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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-methylphenyl)-1,3-oxazole-4-carbohydroxamic acid —— C11H10N2O3
2-(4-methylphenyl)-1,3-oxazole-4-carbohydroxamic acid
—— 2-[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]pyrimidine —— C11H8N6S
2-[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]pyrimidine
—— 1-(4-fluorophenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5H-pyrazolo[3,4-b]quinolin-5-one —— C19H18FN3O
1-(4-fluorophenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5H-pyrazolo[3,4-b]quinolin-5-one
—— 3,7,7-trimethyl-1-phenyl-7,8-dihydrociclohexa[2,3-e]pyrazolo-[3,4-b]pyridin-5(6H)-one —— C19H19N3O
3,7,7-trimethyl-1-phenyl-7,8-dihydrociclohexa[2,3-e]pyrazolo-[3,4-b]pyridin-5(6H)-one
—— 7-cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine —— C21H23N7O
7-cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine
—— 7-cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine —— C20H21N7O
7-cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine
—— 7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine —— C19H21N7O
7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine
—— 2-[2-methyl-4-(2-methyl-pyridin-4-ylethynyl)-imidazol-1-yl]-pyrimidine —— C16H13N5
2-[2-methyl-4-(2-methyl-pyridin-4-ylethynyl)-imidazol-1-yl]-pyrimidine
—— 2-(4-chloro-2-fluoro-5-hydroxyphenyl)hexa-hydro-3-thioxo-1H-[1,2,4]triazolo[1,2-a]pyridazin-1-one —— C12H11ClFN3O2S
2-(4-chloro-2-fluoro-5-hydroxyphenyl)hexa-hydro-3-thioxo-1H-[1,2,4]triazolo[1,2-a]pyridazin-1-one
—— 4-(6,6-dimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)-N-(4-methoxyphenyl)benzenesulfonamide —— C22H23N3O4S
4-(6,6-dimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indazol-1-yl)-N-(4-methoxyphenyl)benzenesulfonamide
—— N-((1-(3-(difluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)methyl)pyrimidin-2-amine —— C14H12F2N6
N-((1-(3-(difluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)methyl)pyrimidin-2-amine
—— 2-({1-[4-(4-chlorophenyl)-5-methyl-4H-1,2,4-triazol-3-yl]-piperidin-4-yl}oxy)pyrimidine —— C18H19ClN6O
2-({1-[4-(4-chlorophenyl)-5-methyl-4H-1,2,4-triazol-3-yl]-piperidin-4-yl}oxy)pyrimidine
—— 2-((1-(4-chloro-3-(difluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)methoxy)pyrimidine —— C14H10ClF2N5O
2-((1-(4-chloro-3-(difluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)methoxy)pyrimidine
—— 2-(3-phenyl-1H-pyrazol-1-yl)pyrimidine —— C13H10N4
2-(3-phenyl-1H-pyrazol-1-yl)pyrimidine
—— N'-hydroxy-4-(1H-pyrazol-1-yl)benzimidamide —— C10H10N4O
N'-hydroxy-4-(1H-pyrazol-1-yl)benzimidamide
—— 5,5-dimethyl-2-[(1H-pyrazol-3-ylamino)-methylene]cyclohexane-1,3-dione —— C12H15N3O2
5,5-dimethyl-2-[(1H-pyrazol-3-ylamino)-methylene]cyclohexane-1,3-dione
—— 2-(4-(1-(2-chlorophenyl)-3-(trifluoromethyl)-1H-pyrazol-5-yl)phenoxy)pyrimidine —— C20H12ClF3N4O
2-(4-(1-(2-chlorophenyl)-3-(trifluoromethyl)-1H-pyrazol-5-yl)phenoxy)pyrimidine
—— 2,4,6-tris[4-(pyrazol-1-yl)phenyl]-1,3,5-triazine —— C30H21N9
2,4,6-tris[4-(pyrazol-1-yl)phenyl]-1,3,5-triazine
—— 2-[4-(3-chloro-phenylethynyl)-2-methyl-imidazol-1-yl]-pyrimidine —— C16H11ClN4
2-[4-(3-chloro-phenylethynyl)-2-methyl-imidazol-1-yl]-pyrimidine
—— 6-(1-(4-cyanophenyl)-1H-pyrazol-5-yl)-N-ethyl-5-methyl-3-oxo-4-(3-(trifluoromethyl)phenyl)-3,4-dihydropyrazine-2-carboxamide —— C24H17F3N6O2
6-(1-(4-cyanophenyl)-1H-pyrazol-5-yl)-N-ethyl-5-methyl-3-oxo-4-(3-(trifluoromethyl)phenyl)-3,4-dihydropyrazine-2-carboxamide
—— 1-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]pyrazole —— C12H12N4
1-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]pyrazole
—— 1-[4-(1H-imidazol-2-yl)phenyl]pyrazole —— C12H10N4
1-[4-(1H-imidazol-2-yl)phenyl]pyrazole
—— 4-{6-bromo-8-[(oxetan-3-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-N-cyclopropyl-2-methylbenzamide —— C21H22BrN5O2
4-{6-bromo-8-[(oxetan-3-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-N-cyclopropyl-2-methylbenzamide
—— 4-[6-bromo-8-(methylsulfanyl)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopropyl-2-methylbenzamide —— C18H17BrN4OS
4-[6-bromo-8-(methylsulfanyl)imidazo[1,2-b]pyridazin-3-yl]-N-cyclopropyl-2-methylbenzamide
—— 3-chloro-N'-[((E)-5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methylidene]benzo[b]thiophene-2-carbohydrazide —— C20H14Cl2N4OS
3-chloro-N'-[((E)-5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methylidene]benzo[b]thiophene-2-carbohydrazide
—— 2-(2-(4-chloro-3-(3-methylpyrazolo[1,5-a]pyridin-2-yl)phenyl)-1,2,3,4-tetrahydroisoquinolin-6-yl)-2-propanol —— C26H26ClN3O
2-(2-(4-chloro-3-(3-methylpyrazolo[1,5-a]pyridin-2-yl)phenyl)-1,2,3,4-tetrahydroisoquinolin-6-yl)-2-propanol
—— 3-(4-((6-methyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino)phenoxy)propyl nitrate —— C21H20N6O4
3-(4-((6-methyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino)phenoxy)propyl nitrate
—— N-(4-(3-bromopropoxy)phenyl)-6-methyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine —— C21H20BrN5O
N-(4-(3-bromopropoxy)phenyl)-6-methyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— 1-phenyl[1]benzothieno[2',3':5,6]pyrano[2,3-c]pyrazol-4(1H)-one —— C18H10N2O2S
1-phenyl[1]benzothieno[2',3':5,6]pyrano[2,3-c]pyrazol-4(1H)-one
—— 3-methyl-1-phenyl[1]benzothieno[2',3':5,6]pyrano[2,3-c]pyrazol-4(1H)-one —— C19H12N2O2S
3-methyl-1-phenyl[1]benzothieno[2',3':5,6]pyrano[2,3-c]pyrazol-4(1H)-one
—— 1-(4-hydroxymethylphenyl)-5-(4-(methylsulfonyl)phenyl)-1H-tetrazole —— C15H14N4O3S
1-(4-hydroxymethylphenyl)-5-(4-(methylsulfonyl)phenyl)-1H-tetrazole
—— Example 3 —— C23H22N6O
Example 3
—— 1-[(1,'3'-dihydroxy-2'-methyl)-2'-propyl]-2-methyl-4-nitro-1H-imidazole —— C8H13N3O4
1-[(1,'3'-dihydroxy-2'-methyl)-2'-propyl]-2-methyl-4-nitro-1H-imidazole
—— 1-(methyl 5'-deoxy-2',3'-O-isopropylidene-β-D-ribofuranosid-5'-yl)-2-methyl-4-nitro-1-[15N]-1H-imidazole —— C13H19N3O6
1-(methyl 5'-deoxy-2',3'-O-isopropylidene-β-D-ribofuranosid-5'-yl)-2-methyl-4-nitro-1-[15N]-1H-imidazole
—— 2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole —— C12H13N3O2
2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole
—— (S)-3-(2-methyl-4-nitro-1H-imidazol-1-yl)propane-1,2-diol —— C7H11N3O4
(S)-3-(2-methyl-4-nitro-1H-imidazol-1-yl)propane-1,2-diol
—— (R)-2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole —— C12H13N3O2
(R)-2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole
—— (S)-2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole —— C12H13N3O2
(S)-2-methyl-4-nitro-1-(1-phenylethyl)-1H-imidazole
—— ethyl 2-benzyloxazole-5-carboxylate —— C13H13NO3
ethyl 2-benzyloxazole-5-carboxylate
—— 2-(2-chlorobenzyl)-8-(morpholinosulfonyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one —— C17H17ClN4O4S
2-(2-chlorobenzyl)-8-(morpholinosulfonyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— 2-amino-5-butyl-4-phenylthiazole —— C13H16N2S
2-amino-5-butyl-4-phenylthiazole
—— 1-(4-bromo-phenyl)-5-(4-methylsulfonyl-phenyl)-3-trifluoromethyl-1H-1,2,4-triazole —— C16H11BrF3N3O2S
1-(4-bromo-phenyl)-5-(4-methylsulfonyl-phenyl)-3-trifluoromethyl-1H-1,2,4-triazole
—— 5-(2-chloro-4-nitrophenyl)-1-methyl-1H-1,2,4-triazole —— C9H7ClN4O2
5-(2-chloro-4-nitrophenyl)-1-methyl-1H-1,2,4-triazole
—— N-(1-(2,6-dimethoxyphenyl)-2-(6-ethoxypyridin-2-yl)-1H-imidazo[4,5-b]pyrazin-5-yl)-2-phenylacetamide —— C28H26N6O4
N-(1-(2,6-dimethoxyphenyl)-2-(6-ethoxypyridin-2-yl)-1H-imidazo[4,5-b]pyrazin-5-yl)-2-phenylacetamide
—— 3-(2-methyl-4-nitro-1H-imidazol-1-yl)propylamine —— C7H12N4O2
3-(2-methyl-4-nitro-1H-imidazol-1-yl)propylamine
—— 5-S-(methyl 2,3,6-tri-O-benzyl-4-deoxy-α-D-galactopyranos-4-yl)-1-phenyl-5-thiotetrazole —— C35H36N4O5S
5-S-(methyl 2,3,6-tri-O-benzyl-4-deoxy-α-D-galactopyranos-4-yl)-1-phenyl-5-thiotetrazole
—— N-propyl-N-[2-(4-chlorophenoxy)ethyl]thiazole-5-carboxamide —— C15H17ClN2O2S
N-propyl-N-[2-(4-chlorophenoxy)ethyl]thiazole-5-carboxamide
—— 1-(2,6-dichloro-4-trifluoromethylphenyl)-3-cyano-4-trifluoromethylsulfenyl-5-(methylthioacetamido)pyrazole —— C15H8Cl2F6N4OS2
1-(2,6-dichloro-4-trifluoromethylphenyl)-3-cyano-4-trifluoromethylsulfenyl-5-(methylthioacetamido)pyrazole
—— 6-methoxy-3-methyl-1-phenylchromeno[2,3-c]pyrazol-4(1H)-one —— C18H14N2O3
6-methoxy-3-methyl-1-phenylchromeno[2,3-c]pyrazol-4(1H)-one
—— 1-(2-methoxyphenyl)-1H-imidazole —— C10H9N2O
1-(2-methoxyphenyl)-1H-imidazole