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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,4-bis(4-phenoxyphenyl)pyridine 1285694-81-6 C29H21NO2
2,4-bis(4-phenoxyphenyl)pyridine
—— 1,5-bis(tert-butyldimethylsilyl)-3-chloropenta-1,4-diyne 1198424-85-9 C17H31ClSi2
1,5-bis(tert-butyldimethylsilyl)-3-chloropenta-1,4-diyne
—— dimethoxyethyl-1,4-dihydro-2,6-dimethyl-4-[2-methylthio-1-(phenylamino)-1H-imidazole-5-yl]-3,5-pyridinedicarboxylate 1345674-63-6 C25H32N4O6S
dimethoxyethyl-1,4-dihydro-2,6-dimethyl-4-[2-methylthio-1-(phenylamino)-1H-imidazole-5-yl]-3,5-pyridinedicarboxylate
—— 6-bromo-3-methylpyrimidin-4(3H)-one 1611464-74-4 C5H5BrN2O
6-bromo-3-methylpyrimidin-4(3H)-one
—— 4-[2-((1S,3S)-3-acetylamino-cyclopentyloxy)-4-fluoro-phenylamino]-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid 1332634-75-9 C21H21FN4O4S
4-[2-((1S,3S)-3-acetylamino-cyclopentyloxy)-4-fluoro-phenylamino]-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid
—— 4-chloro-2-fluoro-5-(1-ethoxycarbonylethoxy)phenyl isothiocyanate 102800-69-1 C12H11ClFNO3S
4-chloro-2-fluoro-5-(1-ethoxycarbonylethoxy)phenyl isothiocyanate
—— ethyl 1-amino-3-p-tolyl-2-naphthoate 1609162-34-6 C20H19NO2
ethyl 1-amino-3-p-tolyl-2-naphthoate
—— 2-(5-p-tolyl-2H-1,2,3-triazol-4-yl)benzonitrile 1192716-89-4 C16H12N4
2-(5-p-tolyl-2H-1,2,3-triazol-4-yl)benzonitrile
—— (1S)-1-(hydroxymethyl)-6-methyl-1,2,5,6-tetrahydro-4H,9H-imidazo[1,2,3-ij]-1,8-naphthyridine-4,9-dione 1221721-46-5 C12H14N2O3
(1S)-1-(hydroxymethyl)-6-methyl-1,2,5,6-tetrahydro-4H,9H-imidazo[1,2,3-ij]-1,8-naphthyridine-4,9-dione
—— 4-[2-((1S,3S)-3-acetylamino-cyclopentyloxy)-4-fluoro-phenylamino]-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid methyl ester 1332634-74-8 C22H23FN4O4S
4-[2-((1S,3S)-3-acetylamino-cyclopentyloxy)-4-fluoro-phenylamino]-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid methyl ester
—— 1,1-dimethylethyl (1-{[(1R)-6-methyl-4,9-dioxo-1,2-dihydro-4H,9H-imidazo[1,2,3-ij]-1,8-naphthyridin-1-yl]methyl}-4-piperidinyl)carbamate 1221721-49-8 C22H30N4O4
1,1-dimethylethyl (1-{[(1R)-6-methyl-4,9-dioxo-1,2-dihydro-4H,9H-imidazo[1,2,3-ij]-1,8-naphthyridin-1-yl]methyl}-4-piperidinyl)carbamate
—— 4,4,7,7,11,11-hexanitropentacyclo<6.3.0.0<sup>2,6</sup>.0<sup>3,10</sup>.0<sup>5,9</sup>>undecane 110270-87-6 C11H8N6O12
4,4,7,7,11,11-hexanitropentacyclo<6.3.0.0<sup>2,6</sup>.0<sup>3,10</sup>.0<sup>5,9</sup>>undecane
—— 1-({5-chloro-2-[(phenylmethyl)oxy]phenyl}methyl)-4-nitro-1H-pyrazole 1373394-95-6 C17H14ClN3O3
1-({5-chloro-2-[(phenylmethyl)oxy]phenyl}methyl)-4-nitro-1H-pyrazole
—— (S)-tert-butyl 1-(1-(5-ethylpyrimidin-2-yl)piperidin-4-yl)-2-oxopyrrolidin-3-ylcarbamate 1351168-12-1 C20H31N5O3
(S)-tert-butyl 1-(1-(5-ethylpyrimidin-2-yl)piperidin-4-yl)-2-oxopyrrolidin-3-ylcarbamate
—— 2-methoxy-5-(3-(piperidin-1-yl)propoxy)aniline 1258492-32-8 C15H24N2O2
2-methoxy-5-(3-(piperidin-1-yl)propoxy)aniline
—— Trifluoro-methanesulfonic acid 3-biphenyl-4-ylmethyl-4-oxo-chroman-7-yl ester 179107-69-8 C23H17F3O5S
Trifluoro-methanesulfonic acid 3-biphenyl-4-ylmethyl-4-oxo-chroman-7-yl ester
—— 4-(4-aminopiperidin-1-yl)-2,2-diphenylbutanenitrile 1412903-11-7 C21H25N3
4-(4-aminopiperidin-1-yl)-2,2-diphenylbutanenitrile
—— ethyl {3-chloro-4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetate 1004513-88-5 C26H22ClF2NO6
ethyl {3-chloro-4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetate
—— 6-(4-nitrophenyl)-1-tosylpiperidine-2,4-dione 1186526-43-1 C18H16N2O6S
6-(4-nitrophenyl)-1-tosylpiperidine-2,4-dione
—— 4-(4-phenylpiperazin-1-yl)isoquinoline-6-carboxamide 1235380-73-0 C20H20N4O
4-(4-phenylpiperazin-1-yl)isoquinoline-6-carboxamide
—— N<sup>3</sup>-(4-methoxyfumaroyl)-L-2,3-diaminopropanoyl-UPOC 130905-37-2 C18H23N5O11
N<sup>3</sup>-(4-methoxyfumaroyl)-L-2,3-diaminopropanoyl-UPOC
—— methyl 1-amino-3-(4-methylphenyl)-2-naphthoate 1581713-36-1 C19H17NO2
methyl 1-amino-3-(4-methylphenyl)-2-naphthoate
—— 2-benzyl-5-methoxy-4-[4-(trifluoromethyl)phenyl]-pyridazin-3(2H)-one 1345839-36-2 C19H15F3N2O2
2-benzyl-5-methoxy-4-[4-(trifluoromethyl)phenyl]-pyridazin-3(2H)-one
—— 4-(2-hydroxyethyl)-5-methyl-2-(3-methylphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-one 1001077-44-6 C12H15N3O2
4-(2-hydroxyethyl)-5-methyl-2-(3-methylphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-one
—— (1S,3S,5R)-2-(tert-butoxycarbonyl)-6,6-difluoro-2-azabicyclo[3.1.0]hexane-3-carboxylic acid 1400990-36-4 C11H15F2NO4
(1S,3S,5R)-2-(tert-butoxycarbonyl)-6,6-difluoro-2-azabicyclo[3.1.0]hexane-3-carboxylic acid
—— bis-(fluorodiphenylsilyl)mercury 104925-64-6 C24H20F2HgSi2
bis-(fluorodiphenylsilyl)mercury
—— Eptastigmine tartrate 121652-76-4 C25H39N3O8
Eptastigmine tartrate
—— (8S)-2-(morpholin-4-yl)-8-(trifluoromethyl)-9-[4-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one 1260585-58-7 C19H18F6N4O2
(8S)-2-(morpholin-4-yl)-8-(trifluoromethyl)-9-[4-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one
—— N-((R)-((S)-3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide 1398511-76-6 C18H14Cl2N2O6S
N-((R)-((S)-3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide
—— ethyl {4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-3-fluorophenyl}acetate 1004513-80-7 C26H22F3NO6
ethyl {4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-3-fluorophenyl}acetate
—— 6-Bromo-2-(phenylsulfonyl)-2,3-dihydroisoquinoline-4(1H)-one 1235382-79-2 C15H12BrNO3S
6-Bromo-2-(phenylsulfonyl)-2,3-dihydroisoquinoline-4(1H)-one
—— 2-(4-nitrophenyl)-4-phenylsulfonyl-1-tosyl-2,5-dihydro-1H-pyrrole 1192593-18-2 C23H20N2O6S2
2-(4-nitrophenyl)-4-phenylsulfonyl-1-tosyl-2,5-dihydro-1H-pyrrole
—— ethyl (3-chloro-4-{4-(ethyloxy)-3-hydroxy-1-oxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetate 1004514-44-6 C26H23ClF3NO6
ethyl (3-chloro-4-{4-(ethyloxy)-3-hydroxy-1-oxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetate
—— (Z,Z)-5-(3-chloro-4-hydroxybenzylidene)-2-isopropylimino-3-m-tolyl-thiazolidin-4-one 1228116-92-4 C20H19ClN2O2S
(Z,Z)-5-(3-chloro-4-hydroxybenzylidene)-2-isopropylimino-3-m-tolyl-thiazolidin-4-one
—— Example 41 1347434-80-3 C26H28ClF3N2O3S
Example 41
—— 2-cyclopropyl-propane-1,2-diamine 1021392-54-0 C6H14N2
2-cyclopropyl-propane-1,2-diamine
—— methyl 1-amino-3-(2-methylphenyl)-2-naphthoate 1581713-37-2 C19H17NO2
methyl 1-amino-3-(2-methylphenyl)-2-naphthoate
—— 6-(furan-2-yl)-1-tosylpiperidine-2,4-dione 1186526-48-6 C16H15NO5S
6-(furan-2-yl)-1-tosylpiperidine-2,4-dione
—— (3-chloro-4-{1,3-dioxo-4,9-bis[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid 1004514-36-6 C24H14ClF6NO6
(3-chloro-4-{1,3-dioxo-4,9-bis[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid
—— 1-{5-[2-oxo-2-(4-trifluoromethylphenyl)ethyl]furan-2-yl}propan-2-one 1195869-76-1 C16H13F3O3
1-{5-[2-oxo-2-(4-trifluoromethylphenyl)ethyl]furan-2-yl}propan-2-one
—— (4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}-3-fluorophenyl)acetic acid 1004514-40-2 C24H17F4NO6
(4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}-3-fluorophenyl)acetic acid
—— methyl 3-((tert-butyldimethylsilyl)oxy)-2-(N-(prop-2-yn-1-yl)vinylsulfonamido)propanoate 1357283-08-9 C15H27NO5SSi
methyl 3-((tert-butyldimethylsilyl)oxy)-2-(N-(prop-2-yn-1-yl)vinylsulfonamido)propanoate
—— (4R,5S)-4-(methoxycarbonyl)-5-(4-nitrophenyl)-N-tosyl-2-imidazoline 1245746-93-3 C18H17N3O6S
(4R,5S)-4-(methoxycarbonyl)-5-(4-nitrophenyl)-N-tosyl-2-imidazoline
—— 3-(2-(2,2,2-trifluoroethoxy)-phenyl)-4-fluorobenzoic acid 1055983-96-4 C15H10F4O3
3-(2-(2,2,2-trifluoroethoxy)-phenyl)-4-fluorobenzoic acid
—— (S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-diphenylcyclopent-1-enyl)methyl)benzenesulfonamide 1397711-83-9 C31H26N2O5S
(S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-diphenylcyclopent-1-enyl)methyl)benzenesulfonamide
—— 4-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole 1257078-38-8 C9H14N4O2
4-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole
—— (S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-bis(4-(trifluoromethyl)phenyl)cyclopent-1-enyl)methyl)benzenesulfonamide 1397711-97-5 C33H24F6N2O5S
(S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-bis(4-(trifluoromethyl)phenyl)cyclopent-1-enyl)methyl)benzenesulfonamide
—— ethyl 6-methyl-5-{[(4-methylphenyl)sulfonyl]amino}-4-oxo-5-azaspiro[2.4]hept-6-ene-7-carboxylate 1177445-87-2 C17H20N2O5S
ethyl 6-methyl-5-{[(4-methylphenyl)sulfonyl]amino}-4-oxo-5-azaspiro[2.4]hept-6-ene-7-carboxylate
—— 4-[(4-nitro-1H-pyrazol-1-yl)methyl]pyridine 1006571-33-0 C9H8N4O2
4-[(4-nitro-1H-pyrazol-1-yl)methyl]pyridine
—— (3-chloro-4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid 1004514-42-4 C24H17ClF3NO6
(3-chloro-4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid