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—— (7S,9aR)-7-(4-amino-3-bromoimidazo[1,5-a]pyrazin-4-ium-1-yl)-1,2,3,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-4-one —— C14H18BrN6O+
(7S,9aR)-7-(4-amino-3-bromoimidazo[1,5-a]pyrazin-4-ium-1-yl)-1,2,3,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-4-one
—— (7S,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one —— C15H16BrClN4O
(7S,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one
—— (7S,9aS)-N-[(3-chloropyrazin-2-yl)methyl]-4-oxo-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazine-7-carboxamide —— C14H17ClN4O3
(7S,9aS)-N-[(3-chloropyrazin-2-yl)methyl]-4-oxo-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazine-7-carboxamide
—— 7-(3-bromo-4H-imidazo[1,5-a]pyrazin-4-ium-1-yl)-2-methyl-4,4a,5,6,7,8-hexahydro-3H-pyrido[1,2-c]pyrimidin-1-one;chloride —— C15H19BrClN5O
7-(3-bromo-4H-imidazo[1,5-a]pyrazin-4-ium-1-yl)-2-methyl-4,4a,5,6,7,8-hexahydro-3H-pyrido[1,2-c]pyrimidin-1-one;chloride
—— 7-(3-bromoimidazo[1,5-a]pyrazin-1-yl)-2-methyl-4,4a,5,6,7,8-hexahydro-3H-pyrido[1,2-c]pyrimidin-1-one —— C15H18BrN5O
7-(3-bromoimidazo[1,5-a]pyrazin-1-yl)-2-methyl-4,4a,5,6,7,8-hexahydro-3H-pyrido[1,2-c]pyrimidin-1-one
—— (7R,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-4-one —— C14H14BrClN4O2
(7R,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-4-one
—— (7R,9aS)-N-[(3-chloropyrazin-2-yl)methyl]-4-oxo-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazine-7-carboxamide —— C14H17ClN4O3
(7R,9aS)-N-[(3-chloropyrazin-2-yl)methyl]-4-oxo-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazine-7-carboxamide
—— (7E)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C45H55F3N6O8S2
(7E)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (7E)-N-cyclopropylsulfonyl-14-[2-(2,6-dimethylpiperidin-1-yl)-2-oxoethyl]-18-(7-methoxy-2-phenylquinolin-4-yl)oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C46H57N5O8S
(7E)-N-cyclopropylsulfonyl-14-[2-(2,6-dimethylpiperidin-1-yl)-2-oxoethyl]-18-(7-methoxy-2-phenylquinolin-4-yl)oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (7R,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one —— C15H16BrClN4O
(7R,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one
—— 7-[4-(imidazo[1,2-c]pyrimidin-2-ylmethoxy)-2-oxopyridin-1-yl]-5-methyl-3,4-dihydro-1H-pyrido[4,3-b]indole-2-carboxylic acid —— C25H22N6O4
7-[4-(imidazo[1,2-c]pyrimidin-2-ylmethoxy)-2-oxopyridin-1-yl]-5-methyl-3,4-dihydro-1H-pyrido[4,3-b]indole-2-carboxylic acid
—— (7R,9aS)-7-(8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one —— C15H18BrN5O
(7R,9aS)-7-(8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl)-1,2,3,6,7,8,9,9a-octahydroquinolizin-4-one
—— 7-Ethoxy-4-(4-fluorophenyl)-2-methyl-5-oxo-[1,3]thiazolo[5,4-b]pyridine-6-carboxylic acid —— C16H13FN2O4S
7-Ethoxy-4-(4-fluorophenyl)-2-methyl-5-oxo-[1,3]thiazolo[5,4-b]pyridine-6-carboxylic acid
—— (7S,9aR)-7-[(2-methylpropan-2-yl)oxycarbonyl]-4-oxo-3,6,7,8,9,9a-hexahydro-1H-pyrido[1,2-a]pyrazine-2-carboxylic acid;bicyclo[4.1.0]hepta-1,3,5-triene —— C21H28N2O5
(7S,9aR)-7-[(2-methylpropan-2-yl)oxycarbonyl]-4-oxo-3,6,7,8,9,9a-hexahydro-1H-pyrido[1,2-a]pyrazine-2-carboxylic acid;bicyclo[4.1.0]hepta-1,3,5-triene
—— 7,7-Dimethyl-3-oxo-1-propan-2-yl-2,5,6,8-tetrahydroisoquinoline-4-carbonitrile —— C15H20N2O
7,7-Dimethyl-3-oxo-1-propan-2-yl-2,5,6,8-tetrahydroisoquinoline-4-carbonitrile
—— (7S,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-4-one —— C14H14BrClN4O2
(7S,9aS)-7-(1-bromo-8-chloroimidazo[1,5-a]pyrazin-3-yl)-1,6,7,8,9,9a-hexahydropyrido[2,1-c][1,4]oxazin-4-one
—— 7-Methoxy-4,4-dimethyl-2-phenylisoquinoline-1,3-dione —— C18H17NO3
7-Methoxy-4,4-dimethyl-2-phenylisoquinoline-1,3-dione
—— 7-(dimethylamino)-1,9-dimethyl-3-(4-methylpiperazin-1-yl)-10H-phenothiazine-4-carboxylic acid —— C22H28N4O2S
7-(dimethylamino)-1,9-dimethyl-3-(4-methylpiperazin-1-yl)-10H-phenothiazine-4-carboxylic acid
—— 7-(4-cyclopentylsulfonylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine —— C27H38N4O2S2
7-(4-cyclopentylsulfonylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine
—— 7-[(E)-2-(6-methylpyridin-3-yl)ethenyl]-3,12-diazatetracyclo[10.2.2.02,10.04,9]hexadeca-2,4,6,9-tetraene —— C22H23N3
7-[(E)-2-(6-methylpyridin-3-yl)ethenyl]-3,12-diazatetracyclo[10.2.2.02,10.04,9]hexadeca-2,4,6,9-tetraene
—— 7-(4-cyclopropylsulfonylpiperazin-1-yl)-1-ethyl-9-methyl-3-pyrrolidin-1-yl-10H-phenothiazine —— C26H34N4O2S2
7-(4-cyclopropylsulfonylpiperazin-1-yl)-1-ethyl-9-methyl-3-pyrrolidin-1-yl-10H-phenothiazine
—— 7-(4-cyclopropylsulfonylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine —— C25H34N4O2S2
7-(4-cyclopropylsulfonylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine
—— 7-(4-cyclopropylsulfonylpiperazin-1-yl)-N,N,1,9-tetramethyl-10H-phenothiazin-3-amine —— C23H30N4O2S2
7-(4-cyclopropylsulfonylpiperazin-1-yl)-N,N,1,9-tetramethyl-10H-phenothiazin-3-amine
—— 7-(4-cyclopropylsulfonylpiperazin-1-yl)-9-ethyl-N,N-dimethyl-1-propan-2-yl-10H-phenothiazin-3-amine —— C26H36N4O2S2
7-(4-cyclopropylsulfonylpiperazin-1-yl)-9-ethyl-N,N-dimethyl-1-propan-2-yl-10H-phenothiazin-3-amine
—— 7-(4-cyclopropylsulfonylpiperazin-1-yl)-N,N,1-trimethyl-9-propan-2-yl-10H-phenothiazin-3-amine —— C25H34N4O2S2
7-(4-cyclopropylsulfonylpiperazin-1-yl)-N,N,1-trimethyl-9-propan-2-yl-10H-phenothiazin-3-amine
—— 7-(4-cyclopentylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine —— C27H38N4S
7-(4-cyclopentylpiperazin-1-yl)-1,9-diethyl-N,N-dimethyl-10H-phenothiazin-3-amine
—— [7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3R,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C33H41N7O5
[7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3R,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-Bromo-2-[[4-[4-[tert-butyl(dimethyl)silyl]oxy-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C33H45BrN6O6Si
[7-Bromo-2-[[4-[4-[tert-butyl(dimethyl)silyl]oxy-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— 7-(1-Methylpiperidin-4-yl)quinoline-2-carboxamide —— C16H19N3O
7-(1-Methylpiperidin-4-yl)quinoline-2-carboxamide
—— 7-bromo-2-{[5-(3,5-dichlorophenyl)-2-furyl]methylene}[1,3]thiazolo[2',3':2,3]imidazo[4,5-b]pyridin-3(2H)-one —— C19H8BrCl2N3O2S
7-bromo-2-{[5-(3,5-dichlorophenyl)-2-furyl]methylene}[1,3]thiazolo[2',3':2,3]imidazo[4,5-b]pyridin-3(2H)-one
—— [7-Bromo-2-[[4-[3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C29H32BrN9O5
[7-Bromo-2-[[4-[3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-bromo-2-[[4-[(3R,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C27H28BrF3N6O5
[7-bromo-2-[[4-[(3R,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— 7-Thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1,3,5,8,11-pentaene-10,12-diamine —— C9H8N4S
7-Thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1,3,5,8,11-pentaene-10,12-diamine
—— 7-(1,1,1-Trifluoropropan-2-yl)-8,9-dihydropyrazino[1,2-c]pyrimidine-4,6-dione —— C10H10F3N3O2
7-(1,1,1-Trifluoropropan-2-yl)-8,9-dihydropyrazino[1,2-c]pyrimidine-4,6-dione
—— 7-chloro-4-hydroxy-2-methylimino-5-phenyl-3H-1,4-benzodiazepine-3-thiol —— C16H14ClN3OS
7-chloro-4-hydroxy-2-methylimino-5-phenyl-3H-1,4-benzodiazepine-3-thiol
—— 7H-pyrazino[1,2-c]pyrimidine-4,6-dione —— C7H5N3O2
7H-pyrazino[1,2-c]pyrimidine-4,6-dione
—— 7-[(R)-(3-phenoxyphenyl)-(pyridin-2-ylamino)methyl]quinolin-8-ol —— C27H21N3O2
7-[(R)-(3-phenoxyphenyl)-(pyridin-2-ylamino)methyl]quinolin-8-ol
—— [7-ethenyl-2-[[4-[(3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C28H32N6O5
[7-ethenyl-2-[[4-[(3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-bromo-2-[[4-[(3R,5S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C27H28BrF3N6O5
[7-bromo-2-[[4-[(3R,5S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-bromo-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C29H32BrN9O5
[7-bromo-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-ethenyl-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C31H35N9O5
[7-ethenyl-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-(3,6-dihydro-2H-pyran-4-yl)-2-[[4-[(3S,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C32H35F3N6O6
[7-(3,6-dihydro-2H-pyran-4-yl)-2-[[4-[(3S,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-formyl-2-[[4-[(3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C27H30N6O6
[7-formyl-2-[[4-[(3S)-3-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— 7-[(R)-(2,5-dimethylphenyl)-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol —— C24H23N3O
7-[(R)-(2,5-dimethylphenyl)-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol
—— 7-[(S)-(3-phenoxyphenyl)-(pyridin-2-ylamino)methyl]quinolin-8-ol —— C27H21N3O2
7-[(S)-(3-phenoxyphenyl)-(pyridin-2-ylamino)methyl]quinolin-8-ol
—— [7-(3,6-dihydro-2H-pyran-4-yl)-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C34H39N9O6
[7-(3,6-dihydro-2H-pyran-4-yl)-2-[[4-[(3S,4S,5R)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]-4-(triazol-1-yl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-bromo-2-[[4-[(3R,5S)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C27H31BrN6O5
[7-bromo-2-[[4-[(3R,5S)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3R,5S)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C33H41N7O5
[7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3R,5S)-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3S,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C33H38F3N7O5
[7-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-[[4-[(3S,5R)-3-[(2-methylpropan-2-yl)oxycarbonylamino]-5-(trifluoromethyl)piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid
—— [7-bromo-2-[[4-[(3S,4R,5R)-4-[tert-butyl(dimethyl)silyl]oxy-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid —— C33H45BrN6O6Si
[7-bromo-2-[[4-[(3S,4R,5R)-4-[tert-butyl(dimethyl)silyl]oxy-3-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]piperidin-1-yl]pyridin-3-yl]carbamoyl]quinolin-3-yl]carbamic acid