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—— (R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,4-dimethyloxazol-5-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide 1616100-75-4 C23H26F2N4O3S
(R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,4-dimethyloxazol-5-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,5-dimethyloxazol-4-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide 1616100-72-1 C23H28F2N4O3S
(R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,5-dimethyloxazol-4-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,5-dimethyloxazol-4-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide 1616100-71-0 C23H26F2N4O3S
(R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,5-dimethyloxazol-4-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(3,5-dimethylisoxazol-4-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide 1616100-68-5 C23H28F2N4O3S
(R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(3,5-dimethylisoxazol-4-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-3,5-dichloro-1-(1-cyclopropyl-2-methoxyethyl)pyrazin-2(1H)-one 1173435-16-9 C10H12Cl2N2O2
(R)-3,5-dichloro-1-(1-cyclopropyl-2-methoxyethyl)pyrazin-2(1H)-one
—— (R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(3,5-dimethylisoxazol-4-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide 1585970-78-0 C23H26F2N4O3S
(R)-N-((S)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(3,5-dimethylisoxazol-4-yl)-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,4-dimethyloxazol-5-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide 1616100-76-5 C23H28F2N4O3S
(R)-N-((2S,4R)-2-(2,4-difluoro-5-(pyrimidin-5-yl)phenyl)-4-(2,4-dimethyloxazol-5-yl)-4-hydroxybutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-8-(1-hydroxy-3-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)propan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one 1548288-48-7 C25H30N2O6
(R)-8-(1-hydroxy-3-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)propan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— (R)-8-(1-hydroxy-2-methyl-1-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)propan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one 1548288-45-4 C26H32N2O6
(R)-8-(1-hydroxy-2-methyl-1-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)propan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— (R)-1'-(2-hydroxy-2-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)ethyl)spiro[indoline-3,4'-piperidin]-2-one 1548296-04-3 C23H24N2O4
(R)-1'-(2-hydroxy-2-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)ethyl)spiro[indoline-3,4'-piperidin]-2-one
—— (R)-2-methoxy-2-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)acetaldehyde 1548289-13-9 C12H12O4
(R)-2-methoxy-2-(4-methyl-1-oxo-1,3-dihydroisobenzofuran-5-yl)acetaldehyde
—— (R)-4-methoxy-6-(oxiran-2-yl)pyridine-3-carbonitrile 1433484-12-8 C9H8N2O2
(R)-4-methoxy-6-(oxiran-2-yl)pyridine-3-carbonitrile
—— (R)-5-(2-hydroxy-1-methoxyethyl)-4-methylisobenzofuran-1(3H)-one 1548289-20-8 C12H14O4
(R)-5-(2-hydroxy-1-methoxyethyl)-4-methylisobenzofuran-1(3H)-one
—— (rac)-2-amino-3-benzofuran-2-yl-propionic acid 748752-63-8 C11H11NO3
(rac)-2-amino-3-benzofuran-2-yl-propionic acid
—— (R)-dimethyl 2-(1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)malonate 1254200-29-7 C21H22O6
(R)-dimethyl 2-(1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)malonate
—— (R)-methyl-4-(4-((1-(1,3,4-oxadiazol-2-yl)propyl)(cyclopentyl)amino)-5-nitropyrimidin-2-ylamino)-3-methoxybenzoate 1278249-15-2 C23H27N7O6
(R)-methyl-4-(4-((1-(1,3,4-oxadiazol-2-yl)propyl)(cyclopentyl)amino)-5-nitropyrimidin-2-ylamino)-3-methoxybenzoate
—— (rac)-2-chloro-9-cyclohexyl-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-20-5 C15H21ClN4O
(rac)-2-chloro-9-cyclohexyl-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one
—— rac-1-{3-[6-(2-fluorophenyl)-4-methoxy-1-methyl-4H[1,2,4]triazolo[4,3-a][1,4] benzodiazepin-8-yl]-2-propynyl}-3,4-dihydro-2(1H)-quinolinone 125031-11-0 C30H24FN5O2
rac-1-{3-[6-(2-fluorophenyl)-4-methoxy-1-methyl-4H[1,2,4]triazolo[4,3-a][1,4] benzodiazepin-8-yl]-2-propynyl}-3,4-dihydro-2(1H)-quinolinone
—— rac-(2S,3R,4R,5R)-2'-chloro-4-(3-chloro-2-fluorophenyl)-N-(4-(2-hydroxyethoxy)-2-methoxyphenyl)-2-neopentyl-5'-oxo-4',5'-dihydrospiro[pyrrolidine-3,6'-thieno[3,2-b]pyrrole]-5-carboxamide —— C30H32Cl2FN3O5S
rac-(2S,3R,4R,5R)-2'-chloro-4-(3-chloro-2-fluorophenyl)-N-(4-(2-hydroxyethoxy)-2-methoxyphenyl)-2-neopentyl-5'-oxo-4',5'-dihydrospiro[pyrrolidine-3,6'-thieno[3,2-b]pyrrole]-5-carboxamide
—— (R)-[6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]acetic acid 905725-42-0 C13H16O3
(R)-[6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl]acetic acid
—— (R)-3-(1H-benzotriazol-1-yl)-3-(4-methoxyphenyl)-1-phenylpropan-1-one 955123-76-9 C22H19N3O2
(R)-3-(1H-benzotriazol-1-yl)-3-(4-methoxyphenyl)-1-phenylpropan-1-one
—— (R)-1-(furan-3-yl)ethan-1-ol 13129-26-5 C6H8O2
(R)-1-(furan-3-yl)ethan-1-ol
—— (R)-5-bromo-4-fluoro-2-nitro-N-(1-phenylethyl)aniline 1416336-43-0 C14H12BrFN2O2
(R)-5-bromo-4-fluoro-2-nitro-N-(1-phenylethyl)aniline
—— <R>-(-)-2,2,4-trimethylhexen-3-one 109529-41-1 C9H18O
<R>-(-)-2,2,4-trimethylhexen-3-one
—— (R)-tert-butyl 2-oxo-5-((S)-1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)-2,5-dihydro-1H-pyrrole-1-carboxylate 1266096-15-4 C25H27NO5
(R)-tert-butyl 2-oxo-5-((S)-1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)-2,5-dihydro-1H-pyrrole-1-carboxylate
—— (R)-2-amino-N-(2-(2-(dimethylamino)ethoxy)-5-fluoro-4-(1H-pyrazol-4-yl)phenyl)-4-phenylbutanamide 1623130-21-1 C23H28FN5O2
(R)-2-amino-N-(2-(2-(dimethylamino)ethoxy)-5-fluoro-4-(1H-pyrazol-4-yl)phenyl)-4-phenylbutanamide
—— (R,Z)-tert-butyl 1-(2-((2,4-dioxothiazolidin-5-ylidene)methyl)phenyl)piperidin-3-ylcarbamate 1204144-10-4 C20H25N3O4S
(R,Z)-tert-butyl 1-(2-((2,4-dioxothiazolidin-5-ylidene)methyl)phenyl)piperidin-3-ylcarbamate
—— (R)-3-hydroxy-3-(4-methoxyphenyl)-1-phenylpropan-1-one 872333-01-2 C16H16O3
(R)-3-hydroxy-3-(4-methoxyphenyl)-1-phenylpropan-1-one
—— (R)-ethyl 3-n-hexyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)propanoate 1373154-31-4 C17H33BO4
(R)-ethyl 3-n-hexyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)propanoate
—— (R)-1-(4-bromophenyl)ethane-1,2-diol 92093-23-7 C8H9BrO2
(R)-1-(4-bromophenyl)ethane-1,2-diol
—— (R)-5-(2-amino-5-fluoro-1-(1-phenylethyl)-1H-benzo[d]imidazol-6-yl)-N-(tert-butyl)-2-methoxypyridine-3-sulfonamide 1416334-11-6 C25H28FN5O3S
(R)-5-(2-amino-5-fluoro-1-(1-phenylethyl)-1H-benzo[d]imidazol-6-yl)-N-(tert-butyl)-2-methoxypyridine-3-sulfonamide
—— (R)-5-[2-(tert-Butyl-dimethyl-silanyloxy)-ethyl]-5-(3,4-dichloro-phenyl)-3-(3,4-dimethoxy-benzenesulfonyl)-oxazolidine 191673-72-0 C25H35Cl2NO6SSi
(R)-5-[2-(tert-Butyl-dimethyl-silanyloxy)-ethyl]-5-(3,4-dichloro-phenyl)-3-(3,4-dimethoxy-benzenesulfonyl)-oxazolidine
—— rac-(2'S,3'R,4'S,5'R)-6-chloro-4'-(3-chloro-2-fluoro-phenyl)-2'-(2,2-dimethyl-propyl)-2-oxo-1,2-dihydro-spiro[indole-3,3'-pyrrolidine]-5'-carboxylic acid —— C23H23Cl2FN2O3
rac-(2'S,3'R,4'S,5'R)-6-chloro-4'-(3-chloro-2-fluoro-phenyl)-2'-(2,2-dimethyl-propyl)-2-oxo-1,2-dihydro-spiro[indole-3,3'-pyrrolidine]-5'-carboxylic acid
—— (R)-3-(4-methoxyphenyl)-1,3-diphenylpropan-1-one 1020172-02-4 C22H20O2
(R)-3-(4-methoxyphenyl)-1,3-diphenylpropan-1-one
—— (R)-tert-butyl 1-((R)-1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)-3-oxo-1,3-dihydroisobenzofuran-1-carboxylate 1451051-31-2 C29H28O6
(R)-tert-butyl 1-((R)-1-(4-methoxyphenyl)-3-oxo-3-phenylpropyl)-3-oxo-1,3-dihydroisobenzofuran-1-carboxylate
—— rac-(2'S,3'R,4'S,5'R)-6-chloro-4'-(3-chloro-2-fluoro-phenyl)-2'-(2,2-dimethyl-propyl)-2-oxo-1,2-dihydro-spiro[indole-3,3'-pyrrolidine]-5'-carboxylic acid 1375747-55-9 C23H23Cl2FN2O3
rac-(2'S,3'R,4'S,5'R)-6-chloro-4'-(3-chloro-2-fluoro-phenyl)-2'-(2,2-dimethyl-propyl)-2-oxo-1,2-dihydro-spiro[indole-3,3'-pyrrolidine]-5'-carboxylic acid
—— (R)-tert-butyl 1-(2-formylphenyl)piperidin-3-ylcarbamate 1204176-44-2 C17H24N2O3
(R)-tert-butyl 1-(2-formylphenyl)piperidin-3-ylcarbamate
—— (R)-tert-butyl 1-(2-chloro-6-formylphenyl)piperidin-3-ylcarbamate 1204176-22-6 C17H23ClN2O3
(R)-tert-butyl 1-(2-chloro-6-formylphenyl)piperidin-3-ylcarbamate
—— rac-(2S,3S,4S,5R)-6'-chloro-4-(3-chloro-2-fluorophenyl)-N-(4-(2-hydroxyethoxy)-2-methoxyphenyl)-2-neopentyl-2'-oxo-1',2'-dihydrospiro[pyrrolidine-3,3'-pyrrolo[3,2-b]pyridine]-5-carboxamide —— C31H33Cl2FN4O5
rac-(2S,3S,4S,5R)-6'-chloro-4-(3-chloro-2-fluorophenyl)-N-(4-(2-hydroxyethoxy)-2-methoxyphenyl)-2-neopentyl-2'-oxo-1',2'-dihydrospiro[pyrrolidine-3,3'-pyrrolo[3,2-b]pyridine]-5-carboxamide
—— (R)-N-((R)-1-(3-chloro-2-fluorophenyl)allyl)-2-methylpropane-2-sulfinamide 1422510-11-9 C13H17ClFNOS
(R)-N-((R)-1-(3-chloro-2-fluorophenyl)allyl)-2-methylpropane-2-sulfinamide
—— rac-(6S,7R,8S,8aR)-8-(3-chloro-2-fluoro-phenyl)-7-(4-chloro-2-fluoro-phenyl)-2-((S)-3,4-dihydroxy-butyl)-6-(2,2-dimethyl-propyl)-1-oxo-octahydro-pyrrolo[1,2-a]pyrazine-7-carbonitrile 1364614-53-8 C29H33Cl2F2N3O3
rac-(6S,7R,8S,8aR)-8-(3-chloro-2-fluoro-phenyl)-7-(4-chloro-2-fluoro-phenyl)-2-((S)-3,4-dihydroxy-butyl)-6-(2,2-dimethyl-propyl)-1-oxo-octahydro-pyrrolo[1,2-a]pyrazine-7-carbonitrile
—— (R,Z)-tert-butyl 1-(2-chloro-6-((2,4-dioxothiazolidin-5-ylidene)methyl)phenyl)piperidin-3-ylcarbamate 1204112-50-4 C20H24ClN3O4S
(R,Z)-tert-butyl 1-(2-chloro-6-((2,4-dioxothiazolidin-5-ylidene)methyl)phenyl)piperidin-3-ylcarbamate
—— (R)-(+)-Methylsulfamic acid 3-(2-methoxyphenoxy)-2-[[(methylamino)sulfonyl]-oxy]propyl ester 128707-43-7 C12H20N2O8S2
(R)-(+)-Methylsulfamic acid 3-(2-methoxyphenoxy)-2-[[(methylamino)sulfonyl]-oxy]propyl ester
—— rac-6-{[(2R,3S,4R,5S)-3-(3-chloro-2-fluoro-phenyl)-4-(4-chloro-2-fluoro-phenyl)-4-cyano-5-(2,2-dimethyl-propyl)-pyrrolidine-2-carbonyl]-amino}-nicotinic acid methyl ester 1229705-02-5 C30H28Cl2F2N4O3
rac-6-{[(2R,3S,4R,5S)-3-(3-chloro-2-fluoro-phenyl)-4-(4-chloro-2-fluoro-phenyl)-4-cyano-5-(2,2-dimethyl-propyl)-pyrrolidine-2-carbonyl]-amino}-nicotinic acid methyl ester
—— r-2,c-7-diphenylhexahydro-1,4-diazepin-5-one 136661-52-4 C17H18N2O
r-2,c-7-diphenylhexahydro-1,4-diazepin-5-one
—— rac-(2S,3R,4S,5R)-N-(4-carbamoyl-2-methoxyphenyl)-4-(3-chloro-2-fluorophenyl)-2-neopentyl-2'-oxo-1',2'-dihydrospiro[pyrrolidine-3,3'-pyrrolo[3,2-c]pyridine]-5-carboxamide 1360821-10-8 C30H31ClFN5O4
rac-(2S,3R,4S,5R)-N-(4-carbamoyl-2-methoxyphenyl)-4-(3-chloro-2-fluorophenyl)-2-neopentyl-2'-oxo-1',2'-dihydrospiro[pyrrolidine-3,3'-pyrrolo[3,2-c]pyridine]-5-carboxamide
—— racemic 4-{[(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-5-(2,2-dimethylpropyl)pyrrolidine-2-carbonyl]amino}benzoic acid t-butyl ester —— C34H35Cl2F2N3O3
racemic 4-{[(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-5-(2,2-dimethylpropyl)pyrrolidine-2-carbonyl]amino}benzoic acid t-butyl ester
—— (R)-ethyl 2-((R)-2-aMino-3-(benzylthio)propanaMido)-2-phenylacetate 874096-43-2 C20H24N2O3S
(R)-ethyl 2-((R)-2-aMino-3-(benzylthio)propanaMido)-2-phenylacetate
—— rac-(2S,3R,4S)-4-(3-chloro-2-fluorophenyl)-3-(4-chloro-2-fluorophenyl)-3-cyano-2-(2,2-dimethylpropyl)pyrrolidine-1-carboxylic acid ((S)-3,4-dihydroxybutyl)amide 1290097-24-3 C27H31Cl2F2N3O3
rac-(2S,3R,4S)-4-(3-chloro-2-fluorophenyl)-3-(4-chloro-2-fluorophenyl)-3-cyano-2-(2,2-dimethylpropyl)pyrrolidine-1-carboxylic acid ((S)-3,4-dihydroxybutyl)amide
—— racemic-4-((2S,3R,4R,5R)-2'-chloro-4-(3-chloro-2-fluorophenyl)-2-neopentyl-5'-oxo-4',5'-dihydrospiro[pyrrolidine-3,6'-thieno[3,2-b]pyrrole]-5-ylcarboxamido)-3-methoxybenzoic acid —— C29H28Cl2FN3O5S
racemic-4-((2S,3R,4R,5R)-2'-chloro-4-(3-chloro-2-fluorophenyl)-2-neopentyl-5'-oxo-4',5'-dihydrospiro[pyrrolidine-3,6'-thieno[3,2-b]pyrrole]-5-ylcarboxamido)-3-methoxybenzoic acid