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—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C26H26F2N4O5
6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-(2-morpholin-4-ylethylamino)-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C22H26F2N4O6
6,7-difluoro-N-[(2S)-3-hydroxy-1-(2-morpholin-4-ylethylamino)-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6-(5-chlorothiophen-2-yl)-5-methyl-2-(propylamino)pyridine-3-carbonitrile —— C14H14ClN3S
6-(5-chlorothiophen-2-yl)-5-methyl-2-(propylamino)pyridine-3-carbonitrile
—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C24H24F2N6O5
6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6-(3-fluoro-4-methoxyphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid —— C14H12FNO3S
6-(3-fluoro-4-methoxyphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid
—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C27H28F2N4O6
6,7-difluoro-N-[(2S)-3-hydroxy-1-[4-(2-methoxyphenyl)piperazin-1-yl]-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6-(3,4-difluorophenyl)-2-(propylamino)pyridine-3-carboxylic acid —— C15H14F2N2O2
6-(3,4-difluorophenyl)-2-(propylamino)pyridine-3-carboxylic acid
—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-(3-methoxyanilino)-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C23H21F2N3O6
6,7-difluoro-N-[(2S)-3-hydroxy-1-(3-methoxyanilino)-1-oxopropan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(1,2,4-triazol-4-ylamino)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide —— C18H16F2N6O5
6,7-difluoro-N-[(2S)-3-hydroxy-1-oxo-1-(1,2,4-triazol-4-ylamino)propan-2-yl]-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-[4-(4-nitrophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C27H34N4O7
6-hydroxy-N-[(2S)-3-hydroxy-1-[4-(4-nitrophenyl)piperazin-1-yl]-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-(2-morpholin-4-ylethylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C23H35N3O6
6-hydroxy-N-[(2S)-3-hydroxy-1-(2-morpholin-4-ylethylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-(1H-indazol-6-ylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C24H28N4O5
6-hydroxy-N-[(2S)-3-hydroxy-1-(1H-indazol-6-ylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C27H35N3O5
6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(quinolin-6-ylamino)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C26H29N3O5
6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(quinolin-6-ylamino)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-[(5-phenyl-1H-pyrazol-3-yl)amino]propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C26H30N4O5
6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-[(5-phenyl-1H-pyrazol-3-yl)amino]propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-(4-methoxyanilino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C24H30N2O6
6-hydroxy-N-[(2S)-3-hydroxy-1-(4-methoxyanilino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-morpholin-4-yl-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C21H30N2O6
6-hydroxy-N-[(2S)-3-hydroxy-1-morpholin-4-yl-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C28H33N3O5
6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-(3-methoxyanilino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C24H30N2O6
6-hydroxy-N-[(2S)-3-hydroxy-1-(3-methoxyanilino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-(1,2-oxazol-3-ylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C20H25N3O6
6-hydroxy-N-[(2S)-3-hydroxy-1-(1,2-oxazol-3-ylamino)-1-oxopropan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(1,2,4-triazol-4-ylamino)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide —— C19H25N5O5
6-hydroxy-N-[(2S)-3-hydroxy-1-oxo-1-(1,2,4-triazol-4-ylamino)propan-2-yl]-2,5,7,8-tetramethyl-3,4-dihydrochromene-2-carboxamide
—— 6-(2,3-dihydro-1H-inden-5-yl)-5-methyl-2-(propan-2-ylamino)pyridine-3-carbonitrile —— C19H21N3
6-(2,3-dihydro-1H-inden-5-yl)-5-methyl-2-(propan-2-ylamino)pyridine-3-carbonitrile
—— 6-(2,4-dimethylphenyl)-2-piperidin-1-ylpyridine-3-carbonitrile —— C19H21N3
6-(2,4-dimethylphenyl)-2-piperidin-1-ylpyridine-3-carbonitrile
—— 6-(4-ethylphenyl)-5-methyl-2-pyrrolidin-1-ylpyridine-3-carbonitrile —— C19H21N3
6-(4-ethylphenyl)-5-methyl-2-pyrrolidin-1-ylpyridine-3-carbonitrile
—— 6-(3,4-dimethylphenyl)-2-piperidin-1-ylpyridine-3-carbonitrile —— C19H21N3
6-(3,4-dimethylphenyl)-2-piperidin-1-ylpyridine-3-carbonitrile
—— 6-[5-(2-aminoethyl)-1,3,4-oxadiazol-2-yl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C12H13N5O2S
6-[5-(2-aminoethyl)-1,3,4-oxadiazol-2-yl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-(4-methoxy-2,5-dimethylphenyl)-2-sulfanylidene-1H-pyridine-3-carboxylic acid —— C15H15NO3S
6-(4-methoxy-2,5-dimethylphenyl)-2-sulfanylidene-1H-pyridine-3-carboxylic acid
—— 6-(2,3-dihydro-1H-inden-5-yl)-2-pyrrolidin-1-ylpyridine-3-carbonitrile —— C19H19N3
6-(2,3-dihydro-1H-inden-5-yl)-2-pyrrolidin-1-ylpyridine-3-carbonitrile
—— 6-(4-methoxy-3-methylphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid —— C15H15NO3S
6-(4-methoxy-3-methylphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid
—— 6-(2-methoxy-5-methylphenyl)-2-methylsulfanylpyridine-3-carboxylic acid —— C15H15NO3S
6-(2-methoxy-5-methylphenyl)-2-methylsulfanylpyridine-3-carboxylic acid
—— 6-(2,4-dimethylphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carbothioamide —— C15H16N2S2
6-(2,4-dimethylphenyl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carbothioamide
—— 6-(2,5-difluorophenyl)-2-(2-methoxyethylamino)pyridine-3-carbonitrile —— C15H13F2N3O
6-(2,5-difluorophenyl)-2-(2-methoxyethylamino)pyridine-3-carbonitrile
—— 6-(4-propylphenyl)-2-sulfanylidene-1H-pyridine-3-carbothioamide —— C15H16N2S2
6-(4-propylphenyl)-2-sulfanylidene-1H-pyridine-3-carbothioamide
—— 6-(3,4-dimethoxyphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid —— C15H15NO5
6-(3,4-dimethoxyphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid
—— 6-(2,5-dimethoxyphenyl)-2-(methylamino)pyridine-3-carboxylic acid —— C15H16N2O4
6-(2,5-dimethoxyphenyl)-2-(methylamino)pyridine-3-carboxylic acid
—— 6-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid —— C15H13NO5
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid
—— 6-[4-[(2S)-butan-2-yl]phenyl]-2-sulfanylidene-1H-pyridine-3-carboxylic acid —— C16H17NO2S
6-[4-[(2S)-butan-2-yl]phenyl]-2-sulfanylidene-1H-pyridine-3-carboxylic acid
—— 6-(4-ethoxyphenyl)-5-methyl-2-(methylamino)pyridine-3-carboxylic acid —— C16H18N2O3
6-(4-ethoxyphenyl)-5-methyl-2-(methylamino)pyridine-3-carboxylic acid
—— 6-(2-methoxyphenyl)-2-(propan-2-ylamino)pyridine-3-carboxylic acid —— C16H18N2O3
6-(2-methoxyphenyl)-2-(propan-2-ylamino)pyridine-3-carboxylic acid
—— 6-(2,5-difluorophenyl)-5-methyl-2-(propylamino)pyridine-3-carbonitrile —— C16H15F2N3
6-(2,5-difluorophenyl)-5-methyl-2-(propylamino)pyridine-3-carbonitrile
—— 6-(4-methoxy-2,5-dimethylphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid —— C16H17NO4
6-(4-methoxy-2,5-dimethylphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid
—— 6-[4-[(2S)-butan-2-yl]phenyl]-2-chloro-5-methylpyridine-3-carbonitrile —— C17H17ClN2
6-[4-[(2S)-butan-2-yl]phenyl]-2-chloro-5-methylpyridine-3-carbonitrile
—— 6-(3-methoxyphenyl)-2-(propylamino)pyridine-3-carboxylic acid —— C16H18N2O3
6-(3-methoxyphenyl)-2-(propylamino)pyridine-3-carboxylic acid
—— 6-methyl-4-(4-methylphenyl)-2-oxo-1-propan-2-ylpyridine-3-carboxylic acid —— C17H19NO3
6-methyl-4-(4-methylphenyl)-2-oxo-1-propan-2-ylpyridine-3-carboxylic acid
—— 6-(4-butylphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid —— C17H19NO3
6-(4-butylphenyl)-5-methyl-2-oxo-1H-pyridine-3-carboxylic acid
—— 6-(5-chlorothiophen-2-yl)-2-methylsulfanylpyridine-3-carboxylic acid —— C11H8ClNO2S2
6-(5-chlorothiophen-2-yl)-2-methylsulfanylpyridine-3-carboxylic acid
—— 6-(4-ethylphenyl)-2-(propan-2-ylamino)pyridine-3-carboxylic acid —— C17H20N2O2
6-(4-ethylphenyl)-2-(propan-2-ylamino)pyridine-3-carboxylic acid
—— 6-(5-chlorothiophen-2-yl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid —— C11H8ClNO2S2
6-(5-chlorothiophen-2-yl)-5-methyl-2-sulfanylidene-1H-pyridine-3-carboxylic acid
—— 6-(4-butylphenyl)-2-(methylamino)pyridine-3-carboxylic acid —— C17H20N2O2
6-(4-butylphenyl)-2-(methylamino)pyridine-3-carboxylic acid
—— 6-(3,4-difluorophenyl)-2-pyrrolidin-1-ylpyridine-3-carbonitrile —— C16H13F2N3
6-(3,4-difluorophenyl)-2-pyrrolidin-1-ylpyridine-3-carbonitrile