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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,2,2-trifluoro-1-(trifluoromethyl)ethyl 4-[(2-(trifluoromethyl)benzenesulphonylamino)-methyl]piperidine-1-carboxylate 1352012-83-9 C17H17F9N2O4S
2,2,2-trifluoro-1-(trifluoromethyl)ethyl 4-[(2-(trifluoromethyl)benzenesulphonylamino)-methyl]piperidine-1-carboxylate
—— 5-bromobenzo[b]selenophene-2-carboxylic acid ethyl ester 1429048-35-0 C11H9BrO2Se
5-bromobenzo[b]selenophene-2-carboxylic acid ethyl ester
—— 8-(pyridin-3-yl)-2-[2-(quinolin-2-yl)ethyl]phthalazin-1(2H)-one 1433196-38-3 C24H18N4O
8-(pyridin-3-yl)-2-[2-(quinolin-2-yl)ethyl]phthalazin-1(2H)-one
—— N-(4-((3S,4S)-3-amino-4-hydroxy-piperidin-1-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide 1187054-18-7 C20H19F2N5O2S
N-(4-((3S,4S)-3-amino-4-hydroxy-piperidin-1-yl)pyridin-3-yl)-2-(2,6-difluorophenyl)thiazole-4-carboxamide
—— tert-butyl 4-(4-isopropyl-1-(2-(methylsulfonyloxy)ethyl)-1H-imidazol-2-yl)piperidine-1-carboxylate 1295519-36-6 C19H33N3O5S
tert-butyl 4-(4-isopropyl-1-(2-(methylsulfonyloxy)ethyl)-1H-imidazol-2-yl)piperidine-1-carboxylate
—— 2-[(2-bromophenyl)methylamino]benzoic acid 1380084-61-6 C14H12BrNO2
2-[(2-bromophenyl)methylamino]benzoic acid
—— 1-methyl-2-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide 1262395-80-1 C19H27N3O2S
1-methyl-2-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
—— N-[2-({1-[1-(4-chlorophenyl)cyclobutyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxy)ethyl]-3,3,3-trifluoropropane-1-sulfonamide hydrochloride 1190642-53-5 C24H28ClF3N2O3S*ClH
N-[2-({1-[1-(4-chlorophenyl)cyclobutyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxy)ethyl]-3,3,3-trifluoropropane-1-sulfonamide hydrochloride
—— 1-[5-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-3-isopropyl-urea 1080827-03-7 C21H26N6O3
1-[5-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-3-isopropyl-urea
—— 2-tert-butyl 10-methyl 8-(4-methoxybenzyl)-9,11-dioxo-2,8-diazaspiro[5.5]undecane-2,10-dicarboxylate 1312814-98-4 C24H32N2O7
2-tert-butyl 10-methyl 8-(4-methoxybenzyl)-9,11-dioxo-2,8-diazaspiro[5.5]undecane-2,10-dicarboxylate
—— 5-(2-methyl-5-trifluoromethyl-phenyl)-2H-pyrazol-3-ylamine 1040724-47-7 C11H10F3N3
5-(2-methyl-5-trifluoromethyl-phenyl)-2H-pyrazol-3-ylamine
—— 1-(4,4-difluorocyclohex-1-enyl)cyclobutanecarbaldehyde 1432493-21-4 C11H14F2O
1-(4,4-difluorocyclohex-1-enyl)cyclobutanecarbaldehyde
—— N-(3-(5-(1H-pyrazol-1-yl)-1H-benzo[d]imidazol-1-yl)-5-(1H-pyrrol-1-yl)-phenyl)propane-2-sulfonamide 1430724-28-9 C23H22N6O2S
N-(3-(5-(1H-pyrazol-1-yl)-1H-benzo[d]imidazol-1-yl)-5-(1H-pyrrol-1-yl)-phenyl)propane-2-sulfonamide
—— 4-((1-(2,4'-bipyridin-3-ylcarbonyl)-4-hydroxypiperidin-4-yl)methyl)benzonitrile 1429505-29-2 C24H22N4O2
4-((1-(2,4'-bipyridin-3-ylcarbonyl)-4-hydroxypiperidin-4-yl)methyl)benzonitrile
—— 2-cyclopentyl-7-methoxy-4-phenyl-3-(1H-tetrazol-5-yl)quinoline 1433902-72-7 C22H21N5O
2-cyclopentyl-7-methoxy-4-phenyl-3-(1H-tetrazol-5-yl)quinoline
—— 5-[(adamantan-1-ylacetyl)amino]-N-(2-hydroxypropyl)imidazo[1,2-a]pyridine-2-carboxamide 1031834-36-2 C23H30N4O3
5-[(adamantan-1-ylacetyl)amino]-N-(2-hydroxypropyl)imidazo[1,2-a]pyridine-2-carboxamide
—— ethyl 2-(3-nitrobenzyl dicambyl)acrylate 1430102-95-6 C20H17Cl2NO7
ethyl 2-(3-nitrobenzyl dicambyl)acrylate
—— 4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)-1-[(2-phenyl-1H-imidazol-4-yl)carbonyl]piperidine 1138330-78-5 C25H26F3N3O3S
4-(1-methyl-1-([3-(trifluoromethyl)phenyl]sulfonyl)ethyl)-1-[(2-phenyl-1H-imidazol-4-yl)carbonyl]piperidine
—— 3-{9H-pyrido[3,4-b]-indol-3-yl-carbonyl}-amino-3-ethyl-1-(4-fluorophenyl)-5-methoxy-2-indolinone 154058-07-8 C29H23FN4O3
3-{9H-pyrido[3,4-b]-indol-3-yl-carbonyl}-amino-3-ethyl-1-(4-fluorophenyl)-5-methoxy-2-indolinone
—— tert.butyl 4'-[(6-benzyloxycarbonylamino-2-n-butyl-benzimidazol-1-yl)-methyl]biphenyl-2-carboxylate 133141-10-3 C37H39N3O4
tert.butyl 4'-[(6-benzyloxycarbonylamino-2-n-butyl-benzimidazol-1-yl)-methyl]biphenyl-2-carboxylate
—— 3-Propylamino-6,7-dimethyl-2-(3-thioallophanoyl)quinoxaline 137932-64-0 C15H19N5OS
3-Propylamino-6,7-dimethyl-2-(3-thioallophanoyl)quinoxaline
—— 2-amino-6,7-bis(benzyloxy)-3,4-dihydronaphthalen-1(2H)-one 139759-56-1 C24H23NO3
2-amino-6,7-bis(benzyloxy)-3,4-dihydronaphthalen-1(2H)-one
—— 1-hydroxy-1-(1-methylethyl)-3-[3-(methylsulfonyl)phenyl]urea 177025-21-7 C11H16N2O4S
1-hydroxy-1-(1-methylethyl)-3-[3-(methylsulfonyl)phenyl]urea
—— 1,9-di-n-butyl-3,7-dimethoxy-2,8,12-trioxatetracyclo[7.2.1.0(4,11).0(6,10)]dodecane 1333497-06-5 C19H32O5
1,9-di-n-butyl-3,7-dimethoxy-2,8,12-trioxatetracyclo[7.2.1.0(4,11).0(6,10)]dodecane
—— 1-(4-bromo-2-fluorophenyl)-3-(4-methyl-2,5-dioxo-4-(phenoxymethyl)imidazolidin-1-yl)urea 1434717-58-4 C18H16BrFN4O4
1-(4-bromo-2-fluorophenyl)-3-(4-methyl-2,5-dioxo-4-(phenoxymethyl)imidazolidin-1-yl)urea
—— 2-(3,5-Diphenylpyrazol-1-yl)-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone 1440950-91-3 C23H20N4OS
2-(3,5-Diphenylpyrazol-1-yl)-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone
—— [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[acetyl(5-phenylpentyl)amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate 1256286-94-8 C34H53N8O11P
[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[acetyl(5-phenylpentyl)amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate
—— 6-(3,5-dicyano-1-cyclobutyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide 1247932-06-4 C21H17F3N6O2S
6-(3,5-dicyano-1-cyclobutyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide
—— 1-(4-bromophenyl)-3-(4-(2-hydroxyethyl)-4-isopropyl-2,5-dioxoimidazolidin-1-yl)urea 1434719-05-7 C15H19BrN4O4
1-(4-bromophenyl)-3-(4-(2-hydroxyethyl)-4-isopropyl-2,5-dioxoimidazolidin-1-yl)urea
—— 6-{[(1,2-dimethyl-1H-imidazol-4-yl)thio]methyl}-N-(2-methoxyethyl)-4-(4-morpholinyl)-2-pyridinamine 1186688-08-3 C18H27N5O2S
6-{[(1,2-dimethyl-1H-imidazol-4-yl)thio]methyl}-N-(2-methoxyethyl)-4-(4-morpholinyl)-2-pyridinamine
—— phenyl 3,4-di-O-acetyl-2-O-benzyl-6-deoxy-5-methyl-α-L-fucopyranosyl-(1->3)-2-(2,2,2-trichloroethoxy)carbonylamino-6-O-benzyl-2-deoxy-1-thio-β-D-glucopyranoside 1174919-36-8 C39H44Cl3NO12S
phenyl 3,4-di-O-acetyl-2-O-benzyl-6-deoxy-5-methyl-α-L-fucopyranosyl-(1->3)-2-(2,2,2-trichloroethoxy)carbonylamino-6-O-benzyl-2-deoxy-1-thio-β-D-glucopyranoside
—— 4-[(3R)-3-(methylamino)pyrrolidin-1-yl]-7-phenylfuro[3,2-d]pyrimidin-2-amine 1188283-34-2 C17H19N5O
4-[(3R)-3-(methylamino)pyrrolidin-1-yl]-7-phenylfuro[3,2-d]pyrimidin-2-amine
—— 2-tert-butoxy-2-(4-(4-chlorophenyl)-1-isobutyl-2,3,6-trimethyl-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid 1436854-87-3 C26H33ClN2O3
2-tert-butoxy-2-(4-(4-chlorophenyl)-1-isobutyl-2,3,6-trimethyl-1H-pyrrolo[2,3-b]pyridin-5-yl)acetic acid
—— ethyl 4-(4-((methoxy(methyl))carbamoyl)piperidin-1-yl)azepane-1-carboxylate 1438242-16-0 C17H31N3O4
ethyl 4-(4-((methoxy(methyl))carbamoyl)piperidin-1-yl)azepane-1-carboxylate
—— 3-amino-6-(4-(2,6-dimethylphenylcarbonyl)piperazin-1-yl)-N-(pyridin-2-yl)pyrazine-2-carboxamide 1225060-86-5 C23H25N7O2
3-amino-6-(4-(2,6-dimethylphenylcarbonyl)piperazin-1-yl)-N-(pyridin-2-yl)pyrazine-2-carboxamide
—— 3-amino-N-(1,3-dimethyl-1H-pyrazol-5-yl)-6-(1-(ethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)pyrazine-2-carboxamide 1225062-17-8 C17H23N7O3S
3-amino-N-(1,3-dimethyl-1H-pyrazol-5-yl)-6-(1-(ethylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)pyrazine-2-carboxamide
—— 5-(2,6-difluorophenoxy)-3-(6-methyl-1H-benzimidazol-2-yl)pyrazin-2-amine 1349686-72-1 C18H13F2N5O
5-(2,6-difluorophenoxy)-3-(6-methyl-1H-benzimidazol-2-yl)pyrazin-2-amine
—— (R)-5-(1-amino-1-oxobutan-2-ylamino)-3-(quinolin-3-ylamino)pyrazine-2-carboxamide 1438419-83-0 C18H19N7O2
(R)-5-(1-amino-1-oxobutan-2-ylamino)-3-(quinolin-3-ylamino)pyrazine-2-carboxamide
—— 1-ethyl-5-(1-oxa-2-azaspiro[4.5]dec-2-en-3-yl)-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine 1057633-56-3 C21H29N5O2
1-ethyl-5-(1-oxa-2-azaspiro[4.5]dec-2-en-3-yl)-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine
—— 3-(3,5-Dimethoxyphenyl)-3-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]propan-1-ol 1431930-19-6 C24H25N3O3
3-(3,5-Dimethoxyphenyl)-3-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]propan-1-ol
—— 4-((5-chloro-4-((2-(methylsulfonamido)phenyl)amino)pyrimidin-2-yl)amino)-2,5-difluorobenzoic acid 1251954-79-6 C18H14ClF2N5O4S
4-((5-chloro-4-((2-(methylsulfonamido)phenyl)amino)pyrimidin-2-yl)amino)-2,5-difluorobenzoic acid
—— 6-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3'-methyl-2'-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylamino)-3,4'-bipyridine-2-carboxylic acid 1430845-53-6 C39H38N6O3S
6-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-3'-methyl-2'-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-ylamino)-3,4'-bipyridine-2-carboxylic acid
—— 2,2,6,10,10-pentamethyl-5,7-dioxatetracyclo[9.2.1.0(1,9).0(4,8)]tetradecane 1203487-34-6 C17H28O2
2,2,6,10,10-pentamethyl-5,7-dioxatetracyclo[9.2.1.0(1,9).0(4,8)]tetradecane
—— 3-(4-piperidin-1-ylbutoxy)-5,6,9,10,11,11a-hexahydro-8H-pyrido[2,1-f][1,6]naphthyridin-8-one 1190440-95-9 C21H31N3O2
3-(4-piperidin-1-ylbutoxy)-5,6,9,10,11,11a-hexahydro-8H-pyrido[2,1-f][1,6]naphthyridin-8-one
—— N-(1-(3-Chlorophenyl)-2-p-tolylethyl)-4,5-dihydro-1H-imidazol-2-amine 1188271-44-4 C18H20ClN3
N-(1-(3-Chlorophenyl)-2-p-tolylethyl)-4,5-dihydro-1H-imidazol-2-amine
—— 2-[[2-(4-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-6-(3-hydroxyazetidin-1-yl)-4-(5-methyl-1H-pyrazol-3-yl)pyridine-3,5-dicarbonitrile 1187543-10-7 C24H18ClN7O2S
2-[[2-(4-chlorophenyl)-1,3-oxazol-4-yl]methylsulfanyl]-6-(3-hydroxyazetidin-1-yl)-4-(5-methyl-1H-pyrazol-3-yl)pyridine-3,5-dicarbonitrile
—— N-(2-(4-(5-(6-amino-5-methoxypyridin-3-yl)-2-(4-fluorophenyl)-1H-imidazol-4-yl)pyrimidin-2-ylamino)ethyl)-2-methoxyacetamide 1188299-54-8 C24H25FN8O3
N-(2-(4-(5-(6-amino-5-methoxypyridin-3-yl)-2-(4-fluorophenyl)-1H-imidazol-4-yl)pyrimidin-2-ylamino)ethyl)-2-methoxyacetamide
—— 2-[3-cyano-1-cyclobutyl-6-(propan-2-yl)-1H-indol-2-yl]-N-(1,3-difluoropropan-2-yl)pyrimidine-5-sulfonamide 1248575-56-5 C23H25F2N5O2S
2-[3-cyano-1-cyclobutyl-6-(propan-2-yl)-1H-indol-2-yl]-N-(1,3-difluoropropan-2-yl)pyrimidine-5-sulfonamide
—— 3-(1H-benzo[d]imidazol-2-yl)-5-(1-(phenylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)pyrazin-2-amine 1225060-22-9 C22H20N6O2S
3-(1H-benzo[d]imidazol-2-yl)-5-(1-(phenylsulfonyl)-1,2,3,6-tetrahydropyridin-4-yl)pyrazin-2-amine
—— 7-[4-(cyclohexylamino)-1-ethyl-1H-pyrazolo[3,4-b]pyridin-5-yl]-5-oxa-6-azaspiro[3.4]oct-6-ene-2-carbonitrile 1057635-02-5 C21H26N6O
7-[4-(cyclohexylamino)-1-ethyl-1H-pyrazolo[3,4-b]pyridin-5-yl]-5-oxa-6-azaspiro[3.4]oct-6-ene-2-carbonitrile