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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(1-Cyclobutyl-4-hydroxybutyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C22H23F3N6O
6-[(1-Cyclobutyl-4-hydroxybutyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-[2-(3,3-Difluorocyclobutyl)ethylamino]-8-(2-methoxy-5-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C28H25F5N6O
6-[2-(3,3-Difluorocyclobutyl)ethylamino]-8-(2-methoxy-5-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-(1-Cyclobutylethylamino)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-8-[5-propan-2-yl-2-(trifluoromethoxy)phenyl]purine-2-carboxylic acid —— C30H28F7N5O3
6-(1-Cyclobutylethylamino)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-8-[5-propan-2-yl-2-(trifluoromethoxy)phenyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-[2-(3-fluorophenyl)ethyl-prop-2-enylamino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C31H32F4N6O2
6-(2-Cyclobutylethylamino)-8-[2-(3-fluorophenyl)ethyl-prop-2-enylamino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-[Methyl(pentan-2-yl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C27H28F3N5O2
6-[Methyl(pentan-2-yl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethoxy)-7-[(4-methylcyclohexyl)methyl]-8-(4-propan-2-ylpyridin-2-yl)purine-2-carboxylic acid —— C28H37N5O3
6-(2-Cyclobutylethoxy)-7-[(4-methylcyclohexyl)methyl]-8-(4-propan-2-ylpyridin-2-yl)purine-2-carboxylic acid
—— 6-{[(1r)-1-Cyclobutylpropyl]amino}-8-[4-[1-methylethyl)pyridin-2-yl]-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C29H31F3N6O2
6-{[(1r)-1-Cyclobutylpropyl]amino}-8-[4-[1-methylethyl)pyridin-2-yl]-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-[(4-Cyclobutyl-4-hydroxybutyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C22H23F3N6O
6-[(4-Cyclobutyl-4-hydroxybutyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-{[(1r)-1-Cyclopropylethyl] amino}-8-(4-methylpiperazin-1-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C24H28F3N7O2
6-{[(1r)-1-Cyclopropylethyl] amino}-8-(4-methylpiperazin-1-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-{[(1R)-1-cyclobutylethyl]amino}-8-(2,5-dichlorophenyl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid 1621541-75-0 C26H22Cl2F3N5O2
6-{[(1R)-1-cyclobutylethyl]amino}-8-(2,5-dichlorophenyl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-(3,3-dimethylpiperidine-1-carbonyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C28H33F3N6O3
6-(2-Cyclobutylethylamino)-8-(3,3-dimethylpiperidine-1-carbonyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-[2-(2-fluorophenyl)-2-hydroxyethyl]-7-[(4-methylcyclohexyl)methyl]purine-2-carbonitrile —— C28H35FN6O
6-(2-Cyclobutylethylamino)-8-[2-(2-fluorophenyl)-2-hydroxyethyl]-7-[(4-methylcyclohexyl)methyl]purine-2-carbonitrile
—— 6-hydroxy-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile —— C21H14F3N5O
6-hydroxy-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile
—— 6-(1-Cyclobutylethylamino)-8-(2-propan-2-ylpyridin-4-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C28H29F3N6O2
6-(1-Cyclobutylethylamino)-8-(2-propan-2-ylpyridin-4-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(1-Cyclobutylethoxy)-7-[3-fluoro-4-(trifluoromethyl)benzyl]-8-[4-(1-methylethyl)pyridin-2-yl]-7h-purine-2-carboxylic acid (racemate) —— C28H27F4N5O3
6-(1-Cyclobutylethoxy)-7-[3-fluoro-4-(trifluoromethyl)benzyl]-8-[4-(1-methylethyl)pyridin-2-yl]-7h-purine-2-carboxylic acid (racemate)
—— 6-{[(1r)-1-Cyclobutylethyl]amino}-8-(2-phenylazetidin-1-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C29H29F3N6O2
6-{[(1r)-1-Cyclobutylethyl]amino}-8-(2-phenylazetidin-1-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-{[(1R)-1-cyclopropylethyl]amino}-8-(2-methoxypyridin-4-yl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid 1621541-83-0 C25H23F3N6O3
6-{[(1R)-1-cyclopropylethyl]amino}-8-(2-methoxypyridin-4-yl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carboxylic acid
—— 6-{[1s)-1-(3-Chlorophenyl)ethyl] amino}-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C29H23ClF3N5O2
6-{[1s)-1-(3-Chlorophenyl)ethyl] amino}-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-{[(1r)-1-Cyclobutylethyl]amino}-8-(3,4-dihydroisoquinolin-2(1h)-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C29H29F3N6O2
6-{[(1r)-1-Cyclobutylethyl]amino}-8-(3,4-dihydroisoquinolin-2(1h)-yl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-[2,2-Dimethylpropyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C27H28F3N5O2
6-[2,2-Dimethylpropyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-{[(1r)-1-Cyclobutyl-4-(4-methylpiperazin-l-yl)butyl]amino}-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C34H40F3N7O2
6-{[(1r)-1-Cyclobutyl-4-(4-methylpiperazin-l-yl)butyl]amino}-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-(2-cyclobutylethylamino)-8-[(1R)-1-(2-fluorophenyl)-2-hydroxyethyl]-7-[(4-methylcyclohexyl)methyl]purine-2-carbonitrile —— C28H35FN6O
6-(2-cyclobutylethylamino)-8-[(1R)-1-(2-fluorophenyl)-2-hydroxyethyl]-7-[(4-methylcyclohexyl)methyl]purine-2-carbonitrile
—— 6-{[(1r)-1-Cyclobutylethyl]amino}-8-methyl-7-[(trans-4-methylcyclohexyl)methyl]-7h-purine-2-carboxylic acid —— C21H31N5O2
6-{[(1r)-1-Cyclobutylethyl]amino}-8-methyl-7-[(trans-4-methylcyclohexyl)methyl]-7h-purine-2-carboxylic acid
—— 6-[[(1R)-1-cyclobutylethyl]-prop-2-enylamino]-8-[1-(3-fluorophenyl)ethylamino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C31H31F4N7
6-[[(1R)-1-cyclobutylethyl]-prop-2-enylamino]-8-[1-(3-fluorophenyl)ethylamino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-(2-Cyclobutylpiperidin-1-yl)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C30H30F3N5O2
6-(2-Cyclobutylpiperidin-1-yl)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-[[(1R)-1-cyclobutylethyl]amino]-7-[(4-methylcyclohexyl)methyl]-8-(1-phenylpropan-2-yl)purine-2-carboxylic acid —— C29H39N5O2
6-[[(1R)-1-cyclobutylethyl]amino]-7-[(4-methylcyclohexyl)methyl]-8-(1-phenylpropan-2-yl)purine-2-carboxylic acid
—— 6-(2-Cyclobutylethoxy)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-8-(4-propan-2-ylpyridin-2-yl)purine-2-carboxylic acid —— C28H27F4N5O3
6-(2-Cyclobutylethoxy)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-8-(4-propan-2-ylpyridin-2-yl)purine-2-carboxylic acid
—— 6-(((R)-1-cyclobutylethyl)amino)-7-((trans-4-(trifluoromethyl)cyclohexyl)methyl)-7H-purine-2-carbonitrile —— C20H25F3N6
6-(((R)-1-cyclobutylethyl)amino)-7-((trans-4-(trifluoromethyl)cyclohexyl)methyl)-7H-purine-2-carbonitrile
—— 6-{[(1r)-1-Cyclobutylethyl]amino}-8-(1-phenoxyethyl)-7-[4-[4 (trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C28H28F3N5O3
6-{[(1r)-1-Cyclobutylethyl]amino}-8-(1-phenoxyethyl)-7-[4-[4 (trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-(1-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C28H28F4N6O2
6-(1-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-[5-(dimethylamino)-2-(trifluoromethoxy)phenyl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C29H28F6N6O3
6-(2-Cyclobutylethylamino)-8-[5-(dimethylamino)-2-(trifluoromethoxy)phenyl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Tert-butylpyrrolidin-1-yl)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C29H30F3N5O2
6-(2-Tert-butylpyrrolidin-1-yl)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-(phenoxymethyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C27H25F3N6O
6-(2-Cyclobutylethylamino)-8-(phenoxymethyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-(2-cyclobutylethylamino)-8-[(2R)-piperidin-2-yl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C25H29F3N6O2
6-(2-cyclobutylethylamino)-8-[(2R)-piperidin-2-yl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-[Benzyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C29H24F3N5O2
6-[Benzyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C28H28F4N6O2
6-(2-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[(4-methylcyclohexyl)methyl]purine-2-carboxylic acid —— C28H37FN6O2
6-(2-Cyclobutylethylamino)-8-(5-fluoro-4-propan-2-ylpyridin-2-yl)-7-[(4-methylcyclohexyl)methyl]purine-2-carboxylic acid
—— 6-{[(1r)-1-Cyclopropylethyl]amino}-8-(3-methylphenyl)-7-{[4-(trifluoromethyl)cyclohexyl]methyl}-7h-purine-2-carboxylic acid —— C26H30F3N5O2
6-{[(1r)-1-Cyclopropylethyl]amino}-8-(3-methylphenyl)-7-{[4-(trifluoromethyl)cyclohexyl]methyl}-7h-purine-2-carboxylic acid
—— 6-{[(1r)-1-Cyclobutylethyl]amino}-8-(1-hydroxyethyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid —— C22H24F3N5O3
6-{[(1r)-1-Cyclobutylethyl]amino}-8-(1-hydroxyethyl)-7-[4-(trifluoromethyl)benzyl]-7h-purine-2-carboxylic acid
—— 6-[2-Cyclopropylethyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C27H26F3N5O2
6-[2-Cyclopropylethyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(cyclopropylmethoxy)-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carbonitrile —— C25H20F3N5O
6-(cyclopropylmethoxy)-8-(3-methylphenyl)-7-[4-(trifluoromethyl)benzyl]-7H-purine-2-carbonitrile
—— 6-(1-Cyclopropylethylamino)-7-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-8-(3-methylphenyl)purine-2-carbonitrile —— C26H22F4N6
6-(1-Cyclopropylethylamino)-7-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-8-(3-methylphenyl)purine-2-carbonitrile
—— 6-[[(1R)-1-cyclobutylethyl]amino]-8-(1-pyridin-2-ylethylamino)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C27H27F3N8
6-[[(1R)-1-cyclobutylethyl]amino]-8-(1-pyridin-2-ylethylamino)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-(2-Cyclobutylethylamino)-8-[2-(2-methylpropoxy)ethyl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C26H32F3N5O3
6-(2-Cyclobutylethylamino)-8-[2-(2-methylpropoxy)ethyl]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(4-Cyclobutylbutylamino)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile —— C29H29F3N6
6-(4-Cyclobutylbutylamino)-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carbonitrile
—— 6-(2-Cyclobutylethylamino)-8-(6-ethoxy-4-propan-2-ylpyridin-2-yl)-7-[(4-methylcyclohexyl)methyl]purine-2-carboxylic acid —— C30H42N6O3
6-(2-Cyclobutylethylamino)-8-(6-ethoxy-4-propan-2-ylpyridin-2-yl)-7-[(4-methylcyclohexyl)methyl]purine-2-carboxylic acid
—— 6-[Cyclopentyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C27H26F3N5O2
6-[Cyclopentyl(methyl)amino]-8-(3-methylphenyl)-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-[cyclopropylmethyl(2-phenylethyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C32H35F3N6O2
6-(2-Cyclobutylethylamino)-8-[cyclopropylmethyl(2-phenylethyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— 6-(2-Cyclobutylethylamino)-8-[formyl-(1-methylcyclohexyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid —— C28H33F3N6O3
6-(2-Cyclobutylethylamino)-8-[formyl-(1-methylcyclohexyl)amino]-7-[[4-(trifluoromethyl)phenyl]methyl]purine-2-carboxylic acid
—— (6S)-6-methyl-2-[(4-piperidin-1-ylsulfonylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C22H27N3O4S2
(6S)-6-methyl-2-[(4-piperidin-1-ylsulfonylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide