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—— (5S)-5-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C19H29N3O3
(5S)-5-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(2R)-2-[2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C18H24N6O2
5-[(2R)-2-[2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— 5-[(2S)-2-[2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C18H24N6O2
5-[(2S)-2-[2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— (5S)-4-(2-aminopyridine-4-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one —— C18H20N4O2
(5S)-4-(2-aminopyridine-4-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
—— (5R)-1-(3-chlorophenyl)-4-[2-(3-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one —— C19H19ClN2O3
(5R)-1-(3-chlorophenyl)-4-[2-(3-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one
—— 5-[3-[(3S)-3-benzoylpiperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C18H20N2O4
5-[3-[(3S)-3-benzoylpiperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— (5S)-1-(3-chlorophenyl)-4-[2-(3-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one —— C19H19ClN2O3
(5S)-1-(3-chlorophenyl)-4-[2-(3-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one
—— (5R)-4-(2-aminopyridine-4-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one —— C18H20N4O2
(5R)-4-(2-aminopyridine-4-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
—— 5-[(2S)-oxolan-2-yl]-3-[[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]methyl]-1,2,4-oxadiazole —— C19H18N6O2
5-[(2S)-oxolan-2-yl]-3-[[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(2R)-oxolan-2-yl]-3-[[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]methyl]-1,2,4-oxadiazole —— C19H18N6O2
5-[(2R)-oxolan-2-yl]-3-[[2-(3-pyrazol-1-ylphenyl)imidazol-1-yl]methyl]-1,2,4-oxadiazole
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-methoxypropyl)piperidin-1-yl]methanone —— C18H26N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2R)-2-(3-methoxypropyl)piperidin-1-yl]methanone
—— (5-fluoro-2-methylphenyl)-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone —— C22H26FNO2
(5-fluoro-2-methylphenyl)-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-methoxypropyl)piperidin-1-yl]methanone —— C18H26N4O2
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(2S)-2-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-Amino-1-(5-anilino-1,3,4-thiadiazol-2-yl)-3-(4-nitrophenyl)thieno[3,4-d]pyridazin-4-one —— C20H13N7O3S2
5-Amino-1-(5-anilino-1,3,4-thiadiazol-2-yl)-3-(4-nitrophenyl)thieno[3,4-d]pyridazin-4-one
—— (5-chlorothiophen-2-yl)-[(3S)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C16H22ClN5OS
(5-chlorothiophen-2-yl)-[(3S)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— [5-(methoxymethyl)thiophen-2-yl]-[(3S)-3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C21H23N3O2S
[5-(methoxymethyl)thiophen-2-yl]-[(3S)-3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone —— C20H22FN5O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone
—— [5-(methoxymethyl)thiophen-2-yl]-[(3R)-3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C21H23N3O2S
[5-(methoxymethyl)thiophen-2-yl]-[(3R)-3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5R)-5-[2-(2-oxopyrrolidin-1-yl)ethylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H26N4O3
(5R)-5-[2-(2-oxopyrrolidin-1-yl)ethylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5-methoxy-3-methyl-1H-indol-2-yl)-[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone —— C23H27N3O2
(5-methoxy-3-methyl-1H-indol-2-yl)-[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methanone
—— 5-butyl-2-[2-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-ethyl-1,2,4-triazol-3-one —— C19H30N6O2
5-butyl-2-[2-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-ethyl-1,2,4-triazol-3-one
—— (5-chlorothiophen-2-yl)-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C16H22ClN5OS
(5-chlorothiophen-2-yl)-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— 5-[(2R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H21F2N3O2
5-[(2R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[5-[[(3R)-3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]furan-2-yl]-1H-pyrazole —— C20H23N3O3
5-[5-[[(3R)-3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]furan-2-yl]-1H-pyrazole
—— 5-[(2S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C17H21F2N3O2
5-[(2S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5R)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C18H21N3O3
(5R)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-phenyl-N-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]-1,2-oxazole-3-carboxamide —— C21H18N4O2
5-phenyl-N-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]-1,2-oxazole-3-carboxamide
—— (5S)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione —— C18H21N3O3
(5S)-7-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
—— 5-[5-[[(3S)-3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]furan-2-yl]-1H-pyrazole —— C20H23N3O3
5-[5-[[(3S)-3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl]furan-2-yl]-1H-pyrazole
—— (5-fluoro-2-methylphenyl)-[4-[(1R)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone —— C22H26FNO2
(5-fluoro-2-methylphenyl)-[4-[(1R)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone
—— 5-[(2S)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H21N7O
5-[(2S)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-butyl-2-[2-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-ethyl-1,2,4-triazol-3-one —— C19H30N6O2
5-butyl-2-[2-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl]-4-ethyl-1,2,4-triazol-3-one
—— (5S)-5-[2-(2-oxopyrrolidin-1-yl)ethylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H26N4O3
(5S)-5-[2-(2-oxopyrrolidin-1-yl)ethylamino]-1-propyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole —— C22H22N4O
5-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole
—— 5-[(2R)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H21N7O
5-[(2R)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— (5R)-5-(4-phenylmethoxypiperidine-1-carbonyl)pyrrolidin-2-one —— C17H22N2O3
(5R)-5-(4-phenylmethoxypiperidine-1-carbonyl)pyrrolidin-2-one
—— 5-[(2S)-2-[2-[(3-chloropyridin-2-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C16H20ClN5O2
5-[(2S)-2-[2-[(3-chloropyridin-2-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone —— C20H22FN5O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone
—— (5S)-5-(4-phenylmethoxypiperidine-1-carbonyl)pyrrolidin-2-one —— C17H22N2O3
(5S)-5-(4-phenylmethoxypiperidine-1-carbonyl)pyrrolidin-2-one
—— 5-[(2R)-2-[2-[(3-chloropyridin-2-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one —— C16H20ClN5O2
5-[(2R)-2-[2-[(3-chloropyridin-2-yl)amino]ethyl]morpholin-4-yl]-2-methylpyridazin-3-one
—— 5-[(2S)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1H-pyrimidin-6-one —— C17H20N4O2
5-[(2S)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1H-pyrimidin-6-one
—— 5-[(2R)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1H-pyrimidin-6-one —— C17H20N4O2
5-[(2R)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1H-pyrimidin-6-one
—— 5-phenyl-N-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]-1,2-oxazole-3-carboxamide —— C21H18N4O2
5-phenyl-N-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]-1,2-oxazole-3-carboxamide
—— 5-(3H-indol-2-ylsulfanylmethyl)-3-pyridin-2-yl-1,2,4-oxadiazole —— C16H12N4OS
5-(3H-indol-2-ylsulfanylmethyl)-3-pyridin-2-yl-1,2,4-oxadiazole
—— 5-fluoro-N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyridin-2-amine —— C10H14FN3O
5-fluoro-N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyridin-2-amine
—— 5-[2-[(3S)-3-(4-methoxyphenyl)pyrrolidin-1-yl]pyridin-4-yl]-3-methyl-1,2,4-oxadiazole —— C19H20N4O2
5-[2-[(3S)-3-(4-methoxyphenyl)pyrrolidin-1-yl]pyridin-4-yl]-3-methyl-1,2,4-oxadiazole
—— (5S)-5-methyl-1-(2-methylphenyl)-4-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one —— C17H18N8O2
(5S)-5-methyl-1-(2-methylphenyl)-4-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
—— 5-fluoro-N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyridin-2-amine —— C10H14FN3O
5-fluoro-N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyridin-2-amine
—— 5-[2-[(3R)-3-(4-methoxyphenyl)pyrrolidin-1-yl]pyridin-4-yl]-3-methyl-1,2,4-oxadiazole —— C19H20N4O2
5-[2-[(3R)-3-(4-methoxyphenyl)pyrrolidin-1-yl]pyridin-4-yl]-3-methyl-1,2,4-oxadiazole
—— 5-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole —— C22H22N4O
5-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole