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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cycloheptylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C25H32FN5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(cycloheptylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-[[(1S)-2-hydroxy-1-phenylethyl]amino]-N-methylpyridine-3-carboxamide —— C22H21N5O2S
6-(1,3-benzothiazol-6-ylamino)-4-[[(1S)-2-hydroxy-1-phenylethyl]amino]-N-methylpyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-ethyl-2-fluoro-3-hydroxypentyl]-4-[(2-fluoro-2-methylpropyl)amino]pyridine-3-carboxamide 1610019-33-4 C24H31F2N5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-ethyl-2-fluoro-3-hydroxypentyl]-4-[(2-fluoro-2-methylpropyl)amino]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-(cyclopentanecarbonylamino)butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-16-0 C26H34N6O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-(cyclopentanecarbonylamino)butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-[(6-cyanoquinolin-2-yl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(propan-2-ylamino)pyridine-3-carboxamide —— C24H27FN6O2
6-[(6-cyanoquinolin-2-yl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(3S)-3-(propan-2-ylcarbamoylamino)butyl]pyridine-3-carboxamide 1610018-13-7 C24H33N7O2S
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(3S)-3-(propan-2-ylcarbamoylamino)butyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-(4-hydroxycyclohexyl)pyridine-3-carboxamide —— C24H29N5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-(4-hydroxycyclohexyl)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[4-(2-hydroxypropan-2-yl)cyclohexyl]-4-(oxan-3-ylamino)pyridine-3-carboxamide —— C27H35N5O3S
6-(1,3-benzothiazol-6-ylamino)-N-[4-(2-hydroxypropan-2-yl)cyclohexyl]-4-(oxan-3-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[[(1S)-2-hydroxy-1-phenylethyl]amino]pyridine-3-carboxamide —— C26H28FN5O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[[(1S)-2-hydroxy-1-phenylethyl]amino]pyridine-3-carboxamide
—— 6-Methyl-1,5-naphthyridine-3-carboxamide —— C10H9N3O
6-Methyl-1,5-naphthyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)pyridine-3-carboxamide —— C23H25N7OS
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)pyridine-3-carboxamide
—— 6-(2,1,3-benzoxadiazol-5-ylamino)-4-(cyclopropylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C20H23FN6O3
6-(2,1,3-benzoxadiazol-5-ylamino)-4-(cyclopropylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-cyclopropyl-2,4,4,4-tetrafluoro-3-hydroxybutyl]-4-(propan-2-ylamino)pyridine-3-carboxamide —— C23H25F4N5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-cyclopropyl-2,4,4,4-tetrafluoro-3-hydroxybutyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[4-(2,2,2-trifluoroethylcarbamoyl)anilino]pyridine-3-carboxamide —— C27H26F4N6O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[4-(2,2,2-trifluoroethylcarbamoyl)anilino]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[4-[(2-hydroxy-2-methylpropyl)carbamoyl]-1-bicyclo[2.2.2]octanyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-58-0 C29H38N6O3S
6-(1,3-benzothiazol-6-ylamino)-N-[4-[(2-hydroxy-2-methylpropyl)carbamoyl]-1-bicyclo[2.2.2]octanyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-Fluoro-5-methyl-[1,3]thiazolo[5,4-b]pyridine —— C7H5FN2S
6-Fluoro-5-methyl-[1,3]thiazolo[5,4-b]pyridine
—— 6-(1,3-benzothiazol-6-ylamino)-4-[2,5-difluoro-4-(methylcarbamoyl)anilino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C26H25F3N6O3S
6-(1,3-benzothiazol-6-ylamino)-4-[2,5-difluoro-4-(methylcarbamoyl)anilino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-(2-morpholin-4-ylethyl)-4-(propan-2-ylamino)pyridine-3-carboxamide —— C22H28N6O2S
6-(1,3-benzothiazol-6-ylamino)-N-(2-morpholin-4-ylethyl)-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cyclopropylamino)-N-[(2R)-2-fluoro-3-hydroxypropyl]pyridine-3-carboxamide 1610016-56-2 C19H20FN5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(cyclopropylamino)-N-[(2R)-2-fluoro-3-hydroxypropyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-[(2R)-2-fluoro-3-hydroxypropyl]pyridine-3-carboxamide —— C21H24FN5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-[(2R)-2-fluoro-3-hydroxypropyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cyclopropylamino)-N-[(2R)-2,4,4,4-tetrafluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C21H21F4N5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(cyclopropylamino)-N-[(2R)-2,4,4,4-tetrafluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(1-hydroxypropan-2-ylamino)pyridine-3-carboxamide —— C21H26FN5O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(1-hydroxypropan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(oxan-3-yl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-26-2 C27H36N6O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(oxan-3-yl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— (6-ethyl-4-methyl-2-oxochromen-7-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]propanoate —— C20H25NO6
(6-ethyl-4-methyl-2-oxochromen-7-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]propanoate
—— 6-(3,4-Dimethoxyphenyl)-1-(3,4-dimethoxy-5-thiophen-2-ylphenyl)-[1]benzofuro[7,6-g][1]benzofuran-2,7-dione —— C34H24O8S
6-(3,4-Dimethoxyphenyl)-1-(3,4-dimethoxy-5-thiophen-2-ylphenyl)-[1]benzofuro[7,6-g][1]benzofuran-2,7-dione
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(oxan-4-yl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-21-7 C27H36N6O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(oxan-4-yl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[[3-(hydroxymethyl)cyclobutyl]amino]pyridine-3-carboxamide —— C23H28FN5O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[[3-(hydroxymethyl)cyclobutyl]amino]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-[[(1S,2S)-1-(3,5-difluorophenyl)-2,3-dihydroxypropyl]amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C27H28F3N5O4S
6-(1,3-benzothiazol-6-ylamino)-4-[[(1S,2S)-1-(3,5-difluorophenyl)-2,3-dihydroxypropyl]amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-[(4-fluorocyclohexyl)amino]-N-(3-hydroxy-3-methylbutyl)pyridine-3-carboxamide —— C24H30FN5O2S
6-(1,3-benzothiazol-6-ylamino)-4-[(4-fluorocyclohexyl)amino]-N-(3-hydroxy-3-methylbutyl)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(2,2-difluorocyclohexyl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-20-6 C28H36F2N6O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[2-(2,2-difluorocyclohexyl)acetyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-(cyanomethyl)-4-(cyclopentylamino)pyridine-3-carboxamide —— C20H20N6OS
6-(1,3-benzothiazol-6-ylamino)-N-(cyanomethyl)-4-(cyclopentylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[(5-hydroxy-5-methylhexanoyl)amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-22-8 C27H38N6O3S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[(5-hydroxy-5-methylhexanoyl)amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(3-methylbutylamino)pyridine-3-carboxamide 1610017-95-2 C23H30FN5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(3-methylbutylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(ethylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C20H24FN5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(ethylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-[(7-cyano-1,5-naphthyridin-2-yl)amino]-4-[(2,2-difluorocyclopentyl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C25H26F3N7O2
6-[(7-cyano-1,5-naphthyridin-2-yl)amino]-4-[(2,2-difluorocyclopentyl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-[(5-hydroxy-2-adamantyl)amino]-N-methylpyridine-3-carboxamide —— C24H27N5O2S
6-(1,3-benzothiazol-6-ylamino)-4-[(5-hydroxy-2-adamantyl)amino]-N-methylpyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(2R)-2,4,4,4-tetrafluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C21H23F4N5O2S
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(2R)-2,4,4,4-tetrafluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— (6Z)-6-{[5-(3-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H15ClN4O2S
(6Z)-6-{[5-(3-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-Bromo-4,5-dimethoxyphenyl)-1-(3-bromo-4-ethoxy-5-methoxyphenyl)-[1]benzofuro[7,6-g][1]benzofuran-2,7-dione —— C31H22Br2O8
6-(3-Bromo-4,5-dimethoxyphenyl)-1-(3-bromo-4-ethoxy-5-methoxyphenyl)-[1]benzofuro[7,6-g][1]benzofuran-2,7-dione
—— 6-[(5-fluoro-1,3-benzothiazol-6-yl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[(2-fluoro-2-methylpropyl)amino]pyridine-3-carboxamide —— C22H26F3N5O2S
6-[(5-fluoro-1,3-benzothiazol-6-yl)amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[(2-fluoro-2-methylpropyl)amino]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(2,2,2-trifluoroethylamino)pyridine-3-carboxamide —— C20H21F4N5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(2,2,2-trifluoroethylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-[4-(difluoromethoxy)anilino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C25H24F3N5O3S
6-(1,3-benzothiazol-6-ylamino)-4-[4-(difluoromethoxy)anilino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[4-(propan-2-ylcarbamoyl)cyclohexyl]pyridine-3-carboxamide —— C26H34N6O2S
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[4-(propan-2-ylcarbamoyl)cyclohexyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-(2-pyrrolidin-1-ylethyl)pyridine-3-carboxamide —— C24H30N6OS
6-(1,3-benzothiazol-6-ylamino)-4-(cyclopentylamino)-N-(2-pyrrolidin-1-ylethyl)pyridine-3-carboxamide
—— 6-(3a,7a-dihydro-1,3-benzothiazol-6-ylamino)-4-[[3-(difluoromethyl)cyclobutyl]amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide —— C23H28F3N5O2S
6-(3a,7a-dihydro-1,3-benzothiazol-6-ylamino)-4-[[3-(difluoromethyl)cyclobutyl]amino]-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(3R)-3-[[2-(triazol-1-yl)acetyl]amino]butyl]pyridine-3-carboxamide 1610018-25-1 C24H29N9O2S
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[(3R)-3-[[2-(triazol-1-yl)acetyl]amino]butyl]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[(1R,3S)-3-fluorocyclopentanecarbonyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide 1610018-30-8 C26H33FN6O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(3R)-3-[[(1R,3S)-3-fluorocyclopentanecarbonyl]amino]butyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[(2-methylphenyl)methylamino]pyridine-3-carboxamide 1610017-98-5 C26H28FN5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-[(2-methylphenyl)methylamino]pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-cyclopropyl-2-fluoro-3-hydroxypropyl]-4-(propan-2-ylamino)pyridine-3-carboxamide —— C22H26FN5O2S
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-cyclopropyl-2-fluoro-3-hydroxypropyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
—— 6-(1,3-benzothiazol-6-ylamino)-N-[4-(methylcarbamoyl)cyclohexyl]-4-(propan-2-ylamino)pyridine-3-carboxamide —— C24H30N6O2S
6-(1,3-benzothiazol-6-ylamino)-N-[4-(methylcarbamoyl)cyclohexyl]-4-(propan-2-ylamino)pyridine-3-carboxamide