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—— (6Z)-6-[[1-(5-chloro-2-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H19ClFN5OS
(6Z)-6-[[1-(5-chloro-2-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-nitro-4-phenyl-3-(4-phenylpiperazin-1-yl)quinolin-2(1H)-one —— C25H22N4O3
6-nitro-4-phenyl-3-(4-phenylpiperazin-1-yl)quinolin-2(1H)-one
—— [(6S,8S,9R,10S,11S,13S,14S,16R,17R)-6,9-difluoro-17-(fluoromethylsulfanylcarbonyl)-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] furan-2-carboxylate;[(6S,8S,9R,10S,11S,13S,14S,16R,17R)-6,9-difluoro-17-(fluoromethylsulfanylcarbonyl)-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] propanoate —— C58H68F6O13S2
[(6S,8S,9R,10S,11S,13S,14S,16R,17R)-6,9-difluoro-17-(fluoromethylsulfanylcarbonyl)-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] furan-2-carboxylate;[(6S,8S,9R,10S,11S,13S,14S,16R,17R)-6,9-difluoro-17-(fluoromethylsulfanylcarbonyl)-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] propanoate
—— (6Z)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-phenyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H23N5O2S
(6Z)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-phenyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-(2-fluorophenyl)-5-imino-6-[[1-(2-methoxy-5-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22FN5O2S
(6Z)-2-(2-fluorophenyl)-5-imino-6-[[1-(2-methoxy-5-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(5-chloro-2-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(2-fluorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H19ClFN5OS
(6E)-6-{[1-(5-chloro-2-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(2-fluorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R,8aS,9S)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6R,8aS,9S)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-chloro-9-(2-fluorobenzyl)-3,4-dimethyl-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one —— C20H17ClFNO3
6-chloro-9-(2-fluorobenzyl)-3,4-dimethyl-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one
—— 6-benzyl-2-(benzylamino)-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one —— C20H19N5O
6-benzyl-2-(benzylamino)-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one
—— (6S,8aR,9S)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6S,8aR,9S)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6Z)-6-{[2,5-dimethyl-1-(2-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-phenyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H21N5OS
(6Z)-6-{[2,5-dimethyl-1-(2-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-phenyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-(2-chlorophenyl)-6-[(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)methylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H18ClN5OS
(6Z)-2-(2-chlorophenyl)-6-[(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)methylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(2,4-dimethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H21N5O4S
(6E)-6-{[1-(2,4-dimethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[1-(2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H21N5O4S
(6Z)-6-[[1-(2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-4-ethyl-9-[2-(4-methoxyphenyl)ethyl]-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one —— C22H22ClNO4
6-chloro-4-ethyl-9-[2-(4-methoxyphenyl)ethyl]-9,10-dihydro-2H,8H-chromeno[8,7-e][1,3]oxazin-2-one
—— 6-chloro-4-ethyl-9-[2-(4-methoxyphenyl)ethyl]-9,10-dihydro-8H-pyrano[2,3-f][1,3]benzoxazin-9-ium-2-one —— C22H23ClNO4+
6-chloro-4-ethyl-9-[2-(4-methoxyphenyl)ethyl]-9,10-dihydro-8H-pyrano[2,3-f][1,3]benzoxazin-9-ium-2-one
—— (6aS)-3-(4-chlorophenyl)-5-[(4-methoxyphenyl)methyl]-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C19H15ClN2O4
(6aS)-3-(4-chlorophenyl)-5-[(4-methoxyphenyl)methyl]-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— (6aS)-5-(1,3-benzodioxol-5-yl)-3-(2-chlorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C18H11ClN2O5
(6aS)-5-(1,3-benzodioxol-5-yl)-3-(2-chlorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— (6S,7R)-5-methylidene-N-(2-methylphenyl)-7-naphthalen-1-yl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H21N5O
(6S,7R)-5-methylidene-N-(2-methylphenyl)-7-naphthalen-1-yl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (6S,8aS,9R)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6S,8aS,9R)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6,7-Dimethoxy-2-(thiophen-2-ylsulfonyl)-1,2,3,4-tetrahydroisoquinoline —— C15H17NO4S2
6,7-Dimethoxy-2-(thiophen-2-ylsulfonyl)-1,2,3,4-tetrahydroisoquinoline
—— (6R,8aS,9R)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6R,8aS,9R)-9-(3-ethoxy-4-hydroxyphenyl)-6-(4-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6E)-2-(2-fluorophenyl)-5-imino-6-{[1-(2-methoxy-5-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22FN5O2S
(6E)-2-(2-fluorophenyl)-5-imino-6-{[1-(2-methoxy-5-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6aS)-5-(4-chloro-2-methoxy-5-methylphenyl)-3-(4-fluorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C19H14ClFN2O4
(6aS)-5-(4-chloro-2-methoxy-5-methylphenyl)-3-(4-fluorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— 6-methyl-2-({[5-(phenylcarbonyl)-1H-benzimidazol-2-yl]methyl}sulfanyl)pyrimidin-4(3H)-one —— C20H16N4O2S
6-methyl-2-({[5-(phenylcarbonyl)-1H-benzimidazol-2-yl]methyl}sulfanyl)pyrimidin-4(3H)-one
—— (6Z)-5-imino-6-[[1-(3-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H20N6O2S
(6Z)-5-imino-6-[[1-(3-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-Benzylpiperazin-4-ium-1-yl)-4,11,13-trimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaene —— C23H27N6+
6-(4-Benzylpiperazin-4-ium-1-yl)-4,11,13-trimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaene
—— 6-chloro-N-(dimethylsulfamoyl)-4,6-difluorocyclohexa-2,4-diene-1-carboxamide —— C9H11ClF2N2O3S
6-chloro-N-(dimethylsulfamoyl)-4,6-difluorocyclohexa-2,4-diene-1-carboxamide
—— (6aS)-5-benzyl-3-(4-fluorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C18H13FN2O3
(6aS)-5-benzyl-3-(4-fluorophenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— 6-methoxy-N-[(3-methoxyphenyl)methylideneamino]-1H-indole-2-carboxamide —— C18H17N3O3
6-methoxy-N-[(3-methoxyphenyl)methylideneamino]-1H-indole-2-carboxamide
—— 6-[5-(bromomethyl)-4-chloro-1H-pyrazol-3-yl]-4,6-dimethylcyclohexa-2,4-diene-1-carboxylic acid —— C13H14BrClN2O2
6-[5-(bromomethyl)-4-chloro-1H-pyrazol-3-yl]-4,6-dimethylcyclohexa-2,4-diene-1-carboxylic acid
—— (6E)-5-imino-6-{[1-(3-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H20N6O2S
(6E)-5-imino-6-{[1-(3-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[3-[(R)-amino(phenyl)methyl]-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl]-4H-1,4-benzoxazin-3-one —— C19H16N6O2S
6-[3-[(R)-amino(phenyl)methyl]-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl]-4H-1,4-benzoxazin-3-one
—— 6-chloro-2-(1H-indol-3-yl)-N-(2-methylphenyl)-1H-imidazo[1,2-a]pyridin-4-ium-3-amine —— C22H18ClN4+
6-chloro-2-(1H-indol-3-yl)-N-(2-methylphenyl)-1H-imidazo[1,2-a]pyridin-4-ium-3-amine
—— [[6-(1,8-diethyl-4,9-dihydro-3H-pyrano[3,4-b]indol-1-yl)-5-oxohexyl]amino]thiourea —— C22H32N4O2S
[[6-(1,8-diethyl-4,9-dihydro-3H-pyrano[3,4-b]indol-1-yl)-5-oxohexyl]amino]thiourea
—— 6-iodo-1H-indole-2-carboxylate —— C9H5INO2-
6-iodo-1H-indole-2-carboxylate
—— (6S,6aR)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C21H21NO2S
(6S,6aR)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— 6-oxo-1,2-dihydrotriazolo[4,5-b]pyridine-7-carboxylic acid —— C6H4N4O3
6-oxo-1,2-dihydrotriazolo[4,5-b]pyridine-7-carboxylic acid
—— (6aS)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C19H15ClN2O3
(6aS)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— 6-iodo-1H-indole-2-carboxylic Acid —— C9H6INO2
6-iodo-1H-indole-2-carboxylic Acid
—— (6Z)-3-(benzylsulfanyl)-6-{[1-(3,5-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,2,4]thiadiazolo[4,5-a]pyrimidin-7-one —— C27H25N5OS2
(6Z)-3-(benzylsulfanyl)-6-{[1-(3,5-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,2,4]thiadiazolo[4,5-a]pyrimidin-7-one
—— (6R,7S)-N-(4-methoxyphenyl)-5-methylidene-7-naphthalen-1-yl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H21N5O2
(6R,7S)-N-(4-methoxyphenyl)-5-methylidene-7-naphthalen-1-yl-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-[4-[(2,4-Dichlorophenyl)methyl]piperazin-4-ium-1-yl]-4,11,13-trimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaene —— C23H25Cl2N6+
6-[4-[(2,4-Dichlorophenyl)methyl]piperazin-4-ium-1-yl]-4,11,13-trimethyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaene
—— (6aS)-3-(2,5-dimethoxyphenyl)-5-(3,5-dimethylphenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione —— C21H20N2O5
(6aS)-3-(2,5-dimethoxyphenyl)-5-(3,5-dimethylphenyl)-2,6a-dihydropyrrolo[3,4-d][1,2]oxazole-4,6-dione
—— 6-Bromo-5-methyl-2-(2-methyl-allylsulfanyl)-3H-imidazo[4,5-b]pyridine —— C11H12BrN3S
6-Bromo-5-methyl-2-(2-methyl-allylsulfanyl)-3H-imidazo[4,5-b]pyridine
—— (6Z)-6-{3-chloro-4-[2-(3-methoxyphenoxy)ethoxy]benzylidene}-5-imino-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H20ClN5O4S
(6Z)-6-{3-chloro-4-[2-(3-methoxyphenoxy)ethoxy]benzylidene}-5-imino-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-{4-[(2,4-Dichlorophenyl)methyl]piperazin-1-yl}-4,11,13-trimethyl-3,7,8,10-tetraazatricyclo[7.4.0.0^{2,7}]trideca-1,3,5,8,10,12-hexaene —— C23H24Cl2N6
6-{4-[(2,4-Dichlorophenyl)methyl]piperazin-1-yl}-4,11,13-trimethyl-3,7,8,10-tetraazatricyclo[7.4.0.0^{2,7}]trideca-1,3,5,8,10,12-hexaene
—— (6R,6aS)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C21H21NO2S
(6R,6aS)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6R,8aR,9S)-9-(3,4-dimethoxyphenyl)-6-(2-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6R,8aR,9S)-9-(3,4-dimethoxyphenyl)-6-(2-methylphenyl)-6,7,8a,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6E)-6-{[1-(2-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H16FN5O2S
(6E)-6-{[1-(2-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one