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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-phenyl-2-hydrazino-7,7-dimethyl-3,4,6,8-tetrahydro-quinazolin-5-one 1188423-25-7 C16H20N4O
4-phenyl-2-hydrazino-7,7-dimethyl-3,4,6,8-tetrahydro-quinazolin-5-one
—— 8-bromo-2-(2-chloro-4-fluorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3H)-one 1169549-87-4 C16H7BrClFN2O2
8-bromo-2-(2-chloro-4-fluorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3H)-one
—— [1-(3-fluorophenyl)-4-methylamino-4-(3-methyl-1H-indol-2-yl)-cyclohexyl]-dimethylamine 1189795-11-6 C24H30FN3
[1-(3-fluorophenyl)-4-methylamino-4-(3-methyl-1H-indol-2-yl)-cyclohexyl]-dimethylamine
—— (R)-ethyl 3-(4-(tert-butyldiphenylsilyloxymethyl)-2,6-dimethoxyphenyl)heptanoate 1192065-12-5 C34H46O5Si
(R)-ethyl 3-(4-(tert-butyldiphenylsilyloxymethyl)-2,6-dimethoxyphenyl)heptanoate
—— 1-(benzo[d][1,3]dioxol-5-yl)-N-(5-methylpyridin-2-yl)cyclopropanecarboxamide 1189328-40-2 C17H16N2O3
1-(benzo[d][1,3]dioxol-5-yl)-N-(5-methylpyridin-2-yl)cyclopropanecarboxamide
—— N-methyl-3-(naphthalene-2-sulfonamido)-3-phenyl-N-(2-(4-phenyl-4-(pyrrolidin-1-yl)cyclohexyl)ethyl)propanamide 1187961-54-1 C38H45N3O3S
N-methyl-3-(naphthalene-2-sulfonamido)-3-phenyl-N-(2-(4-phenyl-4-(pyrrolidin-1-yl)cyclohexyl)ethyl)propanamide
—— 2-[bis[2-(2,3,4,5,6-pentafluorophenyl)azanidylethyl]amino]ethyl-(2,3,4,5,6-pentafluorophenyl)azanide;bromotitanium(3+) 174735-87-6 C24H12BrF15N4Ti
2-[bis[2-(2,3,4,5,6-pentafluorophenyl)azanidylethyl]amino]ethyl-(2,3,4,5,6-pentafluorophenyl)azanide;bromotitanium(3+)
—— 7-(8-N-phenylaminooctyl)amino-2H-anthra[1,9-cd]pyrazol-6-one 1220286-88-3 C28H30N4O
7-(8-N-phenylaminooctyl)amino-2H-anthra[1,9-cd]pyrazol-6-one
—— 5-tert-butyl-3-(2-chloro-4,5-difluoro-benzyl)-7-(3,3-difluoro-pyrrolidin-1-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidine 1433359-54-6 C19H19ClF4N6
5-tert-butyl-3-(2-chloro-4,5-difluoro-benzyl)-7-(3,3-difluoro-pyrrolidin-1-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidine
—— 6-chloro-N-(3-(4,4-dimethylcyclohexyl)-4-oxo-3,4-dihydrophthalazin-6-yl)-2-methoxy-3-(pivalamidomethyl)benzamide 1436502-20-3 C30H37ClN4O4
6-chloro-N-(3-(4,4-dimethylcyclohexyl)-4-oxo-3,4-dihydrophthalazin-6-yl)-2-methoxy-3-(pivalamidomethyl)benzamide
—— N-[3-(2,4-dichlorophenyl)propyl]-3-methylthiophene-2-carboxamide 1050300-60-1 C15H15Cl2NOS
N-[3-(2,4-dichlorophenyl)propyl]-3-methylthiophene-2-carboxamide
—— 5-((1-(2-bromobenzoyl)-5-chloro-1H-indol-3-yl)methylene)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione 1424353-55-8 C20H11BrClN3O3S
5-((1-(2-bromobenzoyl)-5-chloro-1H-indol-3-yl)methylene)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
—— (Z)-4-(3-(2-(2,4-dihydroxyphenyl)-2-phenylvinyl)quinoxalin-2-yl)benzene-1,3-diol 1446432-68-3 C28H20N2O4
(Z)-4-(3-(2-(2,4-dihydroxyphenyl)-2-phenylvinyl)quinoxalin-2-yl)benzene-1,3-diol
—— (Z)-4-(4-aminobenzylidene)-2-ethoxytetrahydrofuran 1141885-00-8 C13H17NO2
(Z)-4-(4-aminobenzylidene)-2-ethoxytetrahydrofuran
—— 6-bromo-N-(2-methoxybenzyl)-4-phenoxypyridin-3-amine 1330574-85-0 C19H17BrN2O2
6-bromo-N-(2-methoxybenzyl)-4-phenoxypyridin-3-amine
—— (E)-5-(3-(2-((tert-butyldimethylsilyl)oxy)phenyl)prop-1-en-1-yl)benzene-1,2,3-triyl trimethanesulfonate 1131849-99-4 C24H34O10S3Si
(E)-5-(3-(2-((tert-butyldimethylsilyl)oxy)phenyl)prop-1-en-1-yl)benzene-1,2,3-triyl trimethanesulfonate
—— 6-chloro-2-(4'-methylphenyl)-3-{(thiophen-2-yl)methoxy}-4-oxo-4H-1-benzo-pyran 1262841-06-4 C21H15ClO3S
6-chloro-2-(4'-methylphenyl)-3-{(thiophen-2-yl)methoxy}-4-oxo-4H-1-benzo-pyran
—— (2S,4R)-N-((S)-1-(cyclopropylamino)-1,2-dioxopentan-3-yl)-1-(1-(trifluoromethyl)cyclopropanecarbonyl)-4-(2-(trifluoromethyl)phenylsulfonyl)pyrrolidine-2-carboxamide 1439403-65-2 C25H27F6N3O6S
(2S,4R)-N-((S)-1-(cyclopropylamino)-1,2-dioxopentan-3-yl)-1-(1-(trifluoromethyl)cyclopropanecarbonyl)-4-(2-(trifluoromethyl)phenylsulfonyl)pyrrolidine-2-carboxamide
—— 1-(4-ethylphenyl)-3-(4,4-diethyl-2,5-dioxoimidazolidin-1-yl)urea 1434716-49-0 C16H22N4O3
1-(4-ethylphenyl)-3-(4,4-diethyl-2,5-dioxoimidazolidin-1-yl)urea
—— 6-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3-{2-cyano-3-[tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylsulfanyl]phenyl}pyridine-2-carboxylic acid 1430845-25-2 C40H35N5O3S2
6-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3-{2-cyano-3-[tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylsulfanyl]phenyl}pyridine-2-carboxylic acid
—— (S)-2-tert-butoxy-2-(4-(4-chlorophenyl)-1-(ethyl)-2,3,6-trimethyl-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid 1436855-02-5 C24H29ClN2O3
(S)-2-tert-butoxy-2-(4-(4-chlorophenyl)-1-(ethyl)-2,3,6-trimethyl-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid
—— 6-(4-fluorophenyl)-2-{5-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]-2-methylphenyl}-N-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide 1438844-18-8 C25H25FN4O3S
6-(4-fluorophenyl)-2-{5-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]-2-methylphenyl}-N-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
—— 1'-Ethyl-1-[[2-fluoro-4-(1-methylpyrazol-4-yl)phenyl]methyl]spiro[indole-3,3'-pyrrolidine]-2-one 1426688-84-7 C24H25FN4O
1'-Ethyl-1-[[2-fluoro-4-(1-methylpyrazol-4-yl)phenyl]methyl]spiro[indole-3,3'-pyrrolidine]-2-one
—— 2-(5-difluoromethyl-furan-2-yl)-6-(3-methoxy-pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-ylamine 1221432-09-2 C18H14F2N4O2S
2-(5-difluoromethyl-furan-2-yl)-6-(3-methoxy-pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-ylamine
—— 4-chloro-N-[N-(2-oxo-3H-1,3-benzoxazol-6-yl)-N'-(4-phenylphenyl)carbamimidoyl]benzamide 1217241-01-4 C27H19ClN4O3
4-chloro-N-[N-(2-oxo-3H-1,3-benzoxazol-6-yl)-N'-(4-phenylphenyl)carbamimidoyl]benzamide
—— 2-[3-[(3S,9S,15S,18S,29S)-18-amino-15-[(3,5-difluorophenyl)methyl]-2,5,8,14,17,28-hexaoxospiro[1,4,7,13,16,27-hexazatricyclo[27.3.0.09,13]dotriacontane-6,1'-cyclobutane]-3-yl]propyl]guanidine 1421029-70-0 C40H60F2N10O6
2-[3-[(3S,9S,15S,18S,29S)-18-amino-15-[(3,5-difluorophenyl)methyl]-2,5,8,14,17,28-hexaoxospiro[1,4,7,13,16,27-hexazatricyclo[27.3.0.09,13]dotriacontane-6,1'-cyclobutane]-3-yl]propyl]guanidine
—— US10280167, Example 15 1434585-64-4 C16H13N7O
US10280167, Example 15
—— 6-[4-(4-acetylphenyl)phenyl]-2-(4-methylphenyl)-4-phenylpyridine-3-carbonitrile 102146-56-5 C33H24N2O
6-[4-(4-acetylphenyl)phenyl]-2-(4-methylphenyl)-4-phenylpyridine-3-carbonitrile
—— 1,1'-p-phenylenediamino-bis-1-deoxy-β(?)-D-glucopyranuronic acid 110443-12-4 C18H24N2O12
1,1'-p-phenylenediamino-bis-1-deoxy-β(?)-D-glucopyranuronic acid
—— N-(4-((7-chloroquinolin-4-yl)amino)phenyl)-2-(2-(4-isopropylbenzylidene)hydrazineyl)-2-oxoacetamide 1647060-38-5 C27H24ClN5O2
N-(4-((7-chloroquinolin-4-yl)amino)phenyl)-2-(2-(4-isopropylbenzylidene)hydrazineyl)-2-oxoacetamide
—— (N-tert-butyldimethylsilyl)[2-(trityloxy)ethyl]amine 1427722-36-8 C27H35NOSi
(N-tert-butyldimethylsilyl)[2-(trityloxy)ethyl]amine
—— trans-2.2.4.4-Tetramethyl-cyclobutan-diamin-(1.3) 10195-50-3 C8H18N2
trans-2.2.4.4-Tetramethyl-cyclobutan-diamin-(1.3)
—— tert-butyl 2-(cyanomethyl)-4-oxo-4-phenylbutanoate 1608491-07-1 C16H19NO3
tert-butyl 2-(cyanomethyl)-4-oxo-4-phenylbutanoate
—— —— 1402751-74-9 C36H54O3Si2
—— tert-butyl 2-[[1-[(3aR,4R,6R,6aR)-6-(hydroxymethyl)-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-2,4-dioxopyrimidin-5-yl]methyl]-3-oxobutanoate 116235-26-8 C21H30N2O9
tert-butyl 2-[[1-[(3aR,4R,6R,6aR)-6-(hydroxymethyl)-2,2-dimethyl-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-4-yl]-2,4-dioxopyrimidin-5-yl]methyl]-3-oxobutanoate
—— 2,2'-(1,4-phenylene)bis(1-(1H-indol-2-yl)buta-2,3-dien-1-ol) 1333068-47-5 C30H24N2O2
2,2'-(1,4-phenylene)bis(1-(1H-indol-2-yl)buta-2,3-dien-1-ol)
—— N-(4-bromophenyl)-exo-4-camphyl-4-hydroxybut-2(Z)-enamide 116053-24-8 C19H24BrNO2
N-(4-bromophenyl)-exo-4-camphyl-4-hydroxybut-2(Z)-enamide
—— [(1R,4R)-4-(3-Hydroxy-2,2-dimethyl-propyl)-cyclopent-2-enyl]-acetic acid 105555-28-0 C12H20O3
[(1R,4R)-4-(3-Hydroxy-2,2-dimethyl-propyl)-cyclopent-2-enyl]-acetic acid
—— 5(3)-Amino-3(5)-<(4-cyanphenyl)amino>pyrazol-4-carbonsaeure-ethylester 158590-97-7 C13H13N5O2
5(3)-Amino-3(5)-<(4-cyanphenyl)amino>pyrazol-4-carbonsaeure-ethylester
—— methyl 2-ethoxy-1,3-bis(2-methoxy-5-methylphenyl)-6-oxo-1,2,3,6-tetrahydropyrimidine-4-carboxylate 1258067-48-9 C24H28N2O6
methyl 2-ethoxy-1,3-bis(2-methoxy-5-methylphenyl)-6-oxo-1,2,3,6-tetrahydropyrimidine-4-carboxylate
—— N-cyclohexyl-3,5-dimethyl-1H-indole-2-carboxamide 1578260-98-6 C17H22N2O
N-cyclohexyl-3,5-dimethyl-1H-indole-2-carboxamide
—— (3Z)-3-[1-(4-chlorophenyl)ethylidene]-2,3-dihydro-1H-pyrrolizin-1-one 1220387-34-7 C15H12ClNO
(3Z)-3-[1-(4-chlorophenyl)ethylidene]-2,3-dihydro-1H-pyrrolizin-1-one
—— 5-Fluoro-1-(isoquinolin-8-ylmethyl)-4-oxoquinoline-3-carboxylic acid 1224510-16-0 C20H13FN2O3
5-Fluoro-1-(isoquinolin-8-ylmethyl)-4-oxoquinoline-3-carboxylic acid
—— (R)-(8-methyl-3-(2-vinylthiazol-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone 1429557-11-8 C22H19N5OS2
(R)-(8-methyl-3-(2-vinylthiazol-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone
—— 4-benzoyl-N-(5-(4-methoxybenzamido)-6-oxo-6-(6-(5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamido)hexylamino)hexyl)benzamide 1383564-33-7 C44H56N6O7S
4-benzoyl-N-(5-(4-methoxybenzamido)-6-oxo-6-(6-(5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamido)hexylamino)hexyl)benzamide
—— 4-benzyl-4-methylmorpholinium 2-ethylbutyrate 1350474-00-8 C6H11O2*C12H18NO
4-benzyl-4-methylmorpholinium 2-ethylbutyrate
—— 4-ethyl-heptane-2,6-dione 1089183-39-0 C9H16O2
4-ethyl-heptane-2,6-dione
—— 6-ethyl-3-(3-methylsulfonylanilino)-5-[[(2R)-oxolan-2-yl]methylamino]pyrazine-2-carboxamide 1254050-22-0 C19H25N5O4S
6-ethyl-3-(3-methylsulfonylanilino)-5-[[(2R)-oxolan-2-yl]methylamino]pyrazine-2-carboxamide
—— N-[1-[4-[2-(1-ethyl-2-oxopyridin-4-yl)ethynyl]phenyl]propan-2-yl]acetamide 1363426-44-1 C20H22N2O2
N-[1-[4-[2-(1-ethyl-2-oxopyridin-4-yl)ethynyl]phenyl]propan-2-yl]acetamide
—— ethyl 3-(4-(2,2-difluorovinyl)phenyl)propanoate 1501969-18-1 C13H14F2O2
ethyl 3-(4-(2,2-difluorovinyl)phenyl)propanoate