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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-fluoro-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]-1H-benzimidazole-4-carboxamide —— C17H13F4N3O2
6-fluoro-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]-1H-benzimidazole-4-carboxamide
—— 6-fluoro-N-[4-(pyridin-3-ylmethylsulfanyl)phenyl]-1H-benzimidazole-4-carboxamide —— C20H15FN4OS
6-fluoro-N-[4-(pyridin-3-ylmethylsulfanyl)phenyl]-1H-benzimidazole-4-carboxamide
—— 6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H40Cl2N4O5
6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H51N3O5
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-methyl-5-[2-oxo-2-[(2S)-2-thiophen-3-ylpyrrolidin-1-yl]ethyl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H20N4O2S
6-methyl-5-[2-oxo-2-[(2S)-2-thiophen-3-ylpyrrolidin-1-yl]ethyl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— (6-fluoro-1H-benzimidazol-4-yl)-[4-(2-nitrophenyl)piperazin-1-yl]methanone —— C18H16FN5O3
(6-fluoro-1H-benzimidazol-4-yl)-[4-(2-nitrophenyl)piperazin-1-yl]methanone
—— 6-fluoro-N-[3-[[5-(trifluoromethyl)pyridin-2-yl]amino]propyl]-1H-benzimidazole-4-carboxamide —— C17H15F4N5O
6-fluoro-N-[3-[[5-(trifluoromethyl)pyridin-2-yl]amino]propyl]-1H-benzimidazole-4-carboxamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H42N4O5S2
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H51N3O5
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C36H47N3O5
6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-[(1R)-1-phenylethoxy]-N-(1H-pyrazol-5-ylmethyl)pyridine-3-carboxamide —— C18H18N4O2
6-[(1R)-1-phenylethoxy]-N-(1H-pyrazol-5-ylmethyl)pyridine-3-carboxamide
—— 6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H42N4O5S2
6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-fluoro-N-[3-[(2-oxopyrrolidin-1-yl)methyl]phenyl]-1H-benzimidazole-4-carboxamide —— C19H17FN4O2
6-fluoro-N-[3-[(2-oxopyrrolidin-1-yl)methyl]phenyl]-1H-benzimidazole-4-carboxamide
—— 6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H43N3O6S
6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H43N3O6S
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H42N4O5S2
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C32H39N3O6S
6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C30H38N4O5S2
6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H53N3O5
6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H43N3O6S
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H49N3O5
6-acetamido-N-[[2-[4-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-fluoro-N'-[3-methoxy-4-(3-methylbutoxy)benzoyl]-1H-benzimidazole-4-carbohydrazide —— C21H23FN4O4
6-fluoro-N'-[3-methoxy-4-(3-methylbutoxy)benzoyl]-1H-benzimidazole-4-carbohydrazide
—— 6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H53N3O5
6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H49N3O5
6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H53N3O5
6-acetamido-N-[[2-[4-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C34H47N3O5
6-acetamido-N-[3-[(2S,4S,6R)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C35H45N3O5
6-acetamido-N-[[4-[(2S,4S,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C39H51N3O6
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H44N4O5
6-acetamido-N-[[3-[4-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C35H42N6O5S
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C33H38N4O5
6-acetamido-N-[3-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C29H38N6O5S
6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H40N4O5
6-acetamido-N-[[4-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H44N4O5
6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C35H42N6O5S
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C29H37N5O5S
6-acetamido-N-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— (6-imidazol-1-ylpyridin-3-yl)-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone —— C17H17N5O2
(6-imidazol-1-ylpyridin-3-yl)-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methanone
—— 6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H43N5O5S
6-acetamido-N-[[3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C37H44N4O5S
6-acetamido-N-[[2-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-enylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H23N3O2
6-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-enylamino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[[methyl-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]amino]methyl]-1H-pyrimidine-2,4-dione —— C15H19N3O3
6-[[methyl-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]amino]methyl]-1H-pyrimidine-2,4-dione
—— 6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C33H47N3O6
6-acetamido-N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-[[(4-tert-butylphenyl)methyl-methylamino]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C24H27N5O
6-[[(4-tert-butylphenyl)methyl-methylamino]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-ethyl-7-hydroxy-4-[[propan-2-yl(pyridin-2-ylmethyl)amino]methyl]chromen-2-one —— C21H24N2O3
6-ethyl-7-hydroxy-4-[[propan-2-yl(pyridin-2-ylmethyl)amino]methyl]chromen-2-one
—— 6-(furan-2-yl)-3-methyl-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C16H16N4O4
6-(furan-2-yl)-3-methyl-N-[(2S)-1-(methylamino)-1-oxopropan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6S)-N-(2-imidazol-1-ylethyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H19N3OS
(6S)-N-(2-imidazol-1-ylethyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C18H21N5O2
6-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C19H23N5O
6-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H43N5O5S
6-acetamido-N-[[3-[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H53N3O5
6-acetamido-N-[[3-[3-[(2S,4S,6R)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide