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—— 5-acetyl-3-[(2S)-2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one —— C22H26N2O4
5-acetyl-3-[(2S)-2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one
—— 5-methyl-1-[2-oxo-2-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethyl]pyrimidine-2,4-dione —— C17H23N5O3
5-methyl-1-[2-oxo-2-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethyl]pyrimidine-2,4-dione
—— 5-[(2S)-1-[(4-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C21H20N6O
5-[(2S)-1-[(4-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-acetyl-3-[(2R)-2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one —— C22H26N2O4
5-acetyl-3-[(2R)-2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl]-6-methyl-1H-pyridin-2-one
—— 5-[[(3S)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C22H27N5O
5-[[(3S)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— 5-[(2R)-1-[(4-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole —— C21H20N6O
5-[(2R)-1-[(4-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-yl]-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-[[(3R)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine —— C22H27N5O
5-[[(3R)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]-2-(methoxymethyl)pyrimidine
—— 5-[2-[4-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]piperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C18H27N5O2
5-[2-[4-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]piperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(3S)-3-phenylpiperazin-1-yl]ethyl]-1,2,4-triazol-3-one —— C20H29N5O2
5-butyl-4-ethyl-2-[2-oxo-2-[(3S)-3-phenylpiperazin-1-yl]ethyl]-1,2,4-triazol-3-one
—— (5S)-5-benzyl-4-(2-hydroxyacetyl)-1-(2-phenylphenyl)piperazin-2-one —— C25H24N2O3
(5S)-5-benzyl-4-(2-hydroxyacetyl)-1-(2-phenylphenyl)piperazin-2-one
—— 5-[(2-Methoxy-5-nitrophenoxy)methyl]-1-propyltetrazole —— C12H15N5O4
5-[(2-Methoxy-5-nitrophenoxy)methyl]-1-propyltetrazole
—— (5S)-3-[(2-methoxy-5-methylphenyl)methyl]-5-methyl-5-naphthalen-1-ylimidazolidine-2,4-dione —— C23H22N2O3
(5S)-3-[(2-methoxy-5-methylphenyl)methyl]-5-methyl-5-naphthalen-1-ylimidazolidine-2,4-dione
—— [5-[[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]furan-2-yl]methanol —— C16H23N3O2
[5-[[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]furan-2-yl]methanol
—— [5-[[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]furan-2-yl]methanol —— C16H23N3O2
[5-[[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl]furan-2-yl]methanol
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(2R)-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one —— C15H23F3N4O2
5-butyl-4-ethyl-2-[2-oxo-2-[(2R)-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one
—— (5S)-7-[2-(3-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C14H16N4O5
(5S)-7-[2-(3-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-phenyl-3-[[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H21N5O2
5-phenyl-3-[[(2S)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5R)-7-[2-(3-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C14H16N4O5
(5R)-7-[2-(3-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-butyl-4-ethyl-2-[2-oxo-2-[(2S)-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one —— C15H23F3N4O2
5-butyl-4-ethyl-2-[2-oxo-2-[(2S)-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]-1,2,4-triazol-3-one
—— 5-methyl-1-[3-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]phenyl]tetrazole —— C15H16N6O
5-methyl-1-[3-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]phenyl]tetrazole
—— 5-methyl-1-[3-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]phenyl]tetrazole —— C15H16N6O
5-methyl-1-[3-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]phenyl]tetrazole
—— 5-phenyl-3-[[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H21N5O2
5-phenyl-3-[[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— [5-[1-[(4R)-2,2,6-trimethyl-3,4-dihydrochromen-4-yl]imidazol-2-yl]furan-2-yl]methanol —— C20H22N2O3
[5-[1-[(4R)-2,2,6-trimethyl-3,4-dihydrochromen-4-yl]imidazol-2-yl]furan-2-yl]methanol
—— [5-[1-[(4S)-2,2,6-trimethyl-3,4-dihydrochromen-4-yl]imidazol-2-yl]furan-2-yl]methanol —— C20H22N2O3
[5-[1-[(4S)-2,2,6-trimethyl-3,4-dihydrochromen-4-yl]imidazol-2-yl]furan-2-yl]methanol
—— 5-acetyl-6-methyl-3-[(2R)-2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H-pyridin-2-one —— C21H25N3O3
5-acetyl-6-methyl-3-[(2R)-2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H-pyridin-2-one
—— 5-[3-[(2R)-2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C20H24FN3O2
5-[3-[(2R)-2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C16H16N6O3
5-[[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-acetyl-6-methyl-3-[(2S)-2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H-pyridin-2-one —— C21H25N3O3
5-acetyl-6-methyl-3-[(2S)-2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H-pyridin-2-one
—— 5-[3-[(2S)-2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C20H24FN3O2
5-[3-[(2S)-2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C16H16N6O3
5-[[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[(2R)-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18N4O5
5-[(2R)-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (5R)-5-[(3-oxospiro[1,4-dihydroquinoxaline-2,4'-piperidine]-1'-yl)methyl]-1,3-oxazolidin-2-one —— C16H20N4O3
(5R)-5-[(3-oxospiro[1,4-dihydroquinoxaline-2,4'-piperidine]-1'-yl)methyl]-1,3-oxazolidin-2-one
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone —— C20H22N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone
—— 5-[(2S)-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18N4O5
5-[(2S)-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C18H16N4O3
5-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C18H16N4O3
5-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[3-[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C21H27N3O3
5-[3-[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone —— C20H22N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone
—— 5-[3-[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C21H27N3O3
5-[3-[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine —— C20H24N6
5-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine
—— 5-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine —— C20H24N6
5-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine
—— (5S)-5-[(3-oxospiro[1,4-dihydroquinoxaline-2,4'-piperidine]-1'-yl)methyl]-1,3-oxazolidin-2-one —— C16H20N4O3
(5S)-5-[(3-oxospiro[1,4-dihydroquinoxaline-2,4'-piperidine]-1'-yl)methyl]-1,3-oxazolidin-2-one
—— 5-[(2S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H19N5OS
5-[(2S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H19N5OS
5-[(2R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5,6-dimethyl-2-[2-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C19H30N4O3
5,6-dimethyl-2-[2-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 5,6-dimethyl-2-[2-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C19H30N4O3
5,6-dimethyl-2-[2-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 5-[3-[(3R)-3-benzoylpiperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C18H20N2O4
5-[3-[(3R)-3-benzoylpiperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[2-[(2R)-1-(1,3-benzodioxol-5-yl)propan-2-yl]imidazol-1-yl]-1H-pyrimidine-2,4-dione —— C17H16N4O4
5-[2-[(2R)-1-(1,3-benzodioxol-5-yl)propan-2-yl]imidazol-1-yl]-1H-pyrimidine-2,4-dione
—— (5R)-5-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H29N3O3
(5R)-5-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5-methoxy-3-methyl-1H-indol-2-yl)-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone —— C23H27N3O2
(5-methoxy-3-methyl-1H-indol-2-yl)-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone