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—— 6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C36H47N3O6
6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-[[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]amino]-2H-1,2,4-triazine-3,5-dione —— C10H19N5O2
6-[[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]amino]-2H-1,2,4-triazine-3,5-dione
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C37H49N3O6
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H53N3O6
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H50N6O5
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C37H49N3O6
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-[[(2S)-1-(ethylamino)-1-oxopropan-2-yl]amino]pyridazine-3-carboxylic acid —— C10H14N4O3
6-[[(2S)-1-(ethylamino)-1-oxopropan-2-yl]amino]pyridazine-3-carboxylic acid
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H53N3O6
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H53N3O6
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H50N6O5
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-chloro-N-[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]pyridine-3-carboxamide —— C13H20ClN3O
6-chloro-N-[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]pyridine-3-carboxamide
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C35H46N6O5
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-amino-1-[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]pyrimidine-2,4-dione —— C11H20N4O2
6-amino-1-[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]pyrimidine-2,4-dione
—— 6-amino-1-[(1R)-1-(5-methylfuran-2-yl)ethyl]pyrimidine-2,4-dione —— C11H13N3O3
6-amino-1-[(1R)-1-(5-methylfuran-2-yl)ethyl]pyrimidine-2,4-dione
—— 6-[[(1R)-1-(5-methylfuran-2-yl)ethyl]amino]pyridine-3-carbothioamide —— C13H15N3OS
6-[[(1R)-1-(5-methylfuran-2-yl)ethyl]amino]pyridine-3-carbothioamide
—— 6-chloro-N-[(2S)-1-(dimethylamino)-3-methylbutan-2-yl]pyridazine-3-carboxamide —— C12H19ClN4O
6-chloro-N-[(2S)-1-(dimethylamino)-3-methylbutan-2-yl]pyridazine-3-carboxamide
—— 6-[[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]amino]-6-oxohexanoic acid —— C13H26N2O3
6-[[(2R)-1-(dimethylamino)-3-methylbutan-2-yl]amino]-6-oxohexanoic acid
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C36H52N4O5
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H56N4O5
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-[[(1S)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridine-3-carbothioamide —— C13H15N3S2
6-[[(1S)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridine-3-carbothioamide
—— 6-[[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridine-3-carbothioamide —— C13H15N3S2
6-[[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]pyridine-3-carbothioamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H56N4O5
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-amino-1-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyrimidine-2,4-dione —— C11H13N3O2S
6-amino-1-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyrimidine-2,4-dione
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H57N3O5
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C37H53N3O5
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-methyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyridazin-3-amine —— C12H15N3S
6-methyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyridazin-3-amine
—— 6-amino-1-[(2R)-1-thiophen-3-ylpropan-2-yl]pyrimidine-2,4-dione —— C11H13N3O2S
6-amino-1-[(2R)-1-thiophen-3-ylpropan-2-yl]pyrimidine-2,4-dione
—— 6-amino-1-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyrimidine-2,4-dione —— C11H13N3O2S
6-amino-1-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyrimidine-2,4-dione
—— 6-methyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyridazin-3-amine —— C12H15N3S
6-methyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyridazin-3-amine
—— 6-amino-1-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyrimidine-2,4-dione —— C11H18N4O2
6-amino-1-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyrimidine-2,4-dione
—— 6-acetamido-N-[[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H47N3O7
6-acetamido-N-[[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C43H57N3O5
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C36H51N3O5
6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-methyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyridin-2-amine —— C13H16N2S
6-methyl-N-[(1S)-1-(5-methylthiophen-2-yl)ethyl]pyridin-2-amine
—— 6-ethyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyrimidin-4-amine —— C13H17N3S
6-ethyl-N-[(1R)-1-(5-methylthiophen-2-yl)ethyl]pyrimidin-4-amine
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H42N2O6S
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-chloro-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyridazin-3-amine —— C11H17ClN4
6-chloro-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyridazin-3-amine
—— (6R)-4-(5-fluoroquinazolin-4-yl)-2,2,6-trimethylmorpholine —— C15H18FN3O
(6R)-4-(5-fluoroquinazolin-4-yl)-2,2,6-trimethylmorpholine
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H46N2O6S
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H46N2O6S
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H51N3O7
6-acetamido-N-[[2-[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H46N2O6S
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide —— C34H44N4O5
6-acetamido-N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C30H36Cl2N4O5
6-acetamido-N-[[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H50N4O5
6-acetamido-N-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C36H40Cl2N4O5
6-acetamido-N-[[3-[4-[(2R,4R,6S)-4-[(4,5-dichloroimidazol-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C35H46N4O5
6-acetamido-N-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H50N4O5
6-acetamido-N-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6S)-2,2,6-trimethyl-4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)morpholine —— C13H19N5O
(6S)-2,2,6-trimethyl-4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)morpholine
—— 6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C41H50N4O5
6-acetamido-N-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide