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—— (7S)-7-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)heptanamide —— C26H27N7O2S
(7S)-7-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)heptanamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide —— C24H27N7O2
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[3-(1-methylpyrazol-4-yl)propanoylamino]heptanamide —— C27H33N7O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[3-(1-methylpyrazol-4-yl)propanoylamino]heptanamide
—— 7-[5-(2-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C21H26N4O2
7-[5-(2-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[3-(1,2,4-triazol-1-yl)propanoylamino]heptanamide —— C25H30N8O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[3-(1,2,4-triazol-1-yl)propanoylamino]heptanamide
—— (7S)-7-[[2-(2-methylhydrazinyl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C23H32N8O2
(7S)-7-[[2-(2-methylhydrazinyl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]amino]heptanamide —— C31H32N6O3S
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]heptanamide —— C25H29N7O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]heptanamide
—— (7S)-7-[(4-aminophenyl)sulfonylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C26H30N6O4S
(7S)-7-[(4-aminophenyl)sulfonylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[(2-phenylacetyl)amino]heptanamide —— C28H30N4O2
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[(2-phenylacetyl)amino]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoylamino]heptanamide —— C26H32N8O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoylamino]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide —— C26H29N7O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide —— C24H28N8O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide
—— 7-[5-(6-fluoronaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide —— C20H22FN3O
7-[5-(6-fluoronaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide —— C23H26N8O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-pyrrolidin-1-yltetrazol-2-yl)acetyl]amino]heptanamide —— C27H33N9O2
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-pyrrolidin-1-yltetrazol-2-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]heptanamide —— C26H31N7O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]heptanamide
—— 7-[5-(4-phenylphenyl)-1H-imidazol-2-yl]heptanamide —— C22H25N3O
7-[5-(4-phenylphenyl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(6-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide —— C21H25N3O2
7-[5-(6-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide
—— (7Z)-3-(4-ethylphenyl)-7-(pyridin-4-ylmethylidene)-3,4-dihydro-2H-[1,3]thiazolo[3,2-a][1,3,5]triazin-6(7H)-one —— C19H18N4OS
(7Z)-3-(4-ethylphenyl)-7-(pyridin-4-ylmethylidene)-3,4-dihydro-2H-[1,3]thiazolo[3,2-a][1,3,5]triazin-6(7H)-one
—— (7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide —— C29H33F3N6O2
(7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(3-morpholin-4-ylpropanoylamino)heptanamide —— C27H36N6O4
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(3-morpholin-4-ylpropanoylamino)heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide —— C25H27N7O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide
—— (7S)-7-[(2-morpholin-4-ylacetyl)amino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide —— C26H33N5O3
(7S)-7-[(2-morpholin-4-ylacetyl)amino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide
—— (7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(4-phenyl-1,3-thiazol-2-yl)acetyl]amino]heptanamide —— C32H33N5O2S
(7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(4-phenyl-1,3-thiazol-2-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)acetyl]amino]heptanamide —— C24H27N7O3
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)acetyl]amino]heptanamide
—— (7S)-7-[(2-indazol-2-ylacetyl)amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C30H34N8O2
(7S)-7-[(2-indazol-2-ylacetyl)amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[[2-[[(Z)-2-aminoethenyl]-methylamino]acetyl]amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C26H36N8O2
(7S)-7-[[2-[[(Z)-2-aminoethenyl]-methylamino]acetyl]amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C32H37N7O3
(7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-[3-(aminomethyl)phenyl]-1H-imidazol-2-yl]heptanamide —— C17H24N4O
7-[5-[3-(aminomethyl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C30H35N9O3
(7S)-7-[3-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoylamino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide —— C27H29N7O2S
(7S)-7-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide
—— (7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide —— C25H29N7O2
(7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(1,2,4-triazol-4-yl)acetyl]amino]heptanamide
—— 7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C20H25N5O
7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— 7-[5-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C19H23N5O
7-[5-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— 7-[5-(2-methoxyquinolin-3-yl)-1,3-oxazol-2-yl]-N-methylheptanamide —— C21H25N3O3
7-[5-(2-methoxyquinolin-3-yl)-1,3-oxazol-2-yl]-N-methylheptanamide
—— (7S)-7-[[2-[[(Z)-2-aminoethenyl]-methylamino]acetyl]amino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C25H34N8O2
(7S)-7-[[2-[[(Z)-2-aminoethenyl]-methylamino]acetyl]amino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C26H32N8O2
(7S)-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide —— C29H31N7O2
(7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide
—— 7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C19H23N5O
7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)acetyl]amino]heptanamide —— C25H29N7O3
(7S)-N-methyl-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)acetyl]amino]heptanamide
—— 7-[5-(5-methoxy-1H-indol-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C20H26N4O2
7-[5-(5-methoxy-1H-indol-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— 7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide —— C20H23N3O
7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide
—— (7S)-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide —— C24H29N9O2
(7S)-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide
—— 7-[5-(4-pyridin-4-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C21H24N4O
7-[5-(4-pyridin-4-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide —— C24H28N8O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(1,2,4-triazol-1-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-([1,2,4]triazolo[1,5-a]pyrimidin-6-yl)acetyl]amino]heptanamide —— C27H28N8O2
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[[2-([1,2,4]triazolo[1,5-a]pyrimidin-6-yl)acetyl]amino]heptanamide
—— 7-[5-(1-benzothiophen-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C19H23N3OS
7-[5-(1-benzothiophen-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— 7-[5-(3-methoxyisoquinolin-7-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C21H26N4O2
7-[5-(3-methoxyisoquinolin-7-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— 7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C20H24N4O2
7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide