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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8S)-N-methoxy-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole-5-carboxamide 1046468-96-5 C21H23N3O3
(8S)-N-methoxy-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole-5-carboxamide
—— (8S)-5-[(3-propoxyazetidin-1-yl)carbonyl]-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole 1046468-93-2 C26H31N3O3
(8S)-5-[(3-propoxyazetidin-1-yl)carbonyl]-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole
—— 2-Diethoxyphosphoryl-1-[4-(2-hydroxyethoxy)-2,3-dimethylphenyl]ethanone 1045863-43-1 C16H25O6P
2-Diethoxyphosphoryl-1-[4-(2-hydroxyethoxy)-2,3-dimethylphenyl]ethanone
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-[2-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-L-phenylalanine 1031342-50-3 C25H22BrF3N4O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-[2-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-L-phenylalanine
—— N-((1S)-2-amino-1-{[2-(trifluoromethyl)phenyl]methyl}ethyl)-2-chloro-1-methyl-5-(1-methyl-1H-pyrazol-5-yl)-1H-pyrrole-3-carboxamide 1044852-31-4 C20H21ClF3N5O
N-((1S)-2-amino-1-{[2-(trifluoromethyl)phenyl]methyl}ethyl)-2-chloro-1-methyl-5-(1-methyl-1H-pyrazol-5-yl)-1H-pyrrole-3-carboxamide
—— 1-{2-fluoro-4-[2-(3-hydroxy-propylamino)-pyrimidin-4-yloxy]-phenyl}-3-(4-chloro-3-trifluoromethylphenyl)-urea 1035558-59-8 C21H18ClF4N5O3
1-{2-fluoro-4-[2-(3-hydroxy-propylamino)-pyrimidin-4-yloxy]-phenyl}-3-(4-chloro-3-trifluoromethylphenyl)-urea
—— (8S)-1-[(2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazol-5-yl)carbonyl]azetidine-2-carboxamide 1046468-94-3 C24H26N4O3
(8S)-1-[(2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazol-5-yl)carbonyl]azetidine-2-carboxamide
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-[2-(methylthio)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine 1031341-48-6 C27H29BrN4O3S
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-{2-[2-(methylthio)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}-L-phenylalanine
—— 1-[4-(2-{4-[4-(2,4-difluoro-phenoxy)-thieno[3,2-d]pyrimidin-2-yl]-phenoxy}-ethyl)-[1,4]diazepan-1-yl]-ethanone 1043929-78-7 C27H26F2N4O3S
1-[4-(2-{4-[4-(2,4-difluoro-phenoxy)-thieno[3,2-d]pyrimidin-2-yl]-phenoxy}-ethyl)-[1,4]diazepan-1-yl]-ethanone
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-[2-(cyclopropylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-L-phenylalanine 1031341-03-3 C28H29BrN4O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-[2-(cyclopropylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-L-phenylalanine
—— (8S)-5-[(3-methoxyazetidin-1-yl)carbonyl]-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole 1046468-92-1 C24H27N3O3
(8S)-5-[(3-methoxyazetidin-1-yl)carbonyl]-2,3-dimethyl-8-(2-methylphenyl)-3,6,7,8-tetrahydrochromeno[7,8-d]imidazole
—— 5'-O-[({2-[(2-cycloheptylcarbonyl)oxy]ethyl}amino)(phenoxy)phosphoryl]-2'-C-methylcytidine 1039052-88-4 C26H37N4O9P
5'-O-[({2-[(2-cycloheptylcarbonyl)oxy]ethyl}amino)(phenoxy)phosphoryl]-2'-C-methylcytidine
—— 3,4-dihydro-3-phenethyl-5-methyl-4-methylene-7-ethylsulfanyl-pyrido[4,3-d]pyrimidine-8-carbonitrile 1097698-99-1 C20H20N4S
3,4-dihydro-3-phenethyl-5-methyl-4-methylene-7-ethylsulfanyl-pyrido[4,3-d]pyrimidine-8-carbonitrile
—— 1-methyl-3-(4-methyl-piperazin-1-yl)-1H-indazole-6-carboxylic acid 4-methoxy-benzylamide 1027257-28-8 C22H27N5O2
1-methyl-3-(4-methyl-piperazin-1-yl)-1H-indazole-6-carboxylic acid 4-methoxy-benzylamide
—— 4-{2-amino-4-[5-(2-fluoro-5-methoxyphenyl)pyridin-3-yl]-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl}phenyl methanesulfonate 1035265-94-1 C23H21FN4O5S
4-{2-amino-4-[5-(2-fluoro-5-methoxyphenyl)pyridin-3-yl]-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl}phenyl methanesulfonate
—— cytidine, 5'-O-[[[2-(benzyloxy)ethyl]amino]phenyloxyphosphinyl]-2'-C-methyl 1039052-84-0 C25H29N4O9P
cytidine, 5'-O-[[[2-(benzyloxy)ethyl]amino]phenyloxyphosphinyl]-2'-C-methyl
—— (+/-)-1-(3,4-dihydro-2,2-dimethyl-2H-1-benzopyran-4-yl)-3-(isoquinolin-5-yl)urea 1026994-09-1 C21H21N3O2
(+/-)-1-(3,4-dihydro-2,2-dimethyl-2H-1-benzopyran-4-yl)-3-(isoquinolin-5-yl)urea
—— 1-{2-chloro-4-[2-(3-hydroxy-propylamino)-pyrimidin-4-yloxy]-phenyl}-3-(4-chloro-3-trifluoromethylphenyl)-urea 1035558-47-4 C21H18Cl2F3N5O3
1-{2-chloro-4-[2-(3-hydroxy-propylamino)-pyrimidin-4-yloxy]-phenyl}-3-(4-chloro-3-trifluoromethylphenyl)-urea
—— 5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-5-methyl-4,5-dihydro-1 H-pyrazole-3-carboxylic acid cycloheptylamide 1040397-94-1 C24H26Cl3N3O
5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-5-methyl-4,5-dihydro-1 H-pyrazole-3-carboxylic acid cycloheptylamide
—— [6-fluoro-2-methyl-3-(4-pyrimidin-5-ylphenylsulfanyl)indolizin-1-yl]acetic acid 1036713-51-5 C21H16FN3O2S
[6-fluoro-2-methyl-3-(4-pyrimidin-5-ylphenylsulfanyl)indolizin-1-yl]acetic acid
—— 8-amino-1-methyl-2-phenyl-4,5-dihydro-1H-1,7,9-triaza-cyclopenta[a]naphthalene-3-carboxylic acid amide 1031441-29-8 C18H17N5O
8-amino-1-methyl-2-phenyl-4,5-dihydro-1H-1,7,9-triaza-cyclopenta[a]naphthalene-3-carboxylic acid amide
—— 1,1-dioxo-5-(3-(trifluoromethyl)benzyl)-2-(3,4-dichlorophenylimino)-1λ6-thiazolidin-4-one 1041671-89-9 C17H11Cl2F3N2O3S
1,1-dioxo-5-(3-(trifluoromethyl)benzyl)-2-(3,4-dichlorophenylimino)-1λ6-thiazolidin-4-one
—— N-(2-chloro-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine 1031341-35-1 C29H26ClN5O3
N-(2-chloro-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-pyridin-3-yl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine
—— 3-[(pyridin-2-yl)sulfonylmethyl]-N(4),N(5)-dibenzylisoxazole-4,5-dicarboxamide 1135402-44-6 C25H22N4O5S
3-[(pyridin-2-yl)sulfonylmethyl]-N(4),N(5)-dibenzylisoxazole-4,5-dicarboxamide
—— 2-(3'-methoxyphenyl)-6,7-methylenedioxyquinolin-4-yl-phosphate 1032315-80-2 C17H14NO7P
2-(3'-methoxyphenyl)-6,7-methylenedioxyquinolin-4-yl-phosphate
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-piperidin-4-yl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine 1031342-41-2 C29H32BrN5O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(2-piperidin-4-yl-3H-imidazo[4,5-b]pyridin-3-yl)-L-phenylalanine
—— [(3aS,4R,6aR)-2,3,3a,4,5,6a-hexahydrofuro[2,3-b]furan-4-yl] N-[(2S,3R)-3-amino-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-1-(4-phenylmethoxyphenyl)butan-2-yl]carbamate 1005324-22-0 C35H45N3O8S
[(3aS,4R,6aR)-2,3,3a,4,5,6a-hexahydrofuro[2,3-b]furan-4-yl] N-[(2S,3R)-3-amino-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-1-(4-phenylmethoxyphenyl)butan-2-yl]carbamate
—— 2-(1-(4-bromophenyl)-2-(2,4-dichlorophenyl)-5-ethyl-1H-imidazol-4-yl)-5-t-butyl-1,3,4-oxadiazole 1049683-22-8 C23H21BrCl2N4O
2-(1-(4-bromophenyl)-2-(2,4-dichlorophenyl)-5-ethyl-1H-imidazol-4-yl)-5-t-butyl-1,3,4-oxadiazole
—— UVI5014 1052247-26-3 C26H26Br2N6O4S2
UVI5014
—— N-(4-{methyl[2-({3-[2-(4-morpholinyl)ethyl]phenyl}amino)-4-pyrimidinyl]amino}phenyl)-N'-[3-(trifluoromethyl)phenyl]urea 1027211-25-1 C31H32F3N7O2
N-(4-{methyl[2-({3-[2-(4-morpholinyl)ethyl]phenyl}amino)-4-pyrimidinyl]amino}phenyl)-N'-[3-(trifluoromethyl)phenyl]urea
—— (R/S)-2-hydroxy-2-methyl-N-((S)-6-oxo-6,7-dihydro-5H-dibenzo[b,d]azepin-7-yl)-N'-(3,3,3-trifluoro-propyl)-malonamide 1043963-64-9 C21H20F3N3O4
(R/S)-2-hydroxy-2-methyl-N-((S)-6-oxo-6,7-dihydro-5H-dibenzo[b,d]azepin-7-yl)-N'-(3,3,3-trifluoro-propyl)-malonamide
—— 7-methoxy-2-oxo-8-propyl-2H-chromene-3-carboxylic acid (4-pyrrolidin-2-yl-phenyl)-amide 1043906-61-1 C24H26N2O4
7-methoxy-2-oxo-8-propyl-2H-chromene-3-carboxylic acid (4-pyrrolidin-2-yl-phenyl)-amide
—— JNJ 39758979 1046447-90-8 C11H19N5
JNJ 39758979
—— methyl 1-hydroxy-6-difluoromethoxybenzo[4,5]furo[3,2-c]pyridine-9-carboxylate 1038400-61-1 C14H9F2NO5
methyl 1-hydroxy-6-difluoromethoxybenzo[4,5]furo[3,2-c]pyridine-9-carboxylate
—— 2-{2-[1-(2,6-dimethylbenzyl)-6-fluoro-1H-benzimidazol-2-yl]-5-methoxy-3-methylphenoxy}acetamide 1050479-28-1 C26H26FN3O3
2-{2-[1-(2,6-dimethylbenzyl)-6-fluoro-1H-benzimidazol-2-yl]-5-methoxy-3-methylphenoxy}acetamide
—— 2-[3-(naphthalene-1-yloxy)-3-thiophen-2-yl-propyl]-isoindole-1,3-dione 1037816-88-8 C25H19NO3S
2-[3-(naphthalene-1-yloxy)-3-thiophen-2-yl-propyl]-isoindole-1,3-dione
—— (R)-tert-butyl 3-(4-(2-butyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl)-2-fluorophenylamino)pyrrolidine-1-carboxylate 1046159-21-0 C27H33FN4O3
(R)-tert-butyl 3-(4-(2-butyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl)-2-fluorophenylamino)pyrrolidine-1-carboxylate
—— benzyl {6-[(3S)-3-(2-fluorophenoxy)pyrrolidin-1-yl]pyridin-3-yl}carbamate 1010398-47-6 C23H22FN3O3
benzyl {6-[(3S)-3-(2-fluorophenoxy)pyrrolidin-1-yl]pyridin-3-yl}carbamate
—— N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(5-fluoro-2-pyridin-3-yl-1H-benzimidazol-1-yl)-L-phenylalanine 1031340-97-2 C30H26BrFN4O3
N-(2-bromo-3-oxospiro[3.5]non-1-en-1-yl)-4-(5-fluoro-2-pyridin-3-yl-1H-benzimidazol-1-yl)-L-phenylalanine
—— 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-methylamino-ethyl)-1H-indol-5-yl]-amide 1042720-32-0 C20H20ClN3O2S2
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-methylamino-ethyl)-1H-indol-5-yl]-amide
—— 2-methylpropyl 2-[[2-(4-chlorophenyl)-3-morpholin-4-yl-3-sulfanylideneprop-1-enyl]amino]acetate 164595-35-1 C19H25ClN2O3S
2-methylpropyl 2-[[2-(4-chlorophenyl)-3-morpholin-4-yl-3-sulfanylideneprop-1-enyl]amino]acetate
—— 4-fluoro-N-(((4R,5R)-3-(4-fluorophenyl)-4-(4-hydroxyphenyl)-2-oxooxazolidin-5-yl)methyl)benzamide 1011265-09-0 C23H18F2N2O4
4-fluoro-N-(((4R,5R)-3-(4-fluorophenyl)-4-(4-hydroxyphenyl)-2-oxooxazolidin-5-yl)methyl)benzamide
—— (2S)-Benzofuran-4-carboxylic acid [1-(biphenyl-2-sulfonyl)-azetidin-2-ylmethyl]-amide 1007873-75-7 C25H22N2O4S
(2S)-Benzofuran-4-carboxylic acid [1-(biphenyl-2-sulfonyl)-azetidin-2-ylmethyl]-amide
—— N-[2-amino-1-(phenylmethyl)ethyl]-5-(1-methyl-1H-imidazol-5-yl)-2-thiophenecarboxamide 1047645-36-2 C18H20N4OS
N-[2-amino-1-(phenylmethyl)ethyl]-5-(1-methyl-1H-imidazol-5-yl)-2-thiophenecarboxamide
—— 4'-(p-fluorobenzenesulfonate)-4-hydroxychalcone 1010118-53-2 C21H15FO5S
4'-(p-fluorobenzenesulfonate)-4-hydroxychalcone
—— 2-[2-Fluoro-4-(methylsulfonyl)phenyl]-5-[({1-[3-(1-methylethyl)-1,2,4-thiadiazol-5-yl]-4-piperidinyl}methyl)oxy]pyridine 1032824-70-6 C23H27FN4O3S2
2-[2-Fluoro-4-(methylsulfonyl)phenyl]-5-[({1-[3-(1-methylethyl)-1,2,4-thiadiazol-5-yl]-4-piperidinyl}methyl)oxy]pyridine
—— 4-[[4-[4-[(E)-2-cyanovinyl]-2,6-dimethyl-anilino]-6-[(2-methoxyethylamino)methyl]pyrimidin-2-yl]amino]benzonitrile 1037445-04-7 C26H27N7O
4-[[4-[4-[(E)-2-cyanovinyl]-2,6-dimethyl-anilino]-6-[(2-methoxyethylamino)methyl]pyrimidin-2-yl]amino]benzonitrile
—— [4-difluoromethoxy-2-ethyl-8-fluoro-3-(4-pyrazol-1-yl-benzyl)quinolin-5-yloxy]acetic acid 1071495-39-0 C24H20F3N3O4
[4-difluoromethoxy-2-ethyl-8-fluoro-3-(4-pyrazol-1-yl-benzyl)quinolin-5-yloxy]acetic acid
—— 1-methyl-2-o-tolyl-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide 1031441-11-8 C20H19N3O
1-methyl-2-o-tolyl-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid amide
—— 4-(benzyloxy)-5-[(3R)-3-hydroxy-3-(2-methylphenyl)propyl]-N-methoxy-N,1,2-trimethyl-1H-benzimidazole-6-carboxamide 1034771-36-2 C29H33N3O4
4-(benzyloxy)-5-[(3R)-3-hydroxy-3-(2-methylphenyl)propyl]-N-methoxy-N,1,2-trimethyl-1H-benzimidazole-6-carboxamide