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—— (Z)-3-(5-bromothiophen-3-yl)-1-[(3R)-3-(methoxymethyl)piperidin-1-yl]prop-2-en-1-one —— C14H18BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-1-[(3R)-3-(methoxymethyl)piperidin-1-yl]prop-2-en-1-one
—— (Z)-3-(5-bromothiophen-3-yl)-N-[2-(methylamino)-2-oxoethyl]-N-propylprop-2-enamide —— C13H17BrN2O2S
(Z)-3-(5-bromothiophen-3-yl)-N-[2-(methylamino)-2-oxoethyl]-N-propylprop-2-enamide
—— (Z)-3-(3-cyanophenyl)-N-[1-(1,3-thiazol-2-yl)cyclopentyl]prop-2-enamide —— C18H17N3OS
(Z)-3-(3-cyanophenyl)-N-[1-(1,3-thiazol-2-yl)cyclopentyl]prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-(2-pyridin-3-ylethyl)prop-2-enamide —— C14H13BrN2OS
(Z)-3-(5-bromothiophen-3-yl)-N-(2-pyridin-3-ylethyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(1S)-1-pyridin-2-ylethyl]prop-2-enamide —— C14H13BrN2OS
(Z)-3-(5-bromothiophen-3-yl)-N-[(1S)-1-pyridin-2-ylethyl]prop-2-enamide
—— (Z)-N-[1-[(1S)-1-phenylethyl]piperidin-4-yl]-3-(1,3-thiazol-4-yl)prop-2-enamide —— C19H23N3OS
(Z)-N-[1-[(1S)-1-phenylethyl]piperidin-4-yl]-3-(1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-N-(2-amino-2-oxoethyl)-3-(5-bromothiophen-3-yl)-N-(2-methylpropyl)prop-2-enamide —— C13H17BrN2O2S
(Z)-N-(2-amino-2-oxoethyl)-3-(5-bromothiophen-3-yl)-N-(2-methylpropyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(2S)-1-imidazol-1-ylpropan-2-yl]prop-2-enamide —— C13H14BrN3OS
(Z)-3-(5-bromothiophen-3-yl)-N-[(2S)-1-imidazol-1-ylpropan-2-yl]prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-ethoxyprop-2-enamide —— C9H10BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-N-ethoxyprop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-(1,3-thiazol-2-ylmethyl)prop-2-enamide —— C11H9BrN2OS2
(Z)-3-(5-bromothiophen-3-yl)-N-(1,3-thiazol-2-ylmethyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-methyl-N-(pyridin-4-ylmethyl)prop-2-enamide —— C14H13BrN2OS
(Z)-3-(5-bromothiophen-3-yl)-N-methyl-N-(pyridin-4-ylmethyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(2R)-oxan-2-yl]oxyprop-2-enamide —— C12H14BrNO3S
(Z)-3-(5-bromothiophen-3-yl)-N-[(2R)-oxan-2-yl]oxyprop-2-enamide
—— (Z)-N-[1-[(1R)-1-phenylethyl]piperidin-4-yl]-3-(1,3-thiazol-4-yl)prop-2-enamide —— C19H23N3OS
(Z)-N-[1-[(1R)-1-phenylethyl]piperidin-4-yl]-3-(1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide —— C14H13BrN2OS
(Z)-3-(5-bromothiophen-3-yl)-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide
—— (Z)-N-(3-acetamidopropyl)-3-(5-bromothiophen-3-yl)prop-2-enamide —— C12H15BrN2O2S
(Z)-N-(3-acetamidopropyl)-3-(5-bromothiophen-3-yl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide —— C12H12BrN3O2S
(Z)-3-(5-bromothiophen-3-yl)-N-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide —— C14H13BrN2OS
(Z)-3-(5-bromothiophen-3-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-1-[(3R)-3-methylmorpholin-4-yl]prop-2-en-1-one —— C12H14BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-1-[(3R)-3-methylmorpholin-4-yl]prop-2-en-1-one
—— (Z)-3-(5-bromothiophen-3-yl)-N-(3-pyrazol-1-ylpropyl)prop-2-enamide —— C13H14BrN3OS
(Z)-3-(5-bromothiophen-3-yl)-N-(3-pyrazol-1-ylpropyl)prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-1-[(3S)-3-methylmorpholin-4-yl]prop-2-en-1-one —— C12H14BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-1-[(3S)-3-methylmorpholin-4-yl]prop-2-en-1-one
—— (Z)-3-(5-bromothiophen-3-yl)-1-(4-ethoxypiperidin-1-yl)prop-2-en-1-one —— C14H18BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-1-(4-ethoxypiperidin-1-yl)prop-2-en-1-one
—— (Z)-3-(5-bromothiophen-3-yl)-N-(3-methoxypropyl)-N-methylprop-2-enamide —— C12H16BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-N-(3-methoxypropyl)-N-methylprop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide —— C12H12BrN3O2S
(Z)-3-(5-bromothiophen-3-yl)-N-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C12H14BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (Z)-3-(5-bromothiophen-3-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C12H14BrNO2S
(Z)-3-(5-bromothiophen-3-yl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (Z)-N-methyl-N-[(3R)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide —— C20H21N3O2
(Z)-N-methyl-N-[(3R)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-3-pyridin-4-ylprop-2-enamide —— C18H19F2N3O
(Z)-N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-[(1R)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-pyridin-4-ylprop-2-enamide —— C22H21N3O
(Z)-N-[(1R)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-3-(1,3-benzothiazol-2-yl)-N-(5-methoxy-1,3-dimethylpyrazol-4-yl)prop-2-enamide —— C16H16N4O2S
(Z)-3-(1,3-benzothiazol-2-yl)-N-(5-methoxy-1,3-dimethylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-methyl-N-[(3S)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide —— C20H21N3O2
(Z)-N-methyl-N-[(3S)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-[(1R)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide —— C20H19N3OS
(Z)-N-[(1R)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-N-methyl-N-[(3R)-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide —— C20H23N3O
(Z)-N-methyl-N-[(3R)-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-3-pyridin-4-ylprop-2-enamide —— C18H19F2N3O
(Z)-N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-methyl-N-[(3S)-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide —— C20H23N3O
(Z)-N-methyl-N-[(3S)-1-phenylpiperidin-3-yl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-[(3R)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-3-ylprop-2-enamide —— C19H19N3O2
(Z)-N-[(3R)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-3-ylprop-2-enamide
—— (Z)-2-methyl-N-[(1S)-2-methyl-1-(3-methylpyridin-2-yl)propyl]pent-2-enamide —— C16H24N2O
(Z)-2-methyl-N-[(1S)-2-methyl-1-(3-methylpyridin-2-yl)propyl]pent-2-enamide
—— (Z)-N-[(S)-(2-fluorophenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide —— C19H16FN3O2
(Z)-N-[(S)-(2-fluorophenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide
—— (Z)-N-[(R)-(2-methoxyphenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide —— C20H19N3O3
(Z)-N-[(R)-(2-methoxyphenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide
—— (Z)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-pyridin-4-ylprop-2-enamide —— C17H13ClN4O2
(Z)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-pyridin-4-ylprop-2-enamide
—— (Z)-N-(3-imidazol-1-ylpropyl)-3-(3-propan-2-yloxyphenyl)prop-2-enamide —— C18H23N3O2
(Z)-N-(3-imidazol-1-ylpropyl)-3-(3-propan-2-yloxyphenyl)prop-2-enamide
—— (Z)-3-(1,3-benzothiazol-2-yl)-N-(1-methyl-2-oxopyridin-3-yl)prop-2-enamide —— C16H13N3O2S
(Z)-3-(1,3-benzothiazol-2-yl)-N-(1-methyl-2-oxopyridin-3-yl)prop-2-enamide
—— (Z)-N-[(3S)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-3-ylprop-2-enamide —— C19H19N3O2
(Z)-N-[(3S)-2-oxo-1-phenylpiperidin-3-yl]-3-pyridin-3-ylprop-2-enamide
—— (Z)-1-[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H19N3O
(Z)-1-[(2S)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-N-[(R)-(2-fluorophenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide —— C19H16FN3O2
(Z)-N-[(R)-(2-fluorophenyl)-(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylprop-2-enamide
—— (Z)-N-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]-3-(3-fluorophenyl)prop-2-enamide —— C15H15FN2O3
(Z)-N-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]-3-(3-fluorophenyl)prop-2-enamide
—— (Z)-3-pyridin-3-yl-N-[2-(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)ethyl]prop-2-enamide —— C17H20N4OS
(Z)-3-pyridin-3-yl-N-[2-(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)ethyl]prop-2-enamide
—— (Z)-N-[(1S)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide —— C20H19N3OS
(Z)-N-[(1S)-2-(4-methylphenyl)-1-pyridin-2-ylethyl]-3-(1,3-thiazol-2-yl)prop-2-enamide
—— (Z)-1-[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H19N3O
(Z)-1-[(2R)-2-(1-methylpyrrol-2-yl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-4,4-dimethyl-N-[2-methyl-3-(thiomorpholine-4-carbonyl)phenyl]pent-2-enamide —— C19H26N2O2S
(Z)-4,4-dimethyl-N-[2-methyl-3-(thiomorpholine-4-carbonyl)phenyl]pent-2-enamide
—— (Z)-N-(3-imidazol-1-ylpropyl)-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C19H24N4O2
(Z)-N-(3-imidazol-1-ylpropyl)-3-(4-morpholin-4-ylphenyl)prop-2-enamide