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—— ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H22N4O2S2
ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 3-amino-2-[5-[hydroxy(phenyl)methyl]-3H-1,3,4-oxadiazol-2-ylidene]-3-sulfanylidenepropanoate —— C14H15N3O4S
ethyl 3-amino-2-[5-[hydroxy(phenyl)methyl]-3H-1,3,4-oxadiazol-2-ylidene]-3-sulfanylidenepropanoate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(1H-indol-3-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H22FN5O2S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(1H-indol-3-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H30N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H21FN4O2S2
ethyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(3-methylthiophen-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H30N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-benzylsulfanyl-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H30N4O3S
ethyl (7S)-2-benzylsulfanyl-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(3-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H23FN4O3S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(3-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[(E)-2-phenylethenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24N4O2S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[(E)-2-phenylethenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29FN4O3S
ethyl (7R)-7-(3-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H32N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H28N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[(E)-2-phenylethenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23FN4O2S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[(E)-2-phenylethenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-7-(4-methoxycarbonylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24N4O4S
ethyl (7R)-2-benzylsulfanyl-7-(4-methoxycarbonylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H32N4O3S
ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H28N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H28N4O3S
ethyl (7S)-2-benzylsulfanyl-5-methyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H30N4O3S
ethyl (7R)-2-benzylsulfanyl-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H27N5O2S
ethyl (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H30N4O2S
ethyl (7R)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25FN4O2S
ethyl (7R)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H31FN4O3S
ethyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H31FN4O3S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-pentoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 4-[4-[[4-(difluoromethylsulfanyl)anilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C26H20F2N2O4S
ethyl 4-[4-[[4-(difluoromethylsulfanyl)anilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— ethyl 2-[4-[(5-chloro-2-methylanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H25ClN2O4S
ethyl 2-[4-[(5-chloro-2-methylanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-[4-[(4-hydroxyanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C25H20N2O5
ethyl 4-[4-[(4-hydroxyanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H31FN4O3S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-[4-(3-methylbutoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 2-[[2-(3,4-dimethylphenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]-4,5-dimethylthiophene-3-carboxylate —— C27H26N2O4S
ethyl 2-[[2-(3,4-dimethylphenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 3,5-dimethyl-4-[2-[4-[(5-methyl-1,2-oxazol-3-yl)carbamoyl]piperidin-1-yl]acetyl]-1H-pyrrole-2-carboxylate —— C21H28N4O5
ethyl 3,5-dimethyl-4-[2-[4-[(5-methyl-1,2-oxazol-3-yl)carbamoyl]piperidin-1-yl]acetyl]-1H-pyrrole-2-carboxylate
—— ethyl 5-[(2R)-1-cyclohexyloxy-1-oxopropan-2-yl]oxy-1-(4-ethoxyphenyl)-2-methylindole-3-carboxylate —— C29H35NO6
ethyl 5-[(2R)-1-cyclohexyloxy-1-oxopropan-2-yl]oxy-1-(4-ethoxyphenyl)-2-methylindole-3-carboxylate
—— ethyl 6-methyl-2-[[2-oxo-2-[2-[(6-oxo-5-prop-2-enylcyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H27N3O5S
ethyl 6-methyl-2-[[2-oxo-2-[2-[(6-oxo-5-prop-2-enylcyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 5-[(2R)-1-butoxy-1-oxopropan-2-yl]oxy-1-(4-ethoxyphenyl)-2-methylindole-3-carboxylate —— C27H33NO6
ethyl 5-[(2R)-1-butoxy-1-oxopropan-2-yl]oxy-1-(4-ethoxyphenyl)-2-methylindole-3-carboxylate
—— ethyl 2-[[2-(2-chlorophenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H23ClN2O4S
ethyl 2-[[2-(2-chlorophenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H21FN4O3S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25FN4O2S
ethyl (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 1-(4-ethoxyphenyl)-2-methyl-5-[(2S)-1-oxo-1-pentoxypropan-2-yl]oxyindole-3-carboxylate —— C28H35NO6
ethyl 1-(4-ethoxyphenyl)-2-methyl-5-[(2S)-1-oxo-1-pentoxypropan-2-yl]oxyindole-3-carboxylate
—— ethyl 1-(4-ethoxyphenyl)-2-methyl-5-[(2R)-1-[(2R)-2-methylbutoxy]-1-oxopropan-2-yl]oxyindole-3-carboxylate —— C28H35NO6
ethyl 1-(4-ethoxyphenyl)-2-methyl-5-[(2R)-1-[(2R)-2-methylbutoxy]-1-oxopropan-2-yl]oxyindole-3-carboxylate
—— ethyl 2-[[2-[(4-ethyl-5-indol-3-ylidene-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H27N5O3S2
ethyl 2-[[2-[(4-ethyl-5-indol-3-ylidene-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (7S)-7-(4-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29FN4O3S
ethyl (7S)-7-(4-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 4-[2-[3-(4-chlorophenyl)-5-imino-1-methylpyrazol-4-ylidene]hydrazinyl]benzoate —— C19H18ClN5O2
ethyl 4-[2-[3-(4-chlorophenyl)-5-imino-1-methylpyrazol-4-ylidene]hydrazinyl]benzoate
—— ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H21FN4O2S
ethyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl N-[3-[[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate —— C18H26N4O3
ethyl N-[3-[[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate
—— ethyl 2-[[2-[[4-(4-fluorophenyl)-5-indol-3-ylidene-1H-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]acetate —— C22H20FN5O3S
ethyl 2-[[2-[[4-(4-fluorophenyl)-5-indol-3-ylidene-1H-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]acetate
—— ethyl N-[3-[[(1S,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate —— C18H26N4O3
ethyl N-[3-[[(1S,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate
—— ethyl N-[3-[[(1R,2S)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate —— C18H26N4O3
ethyl N-[3-[[(1R,2S)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]amino]-3-oxopropyl]carbamate
—— ethyl 4-[[2-(5-chloro-2-morpholin-4-ylphenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]benzoate —— C29H26ClN3O5
ethyl 4-[[2-(5-chloro-2-morpholin-4-ylphenyl)-1,3-dioxoisoquinolin-4-ylidene]methylamino]benzoate
—— ethyl 4-[4-[(2-methoxyanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C26H22N2O5
ethyl 4-[4-[(2-methoxyanilino)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— ethyl 2-[(4-chlorophenyl)hydrazinylidene]-2-[5-[(4-chlorophenyl)hydrazinylidene]-4-oxo-1,3-thiazol-2-yl]acetate —— C19H15Cl2N5O3S
ethyl 2-[(4-chlorophenyl)hydrazinylidene]-2-[5-[(4-chlorophenyl)hydrazinylidene]-4-oxo-1,3-thiazol-2-yl]acetate
—— ethyl (7R)-7-(3-butoxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29ClN4O3S
ethyl (7R)-7-(3-butoxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H19Cl3N4O2S
ethyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate