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—— ((S)-1-{(1S,2R,3R)-1-Benzyl-3-(2.4-dimethoxy-benzylamino)-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-propylcarbamoyl}-2,2-dimethyl-propyl)-carbamic Acid Benzyl Ester —— C47H61N5O10
((S)-1-{(1S,2R,3R)-1-Benzyl-3-(2.4-dimethoxy-benzylamino)-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-propylcarbamoyl}-2,2-dimethyl-propyl)-carbamic Acid Benzyl Ester
—— {(S)-1-[(1S,2R,3R)-1-benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-(3-methoxy-benzylamino)-propylcarbamoyl]-2,2-dimethyl-propyl}-carbamic acid benzyl ester —— C46H59N5O9
{(S)-1-[(1S,2R,3R)-1-benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-(3-methoxy-benzylamino)-propylcarbamoyl]-2,2-dimethyl-propyl}-carbamic acid benzyl ester
—— ((S)-1-{(1S,2R,3R)-1-benzyl-3-(3,5-dimethoxy-benzylamino)-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-propylcarbamoyl}-2,2-dimethyl-propyl)-carbamic acid benzyl ester —— C47H61N5O10
((S)-1-{(1S,2R,3R)-1-benzyl-3-(3,5-dimethoxy-benzylamino)-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-propylcarbamoyl}-2,2-dimethyl-propyl)-carbamic acid benzyl ester
—— (S,E)‐4‐(tert‐butyl)‐3‐(4‐methylpent‐2‐enoyl)oxazolidin‐2‐one —— C13H21NO3
(S,E)‐4‐(tert‐butyl)‐3‐(4‐methylpent‐2‐enoyl)oxazolidin‐2‐one
—— (S)-[1-[[(4,5-dihydro-5-thioxo-1,3,4-thiadiazol-2-yl)amino]carbonyl]-2,2-dimethylpropyl]carbamic acid phenylmethyl ester —— C16H20N4O3S2
(S)-[1-[[(4,5-dihydro-5-thioxo-1,3,4-thiadiazol-2-yl)amino]carbonyl]-2,2-dimethylpropyl]carbamic acid phenylmethyl ester
—— {(S)-1-[(1S,2R,3R)-1-benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-(3,4,5-trimethoxy-benzylamino)-propylcarbamoyl]-2,2-dimethyl-propyl}-carbamic acid benzyl ester —— C48H63N5O11
{(S)-1-[(1S,2R,3R)-1-benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-(3,4,5-trimethoxy-benzylamino)-propylcarbamoyl]-2,2-dimethyl-propyl}-carbamic acid benzyl ester
—— ((S)-1-{(1S,2R,3R)-1-Benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-[(naphthalen-1-ylmethyl)-amino]-propylcarbamoyl}-2.2-dimethyl-propyl)-carbamic Acid Benzyl Ester —— C49H59N5O8
((S)-1-{(1S,2R,3R)-1-Benzyl-2-hydroxy-3-[(S)-1-(2-hydroxy-4-methoxy-benzylcarbamoyl)-2-methyl-propylcarbamoyl]-3-[(naphthalen-1-ylmethyl)-amino]-propylcarbamoyl}-2.2-dimethyl-propyl)-carbamic Acid Benzyl Ester
—— (S)-4-methyl-1-(1-methyl-1H-imidazole-2-yl)-3-(1-methyl-1H-indol-3-yl)pentan-1-one —— C19H23N3O
(S)-4-methyl-1-(1-methyl-1H-imidazole-2-yl)-3-(1-methyl-1H-indol-3-yl)pentan-1-one
—— (S,E)-3-(4'-methylpent-2'-enoyl)-4-benzyloxazolidin-2-one —— C16H19NO3
(S,E)-3-(4'-methylpent-2'-enoyl)-4-benzyloxazolidin-2-one
—— (S)-2-fluorocyclohexylacetaldehyde —— C8H13FO
(S)-2-fluorocyclohexylacetaldehyde
—— (-)-(S)-2-cyano-2-(1H-indol-3-yl)propanoic acid —— C12H10N2O2
(-)-(S)-2-cyano-2-(1H-indol-3-yl)propanoic acid
—— (S)-(-)-1-Phenylethyl 2,2-dimethylpropionate —— C13H18O2
(S)-(-)-1-Phenylethyl 2,2-dimethylpropionate
—— (S*)-N-[[1-[[[(1,1-Dimethylethoxy)carbonyl]amino][[(1,1-dimethylethoxy)carbonyl]imino]methyl]-4-piperidinyl]methyl]-1-[1-[[(1,1-dimethylethoxy)carbonyl]amino]-2-phenylethyl]-L-prolinamide —— C35H56N6O7
(S*)-N-[[1-[[[(1,1-Dimethylethoxy)carbonyl]amino][[(1,1-dimethylethoxy)carbonyl]imino]methyl]-4-piperidinyl]methyl]-1-[1-[[(1,1-dimethylethoxy)carbonyl]amino]-2-phenylethyl]-L-prolinamide
—— (S*)-N-[[1-[[[(1,1-Dimethylethoxy)carbonyl]amino][[(1,1-dimethylethoxy)carbonyl]imino]methyl]-4-piperidinyl]methyl]-1-[1-[[(1,1-dimethylethoxy)carbonyl]amino]-2-phenylethyl]-S-prolinamide —— C35H56N6O7
(S*)-N-[[1-[[[(1,1-Dimethylethoxy)carbonyl]amino][[(1,1-dimethylethoxy)carbonyl]imino]methyl]-4-piperidinyl]methyl]-1-[1-[[(1,1-dimethylethoxy)carbonyl]amino]-2-phenylethyl]-S-prolinamide
—— S-α-methyl-<1-(2-chlorophenyl)-2-(2'-pyrido)-1-ethylidene>benzylamine —— C21H19ClN2
S-α-methyl-<1-(2-chlorophenyl)-2-(2'-pyrido)-1-ethylidene>benzylamine
—— (S)-3-(2-chlorophenyl)-3-hydroxypropanenitrile —— C9H8ClNO
(S)-3-(2-chlorophenyl)-3-hydroxypropanenitrile
—— S-6-ethyl-2-{2-[3-(3-methylpyrazin-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine —— C23H24N8O
S-6-ethyl-2-{2-[3-(3-methylpyrazin-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine
—— (S)-6-chloro-4-(5-methyl-1H-pyrazol-3-ylamino)-2-[2-{3-(pyrimid-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]pyrimidine —— C19H18ClN9O
(S)-6-chloro-4-(5-methyl-1H-pyrazol-3-ylamino)-2-[2-{3-(pyrimid-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]pyrimidine
—— S-6-(2-methoxyethoxy)-2-[2-{3-(4-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C24H25N9O3
S-6-(2-methoxyethoxy)-2-[2-{3-(4-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— (S)-2-[5-(1-tert-butoxycarbonylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid ethyl ester —— C15H24N4O4
(S)-2-[5-(1-tert-butoxycarbonylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid ethyl ester
—— S-6-(3-cyanopropoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C24H26N10O2
S-6-(3-cyanopropoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-(2-methoxyethoxy)-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C24H25N9O3
S-6-(2-methoxyethoxy)-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-chloro-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine —— C21H18ClN7O
S-6-chloro-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine
—— S-6-methoxy-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine —— C22H21N7O2
S-6-methoxy-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine
—— S-6-morpholino-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine —— C25H26N8O2
S-6-morpholino-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine
—— S-2-[2-{3-(2-methylaminopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C21H23N9O
S-2-[2-{3-(2-methylaminopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-(3-methoxypropoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C24H29N9O3
S-6-(3-methoxypropoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-[(1-cyanocyclopropyl)methoxy]-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C25H26N10O2
S-6-[(1-cyanocyclopropyl)methoxy]-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-(2-methoxyethoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C23H27N9O3
S-6-(2-methoxyethoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-2-[2-{3-(2-chloropyrid-3-yl)isoxazol-5-yl}-pyrrolidin-1-yl]-6-methyl-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C21H21ClN8O
S-2-[2-{3-(2-chloropyrid-3-yl)isoxazol-5-yl}-pyrrolidin-1-yl]-6-methyl-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-(2-ethoxyethoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C24H29N9O3
S-6-(2-ethoxyethoxy)-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-methoxy-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C21H23N9O2
S-6-methoxy-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-methoxy-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C22H21N9O2
S-6-methoxy-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-ethyl-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C22H25N9O
S-6-ethyl-2-[2-{3-(3-methylpyrazin-2-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-methyl-2-[2-{3-(2-methylaminopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C22H25N9O
S-6-methyl-2-[2-{3-(2-methylaminopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-2-[2-{3-(2-chloropyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C20H19ClN8O
S-2-[2-{3-(2-chloropyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-methoxy-2-[2-{3-(1-oxopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C21H22N8O3
S-6-methoxy-2-[2-{3-(1-oxopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— (S)-2-((6-(1H-pyrazol-1-yl)pyrimidin-4-yl)amino)-4-(((R)-2-methoxypropyl)(4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butyl)amino)butanoic acid —— C27H38N8O3
(S)-2-((6-(1H-pyrazol-1-yl)pyrimidin-4-yl)amino)-4-(((R)-2-methoxypropyl)(4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)butyl)amino)butanoic acid
—— (S)-2-[5-(1-acetylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid ethyl ester —— C12H18N4O3
(S)-2-[5-(1-acetylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid ethyl ester
—— (S)-2-[4-(1-acetylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid N-methyl amide —— C11H17N5O2
(S)-2-[4-(1-acetylpyrrolidin-2-yl)-(1,2,3)-triazol-1-yl]acetic acid N-methyl amide
—— S-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-(5-methyl-1H-pyrazol-3-ylamino)-6-morpholinopyrimidine —— C25H26N10O2
S-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-(5-methyl-1H-pyrazol-3-ylamino)-6-morpholinopyrimidine
—— S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(4-methylpyrid-2-ylamino)pyrimidine —— C23H23N7O
S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(4-methylpyrid-2-ylamino)pyrimidine
—— S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(4-cyanopyrid-2-ylamino)pyrimidine —— C23H20N8O
S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(4-cyanopyrid-2-ylamino)pyrimidine
—— S-6-chloro-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C21H18ClN9O
S-6-chloro-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-6-methyl-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C22H21N9O
S-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-6-methyl-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(5-cyanopyrid-2-ylamino)pyrimidine —— C23H20N8O
S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(5-cyanopyrid-2-ylamino)pyrimidine
—— S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(5-methylpyrid-2-ylamino)pyrimidine —— C23H23N7O
S-6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(5-methylpyrid-2-ylamino)pyrimidine
—— S-6-ethyl-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine —— C23H23N9O
S-6-ethyl-2-[2-{3-(2-cyanopyrid-3-yl)isoxazol-5-yl}pyrrolidin-1-yl]-4-(5-methyl-1H-pyrazol-3-ylamino)pyrimidine
—— (S)-(Z)-5-[[5-Fluoro-2-oxo-4-[(pyrrolidin-2-yl)ethynyl]-1,2-dihydro-indol-3-ylidene]methyl]-4-methyl-1H-pyrrole-3-carboxylic acid ethyl ester —— C23H22FN3O3
(S)-(Z)-5-[[5-Fluoro-2-oxo-4-[(pyrrolidin-2-yl)ethynyl]-1,2-dihydro-indol-3-ylidene]methyl]-4-methyl-1H-pyrrole-3-carboxylic acid ethyl ester
—— (S)-(Z)-3-[(4-acetyl-1H-pyrrol-2-yl)methylene]-1,3-dihydro-5-fluoro-4-[(pyrrolidin-2-yl)ethynyl]-2H-indol-2-one —— C21H18FN3O2
(S)-(Z)-3-[(4-acetyl-1H-pyrrol-2-yl)methylene]-1,3-dihydro-5-fluoro-4-[(pyrrolidin-2-yl)ethynyl]-2H-indol-2-one