[(2S)-morpholin-2-yl]methyl]-4-propylpyrimidine-5-carboxamide
—— 2-(propan-2-ylamino)-N-[(3R)-thiolan-3-yl]pyrimidine-5-carboxamide —— C12H18N4OS
2-(propan-2-ylamino)-N-[(3R)-thiolan-3-yl]pyrimidine-5-carboxamide
—— N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide —— C20H21N5O2
N-[(2S)-2-(furan-2-yl)-2-pyrrolidin-1-ylethyl]-2-pyridin-4-ylpyrimidine-5-carboxamide
—— 6-[(2-Fluorophenyl)methyl]-4-(3-methoxyphenyl)-5-methyl-2-[2-[methyl(2-pyridin-2-ylethyl)amino]ethyl]pyridazin-3-one —— C29H31FN4O2
6-[(2-Fluorophenyl)methyl]-4-(3-methoxyphenyl)-5-methyl-2-[2-[methyl(2-pyridin-2-ylethyl)amino]ethyl]pyridazin-3-one
—— 6-[(6R)-6-hydroxy-4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C16H20N6O2
6-[(6R)-6-hydroxy-4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide —— C17H22N6O
N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
—— 6-[(6R)-6-hydroxy-4-(3-oxo-1,2-oxazole-5-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C14H16N6O5
6-[(6R)-6-hydroxy-4-(3-oxo-1,2-oxazole-5-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— N-[(2S)-2-(azepan-1-yl)-2-phenylethyl]imidazo[1,2-a]pyrimidine-2-carboxamide —— C21H25N5O
N-[(2S)-2-(azepan-1-yl)-2-phenylethyl]imidazo[1,2-a]pyrimidine-2-carboxamide