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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Chloro-2-[2-[(2,6-diamino-5-methylsulfonylpyrimidin-4-yl)amino]ethyl]-3-(3,5-difluorophenyl)quinazolin-4-one —— C21H18ClF2N7O3S
5-Chloro-2-[2-[(2,6-diamino-5-methylsulfonylpyrimidin-4-yl)amino]ethyl]-3-(3,5-difluorophenyl)quinazolin-4-one
—— 2,4-Diamino-6-[3-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]propylamino]pyrimidine-5-carbonitrile —— C23H20F2N8O
2,4-Diamino-6-[3-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]propylamino]pyrimidine-5-carbonitrile
—— tert-butyl N-[5-chloro-3-(3,5-dimethoxyphenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C23H26ClN3O5
tert-butyl N-[5-chloro-3-(3,5-dimethoxyphenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— tert-butyl N-[2-[3-(3,5-difluorophenyl)-5,6-difluoro-4-oxoquinazolin-2-yl]ethyl]carbamate —— C21H19F4N3O3
tert-butyl N-[2-[3-(3,5-difluorophenyl)-5,6-difluoro-4-oxoquinazolin-2-yl]ethyl]carbamate
—— 2-(2-Aminoethyl)-5-fluoro-3-[3-fluoro-5-(trifluoromethyl)phenyl]quinazolin-4-one —— C17H12F5N3O
2-(2-Aminoethyl)-5-fluoro-3-[3-fluoro-5-(trifluoromethyl)phenyl]quinazolin-4-one
—— tert-butyl N-(5-carbamoyl-4-oxo-3-phenylquinazolin-2-yl)-N-ethylcarbamate —— C22H24N4O4
tert-butyl N-(5-carbamoyl-4-oxo-3-phenylquinazolin-2-yl)-N-ethylcarbamate
—— 2-(2-Aminoethyl)-5-chloro-3-[5-(difluoromethyl)-2-methylphenyl]quinazolin-4-one —— C18H16ClF2N3O
2-(2-Aminoethyl)-5-chloro-3-[5-(difluoromethyl)-2-methylphenyl]quinazolin-4-one
—— 2,4-Diamino-6-[2-[5-chloro-3-(3,4-difluoro-2-methylphenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C22H17ClF2N8O
2,4-Diamino-6-[2-[5-chloro-3-(3,4-difluoro-2-methylphenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 2-[2-[[6-Amino-5-[2-(4-ethylpyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-3-phenylquinazolin-4-one —— C29H24ClN7O
2-[2-[[6-Amino-5-[2-(4-ethylpyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-3-phenylquinazolin-4-one
—— 3-[2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-4-oxoquinazolin-3-yl]benzonitrile —— C28H18ClFN8O
3-[2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-4-oxoquinazolin-3-yl]benzonitrile
—— 2-(2-Aminoethyl)-5-chloro-3-(3-chlorophenyl)quinazolin-4-one —— C16H13Cl2N3O
2-(2-Aminoethyl)-5-chloro-3-(3-chlorophenyl)quinazolin-4-one
—— tert-butyl N-[3-[3-(3,5-difluorophenyl)-5-fluoro-4-oxoquinazolin-2-yl]propyl]carbamate —— C22H22F3N3O3
tert-butyl N-[3-[3-(3,5-difluorophenyl)-5-fluoro-4-oxoquinazolin-2-yl]propyl]carbamate
—— 2-(3-Aminopropyl)-5,8-difluoro-3-phenylquinazolin-4-one —— C17H15F2N3O
2-(3-Aminopropyl)-5,8-difluoro-3-phenylquinazolin-4-one
—— 2,4-Diamino-6-[2-[3-(3,5-difluorophenyl)-5-methylsulfonyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C22H18F2N8O3S
2,4-Diamino-6-[2-[3-(3,5-difluorophenyl)-5-methylsulfonyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— tert-butyl N-(5-chloro-8-methyl-4-oxo-3-phenylquinazolin-2-yl)-N-ethylcarbamate —— C22H24ClN3O3
tert-butyl N-(5-chloro-8-methyl-4-oxo-3-phenylquinazolin-2-yl)-N-ethylcarbamate
—— tert-butyl N-[2-[5-chloro-4-oxo-3-(3-propan-2-ylphenyl)quinazolin-2-yl]ethyl]carbamate —— C24H28ClN3O3
tert-butyl N-[2-[5-chloro-4-oxo-3-(3-propan-2-ylphenyl)quinazolin-2-yl]ethyl]carbamate
—— 2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-8-methyl-3-phenylquinazolin-4-one —— C28H21ClFN7O
2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-8-methyl-3-phenylquinazolin-4-one
—— 2-[5-Chloro-3-(5-fluoro-2-methylphenyl)-4-oxoquinazolin-2-yl]ethylcarbamic acid —— C18H15ClFN3O3
2-[5-Chloro-3-(5-fluoro-2-methylphenyl)-4-oxoquinazolin-2-yl]ethylcarbamic acid
—— 2-(3-Aminopropyl)-3-(3,5-difluorophenyl)-6,8-difluoroquinazolin-4-one —— C17H13F4N3O
2-(3-Aminopropyl)-3-(3,5-difluorophenyl)-6,8-difluoroquinazolin-4-one
—— tert-butyl N-[2-[3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]ethyl]carbamate —— C21H21F2N3O3
tert-butyl N-[2-[3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]ethyl]carbamate
—— 2-(2-Aminoethyl)-3-(3,5-difluorophenyl)-5-fluoro-8-methylquinazolin-4-one —— C17H14F3N3O
2-(2-Aminoethyl)-3-(3,5-difluorophenyl)-5-fluoro-8-methylquinazolin-4-one
—— 3-[2-(2-Aminoethyl)-5-chloro-8-fluoro-4-oxoquinazolin-3-yl]benzonitrile —— C17H12ClFN4O
3-[2-(2-Aminoethyl)-5-chloro-8-fluoro-4-oxoquinazolin-3-yl]benzonitrile
—— 2,4-Diamino-6-[2-[5-chloro-3-[3-(difluoromethyl)-5-methoxyphenyl]-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C23H19ClF2N8O2
2,4-Diamino-6-[2-[5-chloro-3-[3-(difluoromethyl)-5-methoxyphenyl]-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— tert-butyl N-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]-N-propylcarbamate —— C23H25F2N3O3
tert-butyl N-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]-N-propylcarbamate
—— 3-[2-(2-Aminoethyl)-5,8-difluoro-4-oxoquinazolin-3-yl]benzonitrile —— C17H12F2N4O
3-[2-(2-Aminoethyl)-5,8-difluoro-4-oxoquinazolin-3-yl]benzonitrile
—— 2,4-Diamino-6-[2-[3-(3-cyano-5-fluorophenyl)-5-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C23H18FN9O
2,4-Diamino-6-[2-[3-(3-cyano-5-fluorophenyl)-5-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 2,4-Diamino-6-[2-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C22H18F2N8O
2,4-Diamino-6-[2-[3-(3,5-difluorophenyl)-8-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— Tert-butyl-[4-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-3-methylbutyl]carbamic acid —— C24H26ClF2N3O3
Tert-butyl-[4-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-3-methylbutyl]carbamic acid
—— 2,4-Diamino-6-[2-[3-(3-cyano-5-fluorophenyl)-5-fluoro-8-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C23H17F2N9O
2,4-Diamino-6-[2-[3-(3-cyano-5-fluorophenyl)-5-fluoro-8-methyl-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 3-[2-(2-Aminoethyl)-5-chloro-8-fluoro-4-oxoquinazolin-3-yl]-5-fluorobenzonitrile —— C17H11ClF2N4O
3-[2-(2-Aminoethyl)-5-chloro-8-fluoro-4-oxoquinazolin-3-yl]-5-fluorobenzonitrile
—— 6-[2-[4-Amino-6-[2-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidin-5-yl]ethynyl]pyridine-3-carboxamide —— C28H19ClF2N8O2
6-[2-[4-Amino-6-[2-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidin-5-yl]ethynyl]pyridine-3-carboxamide
—— tert-butyl N-[3-[3,5-bis(difluoromethyl)phenyl]-5-chloro-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C23H22ClF4N3O3
tert-butyl N-[3-[3,5-bis(difluoromethyl)phenyl]-5-chloro-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— 2-(2-Aminoethyl)-5-chloro-3-(2,6-difluorophenyl)quinazolin-4-one —— C16H12ClF2N3O
2-(2-Aminoethyl)-5-chloro-3-(2,6-difluorophenyl)quinazolin-4-one
—— tert-butyl N-[2-[3-(3,5-difluorophenyl)-8-ethyl-4-oxoquinazolin-2-yl]ethyl]carbamate —— C23H25F2N3O3
tert-butyl N-[2-[3-(3,5-difluorophenyl)-8-ethyl-4-oxoquinazolin-2-yl]ethyl]carbamate
—— 2,4-Diamino-6-[2-(6-fluoro-4-oxo-3-phenylquinazolin-2-yl)ethylamino]pyrimidine-5-carbonitrile —— C21H17FN8O
2,4-Diamino-6-[2-(6-fluoro-4-oxo-3-phenylquinazolin-2-yl)ethylamino]pyrimidine-5-carbonitrile
—— 2,4-Diamino-6-[2-[3-[3-chloro-5-(difluoromethyl)phenyl]-5-fluoro-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C22H16ClF3N8O
2,4-Diamino-6-[2-[3-[3-chloro-5-(difluoromethyl)phenyl]-5-fluoro-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 2-(2-Aminoethyl)-5-(difluoromethyl)-3-[3-(difluoromethyl)-5-fluorophenyl]quinazolin-4-one —— C18H14F5N3O
2-(2-Aminoethyl)-5-(difluoromethyl)-3-[3-(difluoromethyl)-5-fluorophenyl]quinazolin-4-one
—— tert-butyl N-[3-(3,5-difluorophenyl)-6,8-difluoro-4-oxoquinazolin-2-yl]-N-propylcarbamate —— C22H21F4N3O3
tert-butyl N-[3-(3,5-difluorophenyl)-6,8-difluoro-4-oxoquinazolin-2-yl]-N-propylcarbamate
—— tert-butyl N-[5-carbamoyl-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C22H22F2N4O4
tert-butyl N-[5-carbamoyl-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— tert-butyl N-[3-(3-cyanophenyl)-6-fluoro-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C22H21FN4O3
tert-butyl N-[3-(3-cyanophenyl)-6-fluoro-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— tert-butyl N-[8-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C21H20ClF2N3O3
tert-butyl N-[8-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— 2,4-Diamino-6-[2-[8-(difluoromethyl)-4-oxo-3-phenylquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C22H18F2N8O
2,4-Diamino-6-[2-[8-(difluoromethyl)-4-oxo-3-phenylquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 2,4-Diamino-6-[3-[8-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]propylamino]pyrimidine-5-carbonitrile —— C22H17ClF2N8O
2,4-Diamino-6-[3-[8-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]propylamino]pyrimidine-5-carbonitrile
—— 2-(Oxolan-3-yl)quinazoline —— C12H12N2O
2-(Oxolan-3-yl)quinazoline
—— 2,4-Diamino-6-[[4-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-3-methylbutyl]amino]pyrimidine-5-carbonitrile —— C24H21ClF2N8O
2,4-Diamino-6-[[4-[5-chloro-3-(3,5-difluorophenyl)-4-oxoquinazolin-2-yl]-3-methylbutyl]amino]pyrimidine-5-carbonitrile
—— tert-butyl N-[5-chloro-3-[3-(difluoromethyl)-5-fluorophenyl]-4-oxoquinazolin-2-yl]-N-ethylcarbamate —— C22H21ClF3N3O3
tert-butyl N-[5-chloro-3-[3-(difluoromethyl)-5-fluorophenyl]-4-oxoquinazolin-2-yl]-N-ethylcarbamate
—— 2,4-Diamino-6-[2-[5-chloro-3-(2,3-dimethylphenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile —— C23H21ClN8O
2,4-Diamino-6-[2-[5-chloro-3-(2,3-dimethylphenyl)-4-oxoquinazolin-2-yl]ethylamino]pyrimidine-5-carbonitrile
—— 2,4-Diamino-6-[3-(5,8-difluoro-4-oxo-3-phenylquinazolin-2-yl)propylamino]pyrimidine-5-carbonitrile —— C22H18F2N8O
2,4-Diamino-6-[3-(5,8-difluoro-4-oxo-3-phenylquinazolin-2-yl)propylamino]pyrimidine-5-carbonitrile
—— 2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5,8-dichloro-3-phenylquinazolin-4-one —— C27H18Cl2FN7O
2-[2-[[6-Amino-5-[2-(5-fluoropyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5,8-dichloro-3-phenylquinazolin-4-one
—— 2-[2-[[6-Amino-5-[2-(4-methylpyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-3-phenylquinazolin-4-one —— C28H22ClN7O
2-[2-[[6-Amino-5-[2-(4-methylpyridin-2-yl)ethynyl]pyrimidin-4-yl]amino]ethyl]-5-chloro-3-phenylquinazolin-4-one