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—— ethyl (2Z)-2-[(5E)-5-[(4-fluorophenyl)methylidene]-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C22H25FN2O4S
ethyl (2Z)-2-[(5E)-5-[(4-fluorophenyl)methylidene]-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 6-(2,5-dimethoxyphenyl)-3-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-2-carboxylate —— C20H23NO5
ethyl 6-(2,5-dimethoxyphenyl)-3-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-2-carboxylate
—— Ethyl 2-[5-[(1,2-dimethylindol-3-yl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C19H20N2O4S
Ethyl 2-[5-[(1,2-dimethylindol-3-yl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— ethyl (2Z)-2-[(5E)-5-[(3-methylthiophen-2-yl)methylidene]-4-oxo-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C23H24N2O4S2
ethyl (2Z)-2-[(5E)-5-[(3-methylthiophen-2-yl)methylidene]-4-oxo-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-5-[(3-methylthiophen-2-yl)methylidene]-4-oxo-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C23H24N2O4S2
ethyl (2E)-2-[(5Z)-5-[(3-methylthiophen-2-yl)methylidene]-4-oxo-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 4-amino-2-[(E)-1-chloro-2-(4-methoxycarbonylphenyl)ethenyl]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate —— C20H18ClN3O5
ethyl 4-amino-2-[(E)-1-chloro-2-(4-methoxycarbonylphenyl)ethenyl]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate
—— ethyl (2Z)-2-[(5E)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate —— C21H26N2O4S2
ethyl (2Z)-2-[(5E)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-5-[(3,5-dimethoxyphenyl)methylidene]-3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C25H32N2O6S
ethyl (2E)-2-[(5Z)-5-[(3,5-dimethoxyphenyl)methylidene]-3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5E)-5-(naphthalen-1-ylmethylidene)-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C25H26N2O5S
ethyl (2E)-2-[(5E)-5-(naphthalen-1-ylmethylidene)-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 1-[2-[2-[[(Z)-3-(4-methoxyphenyl)prop-2-enoyl]amino]benzoyl]oxyacetyl]piperidine-4-carboxylate —— C27H30N2O7
ethyl 1-[2-[2-[[(Z)-3-(4-methoxyphenyl)prop-2-enoyl]amino]benzoyl]oxyacetyl]piperidine-4-carboxylate
—— ethyl (2E)-2-[(5E)-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-5-[(2-phenylmethoxyphenyl)methylidene]-1,3-thiazolidin-2-ylidene]acetate —— C27H28N2O5S
ethyl (2E)-2-[(5E)-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-5-[(2-phenylmethoxyphenyl)methylidene]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate —— C21H26N2O4S2
ethyl (2E)-2-[(5Z)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate
—— (E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(1,3-benzothiazol-2-yl)-4-(2-methoxyphenyl)but-3-enamide —— C26H22N2O4S
(E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(1,3-benzothiazol-2-yl)-4-(2-methoxyphenyl)but-3-enamide
—— ethyl (2E)-2-[(5E)-5-[(4-methylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H26N2O5S
ethyl (2E)-2-[(5E)-5-[(4-methylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2Z)-2-[(5E)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethylidene)-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C22H26N2O6S
ethyl (2Z)-2-[(5E)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethylidene)-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-5-[(4-cyanophenyl)methylidene]-3-[2-(furan-2-ylmethylamino)-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C22H19N3O5S
ethyl (2E)-2-[(5Z)-5-[(4-cyanophenyl)methylidene]-3-[2-(furan-2-ylmethylamino)-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-5-[(2-phenylmethoxyphenyl)methylidene]-1,3-thiazolidin-2-ylidene]acetate —— C27H28N2O5S
ethyl (2E)-2-[(5Z)-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-5-[(2-phenylmethoxyphenyl)methylidene]-1,3-thiazolidin-2-ylidene]acetate
—— (E)-N-[(E)-(4-fluorophenyl)methylideneamino]-4-(4-methoxyphenyl)-3-methyl-1,3-thiazol-2-imine —— C18H16FN3OS
(E)-N-[(E)-(4-fluorophenyl)methylideneamino]-4-(4-methoxyphenyl)-3-methyl-1,3-thiazol-2-imine
—— ethyl (4S)-6-[[(Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H27ClN4O5
ethyl (4S)-6-[[(Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[[(2E,5S)-2-(2-anilino-1-cyano-2-oxoethylidene)-4-oxo-3-phenyl-1,3-thiazolidin-5-yl]methyl]benzoate —— C28H23N3O4S
ethyl 4-[[(2E,5S)-2-(2-anilino-1-cyano-2-oxoethylidene)-4-oxo-3-phenyl-1,3-thiazolidin-5-yl]methyl]benzoate
—— ethyl (2E)-2-[(5E)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate —— C21H26N2O4S2
ethyl (2E)-2-[(5E)-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-5-[(4-methylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H26N2O5S
ethyl (2E)-2-[(5Z)-5-[(4-methylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H24F2N2O6S
ethyl (2E)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 4-[[(2E,5R)-2-(2-anilino-1-cyano-2-oxoethylidene)-4-oxo-3-phenyl-1,3-thiazolidin-5-yl]methyl]benzoate —— C28H23N3O4S
ethyl 4-[[(2E,5R)-2-(2-anilino-1-cyano-2-oxoethylidene)-4-oxo-3-phenyl-1,3-thiazolidin-5-yl]methyl]benzoate
—— ethyl (2Z)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H24F2N2O6S
ethyl (2Z)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— (E)-4-methyl-N-[(E)-(3-methylphenyl)methylideneamino]-3-phenyl-1,3-thiazol-2-imine —— C18H17N3S
(E)-4-methyl-N-[(E)-(3-methylphenyl)methylideneamino]-3-phenyl-1,3-thiazol-2-imine
—— ethyl (2Z)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C24H28F2N2O5S
ethyl (2Z)-2-[(5E)-5-[[4-(difluoromethoxy)phenyl]methylidene]-3-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2Z)-2-[(5E)-5-[(3,5-dimethoxyphenyl)methylidene]-3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C25H32N2O6S
ethyl (2Z)-2-[(5E)-5-[(3,5-dimethoxyphenyl)methylidene]-3-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[(5Z)-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidin-2-ylidene]acetate —— C24H23ClN2O5S
ethyl (2E)-2-[(5Z)-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-4-oxo-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2R)-2-[[(E)-3-bromo-4-(4-butoxyphenyl)-4-oxobut-2-enoyl]amino]butanoate —— C20H26BrNO5
ethyl (2R)-2-[[(E)-3-bromo-4-(4-butoxyphenyl)-4-oxobut-2-enoyl]amino]butanoate
—— ethyl (4R)-6-[[(Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H27ClN4O5
ethyl (4R)-6-[[(Z)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 4-{[butyl({[3-methyl-1-(4-methylphenyl)-4-phenyl-1H-pyrazol-5-YL]carbamoyl}methyl)carbamoyl]amino}benzoate —— C33H37N5O4
Ethyl 4-{[butyl({[3-methyl-1-(4-methylphenyl)-4-phenyl-1H-pyrazol-5-YL]carbamoyl}methyl)carbamoyl]amino}benzoate
—— Ethyl 4-[butyl-[1-[3-(2-methoxyphenyl)-4-oxoquinazolin-2-yl]ethyl]amino]-4-oxobutanoate —— C27H33N3O5
Ethyl 4-[butyl-[1-[3-(2-methoxyphenyl)-4-oxoquinazolin-2-yl]ethyl]amino]-4-oxobutanoate
—— Ethyl 2-[[cyclopropyl-(3,4-dichlorobenzoyl)amino]methyl]-1,3-thiazole-4-carboxylate —— C17H16Cl2N2O3S
Ethyl 2-[[cyclopropyl-(3,4-dichlorobenzoyl)amino]methyl]-1,3-thiazole-4-carboxylate
—— ethyl 2-[(Z)-2-[4-(cyanomethoxy)-3-methoxyphenyl]ethenyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C21H19N3O5S
ethyl 2-[(Z)-2-[4-(cyanomethoxy)-3-methoxyphenyl]ethenyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (2S)-2-[[(E)-3-bromo-4-(4-butoxyphenyl)-4-oxobut-2-enoyl]amino]butanoate —— C20H26BrNO5
ethyl (2S)-2-[[(E)-3-bromo-4-(4-butoxyphenyl)-4-oxobut-2-enoyl]amino]butanoate
—— Ethyl 2-[2-[2-(tert-butylcarbamoylamino)-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate —— C14H21N3O4S2
Ethyl 2-[2-[2-(tert-butylcarbamoylamino)-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate
—— ethyl 2-(3,4-dichlorophenyl)-4-hydroxy-1,5,6,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidine-7(2H)-carboxylate —— C18H17Cl2N3O3S
ethyl 2-(3,4-dichlorophenyl)-4-hydroxy-1,5,6,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidine-7(2H)-carboxylate
—— ethyl 4-[(Z)-3-(3-methoxy-4-phenylmethoxyphenyl)prop-2-enoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H27NO5
ethyl 4-[(Z)-3-(3-methoxy-4-phenylmethoxyphenyl)prop-2-enoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-1-[(4aR,8aS)-6-bromo-2-methyl-4-phenyl-4a,8a-dihydroquinolin-3-yl]-3-(4-bromophenyl)prop-2-en-1-one —— C25H19Br2NO
(E)-1-[(4aR,8aS)-6-bromo-2-methyl-4-phenyl-4a,8a-dihydroquinolin-3-yl]-3-(4-bromophenyl)prop-2-en-1-one
—— (E)-N-benzyl-3-(3-bromo-4-hydroxy-5-nitrophenyl)-2-cyanoprop-2-enamide —— C17H12BrN3O4
(E)-N-benzyl-3-(3-bromo-4-hydroxy-5-nitrophenyl)-2-cyanoprop-2-enamide
—— ethyl (3R)-1-[6-(3-aminopropanoylamino)pyridin-3-yl]piperidine-3-carboxylate —— C16H24N4O3
ethyl (3R)-1-[6-(3-aminopropanoylamino)pyridin-3-yl]piperidine-3-carboxylate
—— ethyl (6S)-2-(4-aminobutanoylamino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C16H24N2O3S
ethyl (6S)-2-(4-aminobutanoylamino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (3R)-1-[6-(4-aminobutanoylamino)pyridin-3-yl]piperidine-3-carboxylate —— C17H26N4O3
ethyl (3R)-1-[6-(4-aminobutanoylamino)pyridin-3-yl]piperidine-3-carboxylate
—— ethyl 5-(1,3-benzodioxol-5-yl)-2-[[3-iodo-5-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H29IN2O7S
ethyl 5-(1,3-benzodioxol-5-yl)-2-[[3-iodo-5-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxy-4-methoxyphenyl)prop-2-enamide —— C23H17ClN2O3S
(E)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxy-4-methoxyphenyl)prop-2-enamide
—— Ethyl 2-[[pentyl-[3-(trifluoromethyl)benzoyl]amino]methyl]-1,3-thiazole-4-carboxylate —— C20H23F3N2O3S
Ethyl 2-[[pentyl-[3-(trifluoromethyl)benzoyl]amino]methyl]-1,3-thiazole-4-carboxylate
—— ethyl 5-(3-bromo-4-methoxyphenyl)-2-[[2-(2-ethoxy-2-oxoethoxy)naphthalen-1-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29BrN2O7S
ethyl 5-(3-bromo-4-methoxyphenyl)-2-[[2-(2-ethoxy-2-oxoethoxy)naphthalen-1-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-[butyl-[2-[cyclohexyl-[[1-[(4-fluorophenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]amino]-4-oxobutanoate —— C30H42FN3O4
Ethyl 4-[butyl-[2-[cyclohexyl-[[1-[(4-fluorophenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]amino]-4-oxobutanoate
—— ethyl 4-[[2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]sulfamoyl]benzoate —— C27H29N3O4S
ethyl 4-[[2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]sulfamoyl]benzoate