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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(8-(2,6-difluorophenyl)-2-{[2-(dimethylamino)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methyl-N-propylbenzamide —— C28H30F2N6O2
3-(8-(2,6-difluorophenyl)-2-{[2-(dimethylamino)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methyl-N-propylbenzamide
—— 3-[8-(2,6-difluorophenyl)-2-(methylsulfinyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-(2-phenylethyl)benzamide —— C30H24F2N4O3S
3-[8-(2,6-difluorophenyl)-2-(methylsulfinyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-(2-phenylethyl)benzamide
—— 3-{8-(2,6-difluorophenyl)-2-[[3-(dimethylamino)propyl](methyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-propylbenzamide —— C30H34F2N6O2
3-{8-(2,6-difluorophenyl)-2-[[3-(dimethylamino)propyl](methyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-propylbenzamide
—— N-cyclopentyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C37H42F2N6O2
N-cyclopentyl-3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]benzamide —— C32H36F2N6O2
N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]benzamide
—— 1,1-diniethylethyl (2-{[8-(2,6-difluorophenyl)-4-(2-methyl-5-{[(2-phenylethyl)amino]carbonyl}phenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}ethyl)methylcarbamate —— C37H38F2N6O4
1,1-diniethylethyl (2-{[8-(2,6-difluorophenyl)-4-(2-methyl-5-{[(2-phenylethyl)amino]carbonyl}phenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}ethyl)methylcarbamate
—— 3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrobromide —— BrH*C28H20F2N8O2S
3-{8-(2,6-difluorophenyl)-2-[(1H-imidazol-2-ylmethyl)amino]-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl}-4-methyl-N-1,3-thiazol-2-ylbenzamide hydrobromide
—— N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C33H38F2N6O2
N-cyclopentyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methylbenzamide —— C31H34F2N6O2
N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methylbenzamide
—— 1,1-dimethylethyl {2-[(8-(2,6-difluorophenyl)-4-{2-methyl-5-[(propylamino)carbonyl]phenyl}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]ethyl}methylcarbamate —— C32H36F2N6O4
1,1-dimethylethyl {2-[(8-(2,6-difluorophenyl)-4-{2-methyl-5-[(propylamino)carbonyl]phenyl}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]ethyl}methylcarbamate
—— N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C31H34F2N6O2
N-cyclopropyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-1,3-thiazol-2-ylbenzamide —— C31H31F2N7O2S
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-2-methyl-N-1,3-thiazol-2-ylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1S)-1,2-dimethylpropyl]-4-methylbenzamide —— C33H40F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1S)-1,2-dimethylpropyl]-4-methylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1R)-1,2-dimethylpropyl]-4-methylbenzamide —— C33H40F2N6O2
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[(1R)-1,2-dimethylpropyl]-4-methylbenzamide
—— 4-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide —— C30H29F2N7O2S
4-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide —— C30H29F2N7O2S
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-1,3-thiazol-2-ylbenzamide
—— N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C28H27F2N5O4
N-(cyclopropylmethyl)-3-[8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,N,4-trimethylbenzamide —— C34H38F2N6O2
3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,N,4-trimethylbenzamide
—— 3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[2-(ethylthio)ethyl]-4-methylbenzamide —— C32H38F2N6O2S
3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N-[2-(ethylthio)ethyl]-4-methylbenzamide
—— 3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,4-dimethylbenzamide —— C33H36F2N6O2
3-[8-(2,6-difluorophenyl)-2-(4-methyl-1,4'-bipiperidin-1'-yl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-N,4-dimethylbenzamide
—— N-cyclohexyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C34H40F2N6O2
N-cyclohexyl-3-[2-{[3-(diethylamino)propyl]amino}-8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— N-(cyclopropylmethyl)-3-(8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methylbenzamide —— C25H20F2N4O2
N-(cyclopropylmethyl)-3-(8-(2,6-difluorophenyl)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-4-methylbenzamide
—— N-cyclopropyl-3-[8-(2,6-difluorophenyl)-2-(methylthio)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide —— C25H20F2N4O2S
N-cyclopropyl-3-[8-(2,6-difluorophenyl)-2-(methylthio)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methylbenzamide
—— 4-(5-amino-2-methylphenyl)-8-(2,6-difluorophenyl)-2-(methylsulfonyl)pyrido[2,3-d]pyrimidin-7(8H)-one —— C21H16F2N4O3S
4-(5-amino-2-methylphenyl)-8-(2,6-difluorophenyl)-2-(methylsulfonyl)pyrido[2,3-d]pyrimidin-7(8H)-one
—— N-cyclopropyl-3-(8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-5-fluoro-4-methylbenzamide —— C27H24F3N5O4
N-cyclopropyl-3-(8-(2,6-difluorophenyl)-2-{[2-hydroxy-1-(hydroxymethyl)ethyl]amino}-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl)-5-fluoro-4-methylbenzamide
—— 3-[8-(2,6-difluorophenyl)-2-(methylthio)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-1,3-thiazol-2-4lbenzamide —— C25H17F2N5O2S2
3-[8-(2,6-difluorophenyl)-2-(methylthio)-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-1,3-thiazol-2-4lbenzamide
—— 3-[8-(2,6-difluoro-phenyl)-2-methylsulfanyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-propyl-benzamide —— C25H22F2N4O2S
3-[8-(2,6-difluoro-phenyl)-2-methylsulfanyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-4-yl]-4-methyl-N-propyl-benzamide
—— 2-p-tolyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H16N4
2-p-tolyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
—— 2-phenyl-5-p-chlorophenylpyrazolo[1,5-a]pyrimidin-7-amine —— C18H13ClN4
2-phenyl-5-p-chlorophenylpyrazolo[1,5-a]pyrimidin-7-amine
—— 2-phenyl-5-p-tolylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H16N4
2-phenyl-5-p-tolylpyrazolo[1,5-a]pyrimidin-7-amine
—— 2-phenyl-5-p-bromophenylpyrazolo[1,5-a]pyrimidin-7-amine —— C18H13BrN4
2-phenyl-5-p-bromophenylpyrazolo[1,5-a]pyrimidin-7-amine
—— 4-{4-[N-(N-tert-butoxycarbonylsarcosyl)amino]phenyl}-2-(2-difluoromethylbenzimidazol-1-yl)-6-morpholinopyrimidine —— C30H33F2N7O4
4-{4-[N-(N-tert-butoxycarbonylsarcosyl)amino]phenyl}-2-(2-difluoromethylbenzimidazol-1-yl)-6-morpholinopyrimidine
—— 4-{4-[N-(N-tert-butoxycarbonylsarcosyl)amino]-3-fluorophenyl}-2-(2-difluoromethylbenzimidazol-1-yl)-6-morpholinopyrimidine —— C30H32F3N7O4
4-{4-[N-(N-tert-butoxycarbonylsarcosyl)amino]-3-fluorophenyl}-2-(2-difluoromethylbenzimidazol-1-yl)-6-morpholinopyrimidine
—— 4-amino-6-phenylpyrimidin-2(1H)-one —— C10H9N3O
4-amino-6-phenylpyrimidin-2(1H)-one
—— 1,3-bis[3-(3,6-dimethyluracil-1-yl)propyl]thymine —— C23H30N6O6
1,3-bis[3-(3,6-dimethyluracil-1-yl)propyl]thymine
—— 7,13,21,24,25-pentamethyl-1,5,7,13,15,19-hexaazatetracyclo[17.3.1.1<sup>5,9</sup>.1<sup>11,15</sup>]pentacosa-9(24),11(25),21(22)-triene-6,8,12,14,20,23-hexaone —— C24H30N6O6
7,13,21,24,25-pentamethyl-1,5,7,13,15,19-hexaazatetracyclo[17.3.1.1<sup>5,9</sup>.1<sup>11,15</sup>]pentacosa-9(24),11(25),21(22)-triene-6,8,12,14,20,23-hexaone
—— 1,3-bis[6-(3,6-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)hexyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione —— C29H42N6O6
1,3-bis[6-(3,6-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)hexyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
—— 10,16,27,30,31-pentamethyl-1,8,10,16,18,25-hexaazatetracyclo[23.3.1.1<sup>8,12</sup>.1<sup>14,18</sup>]hentriaconta-12(30),14(31),25(28)-triene-9,11,15,17,25,29-hexaone —— C30H42N6O6
10,16,27,30,31-pentamethyl-1,8,10,16,18,25-hexaazatetracyclo[23.3.1.1<sup>8,12</sup>.1<sup>14,18</sup>]hentriaconta-12(30),14(31),25(28)-triene-9,11,15,17,25,29-hexaone
—— 6-(2,3-difluorophenoxy)-3-(4-methoxyphenyl)-4-phenylpyridazine —— C23H16F2N2O2
6-(2,3-difluorophenoxy)-3-(4-methoxyphenyl)-4-phenylpyridazine
—— 1-{[(4-amino-4-methylpentyl)oxy]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione —— C11H19N3O3
1-{[(4-amino-4-methylpentyl)oxy]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
—— 3,4-bis(4-methoxyphenyl)-6-(2,3-difluorophenoxy)pyridazine —— C24H18F2N2O3
3,4-bis(4-methoxyphenyl)-6-(2,3-difluorophenoxy)pyridazine
—— 1-[3-(piperidin-1-yl)propyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione —— C12H19N3O2
1-[3-(piperidin-1-yl)propyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
—— tert-butyl 5,6-dimethyl-2,4-dioxo-3-({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,2,3,4-tetrahydropyrimidine-1-carboxylate —— C26H37N3O5
tert-butyl 5,6-dimethyl-2,4-dioxo-3-({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,2,3,4-tetrahydropyrimidine-1-carboxylate
—— tert-butyl 2,4-dioxo-3-(4-(3-(piperidin-1-yl)propoxy)benzyl)-3,4-dihydropyrimidine-1(2H)-carboxylate —— C24H33N3O5
tert-butyl 2,4-dioxo-3-(4-(3-(piperidin-1-yl)propoxy)benzyl)-3,4-dihydropyrimidine-1(2H)-carboxylate
—— tert-butyl 5-methyl-2,4-dioxo-3-({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,2,3,4-tetrahydropyrimidine-1-carboxylate —— C25H35N3O5
tert-butyl 5-methyl-2,4-dioxo-3-({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,2,3,4-tetrahydropyrimidine-1-carboxylate
—— 5-Cyano-3-ethyl-1-methyl-6-phenyl-2-thiouracil —— C14H13N3OS
5-Cyano-3-ethyl-1-methyl-6-phenyl-2-thiouracil
—— 5-Cyano-1-ethyl-3-methyl-6-phenyl-2-thiouracil —— C14H13N3OS
5-Cyano-1-ethyl-3-methyl-6-phenyl-2-thiouracil
—— 3-Benzyl-5-cyano-1-methyl-6-phenyl-2-thiouracil —— C19H15N3OS
3-Benzyl-5-cyano-1-methyl-6-phenyl-2-thiouracil
—— 1-Benzyl-5-cyano-3-methyl-6-phenyl-2-thiouracil —— C19H15N3OS
1-Benzyl-5-cyano-3-methyl-6-phenyl-2-thiouracil
—— 5-cyano-1,3-diallyl-6-phenyl-2-thiouracil —— C17H15N3OS
5-cyano-1,3-diallyl-6-phenyl-2-thiouracil