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—— [7-(4-Aminophenyl)-6-chloro-5-(4-chlorophenyl)pyrrolo[2,3-d]pyrimidin-4-yl]carbamic acid —— C19H13Cl2N5O2
[7-(4-Aminophenyl)-6-chloro-5-(4-chlorophenyl)pyrrolo[2,3-d]pyrimidin-4-yl]carbamic acid
—— 7-[2-[1-amino-2-(3,5-difluorophenyl)ethyl]pyridin-3-yl]-1H-quinolin-2-one —— C22H17F2N3O
7-[2-[1-amino-2-(3,5-difluorophenyl)ethyl]pyridin-3-yl]-1H-quinolin-2-one
—— [7-(3-Aminophenyl)-6-chloro-5-(3-methoxy-4-methylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]carbamic acid —— C21H18ClN5O3
[7-(3-Aminophenyl)-6-chloro-5-(3-methoxy-4-methylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]carbamic acid
—— (7R)-2-[3-methoxy-4-(2-phenylsulfanylethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H26N2O3S2
(7R)-2-[3-methoxy-4-(2-phenylsulfanylethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-butoxy-6-ethyl-4-phenyl-2H-chromen-2-one —— C21H22O3
7-butoxy-6-ethyl-4-phenyl-2H-chromen-2-one
—— (7S)-2-[3-chloro-5-methoxy-4-(2-phenoxyethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H25ClN2O4S
(7S)-2-[3-chloro-5-methoxy-4-(2-phenoxyethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1H-imidazol-2-yl]heptanamide —— C18H23N3O3
7-[5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C19H25N3O3
7-[5-(2,3-dihydro-1,4-benzodioxin-5-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide —— C24H28N8O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methyl-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide
—— 7-[5-(3-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C22H27N3O2
7-[5-(3-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(2-pyrazol-1-ylpropanoylamino)heptanamide —— C26H31N7O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(2-pyrazol-1-ylpropanoylamino)heptanamide
—— (7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C29H32N8O2
(7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(4-chloro-3-methylphenyl)-1H-imidazol-2-yl]-N-methylheptanamide —— C18H24ClN3O
7-[5-(4-chloro-3-methylphenyl)-1H-imidazol-2-yl]-N-methylheptanamide
—— 7-(6-Oxabicyclo[3.1.0]hexan-2-ylmethoxy)heptyl 7-oxabicyclo[4.1.0]heptane-3-carboxylate —— C20H32O5
7-(6-Oxabicyclo[3.1.0]hexan-2-ylmethoxy)heptyl 7-oxabicyclo[4.1.0]heptane-3-carboxylate
—— (7S)-7-[[2-(dimethylamino)acetyl]amino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methylheptanamide —— C25H34N6O3
(7S)-7-[[2-(dimethylamino)acetyl]amino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methylheptanamide
—— 7-[2-methyl-6-(pyridin-2-ylcarbamoyl)phenyl]-N-pentyl-6H-furo[2,3-f][1,3]benzodioxole-7-carboxamide —— C28H29N3O5
7-[2-methyl-6-(pyridin-2-ylcarbamoyl)phenyl]-N-pentyl-6H-furo[2,3-f][1,3]benzodioxole-7-carboxamide
—— (7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[(2-piperazin-1-ylacetyl)amino]heptanamide —— C26H34N6O2
(7S)-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)-7-[(2-piperazin-1-ylacetyl)amino]heptanamide
—— (7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C29H36N8O2S
(7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— 7-[5-(3-methoxyisoquinolin-7-yl)-1H-imidazol-2-yl]heptanamide —— C20H24N4O2
7-[5-(3-methoxyisoquinolin-7-yl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methyl-7-[3-(4-methylpiperazin-1-yl)propanoylamino]heptanamide —— C29H41N7O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methyl-7-[3-(4-methylpiperazin-1-yl)propanoylamino]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methyl-7-[3-(1,2,4-triazol-1-yl)propanoylamino]heptanamide —— C26H32N8O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-N-methyl-7-[3-(1,2,4-triazol-1-yl)propanoylamino]heptanamide
—— 7-[5-(1-benzofuran-5-yl)-1H-imidazol-2-yl]heptanamide —— C18H21N3O2
7-[5-(1-benzofuran-5-yl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(4-pyridin-3-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C21H24N4O
7-[5-(4-pyridin-3-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-(3-piperidin-1-ylpropanoylamino)-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide —— C25H34F3N5O2
(7S)-7-(3-piperidin-1-ylpropanoylamino)-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-N-methyl-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide —— C27H34N8O2
(7S)-N-methyl-7-[[2-(3-methylpyrazol-1-yl)acetyl]amino]-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide —— C27H32N8O2
(7S)-N-methyl-7-[5-[4-(1-methylpyrazol-3-yl)phenyl]-1H-imidazol-2-yl]-7-[(2-pyrimidin-2-ylacetyl)amino]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide —— C24H28N8O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide
—— (7S)-7-[5-(1H-indazol-5-yl)-1H-imidazol-2-yl]-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide —— C21H25N9O2
(7S)-7-[5-(1H-indazol-5-yl)-1H-imidazol-2-yl]-7-[[2-(triazol-1-yl)acetyl]amino]heptanamide
—— (7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoylamino]heptanamide —— C25H30N8O2
(7S)-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoylamino]heptanamide
—— (7S)-7-[(2-indazol-2-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide —— C29H31N7O2
(7S)-7-[(2-indazol-2-ylacetyl)amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-N-methylheptanamide
—— 7-(5-isoquinolin-6-yl-1H-imidazol-2-yl)-N-methylheptanamide —— C20H24N4O
7-(5-isoquinolin-6-yl-1H-imidazol-2-yl)-N-methylheptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[(2-pyridin-2-ylacetyl)amino]heptanamide —— C27H30N6O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[(2-pyridin-2-ylacetyl)amino]heptanamide
—— (7S)-7-[[2-(dimethylamino)acetyl]amino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C24H32N6O3
(7S)-7-[[2-(dimethylamino)acetyl]amino]-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(3-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide —— C21H25N3O2
7-[5-(3-methoxynaphthalen-2-yl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-(3-imidazol-1-ylpropanoylamino)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide —— C26H31N7O3
(7S)-7-(3-imidazol-1-ylpropanoylamino)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]heptanamide
—— 7-[5-(4-chloro-2-methoxyphenyl)-1H-imidazol-2-yl]-N-methylheptanamide —— C18H24ClN3O2
7-[5-(4-chloro-2-methoxyphenyl)-1H-imidazol-2-yl]-N-methylheptanamide
—— (7R)-2-[3-chloro-5-methoxy-4-(2-phenoxyethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H25ClN2O4S
(7R)-2-[3-chloro-5-methoxy-4-(2-phenoxyethoxy)phenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-N-methyl-7-(3-piperidin-1-ylpropanoylamino)-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide —— C26H36F3N5O2
(7S)-N-methyl-7-(3-piperidin-1-ylpropanoylamino)-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide
—— 7-[5-[4-(1-Methylpyrazol-3-yl)phenyl]-1,3-oxazol-2-yl]heptanamide —— C20H24N4O2
7-[5-[4-(1-Methylpyrazol-3-yl)phenyl]-1,3-oxazol-2-yl]heptanamide
—— (7S)-7-[3-(1,3-benzothiazol-2-yl)propanoylamino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C30H33N7O2S
(7S)-7-[3-(1,3-benzothiazol-2-yl)propanoylamino]-N-methyl-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C27H32N8O2S
(7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[(2-pyrazin-2-ylacetyl)amino]heptanamide —— C26H29N7O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-[(2-pyrazin-2-ylacetyl)amino]heptanamide
—— (7S)-7-[[2-(benzimidazol-1-yl)acetyl]amino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide —— C29H30N6O2
(7S)-7-[[2-(benzimidazol-1-yl)acetyl]amino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide
—— (7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(3-piperidin-1-ylpropanoylamino)heptanamide —— C28H38N6O3
(7S)-7-[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]-7-(3-piperidin-1-ylpropanoylamino)heptanamide
—— (7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-N-methyl-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide —— C30H35F3N6O2
(7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-N-methyl-7-[5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide —— C28H30N8O2
(7S)-7-[(2-imidazo[1,2-a]pyridin-3-ylacetyl)amino]-7-[5-(4-pyrazol-1-ylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide —— C32H36N6O2
(7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-(5-naphthalen-2-yl-1H-imidazol-2-yl)heptanamide
—— (7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)heptanamide —— C27H31N7O2S
(7S)-7-[[2-(6,7-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl)acetyl]amino]-7-(5-isoquinolin-7-yl-1H-imidazol-2-yl)heptanamide
—— 7-[5-(4-chloro-3-methylphenyl)-1H-imidazol-2-yl]heptanamide —— C17H22ClN3O
7-[5-(4-chloro-3-methylphenyl)-1H-imidazol-2-yl]heptanamide
—— (7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-(5-naphthalen-2-yl-1,3,4-oxadiazol-2-yl)heptanamide —— C31H34N6O3
(7S)-7-[3-(2-ethylbenzimidazol-1-yl)propanoylamino]-7-(5-naphthalen-2-yl-1,3,4-oxadiazol-2-yl)heptanamide