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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-{[1-benzyl-3-(2-dimethylamino-pyrimidin-5-yl)-5-hydroxy-2-oxo-1,2-dihydro-[1,7]naphthyridine-6-carbonyl]-amino}-propionic acid 1392843-20-7 C25H24N6O5
3-{[1-benzyl-3-(2-dimethylamino-pyrimidin-5-yl)-5-hydroxy-2-oxo-1,2-dihydro-[1,7]naphthyridine-6-carbonyl]-amino}-propionic acid
—— rac-2-[(4-Fluoro-benzylamino)-methyl]-3,3-dimethyl-butyric Acid Ethyl Ester 1198470-67-5 C16H24FNO2
rac-2-[(4-Fluoro-benzylamino)-methyl]-3,3-dimethyl-butyric Acid Ethyl Ester
—— N-[1-(2-naphthyl)ethyl]cyclopropylamine hydrochloride 1197803-63-6 C15H17N*ClH
N-[1-(2-naphthyl)ethyl]cyclopropylamine hydrochloride
—— 3-((Z)-((Z)-5-(4-(carboxymethoxy)benzylidene)-3-allyl-4-oxothiazolidin-2-ylidene)amino)benzoic acid 1448677-91-5 C22H18N2O6S
3-((Z)-((Z)-5-(4-(carboxymethoxy)benzylidene)-3-allyl-4-oxothiazolidin-2-ylidene)amino)benzoic acid
—— 1-methyl-3-undecynylamine 138769-82-1 C12H23N
1-methyl-3-undecynylamine
—— N-[(E)-(2R,3R,6S)-3-Benzyl-2-hydroxy-6-methanesulfonylamino-7-(naphthalene-2-sulfinyl)-hept-4-enyl]-N-isobutyl-4-nitro-benzenesulfonamide 1026361-93-2 C35H41N3O8S3
N-[(E)-(2R,3R,6S)-3-Benzyl-2-hydroxy-6-methanesulfonylamino-7-(naphthalene-2-sulfinyl)-hept-4-enyl]-N-isobutyl-4-nitro-benzenesulfonamide
—— 3-ethoxycarbonyl-4-(4-fluorophenyl)-4-(4-methanesulphonylphenyl)-3-butenoic acid 197439-12-6 C20H19FO6S
3-ethoxycarbonyl-4-(4-fluorophenyl)-4-(4-methanesulphonylphenyl)-3-butenoic acid
—— N<sup>3</sup>-[3,5-dichloro-4-(4-methanesulfonylphenoxy)phenyl]-1H-[1,2,4]triazole-3,5-diamine 1620782-69-5 C15H13Cl2N5O3S
N<sup>3</sup>-[3,5-dichloro-4-(4-methanesulfonylphenoxy)phenyl]-1H-[1,2,4]triazole-3,5-diamine
—— 1-(2,2-dimethylpyrrolidin-1-yl)ethan-1-one 1039553-82-6 C8H15NO
1-(2,2-dimethylpyrrolidin-1-yl)ethan-1-one
—— N-(4-fluorobenzyl)-6-fluoro-3-hydroxy-2-oxoquinoline-4-carboxamide 1383628-00-9 C17H12F2N2O3
N-(4-fluorobenzyl)-6-fluoro-3-hydroxy-2-oxoquinoline-4-carboxamide
—— 2-[3-Methoxy-4-(4-methyl-imidazol-1-yl)-phenylamino]-thiazole-4-carboxylic acid 4-fluoro-benzylamide 1225445-45-3 C22H20FN5O2S
2-[3-Methoxy-4-(4-methyl-imidazol-1-yl)-phenylamino]-thiazole-4-carboxylic acid 4-fluoro-benzylamide
—— 4-[4-(4-methanesulfonyl-phenoxy)-3-methyl-pyrazolo[3,4-d]pyrimidin-1-yl]-piperidine-1-carboxylic acid isopropyl ester 1196484-86-2 C22H27N5O5S
4-[4-(4-methanesulfonyl-phenoxy)-3-methyl-pyrazolo[3,4-d]pyrimidin-1-yl]-piperidine-1-carboxylic acid isopropyl ester
—— methyl 2-(3-(tert-butoxycarbonyl(methyl)amino)-6-(1-(tert-butyldimethylsilyloxy)propyl)tetrahydro-2-H-pyran-3-yl)-5,6-dihydroxypyrimidine-4-carboxylate 1239019-53-4 C26H45N3O8Si
methyl 2-(3-(tert-butoxycarbonyl(methyl)amino)-6-(1-(tert-butyldimethylsilyloxy)propyl)tetrahydro-2-H-pyran-3-yl)-5,6-dihydroxypyrimidine-4-carboxylate
—— 2-((3,5-dichlorophenoxy) methyl)-4-(4-fluorophenyl)-5-(4-methylthiophenyl)thiazole 177561-26-1 C23H16Cl2FNOS2
2-((3,5-dichlorophenoxy) methyl)-4-(4-fluorophenyl)-5-(4-methylthiophenyl)thiazole
—— 2-[4-(tert-butyldimethylsilanyloxy)benzenesulfonyl]-1-(4-morpholin-4-ylmethylphenyl)ethanol 1354657-81-0 C25H37NO5SSi
2-[4-(tert-butyldimethylsilanyloxy)benzenesulfonyl]-1-(4-morpholin-4-ylmethylphenyl)ethanol
—— 3,6-diphenyl-4,5-diaza-9,9'-spirobifluorene 1404084-16-7 C35H22N2
3,6-diphenyl-4,5-diaza-9,9'-spirobifluorene
—— rac-2-[(4-fluoro-benzylamino)-methyl]-pentanoic acid ethyl ester 1198470-69-7 C15H22FNO2
rac-2-[(4-fluoro-benzylamino)-methyl]-pentanoic acid ethyl ester
—— 1-[(1S,2S)-4,6-dichloro-1-(4-methanesulfonylphenoxy)indan-2-yl]-4-methylpiperazine 1215274-53-5 C21H24Cl2N2O3S
1-[(1S,2S)-4,6-dichloro-1-(4-methanesulfonylphenoxy)indan-2-yl]-4-methylpiperazine
—— 8-Methyl-2,3,4,5-tetrahydro-cyclopenta[a]naphthalen-1-one 158389-54-9 C14H14O
8-Methyl-2,3,4,5-tetrahydro-cyclopenta[a]naphthalen-1-one
—— INCB-057643 1820889-23-3 C20H21N3O5S
INCB-057643
—— N-(3-amino-3-oxopropyl)-5-chloro-3-[(3,5-dimethylphenyl)-sulfonyl]-4-fluoro-1H-indole-2-carboxamide 1140947-98-3 C20H19ClFN3O4S
N-(3-amino-3-oxopropyl)-5-chloro-3-[(3,5-dimethylphenyl)-sulfonyl]-4-fluoro-1H-indole-2-carboxamide
—— {4-[5-(4-fluoro-phenyl)-[1,3,4]oxadiazol-2-yl]-piperidin-1-yl}-acetic acid 1419961-09-3 C15H16FN3O3
{4-[5-(4-fluoro-phenyl)-[1,3,4]oxadiazol-2-yl]-piperidin-1-yl}-acetic acid
—— 4-{[(4-fluorophenyl)methyl]amino}-3-nitro-N-[(1R)-1-phenylpropyl]benzamide 1168138-57-5 C23H22FN3O3
4-{[(4-fluorophenyl)methyl]amino}-3-nitro-N-[(1R)-1-phenylpropyl]benzamide
—— 2-(3-{4-[(R)-3-(4-methanesulfonylphenoxy)-1-methylpropyl]piperidin-1-yl}-[1,2,4]oxadiazol-5-yl)pyrrolidine-1-carboxylic acid tert-butyl ester 1204301-99-4 C27H40N4O6S
2-(3-{4-[(R)-3-(4-methanesulfonylphenoxy)-1-methylpropyl]piperidin-1-yl}-[1,2,4]oxadiazol-5-yl)pyrrolidine-1-carboxylic acid tert-butyl ester
—— [4-(4-benzyloxy-benzoyl)-piperidin-1-yl]-acetic acid ethyl ester 1419960-52-3 C23H27NO4
[4-(4-benzyloxy-benzoyl)-piperidin-1-yl]-acetic acid ethyl ester
—— ethyl 2-(1-(tert-butyl)-2-(5-fluoro-2-(5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)acetate 1422052-43-4 C20H22F4N6O2
ethyl 2-(1-(tert-butyl)-2-(5-fluoro-2-(5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)acetate
—— rac-2-cyclopentyl-3-(4-fluoro-benzylamino)-propionic acid ethyl ester 1198470-70-0 C17H24FNO2
rac-2-cyclopentyl-3-(4-fluoro-benzylamino)-propionic acid ethyl ester
—— 1-(3-fluorophenyl)-2-[4-(methylsulfanyl)phenyl]-1-ethanone 177560-78-0 C15H13FOS
1-(3-fluorophenyl)-2-[4-(methylsulfanyl)phenyl]-1-ethanone
—— N-[1-[(1-methylethyl)sulfonyl]-1H-indazol-5-yl]-2-(3-methyl-1-piperidinyl)-4-(trifluoromethyl)-5-oxazolecarboxamide 1227932-44-6 C21H24F3N5O4S
N-[1-[(1-methylethyl)sulfonyl]-1H-indazol-5-yl]-2-(3-methyl-1-piperidinyl)-4-(trifluoromethyl)-5-oxazolecarboxamide
—— 1-(6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-yl)-3-ethylurea 1452478-28-2 C18H18Cl2N2O3
1-(6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-yl)-3-ethylurea
—— (E)-3-[(1S,2S,3R)-2-((S)-Cyano-methyl-methyl)-3-methyl-cyclohexyl]-2-((2R,3R,6S)-6-{(E)-(S)-3-[(2R,3S,5R)-5-((S)-1-methoxy-ethyl)-3-methyl-tetrahydro-furan-2-yl]-but-1-enyl}-3-methyl-tetrahydro-pyran-2-yl)-acrylic acid methyl ester 149298-92-0 C32H51NO5
(E)-3-[(1S,2S,3R)-2-((S)-Cyano-methyl-methyl)-3-methyl-cyclohexyl]-2-((2R,3R,6S)-6-{(E)-(S)-3-[(2R,3S,5R)-5-((S)-1-methoxy-ethyl)-3-methyl-tetrahydro-furan-2-yl]-but-1-enyl}-3-methyl-tetrahydro-pyran-2-yl)-acrylic acid methyl ester
—— 2-(1-(tert-butyl)-2-(5-fluoro-2-(5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)acetic acid 1422051-30-6 C18H18F4N6O2
2-(1-(tert-butyl)-2-(5-fluoro-2-(5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)acetic acid
—— 5-(benzyloxy)-N-(4-fluorobenzyl)-4-(hydroxymethyl)-6-methylnicotinamide 1198621-07-6 C22H21FN2O3
5-(benzyloxy)-N-(4-fluorobenzyl)-4-(hydroxymethyl)-6-methylnicotinamide
—— 4-(4-chloro-6-methoxy-pyrazolo[3,4-d]pyrimidin-1-yl)-piperidine-1-carboxylic acid tert-butyl ester 1196487-16-7 C16H22ClN5O3
4-(4-chloro-6-methoxy-pyrazolo[3,4-d]pyrimidin-1-yl)-piperidine-1-carboxylic acid tert-butyl ester
—— 1,1,1-tris[(4,5-diazafluoren-9-yliminoxy)methyl]propane 1263210-89-4 C39H29N9O3
1,1,1-tris[(4,5-diazafluoren-9-yliminoxy)methyl]propane
—— 2-(3-[2-(1,4-dioxan-2-yl)ethyl]-5-{3-ethyl-4-[(triisopropylsilyl)ethynyl]phenyl}-3H-1,2,3-triazol-4-yl)propan-2-ol 1307854-42-7 C30H47N3O3Si
2-(3-[2-(1,4-dioxan-2-yl)ethyl]-5-{3-ethyl-4-[(triisopropylsilyl)ethynyl]phenyl}-3H-1,2,3-triazol-4-yl)propan-2-ol
—— 6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-amine 1452479-70-7 C15H13Cl2NO2
6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-amine
—— 4-(((2R,11aS)-2-hydroxy-5,11-dioxo-2,3,11,11a-tetrahydro-1H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10(5H)-yl)methyl)benzoic acid 1447533-97-2 C20H18N2O5
4-(((2R,11aS)-2-hydroxy-5,11-dioxo-2,3,11,11a-tetrahydro-1H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10(5H)-yl)methyl)benzoic acid
—— trans-Dimethoxycyclopentan 176298-26-3 C7H14O2
trans-Dimethoxycyclopentan
—— 1-[(1S,2S)-4,6-dichloro-1-(4-methanesulfonylphenoxy)indan-2-yl]-4-methyl-1,4-diazepane 1215274-52-4 C22H26Cl2N2O3S
1-[(1S,2S)-4,6-dichloro-1-(4-methanesulfonylphenoxy)indan-2-yl]-4-methyl-1,4-diazepane
—— 1-methyl-4-(4-(methylthio)phenyl)-5-phenyl-1H-imidazole-2(3H)-thione 1446909-33-6 C17H15FN2S2
1-methyl-4-(4-(methylthio)phenyl)-5-phenyl-1H-imidazole-2(3H)-thione
—— Pyrazolo[3,4-b]quinolin-1-yl-acetic acid [3-allyl-4-phenyl-3H-thiazol-(2Z)-ylidene]-hydrazide 132719-78-9 C24H20N6OS
Pyrazolo[3,4-b]quinolin-1-yl-acetic acid [3-allyl-4-phenyl-3H-thiazol-(2Z)-ylidene]-hydrazide
—— 4-[4-(4-methanesulfonylphenoxymethyl)-5-methylthiazol-2-yl]piperidine-1-carboxylic acid tert-butyl ester 1037792-99-6 C22H30N2O5S2
4-[4-(4-methanesulfonylphenoxymethyl)-5-methylthiazol-2-yl]piperidine-1-carboxylic acid tert-butyl ester
—— {1-[10-(1-Ethoxycarbonylmethyl-cyclopropyl)-decyl]-cyclopropyl}-acetic acid ethyl ester 1365571-68-1 C24H42O4
{1-[10-(1-Ethoxycarbonylmethyl-cyclopropyl)-decyl]-cyclopropyl}-acetic acid ethyl ester
—— ethyl N-(6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-yl)glycinate 1452478-37-3 C19H19Cl2NO4
ethyl N-(6-((2,4-dichlorobenzyl)oxy)-2,3-dihydro-1-benzofuran-3-yl)glycinate
—— 2-chloro-5-(4-methanesulfonylphenoxymethyl)pyrazine 1318791-32-0 C12H11ClN2O3S
2-chloro-5-(4-methanesulfonylphenoxymethyl)pyrazine
—— 2-{3-[4-((R)-3-hydroxy-1-methylpropyl)piperidin-1-yl]-[1,2,4]oxadiazol-5-yl}pyrrolidine-1-carboxylic acid tert-butyl ester 1204301-98-3 C20H34N4O4
2-{3-[4-((R)-3-hydroxy-1-methylpropyl)piperidin-1-yl]-[1,2,4]oxadiazol-5-yl}pyrrolidine-1-carboxylic acid tert-butyl ester
—— 4-chloro-6-(6-methoxypyridin-3-yl)-1-methyl-1H-pyrazolo[3,4-b]pyridine 1227089-98-6 C13H11ClN4O
4-chloro-6-(6-methoxypyridin-3-yl)-1-methyl-1H-pyrazolo[3,4-b]pyridine
—— ethyl 2-(1-tert-butyl-2-(2-chloro-5-fluoropyrimidin-4-yl)hydrazinyl)ethanoate 1422052-41-2 C12H18ClFN4O2
ethyl 2-(1-tert-butyl-2-(2-chloro-5-fluoropyrimidin-4-yl)hydrazinyl)ethanoate
—— ethyl 2-(1-tert-butyl-2-(5-fluoro-2-(1-tosyl-5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)ethanoate 1422052-42-3 C27H28F4N6O4S
ethyl 2-(1-tert-butyl-2-(5-fluoro-2-(1-tosyl-5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl)hydrazinyl)ethanoate