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—— (7R)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(2-methoxyethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H35N3O4S
(7R)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(2-methoxyethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[benzyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C29H33N3O3S
(7S)-2-[[benzyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-2-hydroxy-3-propan-2-yloxypropyl]-methylamino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H29N3O3S
(7S)-2-[[[(2S)-2-hydroxy-3-propan-2-yloxypropyl]-methylamino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2R)-3-ethoxy-2-hydroxypropyl]-(furan-2-ylmethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N3O4S
(7R)-2-[[[(2R)-3-ethoxy-2-hydroxypropyl]-(furan-2-ylmethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2R)-2-hydroxy-3-methylbutyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H36N4O3S
(7S)-2-[[[(2R)-2-hydroxy-3-methylbutyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-2-hydroxy-3-propan-2-yloxypropyl]-(2-methoxyethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H33N3O4S
(7R)-2-[[[(2S)-2-hydroxy-3-propan-2-yloxypropyl]-(2-methoxyethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-2-hydroxy-3-(2-methylpropoxy)propyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H40N4O4S
(7R)-2-[[[(2S)-2-hydroxy-3-(2-methylpropoxy)propyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2R)-2-hydroxy-3-methylbutyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H36N4O3S
(7R)-2-[[[(2R)-2-hydroxy-3-methylbutyl]-(2-morpholin-4-ylethyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7,7-Dimethyl-1-(4-methylphenyl)-2-pyridin-3-yl-4,4-bis(trifluoromethyl)-6,8-dihydroquinazolin-5-one —— C24H21F6N3O
7,7-Dimethyl-1-(4-methylphenyl)-2-pyridin-3-yl-4,4-bis(trifluoromethyl)-6,8-dihydroquinazolin-5-one
—— (7R)-7-methyl-2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H21N5O4S2
(7R)-7-methyl-2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H21N5O4S2
(7S)-7-methyl-2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-(3-chloropropylsulfonyl)-3,4-dihydro-2H-1,5-benzodioxepine —— C12H15ClO4S
7-(3-chloropropylsulfonyl)-3,4-dihydro-2H-1,5-benzodioxepine
—— 7-Amino-5-[5-(4-chlorophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11ClN4O3S
7-Amino-5-[5-(4-chlorophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-4-oxo-5-(5-phenylfuran-2-yl)-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H12N4O3S
7-Amino-4-oxo-5-(5-phenylfuran-2-yl)-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(2,5-dichlorophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H10Cl2N4O4
7-Amino-5-[5-(2,5-dichlorophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(2,5-dichlorophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H10Cl2N4O3S
7-Amino-5-[5-(2,5-dichlorophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-chlorophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11ClN4O4
7-Amino-5-[5-(4-chlorophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(3-nitrophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11N5O5S
7-Amino-5-[5-(3-nitrophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-methylphenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C19H14N4O3S
7-Amino-5-[5-(4-methylphenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-bromophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11BrN4O4
7-Amino-5-[5-(4-bromophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-methylphenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C19H14N4O4
7-Amino-5-[5-(4-methylphenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-methoxyphenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C19H14N4O5
7-Amino-5-[5-(4-methoxyphenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-(2-chloroethylsulfonyl)-3,4-dihydro-2H-1,5-benzodioxepine —— C11H13ClO4S
7-(2-chloroethylsulfonyl)-3,4-dihydro-2H-1,5-benzodioxepine
—— 7-Amino-5-[5-(3-nitrophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11N5O6
7-Amino-5-[5-(3-nitrophenyl)furan-2-yl]-2,4-dioxo-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-2,4-dioxo-5-(5-phenylfuran-2-yl)-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H12N4O4
7-Amino-2,4-dioxo-5-(5-phenylfuran-2-yl)-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-Amino-5-[5-(4-bromophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile —— C18H11BrN4O3S
7-Amino-5-[5-(4-bromophenyl)furan-2-yl]-4-oxo-2-sulfanylidene-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile
—— 7-amino-1-[(3R)-3-ethylpiperidin-1-yl]heptan-1-one —— C14H28N2O
7-amino-1-[(3R)-3-ethylpiperidin-1-yl]heptan-1-one
—— (7R,8S)-7-[(3S)-3-ethylpiperidin-1-yl]-1,4-dioxaspiro[4.5]decan-8-amine —— C15H28N2O2
(7R,8S)-7-[(3S)-3-ethylpiperidin-1-yl]-1,4-dioxaspiro[4.5]decan-8-amine
—— 7-(3-chlorophenyl)-5-(4-fluorophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H12ClFN4
7-(3-chlorophenyl)-5-(4-fluorophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(7-azaniumyl-5-azaspiro[2.4]heptan-5-yl)-8-chloro-6-fluoro-1-(2-fluorocyclopropyl)-4-oxoquinoline-3-carboxylate —— C19H18ClF2N3O3
7-(7-azaniumyl-5-azaspiro[2.4]heptan-5-yl)-8-chloro-6-fluoro-1-(2-fluorocyclopropyl)-4-oxoquinoline-3-carboxylate
—— (7S)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C28H37N3O3S
(7S)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[ethyl(methyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C15H21N3OS
(7R)-2-[[ethyl(methyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H33N3O5S
(7S)-2-[[[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2R)-2-hydroxy-2-phenylethyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H31N3O3S
(7R)-2-[[[(2R)-2-hydroxy-2-phenylethyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-2-hydroxy-3-phenoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H33N3O4S
(7R)-2-[[[(2S)-2-hydroxy-3-phenoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2R)-2-hydroxy-2-phenylethyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H31N3O3S
(7S)-2-[[[(2R)-2-hydroxy-2-phenylethyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-propan-2-yloxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H37N3O3S
(7S)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-propan-2-yloxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-2-hydroxy-3-phenoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H33N3O4S
(7S)-2-[[[(2S)-2-hydroxy-3-phenoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2R)-2-hydroxy-3-phenylpropyl]-(3-methylbutyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H35N3O2S
(7S)-2-[[[(2R)-2-hydroxy-3-phenylpropyl]-(3-methylbutyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H37N3O4S
(7S)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H33N3O5S
(7R)-2-[[[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-3-(4-chlorophenoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H32ClN3O4S
(7S)-2-[[[(2S)-3-(4-chlorophenoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2S)-2-hydroxy-3-prop-2-ynoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H31N3O4S
(7S)-2-[[[(2S)-2-hydroxy-3-prop-2-ynoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-3-(4-chlorophenoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H32ClN3O4S
(7R)-2-[[[(2S)-3-(4-chlorophenoxy)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[ethyl(methyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C15H21N3OS
(7S)-2-[[ethyl(methyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-2-hydroxy-3-prop-2-ynoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H31N3O4S
(7R)-2-[[[(2S)-2-hydroxy-3-prop-2-ynoxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H37N3O4S
(7R)-2-[[[(2S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxy]propyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C28H37N3O3S
(7R)-2-[[cyclohexyl-[(2S)-2-hydroxy-3-phenylmethoxypropyl]amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[[(2R)-2-hydroxypentyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H33N3O3S
(7R)-2-[[[(2R)-2-hydroxypentyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[[(2R)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H29N3O3S
(7S)-2-[[[(2R)-2-hydroxypropyl]-(3-methoxypropyl)amino]methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one