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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-2-chloro-5-((1-(3-chlorophenyl)ethylamino)methyl)benzenesulfonamide 1025771-27-0 C15H16Cl2N2O2S
(R)-2-chloro-5-((1-(3-chlorophenyl)ethylamino)methyl)benzenesulfonamide
—— N-(4-tert-butylphenyl)-2-((6,7-dimethoxyquinoline-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide 1035699-64-9 C32H35N3O3
N-(4-tert-butylphenyl)-2-((6,7-dimethoxyquinoline-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide
—— 3-(3,5-difluorophenyl)-2-[1-(9H-purin-6-ylamino)propyl]thieno[3,2-d]pyrimidin-4(3H)-one 1029280-14-5 C20H15F2N7OS
3-(3,5-difluorophenyl)-2-[1-(9H-purin-6-ylamino)propyl]thieno[3,2-d]pyrimidin-4(3H)-one
—— 9-chloro-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride 1000781-40-7 C12H13ClN2O2*ClH
9-chloro-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride
—— 7-phenyl-1-(5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl)-heptan-1-one 1042152-14-6 C19H20N2O2S
7-phenyl-1-(5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl)-heptan-1-one
—— 4-{4-[4-Amino-5-bromo-6-(4-cyano-2,6-dimethyl-phenoxy)-pyrimidin-2-ylamino]-piperidin-1-ylmethyl}-3-chloro-benzamide 1033951-98-2 C26H27BrClN7O2
4-{4-[4-Amino-5-bromo-6-(4-cyano-2,6-dimethyl-phenoxy)-pyrimidin-2-ylamino]-piperidin-1-ylmethyl}-3-chloro-benzamide
—— 1'-[(3-Cyclopropyl-8-methoxyimidazo[1,2-a]pyridin-6-yl)carbonyl]-6-(1H-tetrazol-5-yl)spiro[chroman-2,4'-piperidin]-4-one 1039757-95-3 C26H25N7O4
1'-[(3-Cyclopropyl-8-methoxyimidazo[1,2-a]pyridin-6-yl)carbonyl]-6-(1H-tetrazol-5-yl)spiro[chroman-2,4'-piperidin]-4-one
—— 2-((6,7-dimethoxyquinolin-4-yl)methyl)-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide 1035699-74-1 C29H24F3N3O4
2-((6,7-dimethoxyquinolin-4-yl)methyl)-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide
—— 3-methyl-5-(5-phenyl-2H-tetrazol-2-yl)thiophene-2-carboxylic acid 1034981-90-2 C13H10N4O2S
3-methyl-5-(5-phenyl-2H-tetrazol-2-yl)thiophene-2-carboxylic acid
—— N'-[[3,5-di(pentadecoxy)phenyl]methyl]ethane-1,2-diamine 1033476-19-5 C39H74N2O2
N'-[[3,5-di(pentadecoxy)phenyl]methyl]ethane-1,2-diamine
—— N1-[(5-chloro-8-hydroxyquinolin-7-yl)(4-methylphenyl)methyl]-N2-(4-cyanophenyl)glycinamide 1009840-61-2 C26H21ClN4O2
N1-[(5-chloro-8-hydroxyquinolin-7-yl)(4-methylphenyl)methyl]-N2-(4-cyanophenyl)glycinamide
—— 2-amino-4,6-dichloro-N-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethyl}benzenesulfonamide 1032648-28-4 C21H14Cl2F4N4O2S
2-amino-4,6-dichloro-N-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]ethyl}benzenesulfonamide
—— 8-methyl-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride 1000781-48-5 C13H16N2O2*ClH
8-methyl-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride
—— 4-{5-Bromo-2-[1-(2-chloro-4-methanesulfonyl-benzyl)-piperidin-4-ylamino]-pyrimidin-4-ylamino}-3,5-dimethyl-benzonitrile 1034013-10-9 C26H28BrClN6O2S
4-{5-Bromo-2-[1-(2-chloro-4-methanesulfonyl-benzyl)-piperidin-4-ylamino]-pyrimidin-4-ylamino}-3,5-dimethyl-benzonitrile
—— (4-{[1-(2-Methoxy-5-methyl-benzenesulfonyl)-2,3-dihydro-1H-indole-6-carbonyl]-amino}-phenyl)-acetic acid 1034775-79-5 C25H24N2O6S
(4-{[1-(2-Methoxy-5-methyl-benzenesulfonyl)-2,3-dihydro-1H-indole-6-carbonyl]-amino}-phenyl)-acetic acid
—— 1-{4-[3-(Cyclopentyloxy)-4-methoxyphenyl]pyrimidin-2-yl}-1,3-dihydro-2H-benzimidazol-2-one 1048378-42-2 C23H22N4O3
1-{4-[3-(Cyclopentyloxy)-4-methoxyphenyl]pyrimidin-2-yl}-1,3-dihydro-2H-benzimidazol-2-one
—— 1-{4-[(1,1-dioxido-2-isothiazolidinyl)methyl]phenyl}-6-methyl-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine 1022930-92-2 C18H21F3N4O2S
1-{4-[(1,1-dioxido-2-isothiazolidinyl)methyl]phenyl}-6-methyl-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine
—— N-(8-tert-butyl-3,4-dihydro-2H-chromen-4-yl)-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-13-2 C24H30N2O3
N-(8-tert-butyl-3,4-dihydro-2H-chromen-4-yl)-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— (S)-(1-pyrimidin-2-yl-piperidin-4-yl)-(3,2',4'-trifluoro-biphenyl-4-yl)methanol 1030903-25-3 C22H20F3N3O
(S)-(1-pyrimidin-2-yl-piperidin-4-yl)-(3,2',4'-trifluoro-biphenyl-4-yl)methanol
—— (4-{[(2,9,9-trimethyl-10,10-dioxido-9H-thioxanthen-3-yl)sulfonyl]amino}piperidin-1-yl)acetic acid 1027347-18-7 C23H28N2O6S2
(4-{[(2,9,9-trimethyl-10,10-dioxido-9H-thioxanthen-3-yl)sulfonyl]amino}piperidin-1-yl)acetic acid
—— 1-[4-(2,7-Diazaspiro[3.5]nonan-2-yl)phenyl]-4-[(4-fluorophenyl)methoxy]pyridin-2-one 1032157-74-6 C25H26FN3O2
1-[4-(2,7-Diazaspiro[3.5]nonan-2-yl)phenyl]-4-[(4-fluorophenyl)methoxy]pyridin-2-one
—— N-(3,5-bis(trifluoromethyl)benzyl)-3-(cyclopropylmethyl)pyrrolidine-3-carboxamide 1018990-55-0 C18H20F6N2O
N-(3,5-bis(trifluoromethyl)benzyl)-3-(cyclopropylmethyl)pyrrolidine-3-carboxamide
—— 3-(3,4-dimethoxyphenyl)-7-N,7-N-dimethylisoquinoline-1,7-diamine 1029008-75-0 C19H21N3O2
3-(3,4-dimethoxyphenyl)-7-N,7-N-dimethylisoquinoline-1,7-diamine
—— N-cyclohexyl-N-(2-(2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino)ethyl)-3-phenethoxypropanamide 1035226-91-5 C30H39N3O4
N-cyclohexyl-N-(2-(2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino)ethyl)-3-phenethoxypropanamide
—— N-3,4-dihydro-2H-chromen-3-yl-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-09-6 C20H22N2O3
N-3,4-dihydro-2H-chromen-3-yl-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— 14-(2-{[(4-{[6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}phenyl)methyl]amino}-2-oxoethyl)-16,16,18,18-tetramethyl-6,7,7a,8a,9,10,16,18-octahydrobenzo[2'',3'']indolizino[8'',7'':5',6']pyrano[3',2':3,4]pyrido[1,2-a]indol-5-ium-2-sulfonate 1059171-71-9 C52H47Cl2N7O6S
14-(2-{[(4-{[6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}phenyl)methyl]amino}-2-oxoethyl)-16,16,18,18-tetramethyl-6,7,7a,8a,9,10,16,18-octahydrobenzo[2'',3'']indolizino[8'',7'':5',6']pyrano[3',2':3,4]pyrido[1,2-a]indol-5-ium-2-sulfonate
—— isobutyric acid 3,4,7-trihydroxy-6-oxo-2,3,4,4a,5,6-hexahydro[1,3]dioxolo[4,5-j]phenanthridin-2-yl ester 1019642-67-1 C18H19NO8
isobutyric acid 3,4,7-trihydroxy-6-oxo-2,3,4,4a,5,6-hexahydro[1,3]dioxolo[4,5-j]phenanthridin-2-yl ester
—— rac-2-({[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl}thio)-4-(tetrahydro-2H-pyran-2-yl)pyridine-3,5-dicarbonitrile 1030622-80-0 C22H17ClN4OS2
rac-2-({[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl}thio)-4-(tetrahydro-2H-pyran-2-yl)pyridine-3,5-dicarbonitrile
—— N-(3,4-dihydro-2H-chromen-2-ylmethyl)-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-18-7 C21H24N2O3
N-(3,4-dihydro-2H-chromen-2-ylmethyl)-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— 5,7-dihydro-1,2,3-trimethoxybenzo[d][1,3]dioxolo[4,5-h][2]benzoxepine 1034742-44-3 C18H18O6
5,7-dihydro-1,2,3-trimethoxybenzo[d][1,3]dioxolo[4,5-h][2]benzoxepine
—— 5-[5-(2-{[2-(methylamino)ethyl]amino}-4-pyridinyl)-1H-benzimidazol-1-yl]-3-({(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}oxy)-2-thiophenecarboxamide 1032198-52-9 C29H27F3N6O2S
5-[5-(2-{[2-(methylamino)ethyl]amino}-4-pyridinyl)-1H-benzimidazol-1-yl]-3-({(1R)-1-[2-(trifluoromethyl)phenyl]ethyl}oxy)-2-thiophenecarboxamide
—— 8-(trifluoromethyl)-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride 1000781-43-0 C13H13F3N2O2*ClH
8-(trifluoromethyl)-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride
—— N-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)-N'-(6-methyl-3,4-dihydro-2H-chromen-4-yl)urea 1034770-15-4 C21H24N2O3
N-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)-N'-(6-methyl-3,4-dihydro-2H-chromen-4-yl)urea
—— (4-{[1-(5-Chloro-2-methoxy-benzenesulfonyl)-1H-indole-6-carbonyl]-amino}-phenyl)-acetic acid 1034775-75-1 C24H19ClN2O6S
(4-{[1-(5-Chloro-2-methoxy-benzenesulfonyl)-1H-indole-6-carbonyl]-amino}-phenyl)-acetic acid
—— 6-o-tolylethynyl-2H-chromene-8-carboxylic acid [(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-amide 1033763-45-9 C30H26N2O3
6-o-tolylethynyl-2H-chromene-8-carboxylic acid [(R)-1-hydroxymethyl-2-(1H-indol-3-yl)-ethyl]-amide
—— 5-(3,4-difluoro-5-methoxy-phenyl)-2,3-dihydro-benzofuran-7-carboxylic acid 1033765-46-6 C16H12F2O4
5-(3,4-difluoro-5-methoxy-phenyl)-2,3-dihydro-benzofuran-7-carboxylic acid
—— N-(5,6-dimethyl-4-(morpholinomethyl)pyridin-2-yl)-2,2-dimethylbutanamide 1029126-59-7 C18H29N3O2
N-(5,6-dimethyl-4-(morpholinomethyl)pyridin-2-yl)-2,2-dimethylbutanamide
—— 1-(4-morpholin-4-yl-benzenesulfonyl)-1H-indole-6-carboxylic acid 1046151-70-5 C19H18N2O5S
1-(4-morpholin-4-yl-benzenesulfonyl)-1H-indole-6-carboxylic acid
—— N-[3-((2R)-2-{[4-[(4-Chlorophenyl)methyl]-1-oxo-2(1H)-phthalazinyl]methyl}-1-pyrrolidinyl)propyl]acetamide, trifluoroacetate 1035040-36-8 C2HF3O2*C25H29ClN4O2
N-[3-((2R)-2-{[4-[(4-Chlorophenyl)methyl]-1-oxo-2(1H)-phthalazinyl]methyl}-1-pyrrolidinyl)propyl]acetamide, trifluoroacetate
—— (2R)-2-(aminomethyl)-4-[(1R)-1-(1-benzyl-4-phenyl-1H-imidazol-2-yl)-2,2-dimethylpropyl]-1,4-oxazepan-5-one 1039747-11-9 C27H34N4O2
(2R)-2-(aminomethyl)-4-[(1R)-1-(1-benzyl-4-phenyl-1H-imidazol-2-yl)-2,2-dimethylpropyl]-1,4-oxazepan-5-one
—— 5-allyl-3-methyl-7-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one 1032648-93-3 C25H19F4N5O2
5-allyl-3-methyl-7-{2,2,2-trifluoro-1-[1-(4-fluorophenyl)-1H-indazol-5-yl]-1-hydroxyethyl}-3,5-dihydropyrrolo[3,2-d]pyrimidin-4-one
—— N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-16-5 C20H22N2O3
N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— 2-{2-[2-(4-trifluoromethyl-phenoxymethyl)-1H-benzoimidazol-5-yl]-benzenesulfonyl}-ethanol 1033624-54-2 C23H19F3N2O4S
2-{2-[2-(4-trifluoromethyl-phenoxymethyl)-1H-benzoimidazol-5-yl]-benzenesulfonyl}-ethanol
—— N-{[1-benzyl-7-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-2-yl]methyl}-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-33-6 C29H30F3N3O2
N-{[1-benzyl-7-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-2-yl]methyl}-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— N-{(3S)-3-[4-(dimethylamino)phenyl]cyclopentyl}-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea 1034770-38-1 C24H31N3O2
N-{(3S)-3-[4-(dimethylamino)phenyl]cyclopentyl}-N'-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
—— 1-oxo-2-(quinolin-4-ylmethyl)-N-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide 1035699-63-8 C27H20F3N3O2
1-oxo-2-(quinolin-4-ylmethyl)-N-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline-5-carboxamide
—— (E)-3-(4-{2-[1-(2-Chloro-4-methanesulfonyl-benzyl)-piperidin-4-ylamino]-pyrimidin-4-ylamino}-3,5-dimethyl-phenyl)-acrylonitrile 1033954-30-1 C28H31ClN6O2S
(E)-3-(4-{2-[1-(2-Chloro-4-methanesulfonyl-benzyl)-piperidin-4-ylamino]-pyrimidin-4-ylamino}-3,5-dimethyl-phenyl)-acrylonitrile
—— 7-chloro-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride 1000781-39-4 C12H13ClN2O2*ClH
7-chloro-1,2,3,4,12,12a-hexahydro-6H-pyrazino[2,1-c][1,4]benzoxazepin-6-one hydrochloride
—— 1,4-dihydro-4-[3-[(2-hydroxyethyl)amino]-1H-indazol-5-yl]-2,6-dimethyl-3,5-pyridinedicarbonitrile 1033768-41-0 C18H18N6O
1,4-dihydro-4-[3-[(2-hydroxyethyl)amino]-1H-indazol-5-yl]-2,6-dimethyl-3,5-pyridinedicarbonitrile
—— 5-[6-(cyclopropylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[2-(dimethylamino)ethyl]thiophene-2-carboxamide 1033243-65-0 C19H24N6OS
5-[6-(cyclopropylmethylamino)imidazo[1,2-b]pyridazin-3-yl]-N-[2-(dimethylamino)ethyl]thiophene-2-carboxamide