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—— (9aR)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C14H20N4O2S
(9aR)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9aS)-2-[[1-(benzenesulfonyl)pyrrol-2-yl]methyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C18H22N4O3S
(9aS)-2-[[1-(benzenesulfonyl)pyrrol-2-yl]methyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9aS)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C14H20N4O2S
(9aS)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9aS)-2-(4-methoxycyclohexanecarbonyl)-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C16H27N3O3
(9aS)-2-(4-methoxycyclohexanecarbonyl)-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9aR)-2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione —— C14H17ClN4O4
(9aR)-2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione
—— (9aS)-2-[(2-methoxypyridin-3-yl)methyl]-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine —— C15H24N4O
(9aS)-2-[(2-methoxypyridin-3-yl)methyl]-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine
—— (9aS)-6,9-dioxo-N-(2-phenoxyphenyl)-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-2-carboxamide —— C20H20N4O4
(9aS)-6,9-dioxo-N-(2-phenoxyphenyl)-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-2-carboxamide
—— (9S)-9-(4-methylphenyl)-8,9,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H18N2O
(9S)-9-(4-methylphenyl)-8,9,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9S)-9-pyridin-3-yl-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C16H14N2O3
(9S)-9-pyridin-3-yl-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— (9R)-6-methyl-9-phenyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H18N2O
(9R)-6-methyl-9-phenyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9aR)-2-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C15H25N5O2
(9aR)-2-[[1-(2-methoxyethyl)imidazol-2-yl]methyl]-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9R)-9-pyridin-3-yl-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C16H14N2O3
(9R)-9-pyridin-3-yl-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— (9aR)-2-(3-chloropyridin-2-yl)-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C13H17ClN4O
(9aR)-2-(3-chloropyridin-2-yl)-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9R)-9-(4-fluorophenyl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H17FN2O
(9R)-9-(4-fluorophenyl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9S)-9-(furan-2-yl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C18H16N2O2
(9S)-9-(furan-2-yl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9aR)-8-methyl-2-(4-phenoxybutanoyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C18H25N3O3
(9aR)-8-methyl-2-(4-phenoxybutanoyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9aS)-2-[3-(3-methoxy-4-methylphenyl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione —— C19H25N3O4
(9aS)-2-[3-(3-methoxy-4-methylphenyl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione
—— (9aS)-8-methyl-2-(1,6-naphthyridin-5-yl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine —— C16H21N5
(9aS)-8-methyl-2-(1,6-naphthyridin-5-yl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine
—— (9aR)-2-[3-(3-methoxy-4-methylphenyl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione —— C19H25N3O4
(9aR)-2-[3-(3-methoxy-4-methylphenyl)propanoyl]-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione
—— (9R)-9-(2,1,3-benzothiadiazol-4-yl)-4-ethyl-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione —— C19H16N4O3S
(9R)-9-(2,1,3-benzothiadiazol-4-yl)-4-ethyl-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione
—— (9S)-9-(2,1,3-benzothiadiazol-4-yl)-4-ethyl-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione —— C19H16N4O3S
(9S)-9-(2,1,3-benzothiadiazol-4-yl)-4-ethyl-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione
—— (9aR)-N-(3-ethylphenyl)-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine-2-carboxamide —— C17H26N4O
(9aR)-N-(3-ethylphenyl)-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine-2-carboxamide
—— (9aS)-2-[(2-ethyl-1,2,4-triazol-3-yl)methyl]-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C13H22N6O
(9aS)-2-[(2-ethyl-1,2,4-triazol-3-yl)methyl]-8-methyl-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9aR)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C18H21N5O3
(9aR)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9S)-6,9-dimethyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C15H16N2O
(9S)-6,9-dimethyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9-Ethylcarbazol-3-yl)methyl-(3-morpholin-4-ium-4-ylpropyl)azanium —— C22H31N3O+2
(9-Ethylcarbazol-3-yl)methyl-(3-morpholin-4-ium-4-ylpropyl)azanium
—— (9R)-4-ethyl-9-(2-ethyl-1,2,4-triazol-3-yl)-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione —— C17H19N5O3
(9R)-4-ethyl-9-(2-ethyl-1,2,4-triazol-3-yl)-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione
—— (9aR)-8-methyl-2-[4-(trifluoromethyl)pyridin-2-yl]-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C14H17F3N4O
(9aR)-8-methyl-2-[4-(trifluoromethyl)pyridin-2-yl]-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9aS)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C18H21N5O3
(9aS)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9aR)-6,9-dioxo-N-(2-phenoxyphenyl)-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-2-carboxamide —— C20H20N4O4
(9aR)-6,9-dioxo-N-(2-phenoxyphenyl)-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-2-carboxamide
—— (9aS)-2-[(3-phenylmethoxyphenyl)methyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C21H25N3O2
(9aS)-2-[(3-phenylmethoxyphenyl)methyl]-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9aR)-2-(6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl)-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C18H21N5O3
(9aR)-2-(6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl)-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9S)-4-ethyl-9-(2-ethyl-1,2,4-triazol-3-yl)-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione —— C17H19N5O3
(9S)-4-ethyl-9-(2-ethyl-1,2,4-triazol-3-yl)-8,9-dihydro-6H-pyrido[2,3-g][1,4]benzoxazine-3,7-dione
—— (9aS)-2-(6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl)-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one —— C18H21N5O3
(9aS)-2-(6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl)-3,4,6,7,8,9a-hexahydro-1H-pyrazino[1,2-a]pyrazin-9-one
—— (9R)-9-pyridin-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C14H13N5O
(9R)-9-pyridin-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9R)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H19N5OS
(9R)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9S)-9-[4-(dimethylamino)phenyl]-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H21N5OS
(9S)-9-[4-(dimethylamino)phenyl]-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9S)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H19N5OS
(9S)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 9H-fluoren-9-yl 4-oxo-4-(4-propylphenyl)butanoate —— C26H24O3
9H-fluoren-9-yl 4-oxo-4-(4-propylphenyl)butanoate
—— (9aR)-2-[3-(2-methylphenoxy)propyl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C18H28N2O
(9aR)-2-[3-(2-methylphenoxy)propyl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— (9aR)-2-(5-chlorothiophen-2-yl)sulfonyl-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione —— C12H14ClN3O4S2
(9aR)-2-(5-chlorothiophen-2-yl)sulfonyl-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione
—— (9R)-9-(4-methoxyphenyl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C21H20N2O2
(9R)-9-(4-methoxyphenyl)-6-methyl-5,8,9,10-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9aS)-2-(5-chlorothiophen-2-yl)sulfonyl-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione —— C12H14ClN3O4S2
(9aS)-2-(5-chlorothiophen-2-yl)sulfonyl-8-methyl-3,4,7,9a-tetrahydro-1H-pyrazino[1,2-a]pyrazine-6,9-dione
—— (9R)-2-ethylsulfanyl-6,6-dimethyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H21N5OS
(9R)-2-ethylsulfanyl-6,6-dimethyl-9-pyridin-3-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9R)-9-(4-fluorophenyl)-8,9,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C19H15FN2O
(9R)-9-(4-fluorophenyl)-8,9,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (9R)-9-[4-(diethylamino)phenyl]-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H25N5OS
(9R)-9-[4-(diethylamino)phenyl]-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9R)-9-(2,3-dimethoxyphenyl)-1-ethyl-8,9-dihydro-6H-pyrido[3,2-g][1,4]benzoxazine-2,7-dione —— C21H22N2O5
(9R)-9-(2,3-dimethoxyphenyl)-1-ethyl-8,9-dihydro-6H-pyrido[3,2-g][1,4]benzoxazine-2,7-dione
—— (9S)-9-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C19H23N5OS
(9S)-9-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9S)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-2-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H19N5OS
(9S)-6,6-dimethyl-2-methylsulfanyl-9-pyridin-2-yl-4,5,7,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (9aS)-2-[(3-methyl-4-pyrrolidin-1-ylphenyl)methyl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione —— C19H26N4O2
(9aS)-2-[(3-methyl-4-pyrrolidin-1-ylphenyl)methyl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione