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—— 7-methyl-3-oxo-N-phenyl-2-(1H-pyrrol-2-ylmethylidene)-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C23H18N4O2S2
7-methyl-3-oxo-N-phenyl-2-(1H-pyrrol-2-ylmethylidene)-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 7-[(S)-cyclohexyl(hydroxy)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H23NO2
7-[(S)-cyclohexyl(hydroxy)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(S)-hydroxy-(4-methylphenyl)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C18H19NO2
7-[(S)-hydroxy-(4-methylphenyl)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-methyl-2-[1-(5-methyl-3-nitro-1H-pyrazol-1-yl)ethyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C13H13N9O2
7-methyl-2-[1-(5-methyl-3-nitro-1H-pyrazol-1-yl)ethyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-[(1S)-1-hydroxybutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C14H19NO2
7-[(1S)-1-hydroxybutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(1R)-1-hydroxybutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C14H19NO2
7-[(1R)-1-hydroxybutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(1R)-1-hydroxy-2-phenylethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C18H19NO2
7-[(1R)-1-hydroxy-2-phenylethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(S)-furan-2-yl(hydroxy)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C15H15NO3
7-[(S)-furan-2-yl(hydroxy)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(R)-hydroxy(phenyl)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H17NO2
7-[(R)-hydroxy(phenyl)methyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(1S)-1-hydroxy-2-phenylethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C18H19NO2
7-[(1S)-1-hydroxy-2-phenylethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(S)-(4-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H16ClNO2
7-[(S)-(4-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(1S)-1-hydroxypentyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C15H21NO2
7-[(1S)-1-hydroxypentyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(S)-(4-fluorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H16FNO2
7-[(S)-(4-fluorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(1S)-2,2,2-trifluoro-1-hydroxyethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C12H12F3NO2
7-[(1S)-2,2,2-trifluoro-1-hydroxyethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-Methyl-2-(5-methyl-1H-pyrazol-3-YL)-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C11H10N8
7-Methyl-2-(5-methyl-1H-pyrazol-3-YL)-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-[(S)-(3-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H16ClNO2
7-[(S)-(3-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(R)-(3-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H16ClNO2
7-[(R)-(3-chlorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(R)-(4-fluorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C17H16FNO2
7-[(R)-(4-fluorophenyl)-hydroxymethyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-Methyl-2-[1-(3-methyl-1H-pyrazol-1-YL)ethyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C13H14N8
7-Methyl-2-[1-(3-methyl-1H-pyrazol-1-YL)ethyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-[(1S)-1-hydroxy-3-methylbutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C15H21NO2
7-[(1S)-1-hydroxy-3-methylbutyl]-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-(Difluoromethyl)-5-(3,4-dimethylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C14H12F2N4
7-(Difluoromethyl)-5-(3,4-dimethylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-Phenyl-2-{[3-(2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C24H24N10
7-Phenyl-2-{[3-(2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-methyl-2-{4-[(5-methyl-3-nitro-1H-pyrazol-1-yl)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C18H15N9O2
7-methyl-2-{4-[(5-methyl-3-nitro-1H-pyrazol-1-yl)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-Methyl-2-[3-(5-methyl-2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C19H22N10
7-Methyl-2-[3-(5-methyl-2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-methyl-N-(2-methylphenyl)-3-oxo-2-(1H-pyrrol-2-ylmethylidene)-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C24H20N4O2S2
7-methyl-N-(2-methylphenyl)-3-oxo-2-(1H-pyrrol-2-ylmethylidene)-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 7-methyl-2-{3-[(3-methyl-4-nitrophenoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C21H17N7O3
7-methyl-2-{3-[(3-methyl-4-nitrophenoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-Methyl-2-[1-methyl-5-(trifluoromethyl)-1H-pyrazol-3-YL]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C12H9F3N8
7-Methyl-2-[1-methyl-5-(trifluoromethyl)-1H-pyrazol-3-YL]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-methyl-2-{3-[(2,2,3,3-tetrafluoropropoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C17H14F4N6O
7-methyl-2-{3-[(2,2,3,3-tetrafluoropropoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-difluoromethyl-5-phenyl-1,2,4-triazolo[1,5-a]pyrimidine —— C12H8F2N4
7-difluoromethyl-5-phenyl-1,2,4-triazolo[1,5-a]pyrimidine
—— 7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-2-(1H-pyrrol-2-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C25H22N4O3S
7-methyl-5-(5-methylfuran-2-yl)-N-(2-methylphenyl)-3-oxo-2-(1H-pyrrol-2-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 7-(Difluoromethyl)-5-(4-fluorophenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C12H7F3N4
7-(Difluoromethyl)-5-(4-fluorophenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(Difluoromethyl)-5-(furan-2-yl)[1,2,4]triazolo[1,5-a]pyrimidine —— C10H6F2N4O
7-(Difluoromethyl)-5-(furan-2-yl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-phenyl-2-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C16H9F3N8
7-phenyl-2-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-Methyl-2-(1,2,3,4-tetrahydro-9H-carbazol-9-ylmethyl)-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C20H19N7
7-Methyl-2-(1,2,3,4-tetrahydro-9H-carbazol-9-ylmethyl)-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-methyl-2-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C12H9F3N8
7-methyl-2-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-(Difluoromethyl)-5-(4-methoxyphenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C13H10F2N4O
7-(Difluoromethyl)-5-(4-methoxyphenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-phenyl-2-{4-[(2,2,3,3-tetrafluoropropoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C22H16F4N6O
7-phenyl-2-{4-[(2,2,3,3-tetrafluoropropoxy)methyl]phenyl}-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-methyl-2-[(3-nitro-1H-pyrazol-1-yl)methyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C11H9N9O2
7-methyl-2-[(3-nitro-1H-pyrazol-1-yl)methyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-(difluoromethyl)-2-(1-ethyl-1H-pyrazol-3-yl)-9-phenylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one —— C21H15F2N5OS
7-(difluoromethyl)-2-(1-ethyl-1H-pyrazol-3-yl)-9-phenylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one
—— 7-(Difluoromethyl)-5-(4-methylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C13H10F2N4
7-(Difluoromethyl)-5-(4-methylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-methyl-2-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C11H7F3N8
7-methyl-2-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-Methyl-2-[3-(5-phenyl-2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C24H24N10
7-Methyl-2-[3-(5-phenyl-2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-Methyl-2-{[3-(2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C19H22N10
7-Methyl-2-{[3-(2H-1,2,3,4-tetraazol-2-YL)-1-adamantyl]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-Methyl-2-{[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-YL]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine —— C13H11F3N8
7-Methyl-2-{[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-YL]methyl}-7H-pyrazolo[4,3-E][1,2,4]triazolo[1,5-C]pyrimidine
—— 7-methyl-2-(1-methyl-1H-pyrazol-3-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine —— C11H10N8
7-methyl-2-(1-methyl-1H-pyrazol-3-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
—— 7-(Difluoromethyl)-5-(4-methylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylic acid —— C14H10F2N4O2
7-(Difluoromethyl)-5-(4-methylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylic acid
—— 7-(Difluoromethyl)-5-(3,4-dimethoxyphenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C14H12F2N4O2
7-(Difluoromethyl)-5-(3,4-dimethoxyphenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(Difluoromethyl)-5-(4-ethylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine —— C14H12F2N4
7-(Difluoromethyl)-5-(4-ethylphenyl)[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[({5-[(2,5-Dimethylphenoxy)methyl]furan-2-yl}carbonyl)amino]-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C25H24N4O6S3
7-[({5-[(2,5-Dimethylphenoxy)methyl]furan-2-yl}carbonyl)amino]-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 7-(1-Ethyl-3-methyl-1H-pyrazol-4-yl)-pyrazolo[1,5-a]pyrimidine-2-carboxylic acid —— C13H13N5O2
7-(1-Ethyl-3-methyl-1H-pyrazol-4-yl)-pyrazolo[1,5-a]pyrimidine-2-carboxylic acid