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—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O3S
(7R)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3S
(7R)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3S
(7S)-7-(3,4-dimethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-ethoxy-3-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O3S
(7R)-7-(4-ethoxy-3-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O2S
(7R)-7-(4-butoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(3a,4,5,6,7,7a-Hexahydropyrrolo[2,3-b]pyridin-1-ylmethyl)-1,5,6,7a-tetrahydropyrrolo[2,3-b]pyridine —— C15H22N4
7-(3a,4,5,6,7,7a-Hexahydropyrrolo[2,3-b]pyridin-1-ylmethyl)-1,5,6,7a-tetrahydropyrrolo[2,3-b]pyridine
—— (7R)-2-ethylsulfanyl-7-(4-methoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7R)-2-ethylsulfanyl-7-(4-methoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5O2S
(7S)-2-ethylsulfanyl-7-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7S)-2-ethylsulfanyl-7-(3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5OS
(7R)-2-ethylsulfanyl-5-methyl-N,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H21N5OS2
(7S)-2-ethylsulfanyl-5-methyl-7-(3-methylthiophen-2-yl)-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7R)-2-ethylsulfanyl-7-(3-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(2-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7R)-2-ethylsulfanyl-7-(2-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7R)-7-(4-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-7-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5OS
(7S)-2-ethylsulfanyl-5-methyl-N,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H15FN6O
7-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (7R)-7-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7R)-7-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5OS2
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(4-methoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7S)-2-ethylsulfanyl-7-(4-methoxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7S)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26N6OS
(7S)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26N6OS
(7R)-7-[4-(dimethylamino)phenyl]-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7R)-7-(3-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20ClN5OS
(7R)-7-(3-chlorophenyl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromofuran-2-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H18BrN5O2S
(7R)-7-(5-bromofuran-2-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5OS2
(7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(4-fluorophenyl)-N-phenylpyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H13FN4O
7-(4-fluorophenyl)-N-phenylpyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2S
(7R)-2-ethylsulfanyl-5-methyl-N-phenyl-7-(3-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5O2S
(7R)-2-ethylsulfanyl-7-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(3-fluorophenyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C18H15FN6O
7-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(3-fluorophenyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 7-(difluoromethyl)-N-[1-(3-fluorobenzyl)-1H-1,2,4-triazol-3-yl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H18F3N7O2
7-(difluoromethyl)-N-[1-(3-fluorobenzyl)-1H-1,2,4-triazol-3-yl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(4-fluorophenyl)-N-(2-methylpropyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C17H17FN4O
7-(4-fluorophenyl)-N-(2-methylpropyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (7R)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7R)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— [7-hydroxy-1-[methyl-(4-methylphenyl)sulfonylamino]-2,3,5,6,7,8-hexahydro-1H-pyrrolizin-2-yl] methanesulfonate —— C16H24N2O6S2
[7-hydroxy-1-[methyl-(4-methylphenyl)sulfonylamino]-2,3,5,6,7,8-hexahydro-1H-pyrrolizin-2-yl] methanesulfonate
—— 7-(difluoromethyl)-N-[7-(morpholin-4-yl)-2,1,3-benzoxadiazol-4-yl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H19F2N7O3
7-(difluoromethyl)-N-[7-(morpholin-4-yl)-2,1,3-benzoxadiazol-4-yl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-2-butylsulfanyl-5-methyl-N-phenyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7S)-2-butylsulfanyl-5-methyl-N-phenyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7S)-2-butylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7S)-2-butylsulfanyl-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxy-3-ethoxyphenyl)-2-butylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7S)-7-(4-butoxy-3-ethoxyphenyl)-2-butylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-2-butylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(3,4-diethoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-2-butylsulfanyl-7-(3,4-diethoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O2S
(7S)-2-butylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide