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—— 6-[(2E)-2-[(2E,4E,6E)-7-[5-[5-carboxypentoxy(methyl)carbamoyl]-3,3-dimethyl-7-(3-sulfopropyl)pyrrolo[2,3-b]pyridin-7-ium-2-yl]hepta-2,4,6-trienylidene]-3,3-dimethyl-5-sulfoindol-1-yl]hexanoic acid —— C43H57N4O12S2+
6-[(2E)-2-[(2E,4E,6E)-7-[5-[5-carboxypentoxy(methyl)carbamoyl]-3,3-dimethyl-7-(3-sulfopropyl)pyrrolo[2,3-b]pyridin-7-ium-2-yl]hepta-2,4,6-trienylidene]-3,3-dimethyl-5-sulfoindol-1-yl]hexanoic acid
—— 6-[(4,6-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-(furan-2-yl)-1H-pyrazol-3-yl]-2-(4-methylpiperazin-1-yl)pyrimidin-4-amine —— C25H24F2N8O2
6-[(4,6-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-(furan-2-yl)-1H-pyrazol-3-yl]-2-(4-methylpiperazin-1-yl)pyrimidin-4-amine
—— 6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C25H31FN8O
6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-[2-[3-[(4R,5R,6R)-2-amino-5-fluoro-6-(methoxymethyl)-4-methyl-5,6-dihydro-1,3-oxazin-4-yl]-4-fluorophenyl]acetyl]pyridine-3-carbonitrile —— C21H20F2N4O3
6-[2-[3-[(4R,5R,6R)-2-amino-5-fluoro-6-(methoxymethyl)-4-methyl-5,6-dihydro-1,3-oxazin-4-yl]-4-fluorophenyl]acetyl]pyridine-3-carbonitrile
—— [6-Methoxy-4-methyl-9,10-bis(oxiran-2-ylmethoxy)-5,8-dihydroanthracen-2-yl]methanol —— C23H26O6
[6-Methoxy-4-methyl-9,10-bis(oxiran-2-ylmethoxy)-5,8-dihydroanthracen-2-yl]methanol
—— 6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-propyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C24H29FN8O
6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-propyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— (6S)-4-ethenyl-6-(fluoromethyl)-5,6-dihydro-4H-1,3-oxazin-2-amine —— C7H11FN2O
(6S)-4-ethenyl-6-(fluoromethyl)-5,6-dihydro-4H-1,3-oxazin-2-amine
—— 6-N-[2-(dimethylamino)ethyl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-4-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidine-4,6-diamine —— C23H27FN8O
6-N-[2-(dimethylamino)ethyl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-4-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidine-4,6-diamine
—— 6-(4-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(1H-pyrazol-5-yl)pyrimidin-4-amine —— C22H25FN8O
6-(4-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(1H-pyrazol-5-yl)pyrimidin-4-amine
—— 6-(azetidin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C20H20FN7O
6-(azetidin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-[[2-(2-Aminoethoxymethoxy)acetyl]amino]hexanoic acid —— C11H22N2O5
6-[[2-(2-Aminoethoxymethoxy)acetyl]amino]hexanoic acid
—— 6-[(3R)-3,5-dimethylpiperazin-1-yl]-2-[(4-fluoro-1H-indol-5-yl)oxy]-N-(1H-pyrazol-5-yl)pyrimidin-4-amine —— C21H23FN8O
6-[(3R)-3,5-dimethylpiperazin-1-yl]-2-[(4-fluoro-1H-indol-5-yl)oxy]-N-(1H-pyrazol-5-yl)pyrimidin-4-amine
—— 6-cyclopropyl-2-[(4,7-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C22H20F2N6O
6-cyclopropyl-2-[(4,7-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C24H27ClN8O
6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-cyclopropyl-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C22H21FN6O
6-cyclopropyl-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-(3-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C25H29FN8O
6-(3-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[(4,6-difluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-thiophen-2-yl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C25H24F2N8OS
6-[(4,6-difluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-thiophen-2-yl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-(nitrosomethyl)-1H-pyrazol-3-yl]pyrimidin-4-amine —— C22H24FN9O2
6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-(nitrosomethyl)-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[(4,7-difluoro-2-methyl-1H-pyrrolo[2,3-c]pyridin-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C23H25F2N9O
6-[(4,7-difluoro-2-methyl-1H-pyrrolo[2,3-c]pyridin-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-(1,1-dioxo-1,4-thiazinan-4-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609118-74-2 C23H24FN7O3S
6-(1,1-dioxo-1,4-thiazinan-4-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[2-[(dimethylamino)methyl]morpholin-4-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C24H29FN8O2
6-[2-[(dimethylamino)methyl]morpholin-4-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— [(6E,10E,12Z)-16-hydroxy-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-18-yl] dihydrogen phosphate —— C26H35N2O9P
[(6E,10E,12Z)-16-hydroxy-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-18-yl] dihydrogen phosphate
—— 6-[2-[(dimethylamino)methyl]morpholin-4-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine —— C26H31FN8O2
6-[2-[(dimethylamino)methyl]morpholin-4-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4,7-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609119-07-4 C27H32F2N8O
6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4,7-difluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[(3S,5R)-3,5-dimethylpiperazin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C23H27FN8O
6-[(3S,5R)-3,5-dimethylpiperazin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C22H25FN8O
6-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C22H25ClN8O
6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-chloro-5-ethoxy-2-methyl-1H-indole —— C11H12ClNO
6-chloro-5-ethoxy-2-methyl-1H-indole
—— 6-(4-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609118-83-3 C25H29FN8O
6-(4-ethylpiperazin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[3-(dimethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609118-80-0 C25H29FN8O
6-[3-(dimethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-cyclopropyl-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C20H19FN6O
6-cyclopropyl-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-Fluoro-5-methoxy-1-methylindole —— C10H10FNO
6-Fluoro-5-methoxy-1-methylindole
—— 6-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C25H32FN9O
6-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-(5-methyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-(azetidin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609118-87-7 C22H22FN7O
6-(azetidin-1-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[2-[2-(3,3-Dimethyl-2-oxobutoxy)ethoxy]ethylamino]-6-methyl-2-(methylamino)-5-oxoheptane-1-sulfonic acid —— C19H38N2O7S
6-[2-[2-(3,3-Dimethyl-2-oxobutoxy)ethoxy]ethylamino]-6-methyl-2-(methylamino)-5-oxoheptane-1-sulfonic acid
—— 6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine 1609118-79-7 C27H33FN8O
6-[3-(diethylamino)pyrrolidin-1-yl]-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-N-[5-[(E)-prop-1-enyl]-1H-pyrazol-3-yl]pyrimidin-4-amine
—— 6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-propyl-1H-pyrazol-3-yl)pyrimidin-4-amine —— C24H29ClN8O
6-[(4-chloro-2-methyl-1H-indol-5-yl)oxy]-2-(4-methylpiperazin-1-yl)-N-(5-propyl-1H-pyrazol-3-yl)pyrimidin-4-amine
—— 6-cyclobutyl-N-(5-ethenyl-1H-pyrazol-3-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]pyrimidin-4-amine —— C22H21FN6O
6-cyclobutyl-N-(5-ethenyl-1H-pyrazol-3-yl)-2-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]pyrimidin-4-amine
—— 6-Methoxy-2-methyl-4a,8a-dihydro-3,1-benzoxazin-4-one —— C10H11NO3
6-Methoxy-2-methyl-4a,8a-dihydro-3,1-benzoxazin-4-one
—— 6-Fluoro-5-methoxy-1,2-dimethylindole —— C11H12FNO
6-Fluoro-5-methoxy-1,2-dimethylindole
—— [(6E,10E,12Z)-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-16-phosphonooxy-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-18-yl] dihydrogen phosphate —— C26H36N2O12P2
[(6E,10E,12Z)-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-16-phosphonooxy-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-18-yl] dihydrogen phosphate
—— [(6E,10E,12Z)-18-hydroxy-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-16-yl] dihydrogen phosphate —— C26H35N2O9P
[(6E,10E,12Z)-18-hydroxy-4,10-dimethyl-2-oxo-12-(2-oxo-2-piperidin-1-ylethoxy)imino-3-oxabicyclo[12.4.0]octadeca-1(14),6,10,15,17-pentaen-16-yl] dihydrogen phosphate
—— (6S)-6-(3-bromo-4-methoxyphenyl)-6,8,9,10-tetrahydro-5H-benzo[c]phenanthridin-7-one —— C24H20BrNO2
(6S)-6-(3-bromo-4-methoxyphenyl)-6,8,9,10-tetrahydro-5H-benzo[c]phenanthridin-7-one
—— (6S)-3-[(S)-(4-bromophenyl)-cyclopropylmethyl]-6-(2-methylprop-2-enyl)-6-phenyl-1,3-oxazinan-2-one —— C24H26BrNO2
(6S)-3-[(S)-(4-bromophenyl)-cyclopropylmethyl]-6-(2-methylprop-2-enyl)-6-phenyl-1,3-oxazinan-2-one
—— (6R)-6-(3-bromo-4-methoxyphenyl)-6,8,9,10-tetrahydro-5H-benzo[c]phenanthridin-7-one —— C24H20BrNO2
(6R)-6-(3-bromo-4-methoxyphenyl)-6,8,9,10-tetrahydro-5H-benzo[c]phenanthridin-7-one
—— (6R)-3-[(S)-(4-bromophenyl)-cyclopropylmethyl]-6-(2-methylprop-2-enyl)-6-phenyl-1,3-oxazinan-2-one —— C24H26BrNO2
(6R)-3-[(S)-(4-bromophenyl)-cyclopropylmethyl]-6-(2-methylprop-2-enyl)-6-phenyl-1,3-oxazinan-2-one
—— 6-(4-bromo-2-fluoroanilino)-7-fluoro-3-methyl-N-(2-phosphanyloxyethoxy)benzimidazole-5-carboxamide —— C17H16BrF2N4O3P
6-(4-bromo-2-fluoroanilino)-7-fluoro-3-methyl-N-(2-phosphanyloxyethoxy)benzimidazole-5-carboxamide
—— 6-bromo-N-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C14H8BrF3N4O
6-bromo-N-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 6-tert-butyl-3-[2-(2-tert-butylphenoxy)pyridin-3-yl]-2H-1,3-benzothiazol-2-amine —— C26H31N3OS
6-tert-butyl-3-[2-(2-tert-butylphenoxy)pyridin-3-yl]-2H-1,3-benzothiazol-2-amine
—— 6-bromo-3-[2-(2-tert-butylphenoxy)pyridin-3-yl]-2H-1,3-benzothiazol-2-amine —— C22H22BrN3OS
6-bromo-3-[2-(2-tert-butylphenoxy)pyridin-3-yl]-2H-1,3-benzothiazol-2-amine