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影响免疫功能药

影响免疫功能的药物 1. 免疫抑制剂

免疫抑制剂是一类用于治疗自身免疫性疾病和器官移植排斥反应的药物,通过降低免疫系统的活性来减少炎症反应和组织损伤。

  • 环孢素:主要用于预防器官移植后的排异反应。它选择性地抑制T淋巴细胞的活化。
  • 他克莫司(FK506):与环孢素作用类似,同样用于防止器官移植中的排斥反应,并且也被用来治疗某些自身免疫性疾病。
  • 霉酚酸酯(MMF):通过干扰次黄嘌呤核苷酸脱氢酶和鸟嘌呤核苷酸合成来抑制淋巴细胞增生。
2. 免疫增强剂

这类药物旨在提高机体的免疫力,主要用于改善免疫缺陷患者的状况或预防感染。

  • 胸腺肽α1:有助于调节T淋巴细胞的功能,提升整体免疫应答能力。它被用于治疗某些类型的艾滋病及慢性乙肝病毒感染。
  • 干扰素α(IFN-α):具有抗病毒、抗增殖和免疫调节作用。可以用于治疗多种疾病如HIV感染、乙型肝炎等。
3. 免疫调节剂

这类药物能够双向调节免疫反应,既可增强又可抑制免疫应答。

  • 白细胞介素-2(IL-2):一种重要促炎因子,在低剂量时具有刺激T细胞增殖的作用;而在高浓度下则可能产生抗肿瘤效果或导致自身免疫性疾病的恶化。
  • 环磷酰胺(CTX):通过在DNA上形成交联阻止其复制来发挥细胞毒作用,同时也被用于癌症治疗中的免疫调节。
4. 免疫检查点抑制剂

这些新型抗癌药物通过阻断癌细胞表面的PD-L1与T淋巴细胞上的PD-1受体之间的相互作用,从而解除对肿瘤杀伤性T细胞的抑制。

  • 帕博利珠单抗(Pembrolizumab)纳武利尤单抗(Nivolumab):这两种药物属于人源化单克隆抗体类免疫检查点抑制剂,能够特异性地结合PD-1受体,恢复T细胞对肿瘤细胞的识别与杀伤功能。
5. 免疫吸附疗法

这是一种物理去除血液中有害物质的方法,在某些自身免疫性疾病中应用广泛。

  • 血浆置换:通过移除含有致病因子(如循环抗体、补体成分)的血浆,替换为新鲜冷冻血浆或白蛋白等生理溶液来达到治疗目的。

这些药物在不同类型的疾病中发挥着重要作用,但同时也存在副作用风险,使用时需严格遵循医嘱。

中文名称 英文名称 CAS号 化学式 结构式图片
雷帕霉素 sirolimus 53123-88-9 C51H79NO13
雷帕霉素
褪黑素 5-methoxy-N-acetyl-tryptamine 73-31-4 C13H16N2O2
褪黑素
咪唑立宾 mizoribine 50924-49-7 C9H13N3O6
咪唑立宾
双醋瑞因 diacetylrhein 13739-02-1 C19H12O8
双醋瑞因
依维莫司 everolimus 159351-69-6 C53H83NO14
依维莫司
—— (1R,9S,12S,15R,16Z,18R,19R,21R,23S,24E,26Z,28E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1R,9S,12S,15R,16Z,18R,19R,21R,23S,24E,26Z,28E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— (1R,9S,12S,15R,16Z,18R,19R,21R,23S,24Z,26Z,28Z,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1R,9S,12S,15R,16Z,18R,19R,21R,23S,24Z,26Z,28Z,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— (1R,9S,12S,15R,16E,18R,19R,21R,23R,24Z,26E,28E,30S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1R,9S,12S,15R,16E,18R,19R,21R,23R,24Z,26E,28E,30S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— Pharmakon1600-01504008 53123-88-9 C51H79NO13
Pharmakon1600-01504008
—— (1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— 23,1-c][1,4]oxaazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone, 9,10,12,13,14,21,22,23,24, 25,26,27,32,33,34,34a-hexadecahydro-9,27-dihydroxy-3-[2-(4-hydroxy-3-methoxycyclohexyl)-1-methylethyl]-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-, [3S-[3R*[S* (1R*,3S*,4S*)],6S*,7E,9S*,10S*,12S*,14R*,15E,17E,19E,21R*, 23R*,26S*,27S*,34aR*]]- 53123-88-9 C51H79NO13
23,1-c][1,4]oxaazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone, 9,10,12,13,14,21,22,23,24, 25,26,27,32,33,34,34a-hexadecahydro-9,27-dihydroxy-3-[2-(4-hydroxy-3-methoxycyclohexyl)-1-methylethyl]-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-, [3S-[3R*[S* (1R*,3S*,4S*)],6S*,7E,9S*,10S*,12S*,14R*,15E,17E,19E,21R*, 23R*,26S*,27S*,34aR*]]-
—— 42-O-(2-hydroxyethyl)rapamycin) 159351-69-6 C53H83NO14
42-O-(2-hydroxyethyl)rapamycin)
—— Everolimus (RAD001) 159351-69-6 C53H83NO14
Everolimus (RAD001)
—— (1S,9R,15R,16E,18R,19R,21S,23R,24E,26E,28E,30S,32R,35S)-1,18-dihydroxy-12-[(2S)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1S,9R,15R,16E,18R,19R,21S,23R,24E,26E,28E,30S,32R,35S)-1,18-dihydroxy-12-[(2S)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— 4-acetamidobenzoic acid;9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-purin-6-one;1-(dimethylamino)propan-2-ol 36703-88-5 C24H34N6O9
4-acetamidobenzoic acid;9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1H-purin-6-one;1-(dimethylamino)propan-2-ol
—— (1R,9S,12S,15R,16E,18R,19R,21R,23S,24Z,26E,28E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
(1R,9S,12S,15R,16E,18R,19R,21R,23S,24Z,26E,28E,30S,32S,35R)-1,18-dihydroxy-12-[(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone
—— AP-22594 53123-88-9 C51H79NO13
AP-22594
—— rapamycin 53123-88-9 C51H79NO13
rapamycin
—— melatonin 73-31-4 C13H16N2O2
melatonin
—— bredinin 50924-49-7 C9H13N3O6
bredinin
—— mizoribine 50924-49-7 C9H13N3O6
mizoribine
—— 1,18-Dihydroxy-12-[1-[4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone 159351-69-6 C53H83NO14
1,18-Dihydroxy-12-[1-[4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl]-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo[30.3.1.04,9]hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentone