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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-4-methyl-4-[(R)-(2-methyl-1H-indol-3-yl)-[3-(trifluoromethyl)phenyl]methyl]-2-phenyl-1,3-oxazol-5-one 1443445-30-4 C27H21F3N2O2
(4S)-4-methyl-4-[(R)-(2-methyl-1H-indol-3-yl)-[3-(trifluoromethyl)phenyl]methyl]-2-phenyl-1,3-oxazol-5-one
—— Dimethyl <Hydroxy-(3-pyridazinyl)methyl>malonate 130823-24-4 C10H12N2O5
Dimethyl <Hydroxy-(3-pyridazinyl)methyl>malonate
—— 2-(4-(4,7-dimethylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)acetic acid 1158970-15-0 C16H15N3O2S
2-(4-(4,7-dimethylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)acetic acid
—— ethyl 3-[2-oxo-5-(trifluoromethyl)-2,3-dihydro-1H-benzimidazol-1-yl] benzoate 1106941-16-5 C17H13F3N2O3
ethyl 3-[2-oxo-5-(trifluoromethyl)-2,3-dihydro-1H-benzimidazol-1-yl] benzoate
—— (R)-2-(N-(2-azidoethyl)-4-methoxyphenylsulfonamido)-N-hydroxy-3-methylbutanamide 1449846-45-0 C14H21N5O5S
(R)-2-(N-(2-azidoethyl)-4-methoxyphenylsulfonamido)-N-hydroxy-3-methylbutanamide
—— 2-[1-[4-(2-ethoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-ethyl]-5-fluoro-1H-pyrrolo[2,3-b]pyridine 1312019-74-1 C24H29FN2O4S
2-[1-[4-(2-ethoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-ethyl]-5-fluoro-1H-pyrrolo[2,3-b]pyridine
—— Dimethyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate 130823-27-7 C15H17N3O4
Dimethyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate
—— diphenyldipropynylmethane 1095216-83-3 C19H16
diphenyldipropynylmethane
—— 1-benzenesulfonyl-5-fluoro-2-{1-[4-(2-methoxy-ethanesulfonyl)-phenyl]-3-methyl-but-1-enyl}-1H-pyrrolo[2,3-b]pyridine 1312019-92-3 C27H27FN2O5S2
1-benzenesulfonyl-5-fluoro-2-{1-[4-(2-methoxy-ethanesulfonyl)-phenyl]-3-methyl-but-1-enyl}-1H-pyrrolo[2,3-b]pyridine
—— 1-benzenesulfonyl-5-fluoro-2-[1-[4-(2-methoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-vinyl]-1H-pyrrolo[2,3-b]pyridine 1312019-72-9 C29H29FN2O6S2
1-benzenesulfonyl-5-fluoro-2-[1-[4-(2-methoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-vinyl]-1H-pyrrolo[2,3-b]pyridine
—— 2-[1-[4-(2-ethoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-vinyl]-5-fluoro-1H-pyrrolo[2,3-b]pyridine 1312019-73-0 C24H27FN2O4S
2-[1-[4-(2-ethoxy-ethanesulfonyl)-phenyl]-2-(tetrahydro-pyran-4-yl)-vinyl]-5-fluoro-1H-pyrrolo[2,3-b]pyridine
—— 4-(1-cyanoethyl)phenyl 4-methylbenzenesulfonate 1309660-23-8 C16H15NO3S
4-(1-cyanoethyl)phenyl 4-methylbenzenesulfonate
—— Dimethyl 2-[(2-phenylindol-1-yl)methylidene]propanedioate 1208105-33-2 C20H17NO4
Dimethyl 2-[(2-phenylindol-1-yl)methylidene]propanedioate
—— 2-{4-[1-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-(tetrahydro-pyran-4-yl)-ethyl]-benzenesulfonyl}-ethanol 1312017-21-2 C22H25FN2O4S
2-{4-[1-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-2-yl)-2-(tetrahydro-pyran-4-yl)-ethyl]-benzenesulfonyl}-ethanol
—— 4-chloro-2-[(4,6-dibromo-2-methylpyridin-3-yl)oxy]-7-(1-ethylpropyl)-1-methyl-1H-benzimidazole 1022249-93-9 C19H20Br2ClN3O
4-chloro-2-[(4,6-dibromo-2-methylpyridin-3-yl)oxy]-7-(1-ethylpropyl)-1-methyl-1H-benzimidazole
—— 3β-hydroxyandrosta-1,5-dien-17-one 18088-27-2 C19H26O2
3β-hydroxyandrosta-1,5-dien-17-one
—— rac-1-(7-fluoro-2-methoxyquinolin-8-yl)ethane-1,2-diol 1442465-52-2 C12H12FNO3
rac-1-(7-fluoro-2-methoxyquinolin-8-yl)ethane-1,2-diol
—— methyl 4-phenyl-2-[(phenylsulfonyl)amino]-2-(trifluoromethyl)but-3-ynoate 1222169-90-5 C18H14F3NO4S
methyl 4-phenyl-2-[(phenylsulfonyl)amino]-2-(trifluoromethyl)but-3-ynoate
—— 4-ethylsulfanyl-2-methylphenol 18979-85-6 C9H12OS
4-ethylsulfanyl-2-methylphenol
—— 4-(2-methoxy-ethanesulfonyl)-phenylboronic acid 1312019-68-3 C9H13BO5S
4-(2-methoxy-ethanesulfonyl)-phenylboronic acid
—— 2-chloro-10-propylpyrimido[1,2-a]benzimidazol-4(10H)-one 1430744-91-4 C13H12ClN3O
2-chloro-10-propylpyrimido[1,2-a]benzimidazol-4(10H)-one
—— (S)-2-cyclohexyl-3-nitro-1-(pyridazin-3-yl)propan-1-one 1175052-24-0 C13H17N3O3
(S)-2-cyclohexyl-3-nitro-1-(pyridazin-3-yl)propan-1-one
—— 5-(4'-fluorophenyl)-2-[2-(dimethylamino)ethyl]-1H-benzo[de]isoquinoline-1,3(2H)-dione 1274673-38-9 C22H19FN2O2
5-(4'-fluorophenyl)-2-[2-(dimethylamino)ethyl]-1H-benzo[de]isoquinoline-1,3(2H)-dione
—— Ethyl Methyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate 130823-32-4 C16H19N3O4
Ethyl Methyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate
—— 1-pyridin-4-ylmethyl-1H-pyrazol-4-carboxylic acid [4-((R)-3-aminopiperidin-1-yl)-5-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]amide 1449321-43-0 C23H26N8O
1-pyridin-4-ylmethyl-1H-pyrazol-4-carboxylic acid [4-((R)-3-aminopiperidin-1-yl)-5-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl]amide
—— 4-(2-pyridylmethyl)thiosemicarbazide 142564-64-5 C7H10N4S
4-(2-pyridylmethyl)thiosemicarbazide
—— Diethyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate 130823-30-2 C17H21N3O4
Diethyl 2,6-Dimethyl-4-(3-pyridazinyl)-1,4-dihydropyridine-3,5-dicarboxylate
—— US10280167, Example 9 1434585-39-3 C15H14N8O
US10280167, Example 9
—— (3-(4-bromophenyl)-4,6-dimethoxy-1H-indol-2-yl)(5-(dimethylamino)-1,3,4-thiadiazol-2-yl) ketone 1569643-64-6 C21H19BrN4O3S
(3-(4-bromophenyl)-4,6-dimethoxy-1H-indol-2-yl)(5-(dimethylamino)-1,3,4-thiadiazol-2-yl) ketone
—— N-[3-[(4aS,7aS)-3-amino-2,2-dimethyl-1,1-dioxo-7,7a-dihydro-5H-furo[3,4-b][1,4]thiazin-4a-yl]-4-fluorophenyl]-5-fluoropyridine-2-carboxamide 1616109-45-5 C20H20F2N4O4S
N-[3-[(4aS,7aS)-3-amino-2,2-dimethyl-1,1-dioxo-7,7a-dihydro-5H-furo[3,4-b][1,4]thiazin-4a-yl]-4-fluorophenyl]-5-fluoropyridine-2-carboxamide
—— (R)-2-(N-(2-azidoethyl)-4-methylphenylsulfonamido)-N-hydroxy-3-methylbutanamide 1449846-46-1 C14H21N5O4S
(R)-2-(N-(2-azidoethyl)-4-methylphenylsulfonamido)-N-hydroxy-3-methylbutanamide
—— S-3-(3-cyclopentyloxy-4-methoxyphenyl)-3-[3-(5-methyl[1,2,4]oxadiazol-3-yl)phenylethynyl]propionic acid 188009-95-2 C26H26N2O5
S-3-(3-cyclopentyloxy-4-methoxyphenyl)-3-[3-(5-methyl[1,2,4]oxadiazol-3-yl)phenylethynyl]propionic acid
—— 2-Piperazin-1-yl-10-propylpyrimido[1,2-a]benzimidazol-4-one 1430745-07-5 C17H21N5O
2-Piperazin-1-yl-10-propylpyrimido[1,2-a]benzimidazol-4-one
—— 3-(7-bromo-1-oxo-1H-isoquinolin-2-yl)propionic acid 1519208-20-8 C12H10BrNO3
3-(7-bromo-1-oxo-1H-isoquinolin-2-yl)propionic acid
—— N-[3-[(4aS,7aS)-3-amino-2,2-dimethyl-1,1-dioxo-7,7a-dihydro-5H-furo[3,4-b][1,4]thiazin-4a-yl]-4-fluorophenyl]-1-methylpyrazole-3-carboxamide 1616109-49-9 C19H22FN5O4S
N-[3-[(4aS,7aS)-3-amino-2,2-dimethyl-1,1-dioxo-7,7a-dihydro-5H-furo[3,4-b][1,4]thiazin-4a-yl]-4-fluorophenyl]-1-methylpyrazole-3-carboxamide
—— (R)-2-(4-(2-fluoroethoxy)-N-(2-(4-(3-fluoropropyl)-1H-1,2,3-triazol-1-yl)ethyl)phenylsulfonamido)-N-hydroxy-3-methylbutanamide 1449846-56-3 C20H29F2N5O5S
(R)-2-(4-(2-fluoroethoxy)-N-(2-(4-(3-fluoropropyl)-1H-1,2,3-triazol-1-yl)ethyl)phenylsulfonamido)-N-hydroxy-3-methylbutanamide
—— iso-propylsulfonylethylamine 1179721-73-3 C5H13NO2S
iso-propylsulfonylethylamine
—— {[4-(3-Oxo-1-cyclopenten-1-yl)phenyl]thio}acetic acid ethyl ester 1211474-18-8 C15H16O3S
{[4-(3-Oxo-1-cyclopenten-1-yl)phenyl]thio}acetic acid ethyl ester
—— 2-(6'-aminopyridin-3-yl)-6-methylbenzothiazole 1448780-06-0 C13H11N3S
2-(6'-aminopyridin-3-yl)-6-methylbenzothiazole
—— (R,R)-N-(1-phenylethyl)-4-(2-chloro-4-fluorophenyl)-6-methyl-2-(2-thiazolyl)-1,4-dihydropyrimidin-5-carboxamide 1005459-66-4 C23H20ClFN4OS
(R,R)-N-(1-phenylethyl)-4-(2-chloro-4-fluorophenyl)-6-methyl-2-(2-thiazolyl)-1,4-dihydropyrimidin-5-carboxamide
—— 5-bromo-1-isopropyl-4-(chloromethyl)-1H-pyrazole 1407966-26-0 C7H10BrClN2
5-bromo-1-isopropyl-4-(chloromethyl)-1H-pyrazole
—— ethyl 6-N,N-diethylcarbamoyl-2-methylthiopyrazolo<1,5-a>pyridine-3-carboxylate 120590-43-4 C16H21N3O3S
ethyl 6-N,N-diethylcarbamoyl-2-methylthiopyrazolo<1,5-a>pyridine-3-carboxylate
—— N-(4-(phenylethynyl)pyridin-3-yl)-2,2-dimethylpropanamide 1021444-65-4 C18H18N2O
N-(4-(phenylethynyl)pyridin-3-yl)-2,2-dimethylpropanamide
—— (S)-2-{(4R,5S,6R)-6-[(2S,3R)-3-(tert-butyldimethylsilyloxy)-5-(4-methoxybenzyloxy)pentan-2-yl]-2,2,5-trimethyl-1,3-dioxan-4-yl}propan-1-ol 1180131-40-1 C29H52O6Si
(S)-2-{(4R,5S,6R)-6-[(2S,3R)-3-(tert-butyldimethylsilyloxy)-5-(4-methoxybenzyloxy)pentan-2-yl]-2,2,5-trimethyl-1,3-dioxan-4-yl}propan-1-ol
—— (3S,5S,6S)-1-[(3S)-1,4-dioxaspiro[4.5]decan-3-yl]-5-methoxy-8-[(4-methoxyphenyl)methoxy]-6-phenylmethoxyoct-1-yn-3-ol 1109289-88-4 C32H42O7
(3S,5S,6S)-1-[(3S)-1,4-dioxaspiro[4.5]decan-3-yl]-5-methoxy-8-[(4-methoxyphenyl)methoxy]-6-phenylmethoxyoct-1-yn-3-ol
—— (R)-2-(N-(2-(4-(3-fluoropropyl)-1H-1,2,3-triazol-1-yl)ethyl)-4-methylphenylsulfonamido)-N-hydroxy-3-methylbutanamide 1449846-53-0 C19H28FN5O4S
(R)-2-(N-(2-(4-(3-fluoropropyl)-1H-1,2,3-triazol-1-yl)ethyl)-4-methylphenylsulfonamido)-N-hydroxy-3-methylbutanamide
—— Trimethyl-(1-methylene-hept-2-ynyloxy)-silane 109283-55-8 C11H20OSi
Trimethyl-(1-methylene-hept-2-ynyloxy)-silane
—— 3-(6-(3-Hydroxy-1,5-undecadienyl)-2-pyridinyl)-oxiranebutanol 118867-16-6 C22H33NO3
3-(6-(3-Hydroxy-1,5-undecadienyl)-2-pyridinyl)-oxiranebutanol
—— (R)-2-(N-(2-azidoethyl)-4-(2-fluoroethoxy)phenylsulfonamido)-N-hydroxy-3-methylbutanamide 1449846-47-2 C15H22FN5O5S
(R)-2-(N-(2-azidoethyl)-4-(2-fluoroethoxy)phenylsulfonamido)-N-hydroxy-3-methylbutanamide
—— 4-O-[2-azido-2-deoxy-3,4-O-isopropylidene-6-O-(1-methoxy-1-methylethyl)-β-D-galactopyranosyl]-2,3:5,6-di-O-isopropylidene-aldehydo-D-glucose dimethyl acetate 1139852-85-9 C27H47N3O12
4-O-[2-azido-2-deoxy-3,4-O-isopropylidene-6-O-(1-methoxy-1-methylethyl)-β-D-galactopyranosyl]-2,3:5,6-di-O-isopropylidene-aldehydo-D-glucose dimethyl acetate