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—— 5-(4-methylphenyl)-3-[3-oxo-3-[(2S)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one —— C23H26N4O3S
5-(4-methylphenyl)-3-[3-oxo-3-[(2S)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one
—— 5,7-dimethyl-6-[3-oxo-3-[(2S)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile —— C19H24N6O2
5,7-dimethyl-6-[3-oxo-3-[(2S)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
—— 5-[2-[(2S)-2-[(dimethylamino)methyl]piperidin-1-yl]-2-oxoethyl]-6-methyl-2-pyridin-3-yl-1H-pyrimidin-4-one —— C20H27N5O2
5-[2-[(2S)-2-[(dimethylamino)methyl]piperidin-1-yl]-2-oxoethyl]-6-methyl-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 5-[(1R)-1-(4-ethylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C17H23FN4O
5-[(1R)-1-(4-ethylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5,7-dimethyl-6-[3-oxo-3-[(2R)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile —— C19H24N6O2
5,7-dimethyl-6-[3-oxo-3-[(2R)-3-oxo-2-propan-2-ylpiperazin-1-yl]propyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
—— 5-Butyl-1-(3,5-dimethoxy-2-methoxycarbonylphenyl)-3-[(4-hydroxyphenyl)methyl]-4,6-dioxo-1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3-carboxylic acid —— C28H32N2O9
5-Butyl-1-(3,5-dimethoxy-2-methoxycarbonylphenyl)-3-[(4-hydroxyphenyl)methyl]-4,6-dioxo-1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3-carboxylic acid
—— [5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl-[(3,4-dimethoxyphenyl)methyl]-methylazanium —— C20H28N3O5S+
[5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl-[(3,4-dimethoxyphenyl)methyl]-methylazanium
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(2,6-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(2,6-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO4
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-[(1S)-1-(4-ethylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C17H23FN4O
5-[(1S)-1-(4-ethylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-chlorophenyl)-5-oxopyrrolidine-3-carboxylate —— C21H22ClNO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-chlorophenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO4
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-ethoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(3-chloro-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H24ClNO3
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(3-chloro-2-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-naphthalen-1-yl-5-oxopyrrolidine-3-carboxylate —— C25H25NO3
(5-methyl-2-propan-2-ylphenyl) (3S)-1-naphthalen-1-yl-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(3,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(3,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-naphthalen-1-yl-5-oxopyrrolidine-3-carboxylate —— C25H25NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-naphthalen-1-yl-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H25NO4
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3S)-1-(2-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H25NO4
(5-methyl-2-propan-2-ylphenyl) (3S)-1-(2-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(5-chloro-2-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H24ClNO4
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(5-chloro-2-methoxyphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H25NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(4-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-5-oxo-1-[(1S)-1-phenylethyl]pyrrolidine-3-carboxylate —— C23H27NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-5-oxo-1-[(1S)-1-phenylethyl]pyrrolidine-3-carboxylate
—— 5-cyclohexyl-N-prop-2-enyl-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C12H19N3S
5-cyclohexyl-N-prop-2-enyl-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-benzyl-5-oxopyrrolidine-3-carboxylate —— C22H25NO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-benzyl-5-oxopyrrolidine-3-carboxylate
—— (5-methyl-2-propan-2-ylphenyl) (3R)-1-(3-chloro-4-methylphenyl)-5-oxopyrrolidine-3-carboxylate —— C22H24ClNO3
(5-methyl-2-propan-2-ylphenyl) (3R)-1-(3-chloro-4-methylphenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-methyl-6-[2-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H28N4O4
5-methyl-6-[2-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5-bromothiophen-2-yl)methyl-methyl-[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]azanium —— C14H15BrN3OS2+
(5-bromothiophen-2-yl)methyl-methyl-[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]azanium
—— (5-bromothiophen-2-yl)methyl-[(1S)-2-(cyclopropylamino)-2-oxo-1-phenylethyl]-methylazanium —— C17H20BrN2OS+
(5-bromothiophen-2-yl)methyl-[(1S)-2-(cyclopropylamino)-2-oxo-1-phenylethyl]-methylazanium
—— 5-methyl-6-[2-[(4R)-4-methylazepan-1-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H22N4O2
5-methyl-6-[2-[(4R)-4-methylazepan-1-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-6-[2-[(4S)-4-methylazepan-1-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H22N4O2
5-methyl-6-[2-[(4S)-4-methylazepan-1-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5-bromothiophen-2-yl)methyl-methyl-[(1R)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]azanium —— C14H15BrN3OS2+
(5-bromothiophen-2-yl)methyl-methyl-[(1R)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]azanium
—— 5-chloro-2-methoxy-N'-[(2-oxo-1,3-dihydroindol-5-yl)sulfonyl]benzohydrazide —— C16H14ClN3O5S
5-chloro-2-methoxy-N'-[(2-oxo-1,3-dihydroindol-5-yl)sulfonyl]benzohydrazide
—— (5-Bromothiophen-2-yl)methyl-[2-[4-(cyanomethyl)anilino]-2-oxoethyl]-prop-2-enylazanium —— C18H19BrN3OS+
(5-Bromothiophen-2-yl)methyl-[2-[4-(cyanomethyl)anilino]-2-oxoethyl]-prop-2-enylazanium
—— 5-methyl-6-[2-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H28N4O4
5-methyl-6-[2-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-2-oxoethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-chloro-2-[[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]amino]benzamide —— C25H23ClN4O3
5-chloro-2-[[2-[(3R)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]amino]benzamide
—— 5-chloro-2-[[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]amino]benzamide —— C25H23ClN4O3
5-chloro-2-[[2-[(3S)-3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]amino]benzamide
—— 5-(4-methoxyphenyl)-N-[(1-methyl-1H-benzimidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide —— C20H19N5O2
5-(4-methoxyphenyl)-N-[(1-methyl-1H-benzimidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
—— [5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl-[2-(cyclopropylamino)-2-oxoethyl]-methylazanium —— C16H25N4O4S+
[5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl-[2-(cyclopropylamino)-2-oxoethyl]-methylazanium
—— 5-[(1S)-1-phenylethyl]sulfanyl-2-[(1R)-1-phenylethyl]sulfanyl-1,3,4-thiadiazole —— C18H18N2S3
5-[(1S)-1-phenylethyl]sulfanyl-2-[(1R)-1-phenylethyl]sulfanyl-1,3,4-thiadiazole
—— (5-ethoxycarbonyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl)methyl-[(6-methoxynaphthalen-2-yl)methyl]-methylazanium —— C21H26N3O4+
(5-ethoxycarbonyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl)methyl-[(6-methoxynaphthalen-2-yl)methyl]-methylazanium
—— 5-(4-methoxyphenyl)-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C19H18N6O2
5-(4-methoxyphenyl)-N-[(1R)-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5-Bromo-2-ethoxycarbonyl-1-benzofuran-3-yl)methyl-[2-(cyclopropylamino)-2-oxoethyl]-methylazanium —— C18H22BrN2O4+
(5-Bromo-2-ethoxycarbonyl-1-benzofuran-3-yl)methyl-[2-(cyclopropylamino)-2-oxoethyl]-methylazanium
—— 5-nitro-N-[(2R)-1-piperidin-1-ylpropan-2-yl]thiophene-3-carboxamide —— C13H19N3O3S
5-nitro-N-[(2R)-1-piperidin-1-ylpropan-2-yl]thiophene-3-carboxamide
—— 5-nitro-N-[(2S)-1-piperidin-1-ylpropan-2-yl]thiophene-3-carboxamide —— C13H19N3O3S
5-nitro-N-[(2S)-1-piperidin-1-ylpropan-2-yl]thiophene-3-carboxamide
—— 5-bromo-3-methyl-N-[(2S)-1-piperidin-1-ylpropan-2-yl]furan-2-carboxamide —— C14H21BrN2O2
5-bromo-3-methyl-N-[(2S)-1-piperidin-1-ylpropan-2-yl]furan-2-carboxamide
—— 5-chloro-N-[(2R)-1-piperidin-1-ylpropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide —— C17H26ClN5O
5-chloro-N-[(2R)-1-piperidin-1-ylpropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide
—— 5-methyl-1-phenyl-N-[(2S)-1-piperidin-1-ylpropan-2-yl]pyrazole-3-carboxamide —— C19H26N4O
5-methyl-1-phenyl-N-[(2S)-1-piperidin-1-ylpropan-2-yl]pyrazole-3-carboxamide
—— 5-chloro-N-[(2S)-1-piperidin-1-ylpropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide —— C17H26ClN5O
5-chloro-N-[(2S)-1-piperidin-1-ylpropan-2-yl]-2-pyrrolidin-1-ylpyrimidine-4-carboxamide