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—— (Z)-N-(3-acetamidopropyl)-N-methyl-3-(1-methylindol-3-yl)prop-2-enamide —— C18H23N3O2
(Z)-N-(3-acetamidopropyl)-N-methyl-3-(1-methylindol-3-yl)prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-(prop-2-enoylamino)ethyl]prop-2-enamide —— C15H21N3O2S
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-(prop-2-enoylamino)ethyl]prop-2-enamide
—— (Z)-N-[3-[[(S)-benzylsulfinyl]methyl]phenyl]-3-cyclopropylprop-2-enamide —— C20H21NO2S
(Z)-N-[3-[[(S)-benzylsulfinyl]methyl]phenyl]-3-cyclopropylprop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-1-(1,1-dioxo-1,4-thiazepan-4-yl)prop-2-en-1-one —— C15H22N2O3S2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-1-(1,1-dioxo-1,4-thiazepan-4-yl)prop-2-en-1-one
—— (Z)-N-methyl-3-(1-methylindol-3-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide —— C20H21N3O
(Z)-N-methyl-3-(1-methylindol-3-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide
—— (Z)-N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-(2-tert-butyl-1,3-thiazol-5-yl)prop-2-enamide —— C18H27N3O2S
(Z)-N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-(2-tert-butyl-1,3-thiazol-5-yl)prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C17H27N3O2S
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— (Z)-3-(1-methylindol-3-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide —— C17H18N4O2
(Z)-3-(1-methylindol-3-yl)-N-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]prop-2-enamide
—— (Z)-N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-(2-tert-butyl-1,3-thiazol-5-yl)prop-2-enamide —— C18H27N3O2S
(Z)-N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-3-(2-tert-butyl-1,3-thiazol-5-yl)prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]prop-2-enamide —— C15H22N2O3S2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (Z)-3-(4-bromothiophen-2-yl)-N-[(2-methyl-1,3-thiazol-5-yl)methyl]prop-2-enamide —— C12H11BrN2OS2
(Z)-3-(4-bromothiophen-2-yl)-N-[(2-methyl-1,3-thiazol-5-yl)methyl]prop-2-enamide
—— (Z)-3-(4-bromothiophen-2-yl)-N-(2-methylsulfonylethyl)prop-2-enamide —— C10H12BrNO3S2
(Z)-3-(4-bromothiophen-2-yl)-N-(2-methylsulfonylethyl)prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C17H27N3O2S
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— (Z)-3-(1-methylindol-3-yl)-N-[3-(2-oxopyridin-1-yl)propyl]prop-2-enamide —— C20H21N3O2
(Z)-3-(1-methylindol-3-yl)-N-[3-(2-oxopyridin-1-yl)propyl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]prop-2-enamide —— C17H23N5OS
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-3-cyanothiolan-3-yl]prop-2-enamide —— C15H19N3OS2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-3-cyanothiolan-3-yl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]prop-2-enamide —— C15H22N2O3S2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (Z)-N-[3-(methanesulfonamido)propyl]-3-(1-methylindol-3-yl)prop-2-enamide —— C16H21N3O3S
(Z)-N-[3-(methanesulfonamido)propyl]-3-(1-methylindol-3-yl)prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C14H20N2O3S2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C14H20N2O3S2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-3-cyanothiolan-3-yl]prop-2-enamide —— C15H19N3OS2
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(3S)-3-cyanothiolan-3-yl]prop-2-enamide
—— (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]prop-2-enamide —— C17H23N5OS
(Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[2-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]prop-2-enamide
—— (Z)-3-(4-bromothiophen-2-yl)-N-methyl-N-[(1-methylpyrazol-4-yl)methyl]prop-2-enamide —— C13H14BrN3OS
(Z)-3-(4-bromothiophen-2-yl)-N-methyl-N-[(1-methylpyrazol-4-yl)methyl]prop-2-enamide
—— (Z)-1-[4-[(3R)-1,1-dioxothiolan-3-yl]piperazin-1-yl]-3,4,4-trimethylpent-2-en-1-one —— C16H28N2O3S
(Z)-1-[4-[(3R)-1,1-dioxothiolan-3-yl]piperazin-1-yl]-3,4,4-trimethylpent-2-en-1-one
—— (Z)-1-[4-[(3S)-1,1-dioxothiolan-3-yl]piperazin-1-yl]-3,4,4-trimethylpent-2-en-1-one —— C16H28N2O3S
(Z)-1-[4-[(3S)-1,1-dioxothiolan-3-yl]piperazin-1-yl]-3,4,4-trimethylpent-2-en-1-one
—— (Z)-2-phenyl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]ethenesulfonamide —— C17H23N3O2S
(Z)-2-phenyl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]ethenesulfonamide
—— (Z)-2-phenyl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]ethenesulfonamide —— C17H23N3O2S
(Z)-2-phenyl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]ethenesulfonamide
—— (Z)-N-[2-(5-methyl-1,3-thiazol-2-yl)ethyl]-2-phenylethenesulfonamide —— C14H16N2O2S2
(Z)-N-[2-(5-methyl-1,3-thiazol-2-yl)ethyl]-2-phenylethenesulfonamide
—— (Z)-N-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylethenesulfonamide —— C16H18N2O2S2
(Z)-N-[(R)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylethenesulfonamide
—— (Z)-N-methyl-N-[(3S)-1-methylpiperidin-3-yl]-2-phenylethenesulfonamide —— C15H22N2O2S
(Z)-N-methyl-N-[(3S)-1-methylpiperidin-3-yl]-2-phenylethenesulfonamide
—— (Z)-N-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylethenesulfonamide —— C16H18N2O2S2
(Z)-N-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylethenesulfonamide
—— (Z)-3-(3-fluorophenyl)-N-[4-[(R)-methylsulfinyl]phenyl]prop-2-enamide —— C16H14FNO2S
(Z)-3-(3-fluorophenyl)-N-[4-[(R)-methylsulfinyl]phenyl]prop-2-enamide
—— (Z)-N-[[(1S)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C20H25N3O2
(Z)-N-[[(1S)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— (Z)-2-phenyl-N-thiophen-3-ylethenesulfonamide —— C12H11NO2S2
(Z)-2-phenyl-N-thiophen-3-ylethenesulfonamide
—— (Z)-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one —— C16H21N3O2S
(Z)-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one
—— (Z)-N-[[(1S)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C18H20N2O2S
(Z)-N-[[(1S)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-N-[[(1R)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C18H20N2O2S
(Z)-N-[[(1R)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (Z)-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C16H20N4OS
(Z)-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-2-methyl-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]pent-2-en-1-one —— C14H23N3OS
(Z)-2-methyl-1-[4-[(5S)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]pent-2-en-1-one
—— (Z)-3-(3-fluorophenyl)-N-[4-[(S)-methylsulfinyl]phenyl]prop-2-enamide —— C16H14FNO2S
(Z)-3-(3-fluorophenyl)-N-[4-[(S)-methylsulfinyl]phenyl]prop-2-enamide
—— (Z)-1-[4-[(5R)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one —— C16H21N3O2S
(Z)-1-[4-[(5R)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]-3-(5-methylfuran-2-yl)prop-2-en-1-one
—— (Z)-N-[[(1R)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C20H25N3O2
(Z)-N-[[(1R)-1-hydroxy-3,4-dihydro-2H-naphthalen-1-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— (Z)-1-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H21N3O2
(Z)-1-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-1-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H21N3O2
(Z)-1-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-1-[(3R)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C20H22N2O2
(Z)-1-[(3R)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-3-[2-(trifluoromethyl)phenyl]but-2-enamide —— C16H17F3N4O
(Z)-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]-3-[2-(trifluoromethyl)phenyl]but-2-enamide
—— (Z)-1-[(3S)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C20H22N2O2
(Z)-1-[(3S)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (Z)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-3-[2-(trifluoromethyl)phenyl]but-2-enamide —— C16H17F3N4O
(Z)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-3-[2-(trifluoromethyl)phenyl]but-2-enamide
—— (Z)-N-[(3S,5S)-5-methyl-2-oxo-1-phenylpyrrolidin-3-yl]-3-pyridin-3-ylprop-2-enamide —— C19H19N3O2
(Z)-N-[(3S,5S)-5-methyl-2-oxo-1-phenylpyrrolidin-3-yl]-3-pyridin-3-ylprop-2-enamide
—— (Z)-3-(furan-2-yl)-N-[(2S)-4-(1-methylpyrrol-2-yl)butan-2-yl]prop-2-enamide —— C16H20N2O2
(Z)-3-(furan-2-yl)-N-[(2S)-4-(1-methylpyrrol-2-yl)butan-2-yl]prop-2-enamide