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中文名称 英文名称 CAS号 化学式 结构式图片
—— H-Phe-Gly-Trp-His-OH 1039024-99-1 C28H31N7O5
H-Phe-Gly-Trp-His-OH
—— 7-(2-methoxy-4-methoxymethoxyphenyl)-8-(2-methoxy-5-nitrophenoxymethyl)-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one 1089680-14-7 C28H31N3O8
7-(2-methoxy-4-methoxymethoxyphenyl)-8-(2-methoxy-5-nitrophenoxymethyl)-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— Methyl 3-[4-(phenylcarbamoyl)-2,3-dihydropyrido[3,2-b][1,4]oxazin-6-yl]benzoate 1214927-70-4 C22H19N3O4
Methyl 3-[4-(phenylcarbamoyl)-2,3-dihydropyrido[3,2-b][1,4]oxazin-6-yl]benzoate
—— 1-butyl-3-ethyl-7-methoxy-1H-pyrimido[5,4-c]quinoline-2,4-dione 1174226-38-0 C18H21N3O3
1-butyl-3-ethyl-7-methoxy-1H-pyrimido[5,4-c]quinoline-2,4-dione
—— US8653087, III-124 1213244-09-7 C31H34F5N9O
US8653087, III-124
—— 2-[8-[[3,5-Diethoxy-4-(4-fluorophenyl)phenyl]methyl]-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]acetamide 1254731-16-2 C27H34FN3O4
2-[8-[[3,5-Diethoxy-4-(4-fluorophenyl)phenyl]methyl]-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]acetamide
—— 4-[3-[2-(4-Bromophenyl)-3-methylbutan-2-yl]-1,2,4-oxadiazol-5-yl]-1-methylpiperazin-2-one 1360552-97-1 C18H23BrN4O2
4-[3-[2-(4-Bromophenyl)-3-methylbutan-2-yl]-1,2,4-oxadiazol-5-yl]-1-methylpiperazin-2-one
—— 2-{4-(dimethylamino)-3-[(dimethylamino)methyl]phenyl}-4,5,6,7-tetrahydro-1,3-benzothiazol-7-ol 1189353-88-5 C18H25N3OS
2-{4-(dimethylamino)-3-[(dimethylamino)methyl]phenyl}-4,5,6,7-tetrahydro-1,3-benzothiazol-7-ol
—— 4-methyl-N-[(1S)-1-phenyl-2-[[(1R)-1-phenylethyl]amino]ethyl]benzenesulfonamide 1192481-68-7 C23H26N2O2S
4-methyl-N-[(1S)-1-phenyl-2-[[(1R)-1-phenylethyl]amino]ethyl]benzenesulfonamide
—— dihomopiperidinoacetylene 1257763-21-5 C14H24N2
dihomopiperidinoacetylene
—— di(but-3-enyl)(tert-butyl)phosphine oxide 1011736-01-8 C12H23OP
di(but-3-enyl)(tert-butyl)phosphine oxide
—— 4-(4-fluorophenyl)-1-(1-(trimethylsilyl)-3-phenyl-3-p-tolylpropa-1,2-dienyl)-1H-1,2,3-triazole 1369584-24-6 C27H26FN3Si
4-(4-fluorophenyl)-1-(1-(trimethylsilyl)-3-phenyl-3-p-tolylpropa-1,2-dienyl)-1H-1,2,3-triazole
—— 3-chloro-6-(6-hydroxy-4,7-dimethoxy-1-benzofuran-5-yl)-4-phenyl-1H-pyridin-2-one 128118-52-5 C21H16ClNO5
3-chloro-6-(6-hydroxy-4,7-dimethoxy-1-benzofuran-5-yl)-4-phenyl-1H-pyridin-2-one
—— (R)-(+)-1-methoxymethoxy-4-methyldocosane 130650-51-0 C25H52O2
(R)-(+)-1-methoxymethoxy-4-methyldocosane
—— (1S,2R)-methyl 2-(4-chlorophenethyl)-1-hydroxy-3-methylenecyclohexanecarboxylate 1238619-43-6 C17H21ClO3
(1S,2R)-methyl 2-(4-chlorophenethyl)-1-hydroxy-3-methylenecyclohexanecarboxylate
—— 2-(4-isopropylphenyl)-4H-furo[3,2-b]pyrrole-5-carboxylic acid 1138343-23-3 C16H15NO3
2-(4-isopropylphenyl)-4H-furo[3,2-b]pyrrole-5-carboxylic acid
—— —— 1092929-17-3 C18H16N4O2
—— [(3S,4S,5S)-4-(methoxymethoxy)-2,5-dimethyl-6-oxohexan-3-yl] (3S,4R,5S)-4-[[(2S,3R)-3-[(2S)-3-(4-methoxyphenyl)-2-[methyl-[(2S)-1-[(2S)-4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]oxy-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoyl]amino]-5-methyl-3-tri(propan-2-yl)silyloxyheptanoate 1053630-19-5 C66H107N5O16Si
[(3S,4S,5S)-4-(methoxymethoxy)-2,5-dimethyl-6-oxohexan-3-yl] (3S,4R,5S)-4-[[(2S,3R)-3-[(2S)-3-(4-methoxyphenyl)-2-[methyl-[(2S)-1-[(2S)-4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]oxy-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoyl]amino]-5-methyl-3-tri(propan-2-yl)silyloxyheptanoate
—— 3-Ethyl-1-[4-(4-fluoropiperidin-1-yl)phenyl]-3-azabicyclo[3.1.0]hexane 1259554-49-8 C18H25FN2
3-Ethyl-1-[4-(4-fluoropiperidin-1-yl)phenyl]-3-azabicyclo[3.1.0]hexane
—— US8653087, III-218 1213245-04-5 C31H38N8O
US8653087, III-218
—— 4-[[4-[[1-(4-chlorophenyl)cyclopropyl]amino]-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino]-N-[4-(cyclopropylsulfonylamino)-4-oxobutyl]benzamide 1360826-90-9 C28H29ClF3N7O5S
4-[[4-[[1-(4-chlorophenyl)cyclopropyl]amino]-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino]-N-[4-(cyclopropylsulfonylamino)-4-oxobutyl]benzamide
—— (S)-2-({(S)-3-[4-(3-chloro-4-methyl-benzyloxy)-phenyl]-7-[2-(cyclopentylmethyl-amino)-4-methyl-thiazole-5-sulfonyl]-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline-8-carbonyl}-amino)-3-(4'-cyano-biphenyl-4-yl)-propionic acid 1246824-92-9 C52H50ClN5O8S2
(S)-2-({(S)-3-[4-(3-chloro-4-methyl-benzyloxy)-phenyl]-7-[2-(cyclopentylmethyl-amino)-4-methyl-thiazole-5-sulfonyl]-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline-8-carbonyl}-amino)-3-(4'-cyano-biphenyl-4-yl)-propionic acid
—— C,C,C-trifluoro-N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-methanesulfonamide 1215221-86-5 C18H19F6N7O3S2
C,C,C-trifluoro-N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-methanesulfonamide
—— 1-[(1S)-1-(hydroxymethyl)-2-methyl-propyl]-7-methoxy-4-oxo-6-[(tetralin-1-ylamino)methyl]-1,8-naphthyridine-3-carboxylic acid 1171822-07-3 C26H31N3O5
1-[(1S)-1-(hydroxymethyl)-2-methyl-propyl]-7-methoxy-4-oxo-6-[(tetralin-1-ylamino)methyl]-1,8-naphthyridine-3-carboxylic acid
—— 2-[4-(4-tert-butoxycarbonylaminobenzyl)piperazin-1-yl]-5-fluoro-4-morpholino-6-[4-(2,3-xylyl)piperazin-1-yl]pyrimidine 1190067-27-6 C36H49FN8O3
2-[4-(4-tert-butoxycarbonylaminobenzyl)piperazin-1-yl]-5-fluoro-4-morpholino-6-[4-(2,3-xylyl)piperazin-1-yl]pyrimidine
—— N-(benzenesulfonyl)-5-bromo-3-(2,4-dioxo-1H-quinazolin-3-yl)-1-methylindole-2-carboxamide 1154598-72-7 C24H17BrN4O5S
N-(benzenesulfonyl)-5-bromo-3-(2,4-dioxo-1H-quinazolin-3-yl)-1-methylindole-2-carboxamide
—— (2S)-1-[(2S)-2-amino-3,3-dimethyl-5-oxo-5-[2-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl]pentanoyl]pyrrolidine-2-carbonitrile;2,2,2-trifluoroacetic acid 1150656-79-3 C2HF3O2*C18H24F3N7O2
(2S)-1-[(2S)-2-amino-3,3-dimethyl-5-oxo-5-[2-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl]pentanoyl]pyrrolidine-2-carbonitrile;2,2,2-trifluoroacetic acid
—— Tert-butyl 4-[5-[3-[1-[4-(5-aminopyrazin-2-yl)phenyl]-1-cyclopropylethyl]-1,2,4-oxadiazol-5-yl]pyrazin-2-yl]piperazine-1-carboxylate 1360552-54-0 C30H35N9O3
Tert-butyl 4-[5-[3-[1-[4-(5-aminopyrazin-2-yl)phenyl]-1-cyclopropylethyl]-1,2,4-oxadiazol-5-yl]pyrazin-2-yl]piperazine-1-carboxylate
—— tert-butyl {4-[2-fluoro-5-(trifluoromethyl)phenyl]pyridin-2-yl}carbamate 1354917-81-9 C17H16F4N2O2
tert-butyl {4-[2-fluoro-5-(trifluoromethyl)phenyl]pyridin-2-yl}carbamate
—— 5-[4-(3-methyl-2-{5-[2-(methylsulfonyl)phenyl]-1,2,4-oxadiazol-3-yl}butan-2-yl)phenyl]pyrimidin-2-amine 1360550-37-3 C24H25N5O3S
5-[4-(3-methyl-2-{5-[2-(methylsulfonyl)phenyl]-1,2,4-oxadiazol-3-yl}butan-2-yl)phenyl]pyrimidin-2-amine
—— 3-(oxiranecarbonyl-amino)-benzoic acid tert-butyl ester 1268152-53-9 C14H17NO4
3-(oxiranecarbonyl-amino)-benzoic acid tert-butyl ester
—— —— 1415810-96-6 C20H31NO5S
—— (+-)-5-phenyl-5-trans-stilben-4-yl-imidazolidine-2,4-dione 102546-74-7 C23H18N2O2
(+-)-5-phenyl-5-trans-stilben-4-yl-imidazolidine-2,4-dione
—— tert-butyl 4-[(2R)-2-hydroxy-3-(2-phenylbenzoxazol-5-yloxy)propyl]-piperazinecarboxylate 1055966-79-4 C25H31N3O5
tert-butyl 4-[(2R)-2-hydroxy-3-(2-phenylbenzoxazol-5-yloxy)propyl]-piperazinecarboxylate
—— (S)-1-{2-[(3S,5R)-3,5-dimethylpiperazin-1-yl]-7-fluoro-8-methylquinolin-3-yl}-ethanamine 1242239-75-3 C18H25FN4
(S)-1-{2-[(3S,5R)-3,5-dimethylpiperazin-1-yl]-7-fluoro-8-methylquinolin-3-yl}-ethanamine
—— ethyl 8-methoxy-2-methylsulfonylquinoline-4-carboxylate 143571-89-5 C14H15NO5S
ethyl 8-methoxy-2-methylsulfonylquinoline-4-carboxylate
—— α-cyano-β-oxo-N-(4'-nitro)phenyl-(3-trifluoromethyl)benzenepropanamide 136564-37-9 C17H10F3N3O4
α-cyano-β-oxo-N-(4'-nitro)phenyl-(3-trifluoromethyl)benzenepropanamide
—— 5-[(4'-methoxy-1,1'-biphenyl)-4-yl]-5-methyl-3,4-dihydroxy-2(5H)-furanone 1098479-26-5 C18H16O5
5-[(4'-methoxy-1,1'-biphenyl)-4-yl]-5-methyl-3,4-dihydroxy-2(5H)-furanone
—— [5-[[(2E)-2-[(4-bromophenyl)methylidene]cyclopropyl]methyl-(4-methylphenyl)sulfonylamino]-2-methylpent-3-yn-2-yl] acetate 1350466-52-2 C26H28BrNO4S
[5-[[(2E)-2-[(4-bromophenyl)methylidene]cyclopropyl]methyl-(4-methylphenyl)sulfonylamino]-2-methylpent-3-yn-2-yl] acetate
—— 2-(4-(4-((2-chlorophenyl)sulfonyl)-1-piperazinyl)phenyl)-1,1,1,3,3,3-hexafluoro-2-propanol 1361215-71-5 C19H17ClF6N2O3S
2-(4-(4-((2-chlorophenyl)sulfonyl)-1-piperazinyl)phenyl)-1,1,1,3,3,3-hexafluoro-2-propanol
—— methyl 5-acetyl-2-oct-1-ynyl-2H-pyridine-1-carboxylate 118160-85-3 C17H23NO3
methyl 5-acetyl-2-oct-1-ynyl-2H-pyridine-1-carboxylate
—— 2-(4-(1-hydroxy-4,5,5-trimethyl-2,5-dihydro-1H-imidazol-2-yl)phenoxy)acetonitrile 1193304-42-5 C14H17N3O2
2-(4-(1-hydroxy-4,5,5-trimethyl-2,5-dihydro-1H-imidazol-2-yl)phenoxy)acetonitrile
—— 4-[(4-methylphenyl)methylsulfamoyl]-3-nitrobenzoic acid 197728-18-0 C15H14N2O6S
4-[(4-methylphenyl)methylsulfamoyl]-3-nitrobenzoic acid
—— Methyl 2-<(5-methoxy-1-methyl)indol-2-yl>propionate 144265-36-1 C14H17NO3
Methyl 2-<(5-methoxy-1-methyl)indol-2-yl>propionate
—— 5-tert-Butyl-2-hydroxy-8,8-dimethyl-bicyclo[4.2.0]octa-1,4-dien-3-one O-methyl-oxime 145030-79-1 C15H23NO2
5-tert-Butyl-2-hydroxy-8,8-dimethyl-bicyclo[4.2.0]octa-1,4-dien-3-one O-methyl-oxime
—— 3-([1,1'-biphenyl]-4-yl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-1H-cyclopropa[3,4]cyclopenta[1,2-c]pyrazol-1-yl)prop-2-en-1-one 1208260-67-6 C25H24N2O
3-([1,1'-biphenyl]-4-yl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-1H-cyclopropa[3,4]cyclopenta[1,2-c]pyrazol-1-yl)prop-2-en-1-one
—— cis-4-tert-butyl-1-(α-hydroxybenzyl)-O-(methoxymethyl)cyclohexanol 110615-45-7 C19H30O3
cis-4-tert-butyl-1-(α-hydroxybenzyl)-O-(methoxymethyl)cyclohexanol
—— (3-methoxy-5-methylhex-5-en-1-ynyl)benzene 1309671-06-4 C14H16O
(3-methoxy-5-methylhex-5-en-1-ynyl)benzene
—— N-(3-methyl-1-{[(1S,4S)-5-({[(2-methylphenyl)sulfonyl]amino}acetyl)-2,5-diazabicyclo[2.2.1]hept-2-yl]carbonyl}butyl)-1-benzothiophene-2-carboxamide 1186642-81-8 C29H34N4O5S2
N-(3-methyl-1-{[(1S,4S)-5-({[(2-methylphenyl)sulfonyl]amino}acetyl)-2,5-diazabicyclo[2.2.1]hept-2-yl]carbonyl}butyl)-1-benzothiophene-2-carboxamide
—— 1-{3-[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-ylthio]phenyl}-3-[1-p-tolyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]urea 1188910-48-6 C30H27F3N6O4S
1-{3-[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-ylthio]phenyl}-3-[1-p-tolyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]urea