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—— 5-[[(2S)-2-[2-(1-methylimidazol-2-yl)ethyl]piperidin-1-yl]methyl]-3-(4-methylphenyl)-1,2-oxazole —— C22H28N4O
5-[[(2S)-2-[2-(1-methylimidazol-2-yl)ethyl]piperidin-1-yl]methyl]-3-(4-methylphenyl)-1,2-oxazole
—— 5-[2-[4-[(1S)-1-hydroxy-3-methylbutyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C16H25N3O4
5-[2-[4-[(1S)-1-hydroxy-3-methylbutyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5-phenyl-1,2-oxazol-3-yl)-[(3R)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone —— C21H21N3O3
(5-phenyl-1,2-oxazol-3-yl)-[(3R)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methanone
—— 5-chloro-2-methoxy-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]benzamide —— C21H21ClN4O2
5-chloro-2-methoxy-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]benzamide
—— 5-[2-[4-[(1R)-1-hydroxy-3-methylbutyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C16H25N3O4
5-[2-[4-[(1R)-1-hydroxy-3-methylbutyl]piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— 5-[[(2R)-2-[2-(1-methylimidazol-2-yl)ethyl]piperidin-1-yl]methyl]-3-(4-methylphenyl)-1,2-oxazole —— C22H28N4O
5-[[(2R)-2-[2-(1-methylimidazol-2-yl)ethyl]piperidin-1-yl]methyl]-3-(4-methylphenyl)-1,2-oxazole
—— 5-[1-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C20H19N7S
5-[1-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— 5-[1-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C20H19N7S
5-[1-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— (5S)-5-benzyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]imidazolidine-2,4-dione —— C21H22N4O5
(5S)-5-benzyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]imidazolidine-2,4-dione
—— 5-[1-[(1R)-1-(5-methylpyridin-2-yl)ethyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(1R)-1-(5-methylpyridin-2-yl)ethyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— 5-(1,5-dimethylpyrazol-4-yl)-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-1,2-oxazole-3-carboxamide —— C18H24N4O4
5-(1,5-dimethylpyrazol-4-yl)-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-1,2-oxazole-3-carboxamide
—— 5-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C20H25N3O3
5-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— (5S)-5-butyl-1-(3-chlorophenyl)-4-(5-methyl-1H-imidazole-2-carbonyl)piperazin-2-one —— C19H23ClN4O2
(5S)-5-butyl-1-(3-chlorophenyl)-4-(5-methyl-1H-imidazole-2-carbonyl)piperazin-2-one
—— 5-[2-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H21N5O3
5-[2-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5R)-5-butyl-1-(3-chlorophenyl)-4-(5-methyl-1H-imidazole-2-carbonyl)piperazin-2-one —— C19H23ClN4O2
(5R)-5-butyl-1-(3-chlorophenyl)-4-(5-methyl-1H-imidazole-2-carbonyl)piperazin-2-one
—— 5-[2-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H21N5O3
5-[2-[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— 5-[4-[(1R)-1-hydroxy-3-phenylpropyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C20H25N3O3
5-[4-[(1R)-1-hydroxy-3-phenylpropyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— 5-(1,5-dimethylpyrazol-4-yl)-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-1,2-oxazole-3-carboxamide —— C18H24N4O4
5-(1,5-dimethylpyrazol-4-yl)-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-1,2-oxazole-3-carboxamide
—— 5-[4-[[(6R)-6-hydroxy-1,4-oxazepan-6-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one —— C15H25N5O3
5-[4-[[(6R)-6-hydroxy-1,4-oxazepan-6-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one
—— 5-fluoro-2-methyl-N-[[(3S)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]benzamide —— C18H21FN4O2
5-fluoro-2-methyl-N-[[(3S)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]benzamide
—— 5-fluoro-2-methyl-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]benzamide —— C18H21FN4O2
5-fluoro-2-methyl-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]benzamide
—— 5-chloro-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]thiophene-2-carboxamide —— C14H18ClNO3S
5-chloro-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]thiophene-2-carboxamide
—— 5-[4-[[(6S)-6-hydroxy-1,4-oxazepan-6-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one —— C15H25N5O3
5-[4-[[(6S)-6-hydroxy-1,4-oxazepan-6-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one
—— 5-chloro-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]thiophene-2-carboxamide —— C14H18ClNO3S
5-chloro-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]thiophene-2-carboxamide
—— 5-(imidazol-1-ylmethyl)-2-[(3R)-3-(2-methylphenyl)piperidin-1-yl]pyridine —— C21H24N4
5-(imidazol-1-ylmethyl)-2-[(3R)-3-(2-methylphenyl)piperidin-1-yl]pyridine
—— 5-[(2S)-1-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H22N6O2S
5-[(2S)-1-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one —— C17H25N5O2S
5-butyl-4-ethyl-2-[2-oxo-2-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one
—— 5-chloro-N-[(3S,4S)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide —— C10H13ClN2O3
5-chloro-N-[(3S,4S)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide
—— 5-(imidazol-1-ylmethyl)-2-[(3S)-3-(2-methylphenyl)piperidin-1-yl]pyridine —— C21H24N4
5-(imidazol-1-ylmethyl)-2-[(3S)-3-(2-methylphenyl)piperidin-1-yl]pyridine
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one —— C17H25N5O2S
5-butyl-4-ethyl-2-[2-oxo-2-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one
—— 5-[(2R)-1-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H22N6O2S
5-[(2R)-1-[[5-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl]methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2R)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H21N5OS
5-[(2R)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H21N5OS
5-[(2S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-chloro-N-[2-[di(propan-2-yl)amino]ethyl]-2-methoxybenzamide —— C16H25ClN2O2
5-chloro-N-[2-[di(propan-2-yl)amino]ethyl]-2-methoxybenzamide
—— 5-chloro-N-[(3S,4R)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide —— C10H13ClN2O3
5-chloro-N-[(3S,4R)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide
—— 5-chloro-N-[(3R,4S)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide —— C10H13ClN2O3
5-chloro-N-[(3R,4S)-4-hydroxypyrrolidin-3-yl]-N-methylfuran-2-carboxamide
—— (5Z)-2-cyclopentylimino-5-[[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]methylidene]-1,3-thiazolidin-4-one —— C19H22N4O2S
(5Z)-2-cyclopentylimino-5-[[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]methylidene]-1,3-thiazolidin-4-one
—— 5-[[[2-(4-Cyano-2-ethoxyphenoxy)acetyl]amino]methyl]-2-methoxybenzoate —— C20H19N2O6-
5-[[[2-(4-Cyano-2-ethoxyphenoxy)acetyl]amino]methyl]-2-methoxybenzoate
—— 5-ethyl-3-[(3S)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1,2,4-oxadiazole —— C17H23N3O3
5-ethyl-3-[(3S)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1,2,4-oxadiazole
—— 5-[[(6S)-2-(3-hydroxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C16H25N5O4
5-[[(6S)-2-(3-hydroxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-(4-chloro-2-nitrophenyl)-2-methyl-N-phenylfuran-3-carboxamide —— C18H13ClN2O4
5-(4-chloro-2-nitrophenyl)-2-methyl-N-phenylfuran-3-carboxamide
—— 5-[3-[(3S)-3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C16H17FN2O3
5-[3-[(3S)-3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[[(6S)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H27N5O3
5-[[(6S)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[[(6R)-2-(3-hydroxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C16H25N5O4
5-[[(6R)-2-(3-hydroxypropyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[[(6R)-2-(3-methylbutyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H29N5O3
5-[[(6R)-2-(3-methylbutyl)-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[3-[(3R)-3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C16H17FN2O3
5-[3-[(3R)-3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[[(6R)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H27N5O3
5-[[(6R)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-cyclopropyl-4-ethyl-2-[[4-(3-methylbutyl)piperazin-1-yl]methyl]-1,2,4-triazole-3-thione —— C17H31N5S
5-cyclopropyl-4-ethyl-2-[[4-(3-methylbutyl)piperazin-1-yl]methyl]-1,2,4-triazole-3-thione
—— 5-ethyl-3-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1,2,4-oxadiazole —— C17H23N3O3
5-ethyl-3-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1,2,4-oxadiazole
—— (5R)-4-(6-aminopyridine-3-carbonyl)-5-butyl-1-(3-methylphenyl)piperazin-2-one —— C21H26N4O2
(5R)-4-(6-aminopyridine-3-carbonyl)-5-butyl-1-(3-methylphenyl)piperazin-2-one