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—— (Z)-3-(1-methylpyrazol-4-yl)-1-(1,3,5-trimethylpyrazol-4-yl)prop-2-en-1-one —— C13H16N4O
(Z)-3-(1-methylpyrazol-4-yl)-1-(1,3,5-trimethylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-3-(4-acetamidophenyl)-N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]prop-2-enamide —— C18H21N3O2S
(Z)-3-(4-acetamidophenyl)-N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]prop-2-enamide
—— (Z)-3-(furan-2-yl)-N-[1-(4-methoxyphenyl)piperidin-4-yl]prop-2-enamide —— C19H22N2O3
(Z)-3-(furan-2-yl)-N-[1-(4-methoxyphenyl)piperidin-4-yl]prop-2-enamide
—— (Z)-N-[1-(2-pyridin-4-ylethyl)piperidin-4-yl]-3-thiophen-3-ylprop-2-enamide —— C19H23N3OS
(Z)-N-[1-(2-pyridin-4-ylethyl)piperidin-4-yl]-3-thiophen-3-ylprop-2-enamide
—— (Z)-N-[(2-morpholin-4-ylphenyl)methyl]-3-thiophen-2-ylprop-2-enamide —— C18H20N2O2S
(Z)-N-[(2-morpholin-4-ylphenyl)methyl]-3-thiophen-2-ylprop-2-enamide
—— (Z)-3-(4-fluorophenyl)-N-[4-(oxan-4-ylamino)phenyl]prop-2-enamide —— C20H21FN2O2
(Z)-3-(4-fluorophenyl)-N-[4-(oxan-4-ylamino)phenyl]prop-2-enamide
—— (Z)-N-ethylsulfonyl-N-methyl-3-(5-methylfuran-2-yl)prop-2-enamide —— C11H15NO4S
(Z)-N-ethylsulfonyl-N-methyl-3-(5-methylfuran-2-yl)prop-2-enamide
—— (Z)-N-(7-oxo-5,6-dihydro-4H-1,3-benzothiazol-2-yl)-3-thiophen-3-ylprop-2-enamide —— C14H12N2O2S2
(Z)-N-(7-oxo-5,6-dihydro-4H-1,3-benzothiazol-2-yl)-3-thiophen-3-ylprop-2-enamide
—— (Z)-3-(furan-2-yl)-N-[2-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]prop-2-enamide —— C15H18N2O2S
(Z)-3-(furan-2-yl)-N-[2-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]prop-2-enamide
—— (Z)-1-[(2R)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(2,6-difluorophenyl)prop-2-en-1-one —— C21H18F2N2OS
(Z)-1-[(2R)-2-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(2,6-difluorophenyl)prop-2-en-1-one
—— (Z)-N-[[(2R)-oxan-2-yl]methylsulfonyl]-3-phenylprop-2-enamide —— C15H19NO4S
(Z)-N-[[(2R)-oxan-2-yl]methylsulfonyl]-3-phenylprop-2-enamide
—— (Z)-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylpyridin-3-yl)prop-2-enamide —— C20H23N3O2S
(Z)-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylpyridin-3-yl)prop-2-enamide
—— (Z)-N-[[(2S)-oxan-2-yl]methylsulfonyl]-3-phenylprop-2-enamide —— C15H19NO4S
(Z)-N-[[(2S)-oxan-2-yl]methylsulfonyl]-3-phenylprop-2-enamide
—— (Z)-3-(2,6-difluorophenyl)-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]prop-2-enamide —— C16H17F5N2O
(Z)-3-(2,6-difluorophenyl)-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]prop-2-enamide
—— (Z)-1-[(2R)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]-3-(1-methylpyrazol-4-yl)prop-2-en-1-one —— C20H23N5O
(Z)-1-[(2R)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]-3-(1-methylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylpyridin-3-yl)prop-2-enamide —— C20H23N3O2S
(Z)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylpyridin-3-yl)prop-2-enamide
—— (Z)-3-[4-chloro-3-(trifluoromethyl)phenyl]-N-[4-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]prop-2-enamide —— C18H11ClF3N3O3
(Z)-3-[4-chloro-3-(trifluoromethyl)phenyl]-N-[4-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]prop-2-enamide
—— (Z)-N-[4-(4-methyl-6-oxo-1H-pyrimidin-2-yl)phenyl]-3-thiophen-2-ylprop-2-enamide —— C18H15N3O2S
(Z)-N-[4-(4-methyl-6-oxo-1H-pyrimidin-2-yl)phenyl]-3-thiophen-2-ylprop-2-enamide
—— (Z)-2-(4-methylphenyl)-N-(2-morpholin-4-ylethyl)ethenesulfonamide —— C15H22N2O3S
(Z)-2-(4-methylphenyl)-N-(2-morpholin-4-ylethyl)ethenesulfonamide
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[1-(2-pyridin-4-ylethyl)pyrazol-3-yl]prop-2-enamide —— C17H17N5OS
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-[1-(2-pyridin-4-ylethyl)pyrazol-3-yl]prop-2-enamide
—— (Z)-3-(3-fluoro-4-pyridin-3-yloxyphenyl)-N-methylsulfonylprop-2-enamide —— C15H13FN2O4S
(Z)-3-(3-fluoro-4-pyridin-3-yloxyphenyl)-N-methylsulfonylprop-2-enamide
—— (Z)-N-(2-cyanoethyl)-N-propan-2-yl-3-thiophen-3-ylprop-2-enamide —— C13H16N2OS
(Z)-N-(2-cyanoethyl)-N-propan-2-yl-3-thiophen-3-ylprop-2-enamide
—— (Z)-N-[2-(3-fluorophenoxy)phenyl]-3-thiophen-3-ylprop-2-enamide —— C19H14FNO2S
(Z)-N-[2-(3-fluorophenoxy)phenyl]-3-thiophen-3-ylprop-2-enamide
—— (Z)-3-(5-methylthiophen-2-yl)-1-[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]prop-2-en-1-one —— C20H23NOS
(Z)-3-(5-methylthiophen-2-yl)-1-[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]prop-2-en-1-one
—— (Z)-3-(2,3-dichlorophenyl)-N-[2-[[(3S)-oxolan-3-yl]methyl]pyrazol-3-yl]prop-2-enamide —— C17H17Cl2N3O2
(Z)-3-(2,3-dichlorophenyl)-N-[2-[[(3S)-oxolan-3-yl]methyl]pyrazol-3-yl]prop-2-enamide
—— (Z)-3-[4-methoxy-3-[methyl-(4-methylphenyl)sulfamoyl]phenyl]prop-2-enoic acid —— C18H19NO5S
(Z)-3-[4-methoxy-3-[methyl-(4-methylphenyl)sulfamoyl]phenyl]prop-2-enoic acid
—— (Z)-3-(2,6-difluorophenyl)-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]prop-2-enamide —— C16H17F5N2O
(Z)-3-(2,6-difluorophenyl)-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]prop-2-enamide
—— (Z)-3-phenyl-N-[1-(2-pyridin-4-ylethyl)pyrazol-3-yl]prop-2-enamide —— C19H18N4O
(Z)-3-phenyl-N-[1-(2-pyridin-4-ylethyl)pyrazol-3-yl]prop-2-enamide
—— (Z)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-(1-methyl-3,4-dihydro-2H-quinolin-6-yl)prop-2-enamide —— C18H21N5O2
(Z)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-3-(1-methyl-3,4-dihydro-2H-quinolin-6-yl)prop-2-enamide
—— (Z)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cycloheptyl]prop-2-enamide —— C20H25N5O2S
(Z)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cycloheptyl]prop-2-enamide
—— (Z)-N-cyclopropyl-3-(3,5-dimethoxyphenyl)-N-[(3S)-2,5-dioxopyrrolidin-3-yl]prop-2-enamide —— C18H20N2O5
(Z)-N-cyclopropyl-3-(3,5-dimethoxyphenyl)-N-[(3S)-2,5-dioxopyrrolidin-3-yl]prop-2-enamide
—— (Z)-3-[3-methoxy-4-[(1-methyl-2-oxopyridin-4-yl)methoxy]phenyl]prop-2-enoic acid —— C17H17NO5
(Z)-3-[3-methoxy-4-[(1-methyl-2-oxopyridin-4-yl)methoxy]phenyl]prop-2-enoic acid
—— (Z)-N-[2-[(2,5-dioxopyrrolidin-1-yl)methyl]phenyl]-3-pyridin-2-ylprop-2-enamide —— C19H17N3O3
(Z)-N-[2-[(2,5-dioxopyrrolidin-1-yl)methyl]phenyl]-3-pyridin-2-ylprop-2-enamide
—— (Z)-3-(2-fluorophenyl)-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide —— C20H22FN3O2
(Z)-3-(2-fluorophenyl)-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide
—— (Z)-N-(2-chloro-4-methylphenyl)-3-pyrazin-2-ylprop-2-enamide —— C14H12ClN3O
(Z)-N-(2-chloro-4-methylphenyl)-3-pyrazin-2-ylprop-2-enamide
—— (Z)-N-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]pent-2-enamide —— C16H20N2O2
(Z)-N-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]pent-2-enamide
—— (Z)-3-(3-phenylphenyl)-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide —— C22H20N2O
(Z)-3-(3-phenylphenyl)-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide
—— (Z)-N-(2-amino-2-oxoethyl)-3-(1,3-benzothiazol-2-yl)-N-cyclopentylprop-2-enamide —— C17H19N3O2S
(Z)-N-(2-amino-2-oxoethyl)-3-(1,3-benzothiazol-2-yl)-N-cyclopentylprop-2-enamide
—— (Z)-1-[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]-3-(1,3-thiazol-2-yl)prop-2-en-1-one —— C18H20N2OS
(Z)-1-[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]-3-(1,3-thiazol-2-yl)prop-2-en-1-one
—— (Z)-3-(2,4-dimethylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C20H27NO2S
(Z)-3-(2,4-dimethylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— (Z)-N-[(1R)-1-[2-(methanesulfonamido)phenyl]ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C16H19N3O3S2
(Z)-N-[(1R)-1-[2-(methanesulfonamido)phenyl]ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-1-(1,1-dioxo-1,2-thiazolidin-2-yl)-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C15H15N3O3S
(Z)-1-(1,1-dioxo-1,2-thiazolidin-2-yl)-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (Z)-3-[4-[(1,3-dimethyl-2,6-dioxopyrimidin-4-yl)methoxy]-3-methoxyphenyl]prop-2-enoic acid —— C17H18N2O6
(Z)-3-[4-[(1,3-dimethyl-2,6-dioxopyrimidin-4-yl)methoxy]-3-methoxyphenyl]prop-2-enoic acid
—— (Z)-3-(2-cyanophenyl)-N-[[2-(2,2,2-trifluoroethoxy)pyridin-4-yl]methyl]prop-2-enamide —— C18H14F3N3O2
(Z)-3-(2-cyanophenyl)-N-[[2-(2,2,2-trifluoroethoxy)pyridin-4-yl]methyl]prop-2-enamide
—— (Z)-3-pyridin-3-yl-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]prop-2-en-1-one —— C18H20N4O
(Z)-3-pyridin-3-yl-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]prop-2-en-1-one
—— (Z)-N-[(1S)-1-[2-(methanesulfonamido)phenyl]ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C16H19N3O3S2
(Z)-N-[(1S)-1-[2-(methanesulfonamido)phenyl]ethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-pyridin-4-ylprop-2-enamide —— C20H23N3O
(Z)-N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-3-(2,4-dimethylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide —— C20H27NO2S
(Z)-3-(2,4-dimethylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]prop-2-enamide
—— (Z)-3-(3-methylphenyl)-N-[3-(2-pyridin-2-ylethynyl)phenyl]prop-2-enamide —— C23H18N2O
(Z)-3-(3-methylphenyl)-N-[3-(2-pyridin-2-ylethynyl)phenyl]prop-2-enamide
—— (Z)-1-[4-[(3S)-3-ethylpiperidine-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C22H30N2O2
(Z)-1-[4-[(3S)-3-ethylpiperidine-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one