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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-Methyl-10,20-dioxapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1,3(11),4(9),5,7,12,14,16,18-nonaene —— C19H12O2
6-Methyl-10,20-dioxapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1,3(11),4(9),5,7,12,14,16,18-nonaene
—— 6-(3-oxo-1H-pyrazol-2-yl)pyrimidine-4-carbonitrile —— C8H5N5O
6-(3-oxo-1H-pyrazol-2-yl)pyrimidine-4-carbonitrile
—— 6-[2-Chloro-5-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-8-methyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C29H28ClN7O2
6-[2-Chloro-5-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-8-methyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[5-Methyl-2-(1-methylpyrrol-2-yl)-1,3-thiazol-4-yl]-2-[4-(1-methylpiperidin-3-yl)oxyanilino]-8-(1,3-thiazol-2-ylmethyl)pyrido[2,3-d]pyrimidin-7-one —— C32H32N8O2S2
6-[5-Methyl-2-(1-methylpyrrol-2-yl)-1,3-thiazol-4-yl]-2-[4-(1-methylpiperidin-3-yl)oxyanilino]-8-(1,3-thiazol-2-ylmethyl)pyrido[2,3-d]pyrimidin-7-one
—— (6S,8R,9R)-3-propyl-2,7-dioxatricyclo[6.3.1.01,6]dodec-10-en-9-ol —— C13H20O3
(6S,8R,9R)-3-propyl-2,7-dioxatricyclo[6.3.1.01,6]dodec-10-en-9-ol
—— 6-Hydrazinylpyridazine-4-carboxylic acid —— C5H6N4O2
6-Hydrazinylpyridazine-4-carboxylic acid
—— 6-(3-oxo-1H-pyrazol-2-yl)pyridazine-4-carbonitrile —— C8H5N5O
6-(3-oxo-1H-pyrazol-2-yl)pyridazine-4-carbonitrile
—— 6-Hydrazinylpyrimidine-4-carboxylic acid —— C5H6N4O2
6-Hydrazinylpyrimidine-4-carboxylic acid
—— 6-(5-methyl-3-oxo-1H-pyrazol-2-yl)pyridazine-4-carbonitrile —— C9H7N5O
6-(5-methyl-3-oxo-1H-pyrazol-2-yl)pyridazine-4-carbonitrile
—— 6-(6-Cyclopentyl-4-methylpyridin-3-yl)-2-[4-(1-methylpiperidin-4-yl)anilino]-8-(1,3-thiazol-2-ylmethyl)pyrido[2,3-d]pyrimidin-7-one —— C34H37N7OS
6-(6-Cyclopentyl-4-methylpyridin-3-yl)-2-[4-(1-methylpiperidin-4-yl)anilino]-8-(1,3-thiazol-2-ylmethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Methyl-4-(1,3-thiazol-2-yl)phenyl]-2-[4-(4-methylthiomorpholin-2-yl)anilino]-8-(2-morpholin-4-ylethyl)pyrido[2,3-d]pyrimidin-7-one —— C34H37N7O2S2
6-[2-Methyl-4-(1,3-thiazol-2-yl)phenyl]-2-[4-(4-methylthiomorpholin-2-yl)anilino]-8-(2-morpholin-4-ylethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Chloro-4-[6-(trifluoromethyl)pyrimidin-4-yl]phenyl]-8-ethyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one 1428759-81-2 C32H29ClF3N7O
6-[2-Chloro-4-[6-(trifluoromethyl)pyrimidin-4-yl]phenyl]-8-ethyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-Methyl-6-(1,3-thiazol-4-yl)pyridin-3-yl]-2-(4-piperidin-4-ylanilino)-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C30H26N8OS2
6-[4-Methyl-6-(1,3-thiazol-4-yl)pyridin-3-yl]-2-(4-piperidin-4-ylanilino)-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 6-(2-Cyclohexyl-4-methylpyrimidin-5-yl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one —— C34H41N9O2
6-(2-Cyclohexyl-4-methylpyrimidin-5-yl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-(4-Cyclopenta-1,4-dien-1-yl-1-methylimidazol-2-yl)-2-(3-methyl-4-piperazin-1-ylanilino)-8-(1-methylsulfinylpiperidin-4-yl)pyrido[2,3-d]pyrimidin-7-one —— C33H39N9O2S
6-(4-Cyclopenta-1,4-dien-1-yl-1-methylimidazol-2-yl)-2-(3-methyl-4-piperazin-1-ylanilino)-8-(1-methylsulfinylpiperidin-4-yl)pyrido[2,3-d]pyrimidin-7-one
—— 6-(4-Bromo-2-chlorophenyl)-8-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one —— C15H12BrClN4O
6-(4-Bromo-2-chlorophenyl)-8-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one
—— 6-(2,5-Dimethyl-1,3-thiazol-4-yl)-8-ethyl-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C25H29N7OS
6-(2,5-Dimethyl-1,3-thiazol-4-yl)-8-ethyl-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-(4-Bromo-2-chlorophenyl)-8-methyl-2-methylsulfanylpyrido[2,3-d]pyrimidin-7-one —— C15H11BrClN3OS
6-(4-Bromo-2-chlorophenyl)-8-methyl-2-methylsulfanylpyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Chloro-4-(6-ethylpyrimidin-4-yl)phenyl]-8-ethyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one 1428759-97-0 C33H34ClN7O
6-[2-Chloro-4-(6-ethylpyrimidin-4-yl)phenyl]-8-ethyl-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-(1-Methylpyrrolidin-3-yl)-2-(trifluoromethyl)phenyl]-8-(oxan-4-ylmethyl)-2-(4-piperidin-4-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C36H41F3N6O3
6-[4-(1-Methylpyrrolidin-3-yl)-2-(trifluoromethyl)phenyl]-8-(oxan-4-ylmethyl)-2-(4-piperidin-4-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-(2,4-Dimethyl-1,3-thiazol-5-yl)-8-ethyl-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C25H29N7OS
6-(2,4-Dimethyl-1,3-thiazol-5-yl)-8-ethyl-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[5-Methyl-2-(1-methylimidazol-2-yl)pyrimidin-4-yl]-8-(2-morpholin-4-ylethyl)-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C33H38N10O3
6-[5-Methyl-2-(1-methylimidazol-2-yl)pyrimidin-4-yl]-8-(2-morpholin-4-ylethyl)-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-[3-Chloro-5-(2-methylpyrazol-3-yl)pyridin-2-yl]-8-(cyclopropylmethyl)-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]pyrido[2,3-d]pyrimidin-7-one —— C31H31ClN8O2
6-[3-Chloro-5-(2-methylpyrazol-3-yl)pyridin-2-yl]-8-(cyclopropylmethyl)-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-(5-Cyclohexyl-3-methylpyridin-2-yl)-2-[3-fluoro-4-(3-methylpiperazin-1-yl)anilino]-8-[2-[methyl(methylsulfanyl)amino]ethyl]pyrido[2,3-d]pyrimidin-7-one —— C34H43FN8OS
6-(5-Cyclohexyl-3-methylpyridin-2-yl)-2-[3-fluoro-4-(3-methylpiperazin-1-yl)anilino]-8-[2-[methyl(methylsulfanyl)amino]ethyl]pyrido[2,3-d]pyrimidin-7-one
—— 6-(5-Methyl-2-piperidin-4-yl-1,3-thiazol-4-yl)-8-(oxolan-3-yl)-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one —— C30H36N8O2S
6-(5-Methyl-2-piperidin-4-yl-1,3-thiazol-4-yl)-8-(oxolan-3-yl)-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2,6-Dichloro-4-(1-methylpyrrolidin-2-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-(2-oxo-2-pyrrolidin-1-ylethyl)pyrido[2,3-d]pyrimidin-7-one —— C35H39Cl2N7O3
6-[2,6-Dichloro-4-(1-methylpyrrolidin-2-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-(2-oxo-2-pyrrolidin-1-ylethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Chloro-4-(1-methylpyrazol-4-yl)phenyl]-2-(4-piperidin-4-yloxyanilino)-8-propan-2-ylpyrido[2,3-d]pyrimidin-7-one —— C31H32ClN7O2
6-[2-Chloro-4-(1-methylpyrazol-4-yl)phenyl]-2-(4-piperidin-4-yloxyanilino)-8-propan-2-ylpyrido[2,3-d]pyrimidin-7-one
—— 6-[4-Chloro-2-(1-methylpyrrol-2-yl)phenyl]-8-ethyl-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C31H31ClN6O2
6-[4-Chloro-2-(1-methylpyrrol-2-yl)phenyl]-8-ethyl-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-(4-Bromo-2-chlorophenyl)-8-methyl-2-methylsulfinylpyrido[2,3-d]pyrimidin-7-one —— C15H11BrClN3O2S
6-(4-Bromo-2-chlorophenyl)-8-methyl-2-methylsulfinylpyrido[2,3-d]pyrimidin-7-one
—— 6-[3-Chloro-5-(oxan-4-yl)pyridin-2-yl]-8-ethyl-2-[4-(1-methylpiperidin-3-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C31H35ClN6O2
6-[3-Chloro-5-(oxan-4-yl)pyridin-2-yl]-8-ethyl-2-[4-(1-methylpiperidin-3-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[3-Chloro-5-(1-methylpiperidin-4-yl)pyridin-2-yl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]-8-(2,2,2-trifluoroethyl)pyrido[2,3-d]pyrimidin-7-one —— C31H33ClF3N7O
6-[3-Chloro-5-(1-methylpiperidin-4-yl)pyridin-2-yl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]-8-(2,2,2-trifluoroethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Chloro-4-(4-fluoropyridin-3-yl)phenyl]-8-ethyl-2-[3-fluoro-4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C32H29ClF2N6O
6-[2-Chloro-4-(4-fluoropyridin-3-yl)phenyl]-8-ethyl-2-[3-fluoro-4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-(5-Cyclopenta-1,4-dien-1-ylpyridin-2-yl)-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H30N8OS
6-(5-Cyclopenta-1,4-dien-1-ylpyridin-2-yl)-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[5-Methyl-1-(3-methylimidazol-4-yl)imidazol-4-yl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C30H36N10OS
6-[5-Methyl-1-(3-methylimidazol-4-yl)imidazol-4-yl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-(3-Methyl-5-thiophen-3-ylpyridin-2-yl)-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]-8-(2,2,2-trifluoroethyl)pyrido[2,3-d]pyrimidin-7-one —— C30H25F3N6OS
6-(3-Methyl-5-thiophen-3-ylpyridin-2-yl)-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]-8-(2,2,2-trifluoroethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-(1-Methylpyrrolidin-3-yl)phenyl]-2-[4-(4-methylthiomorpholin-2-yl)anilino]-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H33N7OS2
6-[4-(1-Methylpyrrolidin-3-yl)phenyl]-2-[4-(4-methylthiomorpholin-2-yl)anilino]-8-(1,3-thiazol-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[3,5-Dimethyl-1-(1-methyltetrazol-5-yl)pyrazol-4-yl]-2-[4-(4-methylmorpholin-2-yl)anilino]-8-(1-methylsulfanylpiperidin-4-yl)pyrido[2,3-d]pyrimidin-7-one —— C31H38N12O2S
6-[3,5-Dimethyl-1-(1-methyltetrazol-5-yl)pyrazol-4-yl]-2-[4-(4-methylmorpholin-2-yl)anilino]-8-(1-methylsulfanylpiperidin-4-yl)pyrido[2,3-d]pyrimidin-7-one
—— 6-(2-Chloro-4-pyrazin-2-ylphenyl)-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-(2-oxo-2-pyrrolidin-1-ylethyl)pyrido[2,3-d]pyrimidin-7-one —— C35H36ClN9O2
6-(2-Chloro-4-pyrazin-2-ylphenyl)-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-(2-oxo-2-pyrrolidin-1-ylethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[1-(1-Methylpyrazol-4-yl)imidazol-2-yl]-8-(1-methylsulfinylpiperidin-4-yl)-2-[4-(4-methylthiomorpholin-2-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C31H36N10O2S2
6-[1-(1-Methylpyrazol-4-yl)imidazol-2-yl]-8-(1-methylsulfinylpiperidin-4-yl)-2-[4-(4-methylthiomorpholin-2-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-[3-Methyl-5-(1-methylpiperidin-3-yl)pyridin-2-yl]-2-[4-piperazin-1-yl-3-(trifluoromethyl)anilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one —— C38H38F6N8O
6-[3-Methyl-5-(1-methylpiperidin-3-yl)pyridin-2-yl]-2-[4-piperazin-1-yl-3-(trifluoromethyl)anilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-Methyl-2-(1,3-oxazol-4-yl)pyrimidin-5-yl]-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one —— C35H32F3N9O2
6-[4-Methyl-2-(1,3-oxazol-4-yl)pyrimidin-5-yl]-2-[4-[methyl(piperidin-4-yl)amino]anilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-(1-Acetylpyrrolidin-3-yl)phenyl]-8-[2-(dimethylamino)ethyl]-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C34H42N8O2
6-[4-(1-Acetylpyrrolidin-3-yl)phenyl]-8-[2-(dimethylamino)ethyl]-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 6-(2-Cyclopentyl-4-methylpyrimidin-5-yl)-2-[4-(4-methylmorpholin-2-yl)anilino]-8-phenylpyrido[2,3-d]pyrimidin-7-one —— C34H35N7O2
6-(2-Cyclopentyl-4-methylpyrimidin-5-yl)-2-[4-(4-methylmorpholin-2-yl)anilino]-8-phenylpyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Methyl-4-(1-methylpyrrolidin-2-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]-8-phenylpyrido[2,3-d]pyrimidin-7-one —— C36H38N6O
6-[2-Methyl-4-(1-methylpyrrolidin-2-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)anilino]-8-phenylpyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Methyl-4-(1-methylimidazol-2-yl)phenyl]-2-(4-piperazin-1-ylanilino)-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one —— C36H33F3N8O
6-[2-Methyl-4-(1-methylimidazol-2-yl)phenyl]-2-(4-piperazin-1-ylanilino)-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one
—— 6-[1-(3-Iminopropanimidoyl)imidazol-2-yl]-2-[4-(4-methylmorpholin-2-yl)anilino]-8-(2-morpholin-4-ylethyl)pyrido[2,3-d]pyrimidin-7-one —— C30H36N10O3
6-[1-(3-Iminopropanimidoyl)imidazol-2-yl]-2-[4-(4-methylmorpholin-2-yl)anilino]-8-(2-morpholin-4-ylethyl)pyrido[2,3-d]pyrimidin-7-one
—— 6-[4-Methyl-2-(2-methyl-1,5-dihydropyrazol-3-yl)pyrimidin-5-yl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-(4-piperidin-4-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C31H38N10O2S
6-[4-Methyl-2-(2-methyl-1,5-dihydropyrazol-3-yl)pyrimidin-5-yl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-(4-piperidin-4-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Fluoro-4-(2-methyltetrazol-5-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one —— C34H29F4N9O2
6-[2-Fluoro-4-(2-methyltetrazol-5-yl)phenyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-[[2-(trifluoromethyl)phenyl]methyl]pyrido[2,3-d]pyrimidin-7-one
—— 6-(2-Methyl-4-pyridin-2-ylphenyl)-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-propan-2-ylpyrido[2,3-d]pyrimidin-7-one —— C33H34N6O2
6-(2-Methyl-4-pyridin-2-ylphenyl)-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-8-propan-2-ylpyrido[2,3-d]pyrimidin-7-one
—— 6-[2-Chloro-4-(1,3,4-oxadiazol-2-yl)phenyl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C30H29ClN8O2S
6-[2-Chloro-4-(1,3,4-oxadiazol-2-yl)phenyl]-8-[2-[methyl(methylsulfanyl)amino]ethyl]-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one