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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-N-[4-(2-methyl-4-oxoquinazolin-3-yl)phenyl]-1-pyrrolidin-1-ylsulfonylpiperidine-3-carboxamide —— C25H29N5O4S
(3S)-N-[4-(2-methyl-4-oxoquinazolin-3-yl)phenyl]-1-pyrrolidin-1-ylsulfonylpiperidine-3-carboxamide
—— 2-benzylsulfanyl-6,6-dimethyl-9-phenyl-1,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4OS
2-benzylsulfanyl-6,6-dimethyl-9-phenyl-1,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— N-[(2S)-butan-2-yl]-2-[3-(4-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide —— C22H20FN3O2S2
N-[(2S)-butan-2-yl]-2-[3-(4-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide
—— (3R)-N-[4-(2-methyl-4-oxoquinazolin-3-yl)phenyl]-1-pyrrolidin-1-ylsulfonylpiperidine-3-carboxamide —— C25H29N5O4S
(3R)-N-[4-(2-methyl-4-oxoquinazolin-3-yl)phenyl]-1-pyrrolidin-1-ylsulfonylpiperidine-3-carboxamide
—— 2-[3-(4-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C23H20ClN3O3S2
2-[3-(4-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[3-(2-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C23H20ClN3O3S2
2-[3-(2-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide —— C23H21N3O3S2
N-[[(2R)-oxolan-2-yl]methyl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide
—— N-[(2S)-butan-2-yl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide —— C22H21N3O2S2
N-[(2S)-butan-2-yl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide
—— 2-[3-(2-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C23H20ClN3O3S2
2-[3-(2-chlorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 7,18,19-Trimethoxy-22-oxo-1,3,15-triazapentacyclo[12.8.0.02,11.04,9.016,21]docosa-2(11),3,5,7,9,12,14,16,18,20-decaene-13-carbonitrile —— C23H16N4O4
7,18,19-Trimethoxy-22-oxo-1,3,15-triazapentacyclo[12.8.0.02,11.04,9.016,21]docosa-2(11),3,5,7,9,12,14,16,18,20-decaene-13-carbonitrile
—— 2-[3-(2-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C23H20FN3O3S2
2-[3-(2-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-[(2S)-butan-2-yl]-2-[3-(2-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide —— C22H20FN3O2S2
N-[(2S)-butan-2-yl]-2-[3-(2-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-[3-(4-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide —— C22H20FN3O2S2
N-[(2R)-butan-2-yl]-2-[3-(4-fluorophenyl)-5-oxo-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide —— C22H21N3O2S2
N-[(2R)-butan-2-yl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide —— C23H21N3O3S2
N-[[(2S)-oxolan-2-yl]methyl]-2-(5-oxo-3-phenyl-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-4-yl)acetamide
—— 9-(4-chlorophenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H15ClN4OS
9-(4-chlorophenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— ethyl 1-[(2R)-2-(4-oxo-3-phenylquinazolin-2-yl)sulfanylpropanoyl]piperidine-4-carboxylate —— C25H27N3O4S
ethyl 1-[(2R)-2-(4-oxo-3-phenylquinazolin-2-yl)sulfanylpropanoyl]piperidine-4-carboxylate
—— ethyl 1-[(2S)-2-(4-oxo-3-phenylquinazolin-2-yl)sulfanylpropanoyl]piperidine-4-carboxylate —— C25H27N3O4S
ethyl 1-[(2S)-2-(4-oxo-3-phenylquinazolin-2-yl)sulfanylpropanoyl]piperidine-4-carboxylate
—— [2-oxo-2-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl] 2-(4-oxo-3H-phthalazin-1-yl)acetate —— C21H17N3O5
[2-oxo-2-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl] 2-(4-oxo-3H-phthalazin-1-yl)acetate
—— 3-[2-[[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]amino]-2-oxoethyl]-4-oxophthalazine-1-carboxamide —— C23H26N4O3
3-[2-[[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]amino]-2-oxoethyl]-4-oxophthalazine-1-carboxamide
—— [3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl 2-(4-oxo-3H-phthalazin-1-yl)acetate —— C21H16F2N4O6
[3-[4-(difluoromethoxy)-3-methoxyphenyl]-1,2,4-oxadiazol-5-yl]methyl 2-(4-oxo-3H-phthalazin-1-yl)acetate
—— N-[[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H31N7O4S
N-[[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— [(2R)-1-oxo-1-[4-(trifluoromethoxy)anilino]propan-2-yl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate —— C22H20F3N3O5
[(2R)-1-oxo-1-[4-(trifluoromethoxy)anilino]propan-2-yl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate
—— 2-(6-bromo-4-oxo-3-propylquinazolin-2-yl)sulfanyl-N-methyl-N-[(1R)-1-phenylethyl]acetamide —— C22H24BrN3O2S
2-(6-bromo-4-oxo-3-propylquinazolin-2-yl)sulfanyl-N-methyl-N-[(1R)-1-phenylethyl]acetamide
—— [2-[[(1R)-1-(2-methoxyphenyl)ethyl]amino]-2-oxoethyl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate —— C23H25N3O5
[2-[[(1R)-1-(2-methoxyphenyl)ethyl]amino]-2-oxoethyl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate
—— 2-[(4-benzyl-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]-N-[(1R)-1-phenylbutyl]acetamide —— C28H27N5O2S
2-[(4-benzyl-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]-N-[(1R)-1-phenylbutyl]acetamide
—— N-methyl-2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide —— C26H32N4O3S
N-methyl-2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide
—— 2-[3-(4-methoxyphenyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylbutyl]acetamide —— C27H27N3O3S
2-[3-(4-methoxyphenyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylbutyl]acetamide
—— 2-[(4-benzyl-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]-N-methyl-N-[(1R)-1-phenylethyl]acetamide —— C27H25N5O2S
2-[(4-benzyl-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]-N-methyl-N-[(1R)-1-phenylethyl]acetamide
—— 2-[[4-(3-methoxyphenyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-[(1S)-1-phenylethyl]acetamide —— C27H25N5O3S
2-[[4-(3-methoxyphenyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-[(1S)-1-phenylethyl]acetamide
—— 2-[[4-(3-methoxyphenyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-[(1R)-1-phenylethyl]acetamide —— C27H25N5O3S
2-[[4-(3-methoxyphenyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-[(1R)-1-phenylethyl]acetamide
—— N-methyl-2-[4-oxo-3-[(1R)-1-phenylethyl]quinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylethyl]acetamide —— C27H27N3O2S
N-methyl-2-[4-oxo-3-[(1R)-1-phenylethyl]quinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylethyl]acetamide
—— N-(4-methyl-3-sulfamoylphenyl)-2-[4-oxo-3-[[(2R)-oxolan-2-yl]methyl]quinazolin-2-yl]sulfanylacetamide —— C22H24N4O5S2
N-(4-methyl-3-sulfamoylphenyl)-2-[4-oxo-3-[[(2R)-oxolan-2-yl]methyl]quinazolin-2-yl]sulfanylacetamide
—— 2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylbutyl]acetamide —— C27H34N4O3S
2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylbutyl]acetamide
—— [2-[[(1S)-1-(2-methoxyphenyl)ethyl]amino]-2-oxoethyl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate —— C23H25N3O5
[2-[[(1S)-1-(2-methoxyphenyl)ethyl]amino]-2-oxoethyl] 4-oxo-3-propan-2-ylphthalazine-1-carboxylate
—— 2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylbutyl]acetamide —— C27H34N4O3S
2-[3-(3-morpholin-4-ylpropyl)-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylbutyl]acetamide
—— N-methyl-2-[3-[(4-methylphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylethyl]acetamide —— C27H27N3O2S
N-methyl-2-[3-[(4-methylphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-[(1R)-1-phenylethyl]acetamide
—— N-[2-(3,4-dimethoxyphenyl)ethyl]-6-(4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)hexanamide —— C24H29N3O4S
N-[2-(3,4-dimethoxyphenyl)ethyl]-6-(4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)hexanamide
—— (2S)-2-[[4-(3-methoxypropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-phenylpropanamide —— C23H25N5O3S
(2S)-2-[[4-(3-methoxypropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]-N-methyl-N-phenylpropanamide
—— N-methyl-2-[4-oxo-3-[(1R)-1-phenylethyl]quinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide —— C27H27N3O2S
N-methyl-2-[4-oxo-3-[(1R)-1-phenylethyl]quinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide
—— N-methyl-2-[3-[(4-methylphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide —— C27H27N3O2S
N-methyl-2-[3-[(4-methylphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanyl-N-[(1S)-1-phenylethyl]acetamide
—— 2-[3-(3-chloro-4-fluorophenyl)-4-oxoquinazolin-2-yl]sulfanyl-N-methyl-N-[(1S)-1-phenylethyl]acetamide —— C25H21ClFN3O2S
2-[3-(3-chloro-4-fluorophenyl)-4-oxoquinazolin-2-yl]sulfanyl-N-methyl-N-[(1S)-1-phenylethyl]acetamide
—— N-(4-methyl-3-sulfamoylphenyl)-2-[4-oxo-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-2-yl]sulfanylacetamide —— C22H24N4O5S2
N-(4-methyl-3-sulfamoylphenyl)-2-[4-oxo-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-2-yl]sulfanylacetamide
—— 3-(1,3-benzodioxol-5-ylmethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C24H26N4O4S
3-(1,3-benzodioxol-5-ylmethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— 2-[3-[4-(difluoromethoxy)phenyl]-4-oxoquinazolin-2-yl]sulfanyl-N-methyl-N-[(1R)-1-phenylethyl]acetamide —— C26H23F2N3O3S
2-[3-[4-(difluoromethoxy)phenyl]-4-oxoquinazolin-2-yl]sulfanyl-N-methyl-N-[(1R)-1-phenylethyl]acetamide
—— N-(4-chloro-2-nitrophenyl)-2-quinazolin-4-ylsulfanylacetamide —— C16H11ClN4O3S
N-(4-chloro-2-nitrophenyl)-2-quinazolin-4-ylsulfanylacetamide
—— 2-(7-chloro-4-oxo-3-prop-2-enylquinazolin-2-yl)sulfanyl-N-[(1S)-1-phenylbutyl]acetamide —— C23H24ClN3O2S
2-(7-chloro-4-oxo-3-prop-2-enylquinazolin-2-yl)sulfanyl-N-[(1S)-1-phenylbutyl]acetamide
—— 2-(7-chloro-4-oxo-3-prop-2-enylquinazolin-2-yl)sulfanyl-N-[(1R)-1-phenylbutyl]acetamide —— C23H24ClN3O2S
2-(7-chloro-4-oxo-3-prop-2-enylquinazolin-2-yl)sulfanyl-N-[(1R)-1-phenylbutyl]acetamide
—— 6-bromo-3-(4-ethylphenyl)-4-hydroxy-N-[2-methyl-3-(4-methylpiperidin-1-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinazoline-4-carboxamide —— C27H35BrN4O3
6-bromo-3-(4-ethylphenyl)-4-hydroxy-N-[2-methyl-3-(4-methylpiperidin-1-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinazoline-4-carboxamide
—— 6-bromo-3-(4-chlorophenyl)-N-[3-(diethylamino)-2-methylpropyl]-4-hydroxy-2-oxo-1,2,3,4-tetrahydroquinazoline-4-carboxamide —— C23H28BrClN4O3
6-bromo-3-(4-chlorophenyl)-N-[3-(diethylamino)-2-methylpropyl]-4-hydroxy-2-oxo-1,2,3,4-tetrahydroquinazoline-4-carboxamide